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Benzimidazole Derivatives Useful As Cb-1 Inverse Agonists App 20190031618 - Macielag; Mark J. ;   et al. | 2019-01-31 |
Benzimidazole derivatives useful as CB-1 inverse agonists Grant 10,118,900 - Macielag , et al. November 6, 2 | 2018-11-06 |
Chemically modified quinoline and quinolone derivatives useful as CB-1 inverse agonists Grant 9,815,790 - Macielag , et al. November 14, 2 | 2017-11-14 |
Indazole derivatives useful as CB-1 inverse agonists Grant 9,682,940 - Macielag , et al. June 20, 2 | 2017-06-20 |
Benzimidazole derivatives useful TRPM8 channel modulators Grant 9,636,345 - Macielag , et al. May 2, 2 | 2017-05-02 |
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Benzimidazole Derivatives Useful As Cb-1 Inverse Agonists App 20170057929 - Macielag; Mark J. ;   et al. | 2017-03-02 |
Chemically Modified Quinoline And Quinolone Derivatives Useful As Cb-1 Inverse Agonists App 20170057922 - Macielag; Mark J. ;   et al. | 2017-03-02 |
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Monoacylglycerol lipase inhibitors for the treatment of metabolic diseases and related disorders Grant 8,987,247 - Connelly , et al. March 24, 2 | 2015-03-24 |
Benzimidazole derivatives useful as TRPM8 channel modulators Grant 8,981,113 - Macielag , et al. March 17, 2 | 2015-03-17 |
Sulfonamides As Trpm8 Modulators App 20140315899 - Branum; Shawn T. ;   et al. | 2014-10-23 |
4-substituted-2-phenoxy-phenylamine delta opioid receptor modulators Grant 8,846,655 - Coats , et al. September 30, 2 | 2014-09-30 |
Heteroaromatic and aromatic piperazinyl azetidinyl amides as monoacylglycerol lipase inhibitors Grant 8,815,839 - Chevalier , et al. August 26, 2 | 2014-08-26 |
Sulfonamides as TRPM8 modulators Grant 8,809,327 - Branum , et al. August 19, 2 | 2014-08-19 |
Di-azetidinyl diamide as monoacylglycerol lipase inhibitors Grant 8,759,333 - Connolly , et al. June 24, 2 | 2014-06-24 |
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Amino-pyrrolidine-azetidine diamides as monoacylglycerol lipase inhibitors Grant 8,748,417 - Zhang , et al. June 10, 2 | 2014-06-10 |
Azetidinyl diamides as monoacylglycerol lipase inhibitors Grant 8,697,683 - Bian , et al. April 15, 2 | 2014-04-15 |
Pyrimidine compounds as delta opioid receptor modulators Grant 8,685,990 - Coats , et al. April 1, 2 | 2014-04-01 |
IMIDAZO[1,2-a]PYRIDINE SULFONAMIDES AS TRPM8 MODULATORS App 20140088098 - Macielag; Mark J. ;   et al. | 2014-03-27 |
Oxopiperazine-azetidine amides and oxodiazepine-azetidine amides as monoacylglycerol lipase inhibitors Grant 8,637,498 - Connolly , et al. January 28, 2 | 2014-01-28 |
Imidazo[1,2-.alpha.]pyridine sulfonamides as TRPM8 modulators Grant 8,618,150 - Macielag , et al. December 31, 2 | 2013-12-31 |
Imidazo[1,2-α]pyridine sulfonamides as TRPM8 modulators Grant 08618150 - | 2013-12-31 |
Pyrimidine Compounds As Delta Opioid Receptor Modulators App 20130310358 - Coats; Steven J. ;   et al. | 2013-11-21 |
Amino-pyrrolidine-azetidine diamides as monoacylglycerol lipase inhibitors Grant 8,575,363 - Zhang , et al. November 5, 2 | 2013-11-05 |
Azetidinyl Diamides As Monoacylglycerol Lipase Inhibitors App 20130244997 - Bian; Haiyan ;   et al. | 2013-09-19 |
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Azetidinyl Diamides As Monoacylglycerol Lipase Inhibitors App 20130237517 - Bian; Haiyan ;   et al. | 2013-09-12 |
Pyrimidine compounds as delta opioid receptor modulators Grant 8,513,271 - Coats , et al. August 20, 2 | 2013-08-20 |
Piperidin-4-yl-azetidine diamides as monoacylglycerol lipase inhibitors Grant 8,513,423 - Connolly , et al. August 20, 2 | 2013-08-20 |
Di-azetidinyl Diamide As Monoacylglcerol Lipase Inhibitors App 20130196969 - Connolly; Peter J. ;   et al. | 2013-08-01 |
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Heteroaromatic And Aromatic Piperazinyl Azetidinyl Amides As Monoacylglycerol Lipase Inhibitors App 20130184251 - Chevalier; Kristen ;   et al. | 2013-07-18 |
Benzimidazole derivatives useful as TRPM8 channel modulators Grant 8,450,497 - Macielag , et al. May 28, 2 | 2013-05-28 |
Piperidin-4-yl-azetidine Diamides As Monoacylglycerol Lipase Inhibitors App 20130102584 - Connolly; Peter J. ;   et al. | 2013-04-25 |
Monoacylglycerol Lipase Inhibitors For The Treatment Of Metabolic Diseases And Related Disorders App 20130085129 - Connelly; Margery ;   et al. | 2013-04-04 |
Monoacylglycerol Lipase Inhibitors For The Treatment Of Metabolic Diseases And Related Disorders App 20130085130 - Connelly; Margery ;   et al. | 2013-04-04 |
Hexahydro-cycloheptapyrazole cannabinoid modulators Grant 8,378,117 - Liotta , et al. February 19, 2 | 2013-02-19 |
4-substituted-2-phenoxy-phenylamine Delta Opioid Receptor Modulators App 20120302541 - Coats; Steven J. ;   et al. | 2012-11-29 |
Pyrazines as delta opioid receptor modulators Grant 8,293,750 - Connolly , et al. October 23, 2 | 2012-10-23 |
Benzimidazole derivatives useful as TRPM8 channel modulators Grant 8,242,157 - Jetter , et al. August 14, 2 | 2012-08-14 |
Pyrazines As Delta Opioid Receptor Modulators App 20120202824 - CONNOLLY; Peter J. ;   et al. | 2012-08-09 |
Sulfonamides As Trpm8 Modulators App 20120190674 - Branum; Shawn T. ;   et al. | 2012-07-26 |
IMIDAZO[1,2-a]PYRIDINE SULFONAMIDES AS TRPM8 MODULATORS App 20120149699 - Macielag; Mark J. ;   et al. | 2012-06-14 |
Pyrazines as delta opioid receptor modulators Grant 8,183,371 - Connolly , et al. May 22, 2 | 2012-05-22 |
Amino-pyrrolidine-azetidine Diamides As Monoacylglycerol Lipase Inhibitors App 20120101081 - Zhang; Yue-Mei ;   et al. | 2012-04-26 |
Sulfonamides as TRPM8 modulators Grant 8,153,682 - Branum , et al. April 10, 2 | 2012-04-10 |
Sulfonamides as TRPM8 modulators Grant 8,148,422 - Macielag , et al. April 3, 2 | 2012-04-03 |
Oxopiperazine-azetidine Amides And Oxodiazepine-azetidine Amides As Monoacylglycerol Lipase Inhibitors App 20120077797 - Connolly; Peter J. ;   et al. | 2012-03-29 |
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Pyrazines As Delta Opioid Receptor Modulators App 20110105527 - CONNOLLY; PETER J. ;   et al. | 2011-05-05 |
Pyrimidine Compounds As Delta Opioid Receptor Modulators App 20110105520 - COATS; STEVEN J. ;   et al. | 2011-05-05 |
C-7 isoxazolinyl quinolone / naphthyridine derivatives useful as antibacterial agents Grant 7,902,227 - Macielag , et al. March 8, 2 | 2011-03-08 |
Benzimidazole Derivatives Useful As Trpm8 Channel Modulators App 20110003800 - Macielag; Mark J. ;   et al. | 2011-01-06 |
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Hexahydro-cyclooctyl Pyrazole Cannabinoid Modulators App 20100317633 - Xia; Mingde ;   et al. | 2010-12-16 |
Hexahydro-cyclooctyl pyrazole cannabinoid modulators Grant 7,825,151 - Xia , et al. November 2, 2 | 2010-11-02 |
Antimicrobial oxazolidinone prodrugs Grant 7,776,855 - Macielag , et al. August 17, 2 | 2010-08-17 |
Sulfonamides As Trpm8 Modulators App 20100160289 - Macielag; Mark J. ;   et al. | 2010-06-24 |
Novel Rifamycin 3,4-(3-substituted Aminomethyl) Fused Pyrrolo Derivatives App 20100152267 - MACIELAG; Mark J. ;   et al. | 2010-06-17 |
7-amino alkylidenyl-heterocyclic quinolones and naphthyridones Grant 7,732,612 - Grant , et al. June 8, 2 | 2010-06-08 |
3-(substituted Ethyl)-rifamycin Derivatives Useful As Antimicrobial Agents App 20100029669 - MACIELAG; Mark J. ;   et al. | 2010-02-04 |
3-hydrazone Piperazinyl Rifamycin Derivatives Useful As Antimicrobial Agents App 20090275594 - MACIELAG; Mark J. ;   et al. | 2009-11-05 |
Quinolone Derivatives Useful As Antibacterial Agents App 20090270379 - Macielag; Mark J. ;   et al. | 2009-10-29 |
Sulfonamides As Trpm8 Modulators App 20090264474 - Branum; Shawn T. ;   et al. | 2009-10-22 |
Method For Treating Cb2 Receptor Mediated Pain App 20090215850 - Xia; Mingde ;   et al. | 2009-08-27 |
7-amino Alkylidenyl-heterocyclic Quinolones And Naphthyridones App 20090156577 - Davis; Benjamin ;   et al. | 2009-06-18 |
C-7 Isoxazolinyl Quinolone / Naphthyridine Derivatives Useful as Antibacterial Agents App 20090029980 - Macielag; Mark J. ;   et al. | 2009-01-29 |
Method For Treating Cb2 Receptor Mediated Pain App 20080234347 - Xia; Mingde ;   et al. | 2008-09-25 |
Hexahydro-Cyclooctyl Pyrazole Cannabinoid Modulators App 20080076814 - Xia; Mingde ;   et al. | 2008-03-27 |
Hexahydro-Cycloheptapyrazole Cannabinoid Modulators App 20080070968 - Liotta; Fina ;   et al. | 2008-03-20 |
Antimicrobial Oxazolidinone Prodrugs App 20080027053 - Macielag; Mark J. ;   et al. | 2008-01-31 |
Cyclohexyl derivatives as selective estrogen receptor modulators Grant 7,183,445 - Jain , et al. February 27, 2 | 2007-02-27 |
7-amino alkylidenyl-heterocyclic quinolones and naphthyridones Grant 7,179,805 - Grant, III , et al. February 20, 2 | 2007-02-20 |
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Inhibitors of bacterial Type III protein secretion systems App 20050272784 - Li, Xiaobing ;   et al. | 2005-12-08 |
11,12-Cyclic thiocarbamate macrolide antibacterial agents App 20050250713 - Zhu, Bin ;   et al. | 2005-11-10 |
Triazine compounds as inhibitors of bacterial type III protein secretion systems App 20050250945 - Li, Xiaobing ;   et al. | 2005-11-10 |
Inhibitors of bacterial type III protein secretion systems App 20050250819 - Li, Xiaobing ;   et al. | 2005-11-10 |
Neurotrophic pyrrolidines and piperidines, and related compositions and methods App 20050153951 - Kanojia, Ramesh M. ;   et al. | 2005-07-14 |
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors App 20050113402 - Sui, Zhihua ;   et al. | 2005-05-26 |
7-Amino alkylidenyl-heterocyclic quinolones and naphthyridones App 20050101588 - Grant, Eugene B. III ;   et al. | 2005-05-12 |
Benzo[4,5]thieno[2,3-c]pyridine and Benzo[4,5]furo[2,3-c]pyridine Derivatives Useful as Inhibitors of Phosphodiesterase Grant 6,864,253 - Sui , et al. March 8, 2 | 2005-03-08 |
Cyclohexyl derivatives as selective estrogen receptor modulators App 20050009799 - Jain, Nareshkumar F. ;   et al. | 2005-01-13 |
3-descladinosyl-6-O-carbamoyl and 6-O-carbonoyl macrolide antibacterial agents Grant 6,825,172 - Henninger , et al. November 30, 2 | 2004-11-30 |
6-O-acyl ketolide antibacterials Grant 6,825,170 - Henninger , et al. November 30, 2 | 2004-11-30 |
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors Grant 6,818,646 - Sui , et al. November 16, 2 | 2004-11-16 |
Neurotrophic pyrrolidines and piperidines, and related compositions and methods Grant 6,809,107 - Kanojia , et al. October 26, 2 | 2004-10-26 |
Substituted aminoalkylamide derivatives as antagonists of follicle stimulating hormone App 20040092505 - Coats, Steven J. ;   et al. | 2004-05-13 |
6-O-carbamate-11,12-lacto-ketolide antimicrobials Grant 6,713,455 - Grant, III , et al. March 30, 2 | 2004-03-30 |
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors App 20040044021 - Sui, Zhihua ;   et al. | 2004-03-04 |
3-Descladinosyl-6-O-carbamoyl and 6-O-carbonoyl macrolide antibacterial agents App 20040018994 - Henninger, Todd C. ;   et al. | 2004-01-29 |
6-O-acyl ketolide antibacterials App 20030220272 - Henninger, Todd C. ;   et al. | 2003-11-27 |
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors Grant 6,635,638 - Sui , et al. October 21, 2 | 2003-10-21 |
Beta-carboline derivatives useful as inhibitors of phosphodiesterase App 20030166641 - Sui, Zhihua ;   et al. | 2003-09-04 |
6-O-carbamate-11,12-lacto-ketolide antimicrobials App 20030125267 - Grant, Eugene B. III ;   et al. | 2003-07-03 |
.beta.-carboline derivatives useful as inhibitors of phosphodiesterase Grant 6,492,358 - Sui , et al. December 10, 2 | 2002-12-10 |
Substituted aminoalkylamide derivatives as antagonists of follicle stimulating hormone App 20020058654 - Coats, Steven J. ;   et al. | 2002-05-16 |
beta-carboline derivatives useful as inhibitors of phosphodiesterase App 20020010189 - Sui, Zhihua ;   et al. | 2002-01-24 |
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors App 20020010183 - Sui, Zhihua ;   et al. | 2002-01-24 |
5-heterocyclyl pyrazolo[4,3-d]pyrimidin-7-ones for the treatment of male erectile dysfunction Grant 6,077,841 - Sui , et al. June 20, 2 | 2000-06-20 |
Peptide skeletal muscle relaxants Grant 5,494,898 - Cheng , et al. February 27, 1 | 1996-02-27 |