Patent | Date |
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Polycyclic pyridone derivative Grant 11,453,669 - Taoda September 27, 2 | 2022-09-27 |
SUBSTITUTED 1,2,3,3a,4,5,7,9,13,13a-DECAHYDROPYRIDO[1',2':4,5]PYRAZINO[1,2-a]PYRROLO[- 1,2-c]PYRIMIDINES HAVING HIV INTEGRASE INHIBITORY ACTIVITY App 20220213121 - JOHNS; Brian A. ;   et al. | 2022-07-07 |
Substituted 1,2,3,3a,4,5,7,9,13,13a-decahydropyrido[1',2':4,5]pyrazino[1,2-a]pyrrolo[- 1,2-c]pyrimidines having HIV integrase inhibitory activity Grant 11,267,823 - Johns , et al. March 8, 2 | 2022-03-08 |
Arenavirus Growth Inhibitor Comprising Polycyclic Carbamoyl Pyridone Derivative App 20210292321 - ISHII; Akihiro ;   et al. | 2021-09-23 |
Polycyclic Pyridone Derivative App 20210155622 - TAODA; Yoshiyuki | 2021-05-27 |
Polycyclic Carbamoylpyridone Derivative App 20210122751 - TAODA; Yoshiyuki ;   et al. | 2021-04-29 |
N-[(2,4-difluorophenyl)methyl]-6-hydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a- -hexahydro[1,3] oxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide having HIV integrase inhibitory activity Grant 10,927,129 - Johns , et al. February 23, 2 | 2021-02-23 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20200339598 - JOHNS; Brian A. ;   et al. | 2020-10-29 |
Prodrug Substituted Polycyclic Carbamoyl Pyridone Derivative App 20200339565 - TAKAHASHI; Chika ;   et al. | 2020-10-29 |
N-[(2,4-DIFLUOROPHENYL)METHYL]-6-HYDROXY-3-METHYL-5,7-DIOXO-2,3,5,7,11,11a- -HEXAHYDRO[1,3]OXAZOLO[3,2-a]PYRIDO[1,2-d]PYRAZINE-8 App 20190284208 - JOHNS; Brian A. ;   et al. | 2019-09-19 |
Substituted Polycyclic Carbamoyl Pyridone Derivative Prodrug App 20190248785 - TAKAHASHI; Chika ;   et al. | 2019-08-15 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20190152990 - JOHNS; Brian A. ;   et al. | 2019-05-23 |
Substituted polycyclic carbamoyl pyridone derivative prodrug Grant 10,202,379 - Takahashi , et al. Feb | 2019-02-12 |
Hiv Replication Inhibitor App 20180362543 - TOMITA; Kenji ;   et al. | 2018-12-20 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170369509 - JOHNS; Brian A. ;   et al. | 2017-12-28 |
Substituted Polycyclic Carbamoyl Pyridone Derivative Prodrug App 20170349587 - Takahashi; Chika ;   et al. | 2017-12-07 |
Substituted polycyclic carbamolypyridone derivative Grant 9,815,835 - Akiyama , et al. November 14, 2 | 2017-11-14 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170267693 - JOHNS; Brian A. ;   et al. | 2017-09-21 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170260203 - JOHNS; Brian A. ;   et al. | 2017-09-14 |
Substituted polycyclic carbamoyl pyridone derivative prodrug Grant 9,758,515 - Takahashi , et al. September 12, 2 | 2017-09-12 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170253616 - JOHNS; Brian A. ;   et al. | 2017-09-07 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170224695 - JOHNS; Brian A. ;   et al. | 2017-08-10 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170224694 - JOHNS; Brian A. ;   et al. | 2017-08-10 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170209454 - JOHNS; Brian A. ;   et al. | 2017-07-27 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170145033 - JOHNS; Brian A. ;   et al. | 2017-05-25 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170029438 - JOHNS; Brian A. ;   et al. | 2017-02-02 |
Substituted-quinoxaline-type piperidine compounds and the uses thereof Grant 9,527,840 - Fuchino , et al. December 27, 2 | 2016-12-27 |
Substituted Polycyclic Carbamolypyridone Derivative App 20160368921 - AKIYAMA; Toshiyuki ;   et al. | 2016-12-22 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20160304535 - JOHNS; Brian A. ;   et al. | 2016-10-20 |
Substituted polycyclic carbamoylpyridone derivative Grant 9,469,638 - Akiyama , et al. October 18, 2 | 2016-10-18 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20160207939 - JOHNS; Brian A. ;   et al. | 2016-07-21 |
Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates Grant 9,365,587 - Yoshida , et al. June 14, 2 | 2016-06-14 |
Substituted-quinoxaline-type Piperidine Compounds And The Uses Thereof App 20160159785 - FUCHINO; Kouki ;   et al. | 2016-06-09 |
SUBSTITUTED CYCLOPENTA[4,5]OXAZOLO[3,2-a]PYRIDO[1,2-d]PYRAZINES AS HIV INTEGRASE INHIBITORS App 20160137666 - Johns; Brian Alvin ;   et al. | 2016-05-19 |
Substituted-quinoxaline-type piperidine compounds and the uses thereof Grant 9,278,967 - Fuchino , et al. March 8, 2 | 2016-03-08 |
Synthesis Of Carbamoylpyridone Hiv Integrase Inhibitors And Intermediates App 20160060274 - YOSHIDA; Hiroshi ;   et al. | 2016-03-03 |
Substituted pyrido[1',2':4,5]pyrazino[1,2-a]pyrimidines as HIV integrase inhibitors Grant 9,273,065 - Johns , et al. March 1, 2 | 2016-03-01 |
Hiv Replication Inhibitor App 20150361093 - TOMITA; Kenji ;   et al. | 2015-12-17 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20150232479 - JOHNS; Brian A. ;   et al. | 2015-08-20 |
Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-a]pyrr- olo[1',2':3,4]imidazo[1,2-d]pyrazine-8-carboxamides Grant 9,051,337 - Johns , et al. June 9, 2 | 2015-06-09 |
Substituted-quinoxaline-type Piperidine Compounds And The Uses Thereof App 20150141643 - FUCHINO; Kouki ;   et al. | 2015-05-21 |
Substituted Polycyclic Carbamoyl Pyridone Derivative Prodrug App 20150111854 - TAKAHASHI; Chika ;   et al. | 2015-04-23 |
Substituted polycyclic carbamoyl pyridone derivative prodrug Grant 8,987,441 - Takahashi , et al. March 24, 2 | 2015-03-24 |
Substituted Polycyclic Carbamoylpyridone Derivative App 20150065485 - Akiyama; Toshiyuki ;   et al. | 2015-03-05 |
Substituted polycyclic carbamoylpyridone derivative Grant 8,927,710 - Akiyama , et al. January 6, 2 | 2015-01-06 |
Substituted-quinoxaline-type piperidine compounds and the uses thereof Grant 8,846,929 - Fuchino , et al. September 30, 2 | 2014-09-30 |
Synthesis Of Carbamoylpyridone Hiv Integrase Inhibitors And Intermediates App 20140243521 - YOSHIDA; Hiroshi ;   et al. | 2014-08-28 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20140200209 - JOHNS; Brian A. ;   et al. | 2014-07-17 |
Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-.alpha- .]pyrrolo[1',2':3,4]imidazo[1,2-d]pyrazine-8-carboxamides Grant 8,778,943 - Johns , et al. July 15, 2 | 2014-07-15 |
Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates Grant 8,754,214 - Yoshida , et al. June 17, 2 | 2014-06-17 |
Prodrugs of (4aS, 13ar)-N-[(2,4-difluorophenyl)methyl]-10-hydroxy-9-11-dioxo-2,3,4a,5,9,11,- 13,13a-octahydro-1H-pyrido[1,2-a]pyrrolo[1',2':3:4]imidazo[1,2-d]pyrazine-- 8-carboxamide and their use in the treatment of HIV infection Grant 8,691,823 - Johns , et al. April 8, 2 | 2014-04-08 |
Synthesis Of Carbamoylpyridone Hiv Integrase Inhibitors And Intermediates App 20140094605 - YOSHIDA; Hiroshi ;   et al. | 2014-04-03 |
Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates Grant 8,624,023 - Yoshida , et al. January 7, 2 | 2014-01-07 |
Pyrolinone derivative and pharmaceutical composition comprising the same Grant 8,575,197 - Kai , et al. November 5, 2 | 2013-11-05 |
Substituted Polycyclic Carbamoyl Pyridone Derivative Prodrug App 20130197219 - Takahashi; Chika ;   et al. | 2013-08-01 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20130172559 - JOHNS; Brian A. ;   et al. | 2013-07-04 |
Chemical Compounds App 20130165415 - JOHNS; Brian A. ;   et al. | 2013-06-27 |
(3S,11aR)-N-[2,4-difluorophenyl)methyl]-6-hydroxy-3-methyl-5,7-dioxo-2,3,5- ,7,11,11a-hexahydro[1,3]oxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide useful as anti-HIV agent Grant 8,410,103 - Johns , et al. April 2, 2 | 2013-04-02 |
Chemical Compounds App 20120209000 - JOHNS; Brian Alvin ;   et al. | 2012-08-16 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20120208998 - YOSHIDA; Hiroshi ;   et al. | 2012-08-16 |
Substituted Polycyclic Carbamoylpyridone Derivative App 20120184734 - Akiyama; Toshiyuki ;   et al. | 2012-07-19 |
Polycyclic carbamoylpyridone derivative having HIV integrase inhibitory activity Grant 8,188,271 - Yoshida , et al. May 29, 2 | 2012-05-29 |
Substituted 9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydor-1H-pyrido[1,2-a]pyrrolo[1',2':3- ,4]imidazo[1,2-d]pyrazines Grant 8,183,372 - Johns , et al. May 22, 2 | 2012-05-22 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20120115875 - Johns; Brian Alvin ;   et al. | 2012-05-10 |
Substituted 5-hydroxy-3,4,6,9,9a, 10-hexanhydro-2h-1-oxa04a,8a-diaza-anthracene-6,10-dioness Grant 8,129,385 - Johns , et al. March 6, 2 | 2012-03-06 |
Synthesis Of Carbamoylpyridone Hiv Integrase Inhibitors And Intermediates App 20110282055 - Yoshida; Hiroshi ;   et al. | 2011-11-17 |
Novel Pyrolinone Derivative And Pharmaceutical Composition Comprising The Same App 20110183939 - Kai; Hiroyuki ;   et al. | 2011-07-28 |
Bicyclic carbamoylpyridone derivative having HIV integrase inhibitory activity Grant 7,858,788 - Yoshida , et al. December 28, 2 | 2010-12-28 |
Substituted-Quinoxaline-Type Piperidine Compounds and the Uses Thereof App 20100216726 - FUCHINO; Kouki ;   et al. | 2010-08-26 |
Hydroxypyrimidinone derivatives having inhibitory activity against HIV integrase App 20100204237 - Mikamiyama; Hidenori ;   et al. | 2010-08-12 |
Hydroxypyrimidinone derivatives having inhibitory activity against HIV integrase Grant 7,745,453 - Mikamiyama , et al. June 29, 2 | 2010-06-29 |
Polycyclic carbamoylpyridone derivative having hiv integrase inhibitory activity App 20090318421 - Johns; Brian Alvin ;   et al. | 2009-12-24 |
Polycylclic Carbamoylpyridone Derivative Having HIV Integrase Inhibitory Acitvity App 20090143356 - Yoshida; Hiroshi ;   et al. | 2009-06-04 |
Bicyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20080161271 - Yoshida; Hiroshi ;   et al. | 2008-07-03 |
Hydroxypyrimidinone derivatives having inhibitory activity against hiv integrase App 20070149556 - Mikamiyama; Hidenori ;   et al. | 2007-06-28 |