Patent | Date |
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Compounds Useful In Hiv Therapy App 20220298160 - DE LA ROSA; Martha Alicia ;   et al. | 2022-09-22 |
4'-ethynyl-2'-deoxyadenosine Derivatives And Their Use In Hiv Therapy App 20220259252 - MILLER; John ;   et al. | 2022-08-18 |
SUBSTITUTED 1,2,3,3a,4,5,7,9,13,13a-DECAHYDROPYRIDO[1',2':4,5]PYRAZINO[1,2-a]PYRROLO[- 1,2-c]PYRIMIDINES HAVING HIV INTEGRASE INHIBITORY ACTIVITY App 20220213121 - JOHNS; Brian A. ;   et al. | 2022-07-07 |
Compounds Useful in HIV Therapy App 20220119417 - DE LA ROSA; Martha ;   et al. | 2022-04-21 |
Compounds Useful in HIV Therapy App 20220117993 - MILLER; John Franklin ;   et al. | 2022-04-21 |
Pharmaceutical Compositions App 20220096469 - MUNDHARA; Deepak B. ;   et al. | 2022-03-31 |
Methods For Treating Hiv With Dolutegravir And Lamivudine App 20220096487 - GARTLAND; Martin John | 2022-03-31 |
Substituted 1,2,3,3a,4,5,7,9,13,13a-decahydropyrido[1',2':4,5]pyrazino[1,2-a]pyrrolo[- 1,2-c]pyrimidines having HIV integrase inhibitory activity Grant 11,267,823 - Johns , et al. March 8, 2 | 2022-03-08 |
Antiviral therapy Grant 11,234,985 - Underwood February 1, 2 | 2022-02-01 |
Pharmaceutical compositions Grant 11,224,597 - Mundhra , et al. January 18, 2 | 2022-01-18 |
Antiviral Therapy App 20210401850 - Underwood; Mark Richard | 2021-12-30 |
Compounds Useful in HIV Therapy App 20210323993 - MILLER; John ;   et al. | 2021-10-21 |
Compositions and methods for the delivery of therapeutics Grant 11,117,904 - Edagwa , et al. September 14, 2 | 2021-09-14 |
Compositions And Methods For The Delivery Of Therapeutics App 20210230186 - EDAGWA; Benson J. ;   et al. | 2021-07-29 |
N-[(2,4-difluorophenyl)methyl]-6-hydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a- -hexahydro[1,3] oxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide having HIV integrase inhibitory activity Grant 10,927,129 - Johns , et al. February 23, 2 | 2021-02-23 |
Compounds Useful in HIV Therapy App 20210009609 - DE LA ROSA; Martha ;   et al. | 2021-01-14 |
Medical Use App 20200407393 - DE LA ROSA; Martha Alicia ;   et al. | 2020-12-31 |
Compounds useful in HIV therapy Grant 10,870,663 - Dunham , et al. December 22, 2 | 2020-12-22 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20200339598 - JOHNS; Brian A. ;   et al. | 2020-10-29 |
Compounds Useful in HIV Therapy App 20200299309 - DUNHAM; Richard M ;   et al. | 2020-09-24 |
Regimens and compositions for treating HIV infections and AIDS Grant 10,758,531 - Spreen Sep | 2020-09-01 |
Combinations And Uses And Treatments Thereof App 20200246351 - Kind Code | 2020-08-06 |
Antiviral Therapy App 20200230147 - UNDERWOOD; Mark Richard | 2020-07-23 |
Bi-layer Pharmaceutical Tablet Formulation App 20200230141 - KAYE; Jonathan Louis | 2020-07-23 |
Combinations And Uses And Treatments App 20200171039 - COCKETT; Mark I. ;   et al. | 2020-06-04 |
Process for preparing (3S,11aR)-N-(2,4-difluorobenzyl)-6-hydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,- 11a-hexahydrooxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide Grant 10,654,871 - Goodman , et al. | 2020-05-19 |
Process for preparing substituted pyridinones as intermediates in the preparation of polycyclic carbamoylpyridone derivatives Grant 10,654,870 - Goodman , et al. | 2020-05-19 |
Regimens For Treating Hiv Infections And Aids App 20200147092 - ABOUD; Michael ;   et al. | 2020-05-14 |
Regimens For Treating Hiv Infections And Aids App 20200147079A1 - | 2020-05-14 |
Process for preparing (3S,11aR)-6-methoxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a-Hexahydrooxazolo[3,- 2-a]pyrido[1,2-d]pyrazine-8-carboxylic acid Grant 10,647,728 - Goodman , et al. | 2020-05-12 |
Combination Drug Therapy App 20200138845 - SCOTT; Trevor R. | 2020-05-07 |
Combination And Uses And Treatments Thereof App 20200113838A1 - | 2020-04-16 |
Antiviral therapy Grant 10,426,780 - Underwood October 1, 2 | 2019-10-01 |
N-[(2,4-DIFLUOROPHENYL)METHYL]-6-HYDROXY-3-METHYL-5,7-DIOXO-2,3,5,7,11,11a- -HEXAHYDRO[1,3]OXAZOLO[3,2-a]PYRIDO[1,2-d]PYRAZINE-8 App 20190284208 - JOHNS; Brian A. ;   et al. | 2019-09-19 |
Combinations And Uses And Treatments Thereof App 20190183901 - JOHNS; Brian Alvin | 2019-06-20 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20190152990 - JOHNS; Brian A. ;   et al. | 2019-05-23 |
Regimens And Compositions For Treating Hiv Infections And Aids App 20190142828 - SPREEN; William R. | 2019-05-16 |
Process For Preparing Carbamoylpyridone Derivatives And Intermediates App 20190106435 - GOODMAN; Steven N. ;   et al. | 2019-04-11 |
Process For Preparing Carbamoylpyridone Derivatives And Intermediates App 20190100533 - GOODMAN; Steven N. ;   et al. | 2019-04-04 |
Process For Preparing Pyridinone Carboxylic Acid Derivatives And Intermediates App 20190100532 - Goodman; Steven N. ;   et al. | 2019-04-04 |
Process for preparing substituted pyridinones as intermediates in the preparation of polycyclic carbamoylpyridone derivatives Grant 10,233,196 - Goodman , et al. | 2019-03-19 |
Substituted pyridinones as intermediates in the preparation of polycyclic carbamoylpyridone derivatives Grant 10,174,051 - Goodman , et al. J | 2019-01-08 |
Antiviral Therapy App 20180200254 - UNDERWOOD; Mark Richard | 2018-07-19 |
Process For Preparing Carbamoylpyridone Derivatives Andintermediates App 20180186812 - Goodman; Steven N. ;   et al. | 2018-07-05 |
Process for preparing carbamoylpyridone derivatives and intermediates App 20180186811 - GOODMAN; Steven N. ;   et al. | 2018-07-05 |
Antiviral Therapy App 20180098992 - UNDERWOOD; Mark Richard | 2018-04-12 |
Process for preparing (4R,12aS)-N-(2,4-difluorobenzyl)-7-hydroxy-4-methyl-6,8-dioxo-3,4,6,8,12,- 12a-hexahydro-2H-pyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazine-9-carboxamid- e Grant 9,938,296 - Goodman , et al. April 10, 2 | 2018-04-10 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170369509 - JOHNS; Brian A. ;   et al. | 2017-12-28 |
Antiviral Therapy App 20170281636 - UNDERWOOD; Mark Richard | 2017-10-05 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170267693 - JOHNS; Brian A. ;   et al. | 2017-09-21 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170260203 - JOHNS; Brian A. ;   et al. | 2017-09-14 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170253616 - JOHNS; Brian A. ;   et al. | 2017-09-07 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170224694 - JOHNS; Brian A. ;   et al. | 2017-08-10 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170224695 - JOHNS; Brian A. ;   et al. | 2017-08-10 |
Antiviral Therapy App 20170216284 - UNDERWOOD; Mark Richard | 2017-08-03 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170209454 - JOHNS; Brian A. ;   et al. | 2017-07-27 |
PROCESS FOR PREPARING (4R,12aS)-N-(2,4-DIFLUOROBENZYL)-7-METHOXY-4-METHYL-6,8-DIOXO-3,4,6,8,12,- - 12A-HEXAHYDRO-2H-PYRIDO[1',2':4,5]PYRAZINO[2,1-b][1,3]OXAZINE-9-CARBOXAM- IDE App 20170204117 - GOODMAN; Steven N. ;   et al. | 2017-07-20 |
Substituted (3S,11AR)-N-[(2,4-difluorophenyl)methyl]-6-oxy-3-methyl-5,7-dioxo-2,3,5,7- ,11,11A-hexahydro[1,3]oxazolo[3,2-A]pyrido[1,2-D]pyrazine-8-carboxamides as HIV agents Grant 9,707,246 - Johns , et al. July 18, 2 | 2017-07-18 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170145033 - JOHNS; Brian A. ;   et al. | 2017-05-25 |
Process for preparing (4R,12aS)-N-(2,4-difluorobenzyl)-7-methoxy-4-methyl-6,8-dioxo-3,4,6,8,12,- 12A-hexahydro-2H-pyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazine-9-carboxamid- e Grant 9,643,981 - Goodman , et al. May 9, 2 | 2017-05-09 |
Antiviral Therapy App 20170119777 - UNDERWOOD; Mark Richard | 2017-05-04 |
Antiviral Therapy App 20170079982 - UNDERWOOD; Mark Richard | 2017-03-23 |
Pharmaceutical Compositions App 20170027933 - MUNDHRA; Deepak B. ;   et al. | 2017-02-02 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170029438 - JOHNS; Brian A. ;   et al. | 2017-02-02 |
Antiviral Therapy App 20160339033 - Underwood; Mark Richard | 2016-11-24 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20160304535 - JOHNS; Brian A. ;   et al. | 2016-10-20 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20160207939 - JOHNS; Brian A. ;   et al. | 2016-07-21 |
Antiviral Therapy App 20160199379 - Underwood; Mark Richard | 2016-07-14 |
Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates Grant 9,365,587 - Yoshida , et al. June 14, 2 | 2016-06-14 |
SUBSTITUTED CYCLOPENTA[4,5]OXAZOLO[3,2-a]PYRIDO[1,2-d]PYRAZINES AS HIV INTEGRASE INHIBITORS App 20160137666 - Johns; Brian Alvin ;   et al. | 2016-05-19 |
Synthesis Of Carbamoylpyridone Hiv Integrase Inhibitors And Intermediates App 20160060274 - YOSHIDA; Hiroshi ;   et al. | 2016-03-03 |
Substituted pyrido[1',2':4,5]pyrazino[1,2-a]pyrimidines as HIV integrase inhibitors Grant 9,273,065 - Johns , et al. March 1, 2 | 2016-03-01 |
Chemical Compounds App 20150335667 - JOHNS; Brian Alvin ;   et al. | 2015-11-26 |
PROCESS FOR PREPARING (4R,12aS)-N-(2,4-DIFLUOROBENZYL)-7-METHOXY-4-METHYL-6,8-DIOXO-3,4,6,8,12,- 12A-HEXAHYDRO-2H-PYRIDO[1',2':4,5]PYRAZINO[2,1-b][1,3]OXAZINE-9-CARBOXAMID- E App 20150329559 - GOODMAN; Steven N. ;   et al. | 2015-11-19 |
(3S,11aR)-6-[(phenylmethyl)oxy]-3-methyl-2,3,11,11a-tetrahydrooxazolo[3,2-- a]pyrido[1,2-d]pyrazine-5,7-dione of the formula P-9 and/or (3S,11aR)-6-[(phenymethyl)oxy]-8-bromo-3-methyl-2,3,11,11a-tetrahydrooxaz- olo[3,2-a]pyrido[1,2-d]pyrazine-5,7-dione of the formula P-10 Grant 9,133,216 - Johns , et al. September 15, 2 | 2015-09-15 |
Process for preparing (4R,12aS)-7-methoxy-4-methyl-6,8-dioxo-3,4,6,8,12,12a-hexahydro-2H-pyrido- [1' ,2':4,5]pyrazino[2,1-b][1,3]oxazine-9-carboxylic acid Grant 9,120,817 - Goodman , et al. September 1, 2 | 2015-09-01 |
Antiviral Therapy App 20150238496 - Underwood; Mark Richard | 2015-08-27 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20150232479 - JOHNS; Brian A. ;   et al. | 2015-08-20 |
Hiv Integrase Inhibitors App 20150225399 - JOHNS; Brian Alvin ;   et al. | 2015-08-13 |
(3S,11aR)-6-[(PHENYLMETHYL)OXY]-3-METHYL-2,3,11,11a-TETRAHYDROOXAZOLO[3,2-- a]PYRIDO[1,2-d]PYRAZINE-5,7-DIONE OF THE FORMULA P-9 AND/OR (3S,11aR)-6-[(PHENYLMETHYL)OXY]-8-BROMO-3-METHYL-2,3,11,11a-TETRAHYDROOXA- ZOLO[3,2-a]PYRIDO[1,2-d]PYRAZINE-5,7-DIONE OF THE FORMULA P-10 App 20150183803 - JOHNS; Brian Alvin ;   et al. | 2015-07-02 |
Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-a]pyrr- olo[1',2':3,4]imidazo[1,2-d]pyrazine-8-carboxamides Grant 9,051,337 - Johns , et al. June 9, 2 | 2015-06-09 |
Substituted (3S, 11aR)-N-[(2,4-difluorophenyl)methyl]-6-oxy-3-methyl-5,7-dioxo-2,3,5,7,11,- 11a-hexahydro[1,3]oxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamides of formula (I) useful as HIV agents Grant 9,012,650 - Johns , et al. April 21, 2 | 2015-04-21 |
2-(2-hydroxy-2-phenylethyl)-3-[(phenylmethyl)oxy]-4H-pyran-4-one of the formula P-3 and/or 2-[(E)-2-phenylethenyl]-3-[(phenylmethyl)oxy]-4H-Pyran-4-one of the formula P-4 Grant 8,981,129 - Johns , et al. March 17, 2 | 2015-03-17 |
Process for Preparing Pyridinone Carboxylic Acid Aldehydes App 20150057444 - Goodman; Steven N. ;   et al. | 2015-02-26 |
4-oxo-3-[(phenylmethyl)oxy]-4H-pyran-2-carboxylic acid Grant 8,940,912 - Johns , et al. January 27, 2 | 2015-01-27 |
Processes for preparing pyridinone carboxylic acid aldehydes Grant 8,889,877 - Goodman , et al. November 18, 2 | 2014-11-18 |
Chemical Compounds App 20140256679 - JOHNS; Brian Alvin ;   et al. | 2014-09-11 |
2-oxonaphthyridine-3-carboxamides Hiv Integrase Inhibitors App 20140256713 - JOHNS; Brian Alvin ;   et al. | 2014-09-11 |
Chemical Compounds App 20140256961 - JOHNS; Brian Alvin ;   et al. | 2014-09-11 |
Synthesis Of Carbamoylpyridone Hiv Integrase Inhibitors And Intermediates App 20140243521 - YOSHIDA; Hiroshi ;   et al. | 2014-08-28 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20140200209 - JOHNS; Brian A. ;   et al. | 2014-07-17 |
Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-.alpha- .]pyrrolo[1',2':3,4]imidazo[1,2-d]pyrazine-8-carboxamides Grant 8,778,943 - Johns , et al. July 15, 2 | 2014-07-15 |
1-(2,3-dihydroxypropyl)-4-oxo-3-[(phenylmethyl)oxy]-1,4-dihydro-2-pyridine- carboxylic acid of the formula P-6 and/or methyl 1-(2,3-dihydroxypropyl)-4-oxo-3-[(phenylmethyl)oxy]-1,4-dihydro-2-pyridin- ecarboxylate of the formula P-7 Grant 8,765,965 - Johns , et al. July 1, 2 | 2014-07-01 |
Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates Grant 8,754,214 - Yoshida , et al. June 17, 2 | 2014-06-17 |
2-oxonaphthyridine-3-carboxamides HIV integrase inhibitors Grant 8,691,991 - Johns , et al. April 8, 2 | 2014-04-08 |
Prodrugs of (4aS, 13ar)-N-[(2,4-difluorophenyl)methyl]-10-hydroxy-9-11-dioxo-2,3,4a,5,9,11,- 13,13a-octahydro-1H-pyrido[1,2-a]pyrrolo[1',2':3:4]imidazo[1,2-d]pyrazine-- 8-carboxamide and their use in the treatment of HIV infection Grant 8,691,823 - Johns , et al. April 8, 2 | 2014-04-08 |
Synthesis Of Carbamoylpyridone Hiv Integrase Inhibitors And Intermediates App 20140094605 - YOSHIDA; Hiroshi ;   et al. | 2014-04-03 |
Processes and Intermediates for carbamoylpyridone HIV integrase inhibitors Grant 8,669,362 - Johns , et al. March 11, 2 | 2014-03-11 |
Chemical Compounds App 20140039207 - JOHNS; Brian Alvin ;   et al. | 2014-02-06 |
Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates Grant 8,624,023 - Yoshida , et al. January 7, 2 | 2014-01-07 |
Processes And Intermediates For Carbamoylpyridone Hiv Integrase Inhibitors App 20140005405 - JOHNS; Brian ;   et al. | 2014-01-02 |
Methyl 3-(benzyloxy)-1-(2,2-dihydroxyethyl)-4-oxo-1,4-dihydropyridine-2-ca- rboxylate and processes for the preparation thereof Grant 8,580,967 - Johns , et al. November 12, 2 | 2013-11-12 |
Processes and intermediates for carbamoylpyridone HIV integrase inhibitors Grant 8,552,187 - Johns , et al. October 8, 2 | 2013-10-08 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20130172559 - JOHNS; Brian A. ;   et al. | 2013-07-04 |
Pharmaceutical Compositions App 20130171214 - Mundhra; Deepak B. ;   et al. | 2013-07-04 |
(3S,11aR)-N-[2,4-difluorophenyl)methyl]-6-hydroxy-3-methyl-5,7-dioxo-2,3,5- ,7,11,11a-hexahydro[1,3]oxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide useful as anti-HIV agent Grant 8,410,103 - Johns , et al. April 2, 2 | 2013-04-02 |