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SUBSTITUTED 1,2,3,3a,4,5,7,9,13,13a-DECAHYDROPYRIDO[1',2':4,5]PYRAZINO[1,2-a]PYRROLO[- 1,2-c]PYRIMIDINES HAVING HIV INTEGRASE INHIBITORY ACTIVITY App 20220213121 - JOHNS; Brian A. ;   et al. | 2022-07-07 |
Substituted 1,2,3,3a,4,5,7,9,13,13a-decahydropyrido[1',2':4,5]pyrazino[1,2-a]pyrrolo[- 1,2-c]pyrimidines having HIV integrase inhibitory activity Grant 11,267,823 - Johns , et al. March 8, 2 | 2022-03-08 |
N-[(2,4-difluorophenyl)methyl]-6-hydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a- -hexahydro[1,3] oxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide having HIV integrase inhibitory activity Grant 10,927,129 - Johns , et al. February 23, 2 | 2021-02-23 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20200339598 - JOHNS; Brian A. ;   et al. | 2020-10-29 |
N-[(2,4-DIFLUOROPHENYL)METHYL]-6-HYDROXY-3-METHYL-5,7-DIOXO-2,3,5,7,11,11a- -HEXAHYDRO[1,3]OXAZOLO[3,2-a]PYRIDO[1,2-d]PYRAZINE-8 App 20190284208 - JOHNS; Brian A. ;   et al. | 2019-09-19 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20190152990 - JOHNS; Brian A. ;   et al. | 2019-05-23 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170369509 - JOHNS; Brian A. ;   et al. | 2017-12-28 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170267693 - JOHNS; Brian A. ;   et al. | 2017-09-21 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170260203 - JOHNS; Brian A. ;   et al. | 2017-09-14 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170253616 - JOHNS; Brian A. ;   et al. | 2017-09-07 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170224695 - JOHNS; Brian A. ;   et al. | 2017-08-10 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170224694 - JOHNS; Brian A. ;   et al. | 2017-08-10 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170209454 - JOHNS; Brian A. ;   et al. | 2017-07-27 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170145033 - JOHNS; Brian A. ;   et al. | 2017-05-25 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20170029438 - JOHNS; Brian A. ;   et al. | 2017-02-02 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20160304535 - JOHNS; Brian A. ;   et al. | 2016-10-20 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20160207939 - JOHNS; Brian A. ;   et al. | 2016-07-21 |
SUBSTITUTED CYCLOPENTA[4,5]OXAZOLO[3,2-a]PYRIDO[1,2-d]PYRAZINES AS HIV INTEGRASE INHIBITORS App 20160137666 - Johns; Brian Alvin ;   et al. | 2016-05-19 |
Substituted pyrido[1',2':4,5]pyrazino[1,2-a]pyrimidines as HIV integrase inhibitors Grant 9,273,065 - Johns , et al. March 1, 2 | 2016-03-01 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20150232479 - JOHNS; Brian A. ;   et al. | 2015-08-20 |
Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-a]pyrr- olo[1',2':3,4]imidazo[1,2-d]pyrazine-8-carboxamides Grant 9,051,337 - Johns , et al. June 9, 2 | 2015-06-09 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20140200209 - JOHNS; Brian A. ;   et al. | 2014-07-17 |
Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-.alpha- .]pyrrolo[1',2':3,4]imidazo[1,2-d]pyrazine-8-carboxamides Grant 8,778,943 - Johns , et al. July 15, 2 | 2014-07-15 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20130172559 - JOHNS; Brian A. ;   et al. | 2013-07-04 |
(3S,11aR)-N-[2,4-difluorophenyl)methyl]-6-hydroxy-3-methyl-5,7-dioxo-2,3,5- ,7,11,11a-hexahydro[1,3]oxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide useful as anti-HIV agent Grant 8,410,103 - Johns , et al. April 2, 2 | 2013-04-02 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20120208998 - YOSHIDA; Hiroshi ;   et al. | 2012-08-16 |
Polycyclic carbamoylpyridone derivative having HIV integrase inhibitory activity Grant 8,188,271 - Yoshida , et al. May 29, 2 | 2012-05-29 |
Polycyclic Carbamoylpyridone Derivative Having Hiv Integrase Inhibitory Activity App 20120115875 - Johns; Brian Alvin ;   et al. | 2012-05-10 |
Substituted 5-hydroxy-3,4,6,9,9a, 10-hexanhydro-2h-1-oxa04a,8a-diaza-anthracene-6,10-dioness Grant 8,129,385 - Johns , et al. March 6, 2 | 2012-03-06 |
Naphthyridine derivatives having inhibitory activity against HIV integrase Grant 7,919,623 - Taishi , et al. April 5, 2 | 2011-04-05 |
Polycyclic carbamoylpyridone derivative having hiv integrase inhibitory activity App 20090318421 - Johns; Brian Alvin ;   et al. | 2009-12-24 |
Naphthyridine derivatives having inhibitory activity against hiv integrase App 20090227621 - Taishi; Teruhiko ;   et al. | 2009-09-10 |
Polycylclic Carbamoylpyridone Derivative Having HIV Integrase Inhibitory Acitvity App 20090143356 - Yoshida; Hiroshi ;   et al. | 2009-06-04 |
Heterocyclic compounds having inhibitory activity against HIV integrase App 20090118233 - Murai; Hitoshi ;   et al. | 2009-05-07 |
Heterocyclic compounds having inhibitory activity against HIV integrase Grant 7,358,249 - Murai , et al. April 15, 2 | 2008-04-15 |
Heterocyclic compounds having inhibitory activity against HIV integrase App 20060247212 - Murai; Hitoshi ;   et al. | 2006-11-02 |
Heterocyclic compounds having inhibitory activity against hiv integrase App 20060128669 - Murai; Hitoshi ;   et al. | 2006-06-15 |