Patent | Date |
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Uses Of Salt-inducible Kinase (sik) Inhibitors For Treating Osteoporosis App 20220305016 - Wein; Marc ;   et al. | 2022-09-29 |
Compounds for the degradation of STK4 and treatment of hematologic malignancies Grant 11,447,467 - Buhrlage , et al. September 20, 2 | 2022-09-20 |
Degraders Of Cyclin-dependent Kinase 7 (cdk7) And Uses Thereof App 20220280649 - Gray; Nathanael S. ;   et al. | 2022-09-08 |
Inhibitors Of Cyclin-dependent Kinase 7 And Uses Thereof App 20220281874 - Zhang; Tinghu ;   et al. | 2022-09-08 |
Small Molecule Inhibitors Of Src Tyrosine Kinase App 20220267294 - Gray; Nathanael S. ;   et al. | 2022-08-25 |
Inhibitors Of Cyclin-dependent Kinases App 20220242865 - Gray; Nathanael S. ;   et al. | 2022-08-04 |
Allosteric Egfr Inhibitors And Methods Of Use Thereof App 20220233545 - Gray; Nathanael S. ;   et al. | 2022-07-28 |
Degraders Of Cyclin-dependent Kinase 12 (cdk12) And Uses Thereof App 20220227734 - Che; Jianwei ;   et al. | 2022-07-21 |
Inhibitors Of Cyclin-dependent Kinase 12 (cdk12) And Uses Thereof App 20220213067 - Gray; Nathanael S. ;   et al. | 2022-07-07 |
Pyrrolopyrimidine Inhibitors Of Wild-type And Mutant Forms Of Lrrk2 App 20220204515 - Gray; Nathanael S. ;   et al. | 2022-06-30 |
Taire Family Kinase Inhibitors And Uses Thereof App 20220169631 - Gray; Nathanael S. ;   et al. | 2022-06-02 |
Inhibitors Of C-jun-n-terminal Kinase (jnk) App 20220153730 - Gray; Nathanael S. ;   et al. | 2022-05-19 |
Inhibitors of cyclin-dependent kinases Grant 11,325,910 - Gray , et al. May 10, 2 | 2022-05-10 |
Uses Of Pyrimidopyrimidinones As Sik Inhibitors App 20220133736 - Fisher; David E. ;   et al. | 2022-05-05 |
Small Molecule Myristate Inhibitors Of Bcr-abl And Methods Of Use App 20220135573 - GRAY; Nathanael S. ;   et al. | 2022-05-05 |
Benzimidazole Derivatives And Aza-benzimidazole Derivatives As Janus Kinase 2 Inhibitors And Uses Thereof App 20220127246 - Gray; Nathanael S. ;   et al. | 2022-04-28 |
Benzothiazole Derivatives And 7-aza-benzothiazole Derivatives As Janus Kinase 2 Inhibitors And Uses Thereof App 20220127284 - Gray; Nathanael S. ;   et al. | 2022-04-28 |
Imidazopyridine Derivatives And Aza-imidazopyridine Derivatives As Janus Kinase 2 Inhibitors And Uses Thereof App 20220127260 - Gray; Nathanael S. ;   et al. | 2022-04-28 |
Inhibitors of cyclin-dependent kinase 12 (CDK12) and uses thereof Grant 11,306,070 - Gray , et al. April 19, 2 | 2022-04-19 |
Macrocyclic Inhibitors Of Dyrk1a App 20220112201 - Gray; Nathanael S. ;   et al. | 2022-04-14 |
Degradation Of Cyclin-dependent Kinase 8 (cdk8) By Conjugation Of Cdk8 Inhibitors With E3 Ligase Ligand And Methods Of Use App 20220112191 - Gray; Nathanael S. ;   et al. | 2022-04-14 |
Inhibitors Of Egfr And/or Her2 And Methods Of Use App 20220106310 - Hatcher; John M. ;   et al. | 2022-04-07 |
Uses of pyrimidopyrimidinones as SIK inhibitors Grant 11,285,158 - Fisher , et al. March 29, 2 | 2022-03-29 |
SMALL MOLECULE DEGRADERS OF FKBP12 VIA RECRUITMENT OF VON HIPPEL-LINDAU E3 UBIQUITIN LIGASE (VHL) E3 UBIQUITIN LIGASE, AND USES IN dTAG SYSTEMS App 20220089589 - Gray; Nathanael S. ;   et al. | 2022-03-24 |
Inhibitors Of Cyclin-dependent Kinase 7 And Uses Thereof App 20220089611 - Gray; Nathanael S. ;   et al. | 2022-03-24 |
NEK inhibitors and methods of use Grant 11,279,707 - Gray , et al. March 22, 2 | 2022-03-22 |
Pyrazolopyridine Inhibitors Of C-jun-n-terminal Kinases And Uses Thereof App 20220073512 - Gray; Nathanael S. ;   et al. | 2022-03-10 |
Compositions And Methods Of Treating Cancers By Administering A Phenothiazine-related Drug That Activates Protein Phosphatase 2a (pp2a) With Reduced Inhibitory Activity Targeted To The Dopamine D2 Receptor And Accompanying Toxicity App 20220062291 - Look; Alfred T. ;   et al. | 2022-03-03 |
Inhibitors Of Cyclin-dependent Kinases App 20220055998 - Gray; Nathanael S. ;   et al. | 2022-02-24 |
Small molecule myristate inhibitors of Bcr-abl and methods of use Grant 11,254,682 - Gray , et al. February 22, 2 | 2022-02-22 |
Degraders Of Wee1 Kinase App 20220047709 - Gray; Nathanael S. ;   et al. | 2022-02-17 |
Inhibitors of MALT1 and uses thereof Grant 11,248,007 - Gray , et al. February 15, 2 | 2022-02-15 |
Degradation of cyclin-dependent kinase 8 (CDK8) by conjugation of CDK8 inhibitors with E3 ligase ligand and methods of use Grant 11,247,991 - Gray , et al. February 15, 2 | 2022-02-15 |
Degradation Of Fak Or Fak And Alk By Conjugation Of Fak And Alk Inhibitors With E3 Ligase Ligands And Methods Of Use App 20220040317 - Gray; Nathanael S. ;   et al. | 2022-02-10 |
Uses of salt-inducible kinase (SIK) inhibitors for treating osteoporosis Grant 11,241,435 - Wein , et al. February 8, 2 | 2022-02-08 |
Macrocyclic Inhibitors Of Alk, Trka, Trkb, And Ros1 App 20220033402 - Gray; Nathanael S. ;   et al. | 2022-02-03 |
Inhibitors Of Cyclin-dependent Kinase 7 (cdk7) App 20220024929 - Gray; Nathanael S. ;   et al. | 2022-01-27 |
Bifunctional Molecules For Degradation Of Egfr And Methods Of Use App 20220017510 - GRAY; NATHANAEL S. ;   et al. | 2022-01-20 |
Inhibitors of EGFR and/or HER2 and methods of use Grant 11,186,574 - Hatcher , et al. November 30, 2 | 2021-11-30 |
Degraders Of Wild-type And Mutant Forms Of Lrrk2 App 20210361774 - Gray; Nathanael S. ;   et al. | 2021-11-25 |
Cyano Quinoline Amide Compounds As Her2 Inhibitors And Methods Of Use App 20210355119 - GRAY; NATHANAEL S. ;   et al. | 2021-11-18 |
Azaindole Inhibitors Of Wild-type And Mutant Forms Of Lrrk2 App 20210347772 - Gray; Nathanael S. ;   et al. | 2021-11-11 |
Inhibitors Of Egfr And Methods Of Use Thereof App 20210346395 - GRAY; NATHANAEL S. ;   et al. | 2021-11-11 |
Degraders Of Hepatitis C Virus Ns3/4a Protein App 20210338825 - Gray; Nathanael S. ;   et al. | 2021-11-04 |
Degradation Of Cyclin-dependent Kinase 4/6 (cdk4/6) By Conjugation Of Cdk4/6 Inhibitors With E3 Ligase Ligand And Methods Of Use App 20210340140 - GRAY; NATHANAEL S. ;   et al. | 2021-11-04 |
Substituted 6,11-dihydro-5h-benzo[b]carbazoles As Inhibitors Of Alk And Srpk App 20210340102 - Hatcher; John ;   et al. | 2021-11-04 |
Modulators Of Pin1 Activity And Uses Thereof App 20210332024 - LONDON; Nir ;   et al. | 2021-10-28 |
Pyrimido-diazepinone kinase scaffold compounds and methods for treating PI3K-mediated disorders Grant 11,155,556 - Gray , et al. October 26, 2 | 2021-10-26 |
Inhibitors Of Cyclin-dependent Kinase 12 (cdk12) And Uses Thereof App 20210317105 - Gray; Nathanael S. ;   et al. | 2021-10-14 |
4,6-pyrimidinylene Derivatives And Uses Thereof App 20210315894 - Gray; Nathanael S. ;   et al. | 2021-10-14 |
Inhibitors of cyclin-dependent kinases Grant 11,142,507 - Gray , et al. October 12, 2 | 2021-10-12 |
Inhibitors Of C-jun-n-terminal Kinase (jnk) App 20210300911 - Gray; Nathanael S. ;   et al. | 2021-09-30 |
Taire Family Kinase Inhibitors And Uses Thereof App 20210292299 - Gray; Nathanael S. ;   et al. | 2021-09-23 |
Degraders That Target Proteins Via Keap1 App 20210276996 - Gray; Nathanael S. ;   et al. | 2021-09-09 |
Inhibitors Of Cyclin-dependent Kinases App 20210261551 - Gray; Nathanael S. ;   et al. | 2021-08-26 |
Irak Degraders And Uses Thereof App 20210230144 - Gray; Nathanael S. ;   et al. | 2021-07-29 |
Compounds For Treating Dengue Virus Infections And Other Infections App 20210230101 - Yang; Priscilla L. ;   et al. | 2021-07-29 |
Uses Of Kinase Inhibitors For Inducing And Maintaining Pluripotency App 20210230538 - Theunissen; Thorold W. ;   et al. | 2021-07-29 |
Substituted 6,11-dihydro-5H-benzo[B]carbazoles as inhibitors of ALK and SRPK Grant 11,066,363 - Hatcher , et al. July 20, 2 | 2021-07-20 |
Pyrimido-diazepinone kinase scaffold compounds and methods of treating DCLK1/2-mediated disorders Grant 11,028,089 - Ferguson , et al. June 8, 2 | 2021-06-08 |
Compounds For Tau Protein Degradation App 20210154184 - Gray; Nathanael S. ;   et al. | 2021-05-27 |
Imidazolyl Kinase Inhibitors And Uses Thereof App 20210147388 - Gray; Nathanael S. ;   et al. | 2021-05-20 |
Bicyclic Urea Kinase Inhibitors And Uses Thereof App 20210147425 - Gray; Nathanael S. ;   et al. | 2021-05-20 |
Heterobifunctional Compounds With Improved Specificity App 20210130368 - NOWAK; Radoslaw P. ;   et al. | 2021-05-06 |
Inhibitors Of Cyclin-dependent Kinase 7 (cdk7) App 20210115051 - Gray; Nathanael S. ;   et al. | 2021-04-22 |
Lrrk2 Inhibitors And Methods Of Making And Using The Same App 20210115055 - Gray; Nathanael S. ;   et al. | 2021-04-22 |
Inhibitors of c-Jun-N-terminal kinase (JNK) Grant 10,981,903 - Gray , et al. April 20, 2 | 2021-04-20 |
Imidazolyl kinase inhibitors and uses thereof Grant 10,975,058 - Gray , et al. April 13, 2 | 2021-04-13 |
Inhibitors of interleukin-1 receptor-associated kinases and uses thereof Grant 10,975,055 - Gray , et al. April 13, 2 | 2021-04-13 |
Degradation Of Bruton's Tyrosine Kinase (btk) By Conjugation Of Btk Inhibitors With E3 Ligase Ligand And Methods Of Use App 20210100908 - Gray; Nathanael S. ;   et al. | 2021-04-08 |
Inhibitors Of Egfr And Methods Of Use Thereof App 20210094913 - GRAY; Nathanael S. ;   et al. | 2021-04-01 |
Pharmaceutical Combinations Of Egfr Inhibitors And Methods Of Use Thereof App 20210085688 - GRAY; NATHANAEL S. ;   et al. | 2021-03-25 |
Bicyclic urea kinase inhibitors and uses thereof Grant 10,954,242 - Gray , et al. March 23, 2 | 2021-03-23 |
Novel Pyrimidines As Egfr Inhibitors And Methods Of Treating Disorders App 20210078977 - GRAY; Nathanael S. ;   et al. | 2021-03-18 |
Pharmaceutical Combinations Of Egfr Inhibitors And Methods Of Use Thereof App 20210077469 - GRAY; NATHANAEL S. ;   et al. | 2021-03-18 |
Cyclin-dependent Kinase Degraders And Methods Of Use App 20210054020 - Gray; Nathanael S. ;   et al. | 2021-02-25 |
Degradation of protein kinases by conjugation of protein kinase inhibitors with E3 ligase ligand and methods of use Grant 10,925,868 - Gray , et al. February 23, 2 | 2021-02-23 |
Degradation of Bruton's tyrosine kinase (BTK) by conjugation of BTK inhibitors with E3 ligase ligand and methods of use Grant 10,925,967 - Gray , et al. February 23, 2 | 2021-02-23 |
Inhibitors Of Egfr And Methods Of Use Thereof App 20210040088 - GRAY; NATHANAEL S. ;   et al. | 2021-02-11 |
Degradation Of Cyclin-dependent Kinase 8 (cdk8) By Conjugation Of Cdk8 Inhibitors With E3 Ligase Ligand And Methods Of Use App 20210040093 - GRAY; Nathanael S. ;   et al. | 2021-02-11 |
LRRK2 inhibitors and methods of making and using the same Grant 10,913,744 - Gray , et al. February 9, 2 | 2021-02-09 |
Degradation Of Bruton's Tyrosine Kinase (btk) By Conjugation Of Btk Inhibitors With E3 Ligase Ligand And Methods Of Use App 20210030832 - Gray; Nathanael S. ;   et al. | 2021-02-04 |
Kinase inhibitors for the treatment of disease Grant 10,906,878 - Gray , et al. February 2, 2 | 2021-02-02 |
Small Molecule Degraders That Recruit Dcaf15 App 20210002295 - Gray; Nathanael S. ;   et al. | 2021-01-07 |
Inhibitors of cyclin-dependent kinase 7 (CDK7) Grant 10,870,651 - Gray , et al. December 22, 2 | 2020-12-22 |
Pyrimidines as EGFR inhibitors and methods of treating disorders Grant 10,870,636 - Gray , et al. December 22, 2 | 2020-12-22 |
Inhibitors Of Egfr And Methods Of Use Thereof App 20200390783 - GRAY; NATHANAEL S. ;   et al. | 2020-12-17 |
Degradation of cyclin-dependent kinase 8 (CDK8) by conjugation of CDK8 inhibitors with E3 ligase ligand and methods of use Grant 10,865,205 - Gray , et al. December 15, 2 | 2020-12-15 |
Degradation of cyclin-dependent kinase 4/6 (CDK4/6) by conjugation of CDK4/6 inhibitors with E3 ligase ligand and methods of use Grant 10,865,204 - Gray , et al. December 15, 2 | 2020-12-15 |
Inhibitors Of Malt1 And Uses Thereof App 20200385405 - Gray; Nathanael S. ;   et al. | 2020-12-10 |
Degraders Of Egfr And Methods Of Use Thereof App 20200377477 - GRAY; NATHANAEL S. ;   et al. | 2020-12-03 |
Pharmaceutical Combinations Of Egfr Inhibitors And Methods Of Use Thereof App 20200375999 - GRAY; NATHANAEL S. ;   et al. | 2020-12-03 |
Degraders Of Egfr And Methods Of Use Thereof App 20200377501 - GRAY; NATHANAEL S. ;   et al. | 2020-12-03 |
Cyclin-dependent Kinase Inhibitors And Methods Of Use App 20200369715 - Gray; Nathanael S. ;   et al. | 2020-11-26 |
Degradation of Bruton's tyrosine kinase (BTK) by conjugation of BTK inhibitors with E3 ligase ligand and methods of use Grant 10,842,878 - Gray , et al. November 24, 2 | 2020-11-24 |
Thiazolyl-containing compounds for treating proliferative diseases Grant 10,844,077 - Gray , et al. November 24, 2 | 2020-11-24 |
Compounds For Treating Dengue Virus Infection And Other Viral Infections App 20200360381 - Yang; Priscilla L. ;   et al. | 2020-11-19 |
Nek Inhibitors And Methods Of Use App 20200361948 - GRAY; NATHANAEL S. ;   et al. | 2020-11-19 |
Inhibitors Of Cyclin-dependent Kinase 12 (cdk12) And Uses Thereof App 20200361906 - Gray; Nathanael S. ;   et al. | 2020-11-19 |
Inhibitors of EGFR and methods of use thereof Grant 10,836,722 - Gray , et al. November 17, 2 | 2020-11-17 |
Small Molecule Myristate Inhibitors Of Bcr-abl And Methods Of Use App 20200347068 - GRAY; Nathanael S. ;   et al. | 2020-11-05 |
4,6-pyrimidinylene Derivatives And Uses Thereof App 20200338075 - Gray; Nathanael S. ;   et al. | 2020-10-29 |
Uses Of Salt-inducible Kinase (sik) Inhibitors App 20200338087 - Shamji; Alykhan ;   et al. | 2020-10-29 |
Combination Therapy Of Transcription Inhibitors And Kinase Inhibitors App 20200338074 - Hammerman; Peter ;   et al. | 2020-10-29 |
Compounds For The Degradation Of Stk4 And Treatment Of Hematologic Malignancies App 20200331889 - Buhrlage; Sara ;   et al. | 2020-10-22 |
Bicyclic Urea Kinase Inhibitors And Uses Thereof App 20200317675 - GRAY; Nathanael S. ;   et al. | 2020-10-08 |
Uses of diazepane derivatives Grant 10,793,571 - Bradner , et al. October 6, 2 | 2020-10-06 |
Pyrimido-diazepinone compounds and methods of treating disorders Grant 10,787,461 - Gray , et al. September 29, 2 | 2020-09-29 |
Inhibitors Of Interleukin-1 Receptor-associated Kinases And Uses Thereof App 20200299257 - Gray; Nathanael S. ;   et al. | 2020-09-24 |
Type Ii Raf Kinase Inhibitors App 20200297721 - Gray; Nathanael S. ;   et al. | 2020-09-24 |
Sulfonamide Derivatives For Protein Degradation App 20200290964 - Gray; Nathanael S. ;   et al. | 2020-09-17 |
Inhibitors Of Cyclin-dependent Kinases App 20200277292 - Gray; Nathanael S. ;   et al. | 2020-09-03 |
Uses Of Pyrimidopyrimidinones As Sik Inhibitors App 20200253981 - Kind Code | 2020-08-13 |
6,11-dihydro-5h-benzo[b]carbazole Inhibitors Of Alk And Srpk And Methods Of Use App 20200223798 - HATCHER; John ;   et al. | 2020-07-16 |
STK4 inhibitors for treatment of hematologic malignancies Grant 10,710,978 - Gray , et al. | 2020-07-14 |
MALT1 inhibitors and uses thereof Grant 10,711,036 - Gray , et al. | 2020-07-14 |
Bifunctional Molecules For Her3 Degradation And Methods Of Use App 20200216454 - GRAY; Nathanael S. ;   et al. | 2020-07-09 |
Combination therapy of transcription inhibitors and kinase inhibitors Grant 10,702,527 - Hammerman , et al. | 2020-07-07 |
4,6-pyrimidinylene derivatives and uses thereof Grant 10,695,346 - Gray , et al. | 2020-06-30 |
Inhibitors Of Egfr And/or Her2 And Methods Of Use App 20200199121 - HATCHER; JOHN M. ;   et al. | 2020-06-25 |
Compounds for MALT1 degredation Grant 10,689,366 - Melnick , et al. | 2020-06-23 |
Uses Of Salt-inducible Kinase (sik) Inhibitors For Treating Osteoporosis App 20200179387 - Wein; Marc ;   et al. | 2020-06-11 |
Inhibitors Of Cyclin-dependent Kinases App 20200172499 - Gray; Nathanael S. ;   et al. | 2020-06-04 |
Thiazolyl-containing Compounds For Treating Proliferative Diseases App 20200165267 - Gray; Nathanael S. ;   et al. | 2020-05-28 |
Methods to treat lymphoplasmacytic lymphoma Grant 10,633,348 - Treon , et al. | 2020-04-28 |
Methods to treat lymphoplasmacytic lymphoma Grant 10,597,387 - Treon , et al. | 2020-03-24 |
Inhibitors Of C-jun-n-terminal Kinase (jnk) App 20200087295 - Gray; Nathanael S. ;   et al. | 2020-03-19 |
Pyrimido-diazepinone Compounds And Methods Of Treating Disorders App 20200071340 - Gray; Nathanael S. ;   et al. | 2020-03-05 |
Pyrimido-diazepinone kinase scaffold compounds and methods of treating disorders Grant 10,570,154 - Gray , et al. Feb | 2020-02-25 |
Inhibitors of cyclin-dependent kinases Grant 10,550,121 - Gray , et al. Fe | 2020-02-04 |
Pyrimidines as EGFR inhibitors and methods of treating disorders Grant 10,550,112 - Gray , et al. Fe | 2020-02-04 |
Degradation of cyclin-dependent kinase 9 (CDK9) by conjugation of CDK9 inhibitors with E3 ligase ligand and methods of use Grant 10,532,103 - Gray , et al. Ja | 2020-01-14 |
HCK as a therapeutic target in MYD88 mutated diseases Grant 10,525,060 - Treon , et al. J | 2020-01-07 |
Inhibitors Of Egfr And Methods Of Use Thereof App 20200002279 - GRAY; Nathanael S. ;   et al. | 2020-01-02 |
Malt1 Inhibitors And Uses Thereof App 20190389904 - Gray; Nathanael S. ;   et al. | 2019-12-26 |
Substituted 6,11-dihydro-5H-benzo[b]carbazoles as inhibitors of ALK and SRPK Grant 10,508,082 - Hatcher , et al. Dec | 2019-12-17 |
Degradation Of Protein Kinases By Conjugation Of Protein Kinase Inhibitors With E3 Ligase Ligand And Methods Of Use App 20190374528 - GRAY; Nathanael S. ;   et al. | 2019-12-12 |
Imidazolyl Kinase Inhibitors And Uses Thereof App 20190367487 - Gray; Nathanael S. ;   et al. | 2019-12-05 |
Uses Of Salt-inducible Kinase (sik) Inhibitors App 20190343842 - Shamji; Alykhan ;   et al. | 2019-11-14 |
Thiazolyl-containing compounds for treating proliferative diseases Grant 10,464,949 - Gray , et al. No | 2019-11-05 |
Macrocyclic kinase inhibitors and uses thereof Grant 10,457,691 - Gray , et al. Oc | 2019-10-29 |
Pyrimido-diazepinone compounds and methods of treating disorders Grant 10,457,692 - Gray , et al. Oc | 2019-10-29 |
Compounds and methods for treating cancer Grant 10,450,281 - D'Andrea , et al. Oc | 2019-10-22 |
Bicyclic Urea Kinase Inhibitors And Uses Thereof App 20190315752 - GRAY; Nathanael S. ;   et al. | 2019-10-17 |
Inhibitors Of Cyclin-dependent Kinases App 20190315747 - Gray; Nathanael S. ;   et al. | 2019-10-17 |
Pyrimido-diazepinone Kinase Scaffold Compounds And Methods Of Treating Dclk1/2-mediated Disorders App 20190315753 - Ferguson; Fleur M. ;   et al. | 2019-10-17 |
Host Targeted Inhibitors Of Dengue Virus And Other Viruses App 20190292178 - Gray; Nathanael S. ;   et al. | 2019-09-26 |
Inhibitors Of Interleukin-1 Receptor-associated Kinases And Uses Thereof App 20190276426 - Gray; Nathanael S. ;   et al. | 2019-09-12 |
Degradation Of Bruton's Tyrosine Kinase (btk) By Conjugation Of Btk Inhibitors With E3 Ligase Ligand And Methods Of Use App 20190262458 - GRAY; Nathanael S. ;   et al. | 2019-08-29 |
Compounds For Malt1 Degradation App 20190263785 - Melnick; Ari M. ;   et al. | 2019-08-29 |
Degradation Of Bruton's Tyrosine Kinase (btk) By Conjugation Of Btk Inhibitors With E3 Ligase Ligand And Methods Of Use App 20190262459 - GRAY; Nathanael S. ;   et al. | 2019-08-29 |
Kinase Inhibitors For The Treatment Of Disease App 20190256475 - GRAY; Nathanael S. ;   et al. | 2019-08-22 |
Inhibitors of EGFR and methods of use thereof Grant 10,385,019 - Gray , et al. A | 2019-08-20 |
Inhibitors Of C-jun-n-terminal Kinase (jnk) App 20190248778 - Gray; Nathanael S. ;   et al. | 2019-08-15 |
Fused bicyclic pyrimidine derivatives and uses thereof Grant 10,342,798 - Gray , et al. July 9, 2 | 2019-07-09 |
Novel Pyrimidines As Egfr Inhibitors And Methods Of Treating Disorders App 20190194169 - GRAY; Nathanael S. ;   et al. | 2019-06-27 |
Imidazolyl kinase inhibitors and uses thereof Grant 10,287,268 - Gray , et al. | 2019-05-14 |
Thiazolyl-containing Compounds For Treating Proliferative Diseases App 20190119301 - Gray; Nathanael S. ;   et al. | 2019-04-25 |
Pyrimidines as EGFR inhibitors and methods of treating disorders Grant 10,266,517 - Gray , et al. | 2019-04-23 |
Uses of salt-inducible kinase (SIK) inhibitors Grant 10,265,321 - Shamji , et al. | 2019-04-23 |
Degradation Of Cyclin-dependent Kinase 9 (cdk9) By Conjugation Of Cdk9 Inhibitors With E3 Ligase Ligand And Methods Of Use App 20190111143 - GRAY; Nathanael S. ;   et al. | 2019-04-18 |
Degradation Of Cyclin-dependent Kinase 8 (cdk8) By Conjugation Of Cdk8 Inhibitors With E3 Ligase Ligand And Methods Of Use App 20190112307 - GRAY; Nathanael S. ;   et al. | 2019-04-18 |
Pyrimido-diazepinon Kinase Scaffold Compounds And Methods For Treating P13k-mediated Disorders App 20190106424 - Gray; Nathanael S. ;   et al. | 2019-04-11 |
Degradation Of Cyclin-dependent Kinase 4/6 (cdk4/6) By Conjugation Of Cdk4/6 Inhibitors With E3 Ligase Ligand And Methods Of Use App 20190092768 - GRAY; Nathanael S. ;   et al. | 2019-03-28 |
Small Molecule Myristate Inhibitors Of Bcr-abl And Methods Of Use App 20190084990 - Gray; Nathanael S. ;   et al. | 2019-03-21 |
Pyrimido-diazepinone Compounds And Methods Of Treating Disorders App 20190084998 - Gray; Nathanael S. ;   et al. | 2019-03-21 |
SIK inhibitor for use in a method of treating an inflammatory and/or immune disorder Grant 10,233,157 - Cohen , et al. | 2019-03-19 |
Inhibitors Of Cyclindependent Kinase 7 (cdk7) App 20190055248 - Gray; Nathanael S. ;   et al. | 2019-02-21 |
EGFR Inhibitors and Methods of Treating Disorders App 20190040065 - Gray; Nathanael S. ;   et al. | 2019-02-07 |
Pyrimido-diazepinone compounds and methods of treating disorders Grant 10,189,861 - Gray , et al. Ja | 2019-01-29 |
Bifunctional Compounds For Her3 Degradation And Methods Of Use App 20190016703 - GRAY; Nathanael S. ;   et al. | 2019-01-17 |
Combination Therapy Of Transcription Inhibitors And Kinase Inhibitors App 20190015411 - Hammerman; Peter ;   et al. | 2019-01-17 |
Fused Bicyclic Pyrimidine Derivatives And Uses Thereof App 20180369243 - Gray; Nathanael S. ;   et al. | 2018-12-27 |
Pyrimido-diazepinone Kinase Scaffold Compounds And Methods Of Treating Disorders App 20180362545 - Gray; Nathanael S. ;   et al. | 2018-12-20 |
Inhibitors Of Cyclin-dependent Kinases App 20180362483 - Gray; Nathanael S. ;   et al. | 2018-12-20 |
Hydrophobically Tagged Small Molecules As Inducers Of Protein Degradation App 20180354954 - Gray; Nathanael S. ;   et al. | 2018-12-13 |
Substituted heterocyclic compounds for treating or preventing viral infections Grant 10,150,742 - Yang , et al. Dec | 2018-12-11 |
4,6-pyrimidinylene Derivatives And Uses Thereof App 20180344733 - Gray; Nathanael S. ;   et al. | 2018-12-06 |
Inhibitors Of Cyclin-dependent Kinases App 20180319801 - Gray; Nathanael S. ;   et al. | 2018-11-08 |
Thiazolyl-containing compounds for treating proliferative diseases Grant 10,112,957 - Gray , et al. October 30, 2 | 2018-10-30 |
Inhibitors Of Egfr And Methods Of Use Thereof App 20180290975 - GRAY; Nathanael S. ;   et al. | 2018-10-11 |
Pyrimido-diazepinone kinase scaffold compounds and methods of treating disorders Grant 10,081,639 - Gray , et al. September 25, 2 | 2018-09-25 |
Host Targeted Inhibitors Of Dengue Virus And Other Viruses App 20180265507 - Gray; Nathanael S. ;   et al. | 2018-09-20 |
Inhibitors Of Alk And Srpk And Methods Of Use App 20180258040 - HATCHER; John ;   et al. | 2018-09-13 |
Malt1 Inhibitors And Uses Thereof App 20180251489 - Gray; Nathanael S. ;   et al. | 2018-09-06 |
Lrrk2 Inhibitors And Methods Of Making And Using The Same App 20180244676 - GRAY; Nathanael S. ;   et al. | 2018-08-30 |
Sik Inhibitor For Use In A Method Of Treating An Inflammatory And/or Immune Disorder App 20180215719 - Cohen; Philip ;   et al. | 2018-08-02 |
Novel Pyrimidines As Egfr Inhibitors And Methods Of Treating Disorders App 20180194758 - GRAY; Nathanael S. ;   et al. | 2018-07-12 |
Methods To Treat Lymphoplasmacytic Lymphoma App 20180194739 - Treon; Steven P. ;   et al. | 2018-07-12 |
Janus kinase inhibitors and uses thereof Grant 10,017,477 - Gray , et al. July 10, 2 | 2018-07-10 |
Methods To Treat Lymphoplasmacytic Lymphoma App 20180186780 - Treon; Steven P. ;   et al. | 2018-07-05 |
Combination Therapy Of Transcription Inhibitors And Kinase Inhibitors App 20180169097 - Hammerman; Peter ;   et al. | 2018-06-21 |
Fused Bicyclic Pyrimidine Derivatives And Uses Thereof App 20180153894 - Gray; Nathanael S. ;   et al. | 2018-06-07 |
4,6-pyrimidinylene Derivatives And Uses Thereof App 20180110778 - Gray; Nathanael S. ;   et al. | 2018-04-26 |
Stk4 Inhibitors For Treatment Of Hematologic Malignancies App 20180111916 - GRAY; Nathanael S. ;   et al. | 2018-04-26 |
Hydrophobically Tagged Small Molecules As Inducers Of Protein Degradation App 20180093990 - Gray; Nathanael S. ;   et al. | 2018-04-05 |
Methods to treat lymphoplasmacytic lymphoma Grant 9,908,872 - Treon , et al. March 6, 2 | 2018-03-06 |
EGFR inhibitors and methods of treating disorders Grant 9,908,884 - Gray , et al. March 6, 2 | 2018-03-06 |
Compounds that modulate EGFR activity and methods for treating or preventing conditions therewith Grant 9,879,028 - Gray , et al. January 30, 2 | 2018-01-30 |
Hydrophobically tagged janus kinase inhibitors and uses thereof Grant 9,862,688 - Gray , et al. January 9, 2 | 2018-01-09 |
Methods to treat lymphoplasmacytic lymphoma Grant 9,856,223 - Treon , et al. January 2, 2 | 2018-01-02 |
Novel Pyrimidines As Egfr Inhibitors And Methods Of Treating Disorders App 20170362204 - GRAY; Nathanael S. ;   et al. | 2017-12-21 |
Small Molecule Myristate Inhibitors Of Bcr-abl And Abl And Methods Of Use App 20170349595 - GRAY; Nathanael S. ;   et al. | 2017-12-07 |
Sik Inhibitor For Use In A Method Of Treating An Inflammatory And/or Immune Disorder App 20170342036 - Cohen; Philip ;   et al. | 2017-11-30 |
Hck As A Therapeutic Target In Myd88 Mutated Diseases App 20170333436 - Treon; Steven P. ;   et al. | 2017-11-23 |
Pyrimido-diazepinone Compounds And Methods Of Treating Disorders App 20170283422 - Gray; Nathanael S. ;   et al. | 2017-10-05 |
Pyrimido-diazepinone Kinase Scaffold Compounds And Methods Of Treating Disorders App 20170260208 - Gray; Nathanael S. ;   et al. | 2017-09-14 |
Thiazolyl-containing Compounds For Treating Proliferative Diseases App 20170233411 - Gray; Nathanael S. ;   et al. | 2017-08-17 |
Uses Of Salt-inducible Kinase (sik) Inhibitors App 20170224700 - Shamji; Alykhan ;   et al. | 2017-08-10 |
Imidazolyl Kinase Inhibitors And Uses Thereof App 20170204082 - Gray; Nathanael S. ;   et al. | 2017-07-20 |
Macrocyclic Kinase Inhibitors And Uses Thereof App 20170204116 - Gray; Nathanael S. ;   et al. | 2017-07-20 |
Pyrimido-diazepinone kinase scaffold compounds and methods of treating disorders Grant 9,701,683 - Gray , et al. July 11, 2 | 2017-07-11 |
Diazepane derivatives and uses thereof Grant 9,695,172 - Bradner , et al. July 4, 2 | 2017-07-04 |
Pyrimido-diazepinone compounds and methods of treating disorders Grant 9,676,792 - Gray , et al. June 13, 2 | 2017-06-13 |
Small molecule myristate inhibitors of Bcr-abl and methods of use Grant 9,670,214 - Gray , et al. June 6, 2 | 2017-06-06 |
Uses Of Kinase Inhibitors For Inducing And Maintaining Pluripotency App 20170114323 - Theunissen; Thorold W. ;   et al. | 2017-04-27 |
Hydrophobically Tagged Janus Kinase Inhibitors And Uses Thereof App 20170044112 - Gray; Nathanael S. ;   et al. | 2017-02-16 |
Janus Kinase Inhibitors And Uses Thereof App 20170044111 - Gray; Nathanael S. ;   et al. | 2017-02-16 |
Uses Of Diazepane Derivatives App 20170008895 - Bradner; James E. ;   et al. | 2017-01-12 |
Inhibitors Of C-jun-n-terminal Kinase (jnk) App 20160368910 - Gray; Nathanael S. ;   et al. | 2016-12-22 |
Pyrimido-diazepinone Kinase Scaffold Compounds And Methods Of Treating Disorders App 20160347755 - Gray; Nathanael S. ;   et al. | 2016-12-01 |
Diazepane Derivatives And Uses Thereof App 20160347749 - Bradner; James E. ;   et al. | 2016-12-01 |
Dihydropteridinone Derivatives And Uses Thereof App 20160347750 - Bradner; James E. ;   et al. | 2016-12-01 |
Methods To Treat Lymphoplasmacytic Lymphoma App 20160318878 - Treon; Steven P. ;   et al. | 2016-11-03 |
Methods To Treat Lymphoplasmacytic Lymphoma App 20160311807 - Treon; Steven P. ;   et al. | 2016-10-27 |
Pyrimido-diazepinone kinase scaffold compounds and methods of treating disorders Grant 9,464,091 - Gray , et al. October 11, 2 | 2016-10-11 |
Compounds that Modulate EGFR Activity and Methods for Treating or Preventing Conditions Therewith App 20160137610 - Gray; Nathanael S. ;   et al. | 2016-05-19 |
Pyrimido-diazepinone Kinase Scaffold Compounds And Methods Of Treating Disorders App 20160122357 - Gray; Nathanael S. ;   et al. | 2016-05-05 |
Pyrimido-diazepinone kinase scaffold compounds and methods of treating disorders Grant 9,266,890 - Gray , et al. February 23, 2 | 2016-02-23 |
Type Ii Raf Kinase Inhibitors App 20160046636 - Gray; Nathanael S. ;   et al. | 2016-02-18 |
Substituted Heterocyclic Compounds for Treating or Preventing Viral Infections App 20160031826 - Yang; Priscilla ;   et al. | 2016-02-04 |
Pyrimido-diazepinone Compounds And Methods Of Treating Disorders App 20160024115 - Gray; Nathanael S. ;   et al. | 2016-01-28 |
Type II Raf kinase inhibitors Grant 9,180,127 - Gray , et al. November 10, 2 | 2015-11-10 |
Small Molecule Myristate Inhibitors Of Bcr-abl And Methods Of Use App 20150094275 - GRAY; Nathanael S. ;   et al. | 2015-04-02 |
Compounds that Modulate EGFR Activity and Methods for Treating or Preventing Conditions Therewith App 20140011810 - Gray; Nathanael S. ;   et al. | 2014-01-09 |
Compounds and compositions as protein kinase inhibitors Grant 8,592,433 - Nagle , et al. November 26, 2 | 2013-11-26 |
Compounds that modulate EGFR activity and methods for treating or preventing conditions therewith App 20130137709 - Gray; Nathanael S. ;   et al. | 2013-05-30 |
Type Ii Raf Kinase Inhibitors App 20130040949 - Gray; Nathanael S. ;   et al. | 2013-02-14 |
Egfr Inhibitors And Methods Of Treating Disorders App 20120094999 - Gray; Nathanael S. ;   et al. | 2012-04-19 |
Pyrimido-diazepinone Kinase Scaffold Compounds And Methods Of Treating Disorders App 20120040961 - Gray; Nathanael S. ;   et al. | 2012-02-16 |
Compounds and compositions as protein kinase inhibitors Grant 8,101,608 - Wan , et al. January 24, 2 | 2012-01-24 |
Small Molecule Myristate Inhibitors Of Bcr-abl And Methods Of Use App 20110312908 - Gray; Nathanael S. ;   et al. | 2011-12-22 |
Compounds That Modulate Egfr Activity And Methods For Treating Or Preventing Conditions Therewith App 20110207736 - GRAY; Nathanael S. ;   et al. | 2011-08-25 |
Compounds And Compositions Useful For The Treatment Of Malaria App 20110144107 - Chatterjee; Arnab K. ;   et al. | 2011-06-16 |
Immunosuppresant compounds and compositions Grant 7,939,519 - Pan , et al. May 10, 2 | 2011-05-10 |
Compounds and Compositions as Inhibitors of Receptor Tyrosine Kinase Activity App 20110092491 - CHENG; Dai ;   et al. | 2011-04-21 |
Compositions And Methods For Treating Cancers App 20110021524 - Adrian; Francisco ;   et al. | 2011-01-27 |
Compounds and compositions as protein kinase inhibitors Grant 7,868,018 - Xie , et al. January 11, 2 | 2011-01-11 |
Compounds And Compositions As Protein Kinase Inhibitors App 20100324062 - Nagle; Advait ;   et al. | 2010-12-23 |
2-biphenylamino-4-aminopyrimidine Derivatives As Kinase Inhibitors App 20100298295 - Marsilje; Thomas H. ;   et al. | 2010-11-25 |
Compounds and compositions as protein kinase inhibitors Grant 7,713,958 - Wan , et al. May 11, 2 | 2010-05-11 |
Purine Compounds And Compositions As Kinase Inhibitors For The Treatment Of Plasmodium Related Diseases App 20100056494 - Winzeler; Elizabeth ;   et al. | 2010-03-04 |
Compositions And Methods For Fgf Receptor Kinases Inhibitors App 20090312321 - Ren; Pingda ;   et al. | 2009-12-17 |
Compounds And Compositions As Protein Kinase Inhibitors App 20090258910 - Gray; Nathanael S. ;   et al. | 2009-10-15 |
Compounds and compositions as protein kinase inhibitors Grant 7,589,101 - Okram , et al. September 15, 2 | 2009-09-15 |
Immunosuppressant Compounds and Compositions App 20090221547 - Gao; Wenqi ;   et al. | 2009-09-03 |
Compounds And Compositions As Protein Kinase Inhibitors App 20090181991 - Zhang; Qiong ;   et al. | 2009-07-16 |
Compounds and Compositions as Protein Kinase Inhibitors App 20090137555 - Wan; Yongqin ;   et al. | 2009-05-28 |
Compounds And Compositions As Protein Kinase Inhibitors App 20090069327 - Ding; Qiang ;   et al. | 2009-03-12 |
Immunosuppresant Compounds And Compositions App 20090036423 - Pan; Shifeng ;   et al. | 2009-02-05 |
Immunosuppressant compounds and compositions Grant 7,462,629 - Pan , et al. December 9, 2 | 2008-12-09 |
Compounds and Compositions as Protein Kinase Inhibitors App 20080300246 - Xie; Yongping ;   et al. | 2008-12-04 |
Compounds and Compositions as Protein Kinase Inhibitors App 20080300267 - Okram; Barun ;   et al. | 2008-12-04 |
Compounds and Compositions as Protein Kinase Inhibitors App 20080287432 - Okram; Barun ;   et al. | 2008-11-20 |
Compounds and compositions as protein kinase inhibitors Grant 7,449,582 - Ding , et al. November 11, 2 | 2008-11-11 |
5-Substituted Thiazol-2-Yl Amino Compounds and Compositions as Protein Kinase Inhibitors App 20080227783 - Wan; Yongqin ;   et al. | 2008-09-18 |
Compounds and Compositions as Protein Kinase Inhibitors App 20080221192 - Wan; Yongqin ;   et al. | 2008-09-11 |
Compositions And Methods For Inducing Osteogenesis App 20080214541 - Wu; Xu ;   et al. | 2008-09-04 |
Compounds And Compositions As Protein Kinase Inhibitors App 20080108616 - Ding; Qiang ;   et al. | 2008-05-08 |
Compositions and methods for inducing osteogenesis Grant 7,273,864 - Wu , et al. September 25, 2 | 2007-09-25 |
Kinase Inhibitor Scaffolds And Methods For Their Preparation App 20070191380 - Ding; Sheng ;   et al. | 2007-08-16 |
Bicyclic compounds and compositions Grant 7,256,206 - Pan , et al. August 14, 2 | 2007-08-14 |
6-phenyl-7H-pyrrolo[2,3-d]pyrimidine compounds that induce neuronal differentiation in embryonic stem cells Grant 7,253,166 - Ding , et al. August 7, 2 | 2007-08-07 |
Kinase inhibitor scaffolds and methods for their preparation Grant 7,176,312 - Ding , et al. February 13, 2 | 2007-02-13 |
Bis-aromatic alkanols Grant 7,169,817 - Pan , et al. January 30, 2 | 2007-01-30 |
Cyclic compounds and compositions as protein kinase inhibitors Grant 7,151,096 - Ren , et al. December 19, 2 | 2006-12-19 |
Immunosuppressant compounds and compositions Grant 7,060,697 - Marsilje , et al. June 13, 2 | 2006-06-13 |
Methods for the synthesis of substituted purines App 20060009642 - Ding; Sheng ;   et al. | 2006-01-12 |
Methods for the synthesis of substituted purines Grant 6,949,644 - Ding , et al. September 27, 2 | 2005-09-27 |
Compounds and compositions as protein kinase inhibitors App 20050209285 - Gray, Nathanael S. ;   et al. | 2005-09-22 |
Compounds and compositions as protein kinase inhibitors App 20050187230 - Ding, Qiang ;   et al. | 2005-08-25 |
Purine inhibitors of protein kinases, G proteins and polymerases Grant 6,803,371 - Gray , et al. October 12, 2 | 2004-10-12 |
Purine inhibitors of protein kinases, G proteins and polymerases Grant 6,617,331 - Gray , et al. September 9, 2 | 2003-09-09 |