loadpatents
name:-0.067487001419067
name:-0.054548978805542
name:-0.0061650276184082
Macielag; Mark J. Patent Filings

Macielag; Mark J.

Patent Applications and Registrations

Patent applications and USPTO patent grants for Macielag; Mark J..The latest application filed is for "acylsufonamide compounds useful as ep3 receptor antagonists".

Company Profile
6.58.68
  • Macielag; Mark J. - Gwynedd Valley PA
  • Macielag; Mark J - Gwynedd Valley PA
  • Macielag; Mark J - Spring House PA
  • Macielag; Mark J. - Cranbury NJ US
  • Macielag; Mark J. - Branchburg NJ US
  • - Branchburg NJ US
  • Macielag; Mark J. - Spring House PA
  • Macielag; Mark J. - Raritan NJ
  • Macielag; Mark J. - New Brunswick NJ
*profile and listings may contain filings by different individuals or companies with the same name. Review application materials to confirm ownership/assignment.
Patent Activity
PatentDate
Cylcoalkenyl derivatives useful as agonists of the GPR120 and/or GPR40 receptors
Grant 11,230,526 - Lanter , et al. January 25, 2
2022-01-25
Acylsufonamide Compounds Useful As Ep3 Receptor Antagonists
App 20210253562 - Zhu; Bin ;   et al.
2021-08-19
Pyridin-2-one derivatives of formula (I) useful as EP3 receptor antagonists
Grant 10,590,083 - Zhang , et al.
2020-03-17
Pyridin-2-one derivatives of formula (III) useful as EP3 receptor antagonists
Grant 10,399,944 - Zhang , et al. Sep
2019-09-03
Pyridin-2-one derivatives of formula (II) useful as EP3 receptor antagonists
Grant 10,336,701 - Zhang , et al.
2019-07-02
Pyridin-2-one Derivatives Of Formula (iii) Useful As Ep3 Receptor Antagonists
App 20190047961 - Zhang; Xuqing ;   et al.
2019-02-14
Pyridin-2-one Derivatives Of Formula (ii) Useful As Ep3 Receptor Antagonists
App 20190047960 - Zhang; Xuqing ;   et al.
2019-02-14
Pyridin-2-one Derivatives Of Formula (i) Useful As Ep3 Receptor Antagonists
App 20190047959 - Zhang; Xuqing ;   et al.
2019-02-14
Benzimidazole Derivatives Useful As Cb-1 Inverse Agonists
App 20190031618 - Macielag; Mark J. ;   et al.
2019-01-31
Benzimidazole derivatives useful as CB-1 inverse agonists
Grant 10,118,900 - Macielag , et al. November 6, 2
2018-11-06
Chemically modified quinoline and quinolone derivatives useful as CB-1 inverse agonists
Grant 9,815,790 - Macielag , et al. November 14, 2
2017-11-14
Indazole derivatives useful as CB-1 inverse agonists
Grant 9,682,940 - Macielag , et al. June 20, 2
2017-06-20
Benzimidazole derivatives useful TRPM8 channel modulators
Grant 9,636,345 - Macielag , et al. May 2, 2
2017-05-02
Indazole Derivatives Useful As Cb-1 Inverse Agonists
App 20170057925 - Macielag; Mark J. ;   et al.
2017-03-02
Benzimidazole Derivatives Useful As Cb-1 Inverse Agonists
App 20170057929 - Macielag; Mark J. ;   et al.
2017-03-02
Chemically Modified Quinoline And Quinolone Derivatives Useful As Cb-1 Inverse Agonists
App 20170057922 - Macielag; Mark J. ;   et al.
2017-03-02
Sulfonamides as TRPM8 modulators
Grant 9,434,711 - Branum , et al. September 6, 2
2016-09-06
Monoacylglycerol lipase inhibitors for the treatment of metabolic diseases and related disorders
Grant 9,375,430 - Connelly , et al. June 28, 2
2016-06-28
Imidazo[1,2-.alpha.]pyridine sulfonamides as TRPM8 modulators
Grant 9,067,935 - Macielag , et al. June 30, 2
2015-06-30
Benzimidazole Derivatives Useful Trpm8 Channel Modulators
App 20150150882 - Macielag; Mark J. ;   et al.
2015-06-04
Monoacylglycerol lipase inhibitors for the treatment of metabolic diseases and related disorders
Grant 8,987,247 - Connelly , et al. March 24, 2
2015-03-24
Benzimidazole derivatives useful as TRPM8 channel modulators
Grant 8,981,113 - Macielag , et al. March 17, 2
2015-03-17
Sulfonamides As Trpm8 Modulators
App 20140315899 - Branum; Shawn T. ;   et al.
2014-10-23
4-substituted-2-phenoxy-phenylamine delta opioid receptor modulators
Grant 8,846,655 - Coats , et al. September 30, 2
2014-09-30
Heteroaromatic and aromatic piperazinyl azetidinyl amides as monoacylglycerol lipase inhibitors
Grant 8,815,839 - Chevalier , et al. August 26, 2
2014-08-26
Sulfonamides as TRPM8 modulators
Grant 8,809,327 - Branum , et al. August 19, 2
2014-08-19
Di-azetidinyl diamide as monoacylglycerol lipase inhibitors
Grant 8,759,333 - Connolly , et al. June 24, 2
2014-06-24
Di-azetidinyl diamide as monoacylglcerol lipase inhibitors
Grant 8,759,533 - Connolly , et al. June 24, 2
2014-06-24
Amino-pyrrolidine-azetidine diamides as monoacylglycerol lipase inhibitors
Grant 8,748,417 - Zhang , et al. June 10, 2
2014-06-10
Azetidinyl diamides as monoacylglycerol lipase inhibitors
Grant 8,697,683 - Bian , et al. April 15, 2
2014-04-15
Pyrimidine compounds as delta opioid receptor modulators
Grant 8,685,990 - Coats , et al. April 1, 2
2014-04-01
IMIDAZO[1,2-a]PYRIDINE SULFONAMIDES AS TRPM8 MODULATORS
App 20140088098 - Macielag; Mark J. ;   et al.
2014-03-27
Oxopiperazine-azetidine amides and oxodiazepine-azetidine amides as monoacylglycerol lipase inhibitors
Grant 8,637,498 - Connolly , et al. January 28, 2
2014-01-28
Imidazo[1,2-.alpha.]pyridine sulfonamides as TRPM8 modulators
Grant 8,618,150 - Macielag , et al. December 31, 2
2013-12-31
Imidazo[1,2-α]pyridine sulfonamides as TRPM8 modulators
Grant 08618150 -
2013-12-31
Pyrimidine Compounds As Delta Opioid Receptor Modulators
App 20130310358 - Coats; Steven J. ;   et al.
2013-11-21
Amino-pyrrolidine-azetidine diamides as monoacylglycerol lipase inhibitors
Grant 8,575,363 - Zhang , et al. November 5, 2
2013-11-05
Azetidinyl Diamides As Monoacylglycerol Lipase Inhibitors
App 20130244997 - Bian; Haiyan ;   et al.
2013-09-19
Piperidin-4-yl-azetidine Diamides As Monoacylglcerol Lipase Inhibitors
App 20130244998 - Connolly; Peter J. ;   et al.
2013-09-19
Benzimidazole Derivatives Useful As Trpm8 Channel Modulators
App 20130245085 - Macielag; Mark J. ;   et al.
2013-09-19
Azetidinyl Diamides As Monoacylglycerol Lipase Inhibitors
App 20130237517 - Bian; Haiyan ;   et al.
2013-09-12
Pyrimidine compounds as delta opioid receptor modulators
Grant 8,513,271 - Coats , et al. August 20, 2
2013-08-20
Piperidin-4-yl-azetidine diamides as monoacylglycerol lipase inhibitors
Grant 8,513,423 - Connolly , et al. August 20, 2
2013-08-20
Di-azetidinyl Diamide As Monoacylglcerol Lipase Inhibitors
App 20130196969 - Connolly; Peter J. ;   et al.
2013-08-01
Amino-pyrrolidine-azetidine Diamides As Monoacylglycerol Lipase Inhibitors
App 20130196970 - Zhang; Yue-Mei ;   et al.
2013-08-01
Di-azetidinyl Diamide As Monoacylglcerol Lipase Inhibitors
App 20130196968 - Connolly; Peter J. ;   et al.
2013-08-01
Heteroaromatic And Aromatic Piperazinyl Azetidinyl Amides As Monoacylglycerol Lipase Inhibitors
App 20130184251 - Chevalier; Kristen ;   et al.
2013-07-18
Benzimidazole derivatives useful as TRPM8 channel modulators
Grant 8,450,497 - Macielag , et al. May 28, 2
2013-05-28
Piperidin-4-yl-azetidine Diamides As Monoacylglycerol Lipase Inhibitors
App 20130102584 - Connolly; Peter J. ;   et al.
2013-04-25
Monoacylglycerol Lipase Inhibitors For The Treatment Of Metabolic Diseases And Related Disorders
App 20130085129 - Connelly; Margery ;   et al.
2013-04-04
Monoacylglycerol Lipase Inhibitors For The Treatment Of Metabolic Diseases And Related Disorders
App 20130085130 - Connelly; Margery ;   et al.
2013-04-04
Hexahydro-cycloheptapyrazole cannabinoid modulators
Grant 8,378,117 - Liotta , et al. February 19, 2
2013-02-19
4-substituted-2-phenoxy-phenylamine Delta Opioid Receptor Modulators
App 20120302541 - Coats; Steven J. ;   et al.
2012-11-29
Pyrazines as delta opioid receptor modulators
Grant 8,293,750 - Connolly , et al. October 23, 2
2012-10-23
Benzimidazole derivatives useful as TRPM8 channel modulators
Grant 8,242,157 - Jetter , et al. August 14, 2
2012-08-14
Pyrazines As Delta Opioid Receptor Modulators
App 20120202824 - CONNOLLY; Peter J. ;   et al.
2012-08-09
Sulfonamides As Trpm8 Modulators
App 20120190674 - Branum; Shawn T. ;   et al.
2012-07-26
IMIDAZO[1,2-a]PYRIDINE SULFONAMIDES AS TRPM8 MODULATORS
App 20120149699 - Macielag; Mark J. ;   et al.
2012-06-14
Pyrazines as delta opioid receptor modulators
Grant 8,183,371 - Connolly , et al. May 22, 2
2012-05-22
Amino-pyrrolidine-azetidine Diamides As Monoacylglycerol Lipase Inhibitors
App 20120101081 - Zhang; Yue-Mei ;   et al.
2012-04-26
Sulfonamides as TRPM8 modulators
Grant 8,153,682 - Branum , et al. April 10, 2
2012-04-10
Sulfonamides as TRPM8 modulators
Grant 8,148,422 - Macielag , et al. April 3, 2
2012-04-03
Oxopiperazine-azetidine Amides And Oxodiazepine-azetidine Amides As Monoacylglycerol Lipase Inhibitors
App 20120077797 - Connolly; Peter J. ;   et al.
2012-03-29
Di-azetidinyl Diamide As Monoacylglycerol Lipase Inhibitors
App 20120058986 - Connolly; Peter J. ;   et al.
2012-03-08
Pyrimidine Compounds As Delta Opioid Receptor Modulators
App 20110269759 - COATS; Steven J. ;   et al.
2011-11-03
Pyrazines As Delta Opioid Receptor Modulators
App 20110105527 - CONNOLLY; PETER J. ;   et al.
2011-05-05
Pyrimidine Compounds As Delta Opioid Receptor Modulators
App 20110105520 - COATS; STEVEN J. ;   et al.
2011-05-05
C-7 isoxazolinyl quinolone / naphthyridine derivatives useful as antibacterial agents
Grant 7,902,227 - Macielag , et al. March 8, 2
2011-03-08
Benzimidazole Derivatives Useful As Trpm8 Channel Modulators
App 20110003800 - Macielag; Mark J. ;   et al.
2011-01-06
Benzimidazole Derivatives Useful As Trpm8 Channel Modulators
App 20110003801 - Jetter; Michele C. ;   et al.
2011-01-06
Hexahydro-cyclooctyl Pyrazole Cannabinoid Modulators
App 20100317633 - Xia; Mingde ;   et al.
2010-12-16
Hexahydro-cyclooctyl pyrazole cannabinoid modulators
Grant 7,825,151 - Xia , et al. November 2, 2
2010-11-02
Antimicrobial oxazolidinone prodrugs
Grant 7,776,855 - Macielag , et al. August 17, 2
2010-08-17
Sulfonamides As Trpm8 Modulators
App 20100160289 - Macielag; Mark J. ;   et al.
2010-06-24
Novel Rifamycin 3,4-(3-substituted Aminomethyl) Fused Pyrrolo Derivatives
App 20100152267 - MACIELAG; Mark J. ;   et al.
2010-06-17
7-amino alkylidenyl-heterocyclic quinolones and naphthyridones
Grant 7,732,612 - Grant , et al. June 8, 2
2010-06-08
3-(substituted Ethyl)-rifamycin Derivatives Useful As Antimicrobial Agents
App 20100029669 - MACIELAG; Mark J. ;   et al.
2010-02-04
3-hydrazone Piperazinyl Rifamycin Derivatives Useful As Antimicrobial Agents
App 20090275594 - MACIELAG; Mark J. ;   et al.
2009-11-05
Quinolone Derivatives Useful As Antibacterial Agents
App 20090270379 - Macielag; Mark J. ;   et al.
2009-10-29
Sulfonamides As Trpm8 Modulators
App 20090264474 - Branum; Shawn T. ;   et al.
2009-10-22
Method For Treating Cb2 Receptor Mediated Pain
App 20090215850 - Xia; Mingde ;   et al.
2009-08-27
7-amino Alkylidenyl-heterocyclic Quinolones And Naphthyridones
App 20090156577 - Davis; Benjamin ;   et al.
2009-06-18
C-7 Isoxazolinyl Quinolone / Naphthyridine Derivatives Useful as Antibacterial Agents
App 20090029980 - Macielag; Mark J. ;   et al.
2009-01-29
Method For Treating Cb2 Receptor Mediated Pain
App 20080234347 - Xia; Mingde ;   et al.
2008-09-25
Hexahydro-Cyclooctyl Pyrazole Cannabinoid Modulators
App 20080076814 - Xia; Mingde ;   et al.
2008-03-27
Hexahydro-Cycloheptapyrazole Cannabinoid Modulators
App 20080070968 - Liotta; Fina ;   et al.
2008-03-20
Antimicrobial Oxazolidinone Prodrugs
App 20080027053 - Macielag; Mark J. ;   et al.
2008-01-31
Cyclohexyl derivatives as selective estrogen receptor modulators
Grant 7,183,445 - Jain , et al. February 27, 2
2007-02-27
7-amino alkylidenyl-heterocyclic quinolones and naphthyridones
Grant 7,179,805 - Grant, III , et al. February 20, 2
2007-02-20
7-Amino alkylidenyl-heterocyclic quinolones and naphthyridones
App 20060052359 - Grant; Eugene B. ;   et al.
2006-03-09
Inhibitors of bacterial Type III protein secretion systems
App 20050272784 - Li, Xiaobing ;   et al.
2005-12-08
11,12-Cyclic thiocarbamate macrolide antibacterial agents
App 20050250713 - Zhu, Bin ;   et al.
2005-11-10
Triazine compounds as inhibitors of bacterial type III protein secretion systems
App 20050250945 - Li, Xiaobing ;   et al.
2005-11-10
Inhibitors of bacterial type III protein secretion systems
App 20050250819 - Li, Xiaobing ;   et al.
2005-11-10
Neurotrophic pyrrolidines and piperidines, and related compositions and methods
App 20050153951 - Kanojia, Ramesh M. ;   et al.
2005-07-14
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors
App 20050113402 - Sui, Zhihua ;   et al.
2005-05-26
7-Amino alkylidenyl-heterocyclic quinolones and naphthyridones
App 20050101588 - Grant, Eugene B. III ;   et al.
2005-05-12
Benzo[4,5]thieno[2,3-c]pyridine and Benzo[4,5]furo[2,3-c]pyridine Derivatives Useful as Inhibitors of Phosphodiesterase
Grant 6,864,253 - Sui , et al. March 8, 2
2005-03-08
Cyclohexyl derivatives as selective estrogen receptor modulators
App 20050009799 - Jain, Nareshkumar F. ;   et al.
2005-01-13
3-descladinosyl-6-O-carbamoyl and 6-O-carbonoyl macrolide antibacterial agents
Grant 6,825,172 - Henninger , et al. November 30, 2
2004-11-30
6-O-acyl ketolide antibacterials
Grant 6,825,170 - Henninger , et al. November 30, 2
2004-11-30
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors
Grant 6,818,646 - Sui , et al. November 16, 2
2004-11-16
Neurotrophic pyrrolidines and piperidines, and related compositions and methods
Grant 6,809,107 - Kanojia , et al. October 26, 2
2004-10-26
Substituted aminoalkylamide derivatives as antagonists of follicle stimulating hormone
App 20040092505 - Coats, Steven J. ;   et al.
2004-05-13
6-O-carbamate-11,12-lacto-ketolide antimicrobials
Grant 6,713,455 - Grant, III , et al. March 30, 2
2004-03-30
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors
App 20040044021 - Sui, Zhihua ;   et al.
2004-03-04
3-Descladinosyl-6-O-carbamoyl and 6-O-carbonoyl macrolide antibacterial agents
App 20040018994 - Henninger, Todd C. ;   et al.
2004-01-29
6-O-acyl ketolide antibacterials
App 20030220272 - Henninger, Todd C. ;   et al.
2003-11-27
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors
Grant 6,635,638 - Sui , et al. October 21, 2
2003-10-21
Beta-carboline derivatives useful as inhibitors of phosphodiesterase
App 20030166641 - Sui, Zhihua ;   et al.
2003-09-04
6-O-carbamate-11,12-lacto-ketolide antimicrobials
App 20030125267 - Grant, Eugene B. III ;   et al.
2003-07-03
.beta.-carboline derivatives useful as inhibitors of phosphodiesterase
Grant 6,492,358 - Sui , et al. December 10, 2
2002-12-10
Substituted aminoalkylamide derivatives as antagonists of follicle stimulating hormone
App 20020058654 - Coats, Steven J. ;   et al.
2002-05-16
beta-carboline derivatives useful as inhibitors of phosphodiesterase
App 20020010189 - Sui, Zhihua ;   et al.
2002-01-24
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors
App 20020010183 - Sui, Zhihua ;   et al.
2002-01-24
5-heterocyclyl pyrazolo[4,3-d]pyrimidin-7-ones for the treatment of male erectile dysfunction
Grant 6,077,841 - Sui , et al. June 20, 2
2000-06-20
Peptide skeletal muscle relaxants
Grant 5,494,898 - Cheng , et al. February 27, 1
1996-02-27
Company Registrations

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