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Annelated N-heterocyclic sulfonamides with oxadiazolone headgroup, processes for their preparation and their use as pharmaceuticals Grant 8,946,212 - Keil , et al. February 3, 2 | 2015-02-03 |
Use of substituted pyranone acid derivatives for the treatment of metabolic syndrome Grant 8,748,483 - Brummerhop , et al. June 10, 2 | 2014-06-10 |
Regioselective copper catalyzed synthesis of benzimidazoles and azabenzimidazoles Grant 8,735,586 - Alonso , et al. May 27, 2 | 2014-05-27 |
Sulfonamides with heterocycle and oxadiazolone headgroup, processes for their preparation and their use as pharmaceuticals Grant 8,716,317 - Keil , et al. May 6, 2 | 2014-05-06 |
Process for the palladium-catalyzed coupling of terminal alkynes with aryl tosylates Grant 8,487,109 - Rkyek , et al. July 16, 2 | 2013-07-16 |
Process for the palladium-catalyzed coupling of terminal alkynes with heteroaryl tosylates and heteroaryl benzenesulfonates Grant 8,420,812 - Rkyek , et al. April 16, 2 | 2013-04-16 |
Cyclic pyridyl-N-[1,3,4]-thiadiazol-2-yl-benzene sulfonamides, processes for their preparation and their use as pharmaceuticals Grant 8,344,004 - Schoenafinger , et al. January 1, 2 | 2013-01-01 |
Annelated pyrrolidin sulfonamides with oxadiazolone headgroup, processes for their preparation and their use as pharmaceuticals Grant 8,329,725 - Keil , et al. December 11, 2 | 2012-12-11 |
Transition metal catalyzed synthesis of 2H-indazoles Grant 8,283,476 - Halland , et al. October 9, 2 | 2012-10-09 |
Sulfonamides With Heterocycle And Oxadiazolone Headgroup, Processes For Their Preparation And Their Use As Pharmaceuticals App 20120172400 - Keil; Stefanie ;   et al. | 2012-07-05 |
Regioselective palladium catalyzed synthesis of benzimidazoles and azabenzimidazoles Grant 8,188,282 - Alonso , et al. May 29, 2 | 2012-05-29 |
Annelated N-heterocyclic Sulfonamides With Oxadiazolone Headgroup, Processes For Their Preparation And Their Use As Pharmaceuticals App 20120122853 - Keil; Stefanie ;   et al. | 2012-05-17 |
Sulfonyl-phenyl-2H-[1,2,4]oxadiazol-5-one derivatives, processes for their preparation and their use as pharmaceuticals Grant 8,173,674 - Keil , et al. May 8, 2 | 2012-05-08 |
Heteroaryl-carboxylic acid (sulfamoyl alkyl) amide-derivatives as factor Xa inhibitors Grant 8,088,925 - Wagner , et al. January 3, 2 | 2012-01-03 |
Transition metal catalyzed synthesis of N-aminoindoles Grant 8,026,375 - Halland , et al. September 27, 2 | 2011-09-27 |
Cyclic pyridyl-N-[1,3,4]-thiadiazol-2-yl-benzene sulfonamides, processes for their preparation and their use as pharmaceuticals App 20110224263 - SCHOENAFINGER; Karl ;   et al. | 2011-09-15 |
Annelated Pyrrolidin Sulfonamides With Oxadiazolone Headgroup, Processes For Their Preparation And Their Use As Pharmaceuticals App 20110207738 - Keil; Stefanie ;   et al. | 2011-08-25 |
4-oxy-N-[1,3,4]-thiadiazol-2-yl-benzene sulfonamides, pharmaceutical compositions and methods for their therapeutic use Grant 7,910,612 - Keil , et al. March 22, 2 | 2011-03-22 |
N-[1,3,4]-thiadiazol-2-yl-benzene sulfonamides, pharmaceutical compositions thereof and methods for their therapeutic use Grant 7,858,647 - Keil , et al. December 28, 2 | 2010-12-28 |
Phenyl-1,2,4-oxadiazolone derivatives with phenyl group, processes for their preparation and their use as pharmaceuticals Grant 7,851,493 - Bernardelli , et al. December 14, 2 | 2010-12-14 |
Phenyl-[1,2,4]-oxadiazol-5-one derivatives, pharmaceutical compositions and therapeutic use thereof Grant 7,834,030 - Keil , et al. November 16, 2 | 2010-11-16 |
Regioselective copper catalyzed synthesis of benzimidazoles and azabenzimidazoles App 20100261909 - ALONSO; Jorge ;   et al. | 2010-10-14 |
Process for the palladium-catalyzed coupling of terminal alkynes with aryl tosylates App 20100261910 - RKYEK; Omar ;   et al. | 2010-10-14 |
Process for the palladium-catalyzed coupling of terminal alkynes with heteroaryl tosylates and heteroaryl benzenesulfonates App 20100261900 - RKYEK; Omar ;   et al. | 2010-10-14 |
Transition metal catalyzed synthesis of 2H-indazoles App 20100234601 - HALLAND; Nis ;   et al. | 2010-09-16 |
Regioselective metal catalyzed synthesis of annelated benzimidazoles and azabenzimidazoles App 20100216988 - ALONSO; Jorge ;   et al. | 2010-08-26 |
Bicyclic aryl-sulfonic acid [1,3,4]-thiadiazol-2-yl-amides, processes for their preparation, pharmaceutical compositions and methods for their use Grant 7,772,257 - Schoenafinger , et al. August 10, 2 | 2010-08-10 |
Heterocyclic substituted carbonyl derivatives and their use as dopamine D.sub.3 receptor ligands Grant 7,772,252 - Hendrix , et al. August 10, 2 | 2010-08-10 |
Transition metal catalyzed synthesis of N-aminoindoles App 20100168429 - HALLAND; Nis ;   et al. | 2010-07-01 |
Benzimidazole-derivatives as factor Xa inhibitors Grant 7,741,341 - Nazare , et al. June 22, 2 | 2010-06-22 |
Use Of Substituted Pyranone Acid Derivatives For The Treatment Of Metabolic Syndrome App 20100144862 - BRUMMERHOP; Harm ;   et al. | 2010-06-10 |
Phenyl-1,2,4-oxadiazolone derivatives, processes for their preparation and methods for their use as pharmaceuticals Grant 7,709,481 - Keil , et al. May 4, 2 | 2010-05-04 |
Cyclic N-[1,3,4]-thiadiazol-2-yl-benzene sulfonamides, pharmaceutical compositions and methods for the therapeutic use thereof Grant 7,683,181 - Schoenafinger , et al. March 23, 2 | 2010-03-23 |
Derivatives of 2-aminothiazoles and 2-amino-oxazoles, processes for their preparation and their use as pharmaceutical compositions Grant 7,655,679 - Keil , et al. February 2, 2 | 2010-02-02 |
Bicyclic Aryl-sulfonic Acid [1,3,4]-thiadiazol-2-yl-amides, Processes For Their Preparation, Pharmaceutical Compositions And Methods For Their Use App 20100022603 - SCHOENAFINGER; Karl ;   et al. | 2010-01-28 |
Sulfonyl-phenyl-2h-[1,2,4]oxadiazol-5-one Derivatives , Processes For Their Preparation And Their Use As Pharmaceuticals App 20090298871 - KEIL; Stefanie ;   et al. | 2009-12-03 |
Phenyl-1,2,4-oxadiazolone Derivatives With Phenyl Group, Processes For Their Preparation And Their Use As Pharmaceuticals App 20090281084 - Bernardelli; Patrick ;   et al. | 2009-11-12 |
Bicyclic aryl-sulfonic acid [1,3,4]-thiadiazol-2-yl-amides, processes for their preparation, pharmaceutical compositions and methods for their use Grant 7,612,104 - Schoenafinger , et al. November 3, 2 | 2009-11-03 |
Novel Heterocyclic Substituted Carbonyl Derivatives and Their Use as Dopamine D3 Receptor Ligands App 20090247509 - Hendrix; James A. ;   et al. | 2009-10-01 |
Regioselective palladium catalyzed synthesis of benzimidazoles and azabenzimidazoles App 20090203912 - ALONSO; Jorge ;   et al. | 2009-08-13 |
Heterocyclic amide derivatives and their use as dopamine D3 receptor ligands Grant 7,550,469 - Hendrix , et al. June 23, 2 | 2009-06-23 |
Heterocyclic substituted carbonyl derivatives and their use as dopamine D.sub.3 receptor ligands Grant 7,521,445 - Hendrix , et al. April 21, 2 | 2009-04-21 |
4-oxy-n-[1,3,4]-thiadiazol-2-yl-benzene Sulfonamides, Pharmaceutical Compositions And Methods For Their Therapeutic Use App 20090012131 - KEIL; Stefanie ;   et al. | 2009-01-08 |
Pyrrole-derivatives as factor Xa inhibitors Grant 7,465,806 - Bauer , et al. December 16, 2 | 2008-12-16 |
Bicyclic Aryl-sulfonic Acid [1,3,4]-thiadiazol-2-yl-amides, Processes For Their Preparation, Pharmaceutical Compositions And Methods For Their Use App 20080293780 - SCHOENAFINGER; Karl ;   et al. | 2008-11-27 |
Phenyl And Pyridinyl-1,2,4-oxadiazolone Derivatives, Processes For Their Preparation And Their Use As Pharmaceutical Compositions App 20080287409 - Bernardelli; Patrick ;   et al. | 2008-11-20 |
Azaindole-Derivatives As Factor Xa Inhibitors App 20080280946 - NAZARE; Marc ;   et al. | 2008-11-13 |
Cyclic N-[1,3,4]-thiadiazol-2-yl-benzene Sulfonamides, Pharmaceutical Compositions And Methods For The Therapeutic Use Thereof App 20080280959 - SCHOENAFINGER; Karl ;   et al. | 2008-11-13 |
Phosophoinositoglycan binding proteins Grant 7,449,560 - Mueller , et al. November 11, 2 | 2008-11-11 |
Phenyl-[1,2,4]-oxadiazol-5-one Derivatives, Pharmaceutical Compositions and Therapeutic Use Thereof App 20080262036 - Keil; Stefanie ;   et al. | 2008-10-23 |
Phenyl-1,2,4-Oxadiazolone Derivatives, Processes For Their Preparation and Methods For Their Use as Pharmaceuticals App 20080261979 - Keil; Stefanie ;   et al. | 2008-10-23 |
Derivatives Of 2-aminothiazoles And 2-amino-oxazoles, Processes For Their Preparation And Their Use As Pharmaceutical Compositions App 20080227834 - Keil; Stefanie ;   et al. | 2008-09-18 |
Heteroaryl-carboxylic Acid (sulfamoyl Alkyl) Amide - Derivatives As Factor Xa Inhibitors App 20080167346 - WAGNER; Michael ;   et al. | 2008-07-10 |
Indazole-derivatives as factor Xa inhibitors Grant 7,365,088 - Nazare , et al. April 29, 2 | 2008-04-29 |
Azaindole-derivatives as factor Xa inhibitors Grant 7,317,027 - Nazare , et al. January 8, 2 | 2008-01-08 |
Beta-Aminoacid-Derivatives As Factor Xa Inhibitors App 20070179122 - Urmann; Matthias ;   et al. | 2007-08-02 |
Novel heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands App 20070161641 - Hendrix; James A. ;   et al. | 2007-07-12 |
Novel heterocyclic amide derivatives and their use as dopamine D3 receptor ligands App 20070142351 - Hendrix; James A. ;   et al. | 2007-06-21 |
Heterocyclic substituted carbonyl derivatives and their use as dopamine D.sub.3 receptor ligands Grant 7,186,724 - Hendrix , et al. March 6, 2 | 2007-03-06 |
Pyrrole-Derivatives as Factor Xa Inhibitors App 20070049573 - BAUER; Armin ;   et al. | 2007-03-01 |
Phosophoinositoglycan binding proteins App 20060160142 - Mueller; Guenter ;   et al. | 2006-07-20 |
Phosophoinositoglycan binding proteins Grant 7,049,416 - Mueller , et al. May 23, 2 | 2006-05-23 |
Novel heterocyclic amide derivatives and their use as dopamine D3 receptor ligands App 20050107389 - Hendrix, James A. ;   et al. | 2005-05-19 |
Benzimidazole-derivatives as factor Xa inhibitors App 20050009829 - Nazare, Marc ;   et al. | 2005-01-13 |
Azaindole-derivatives as factor Xa inhibitors App 20050009828 - Nazare, Marc ;   et al. | 2005-01-13 |
Indazole-derivatives as factor Xa inhibitors App 20040235824 - Nazare, Marc ;   et al. | 2004-11-25 |
Phosophoinositoglycan binding proteins App 20040229278 - Mueller, Guenter ;   et al. | 2004-11-18 |
Novel heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor App 20040220173 - Hendrix, James A. ;   et al. | 2004-11-04 |
Novel heterocyclic amide derivatives and their use as dopamine D3 receptor ligands App 20040030137 - Hendrix, James A. ;   et al. | 2004-02-12 |
Novel heterocyclic urea derivatives and their use as dopamine D3 receptor ligands App 20030229066 - Hendrix, James A. ;   et al. | 2003-12-11 |