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Heterobicyclic Inhibitors Of Mat2a And Methods Of Use For Treating Cancer App 20220251081 - KONTEATIS; Zenon D. ;   et al. | 2022-08-11 |
Pyruvate Kinase Modulators And Use Thereof App 20220233541 - Cianchetta; Giovanni ;   et al. | 2022-07-28 |
Pyruvate kinase activators for use in treating blood disorders Grant 11,364,240 - Cianchetta , et al. June 21, 2 | 2022-06-21 |
New Organic Compounds App 20220169654 - KONTEATIS; Zenon D. ;   et al. | 2022-06-02 |
Aza-heterobicyclic Inhibitors Of Mat2a And Methods Of Use For Treating Cancer App 20220144820 - KONTEATIS; Zenon D. ;   et al. | 2022-05-12 |
Inhibitors of cellular metabolic processes Grant 11,325,914 - Konteatis , et al. May 10, 2 | 2022-05-10 |
Thieno[3,2-b] Pyrrole[3,2-d]pyridazinone Derivatives And Their Use As Pkm2 Derivatives For The Treatment Of Cancer, Obesity And Diabetes Related Disorders App 20220127267 - Liu; Tao ;   et al. | 2022-04-28 |
Aza-heterobicyclic Inhibitors Of Mat2a And Methods Of Use For Treating Cancer App 20220098203 - KONTEATIS; Zenon D. ;   et al. | 2022-03-31 |
Benzo-fused heterocyclic derivatives useful as agonists of GPR120 Grant 11,254,647 - Sui , et al. February 22, 2 | 2022-02-22 |
Cylcoalkenyl derivatives useful as agonists of the GPR120 and/or GPR40 receptors Grant 11,230,526 - Lanter , et al. January 25, 2 | 2022-01-25 |
Pyruvate kinase activators for use in treating blood disorders Grant 11,040,036 - Cianchetta , et al. June 22, 2 | 2021-06-22 |
Pyruvate Kinase Activators For Use In Treating Blood Disorders App 20210130371 - Cianchetta; Giovanni ;   et al. | 2021-05-06 |
Heterobicyclic Inhibitors Of Mat2a And Methods Of Use For Treating Cancer App 20210115045 - KONTEATIS; Zenon D. ;   et al. | 2021-04-22 |
Pyruvate Kinase Activators For Use In Treating Blood Disorders App 20210077490 - Cianchetta; Giovanni ;   et al. | 2021-03-18 |
Heterocylcoalkenyl Derivatives Useful As Agonists Of The Gpr120 And / Or Gpr40 App 20210024483 - Lanter; James C. ;   et al. | 2021-01-28 |
Inhibitors of cellular metabolic processes Grant 10,800,782 - Konteatis , et al. October 13, 2 | 2020-10-13 |
Benzo-fused Heterocyclic Derivatives Useful As Agonists Of Gpr120 App 20200317629 - Sui; Zhihua ;   et al. | 2020-10-08 |
Benzo-fused heterocyclic derivatives useful as agonists of GPR120 Grant 10,730,847 - Sui , et al. | 2020-08-04 |
Pyruvate Kinase Activators For Use In Treating Blood Disorders App 20200207785 - Cianchetta; Giovanni ;   et al. | 2020-07-02 |
Pyruvate Kinase Modulators And Use Thereof App 20200206225 - Cianchetta; Giovanni ;   et al. | 2020-07-02 |
GPR120 agonists for the treatment of type II diabetes Grant 10,618,893 - Sui , et al. | 2020-04-14 |
Deuterated Analogs Of An Organic Compound App 20200085832 - Sui; Zhihua ;   et al. | 2020-03-19 |
Inhibitors Of Cellular Metabolic Processes App 20190233424 - Konteatis; Zenon D. ;   et al. | 2019-08-01 |
Inhibitors of cellular metabolic processes Grant 10,329,298 - Konteatis , et al. | 2019-06-25 |
Benzo-fused Heterocyclic Derivatives Useful As Agonists Of Gpr120 App 20190152937 - Sui; Zhihua ;   et al. | 2019-05-23 |
Gpr120 Agonists For The Treatment Of Type Ii Diabetes App 20190071435 - Sui; Zhihua ;   et al. | 2019-03-07 |
Benzo-fused heterocyclic derivatives useful as agonists of GPR120 Grant 10,155,737 - Sui , et al. Dec | 2018-12-18 |
GPR120 agonists for the treatment of type II diabetes Grant 10,118,922 - Sui , et al. November 6, 2 | 2018-11-06 |
Tetrahydro-benzoimidazolyl modulators of TGR5 Grant 10,077,241 - Zhang , et al. September 18, 2 | 2018-09-18 |
Inhibitors Of Cellular Metabolic Processes App 20180079753 - Konteatis; Zenon D. ;   et al. | 2018-03-22 |
Indazole compounds useful as ketohexokinase inhibitors Grant 9,771,375 - Zhang , et al. September 26, 2 | 2017-09-26 |
Benzo-fused Heterocyclic Derivatives Useful As Agonists Of Gpr120 App 20170088531 - Sui; Zhihua ;   et al. | 2017-03-30 |
Benzo-fused heterocyclic derivatives useful as agonists of GPR120 Grant 9,562,053 - Sui , et al. February 7, 2 | 2017-02-07 |
Tetrahydro-benzoimidazolyl Modulators Of Tgr5 App 20170029381 - Zhang; Xuqing ;   et al. | 2017-02-02 |
Substituted pyrazoles as N-type calcium channel blockers Grant 9,434,693 - Wall , et al. September 6, 2 | 2016-09-06 |
Indole derivatives as selective androgen receptor modulators (SARMS) Grant 9,434,688 - Lanter , et al. September 6, 2 | 2016-09-06 |
Tetracyclic heteroatom containing derivatives useful as sex steroid hormone receptor modulators Grant 9,303,037 - Sui , et al. April 5, 2 | 2016-04-05 |
Cyclohexyl-azetidinyl antagonists of CCR2 Grant 9,062,048 - Lanter , et al. June 23, 2 | 2015-06-23 |
Bicyclic pyrrole derivatives useful as agonists of GPR120 Grant 9,045,454 - Sui , et al. June 2, 2 | 2015-06-02 |
Octahydro-cyclopentapyrrolyl antagonists of CCR2 Grant 9,024,017 - Cai , et al. May 5, 2 | 2015-05-05 |
4-substituted-cyclohexylamino-4-piperidinyl-acetamide antagonists of CCR2 Grant 8,921,559 - Lanter , et al. December 30, 2 | 2014-12-30 |
Bicyclic pyrrole derivatives useful as agonists of GPR120 Grant 8,912,227 - Sui , et al. December 16, 2 | 2014-12-16 |
Substituted pyrazoles as N-type calcium channel blockers Grant 8,901,314 - Wall , et al. December 2, 2 | 2014-12-02 |
Indazole Compounds Useful As Ketohexokinase Inhibitors App 20140336170 - Zhang; Xuqing ;   et al. | 2014-11-13 |
Cyclopentylpyrazoles as N-type calcium channel blockers Grant 8,853,418 - Winters , et al. October 7, 2 | 2014-10-07 |
Pyrrolopyrazoles as N-type calcium channel blockers Grant 8,846,949 - Winters , et al. September 30, 2 | 2014-09-30 |
Benzo-fused Heterocyclic Derivatives Useful As Agonists Of Gpr120 App 20140275172 - Sui; Zhihua ;   et al. | 2014-09-18 |
Gpr120 Agonists For The Treatment Of Type Ii Diabetes App 20140275179 - Sui; Zhihua ;   et al. | 2014-09-18 |
Bicyclic Pyrrole Derivatives Useful As Agonists Of Gpr120 App 20140275182 - Sui; Zhihua ;   et al. | 2014-09-18 |
Novel Indole Derivatives As Selective Androgen Receptor Modulators (sarms) App 20140249197 - Lanter; James C. ;   et al. | 2014-09-04 |
Fused cyclopentyl antagonists of CCR2 Grant 8,822,460 - Winters , et al. September 2, 2 | 2014-09-02 |
Indazole compounds useful as ketohexokinase inhibitors Grant 8,822,447 - Zhang , et al. September 2, 2 | 2014-09-02 |
Indole derivatives as selective androgen receptor modulators (SARMS) Grant 8,765,782 - Lanter , et al. July 1, 2 | 2014-07-01 |
Substituted Pyrazoles As N-type Calcium Channel Blockers App 20140162997 - Wall; Mark ;   et al. | 2014-06-12 |
Substituted Pyrazoles As N-type Calcium Channel Blockers App 20140163031 - Wall; Mark ;   et al. | 2014-06-12 |
Novel Tetracyclic Heteroatom Containing Derivatives Useful As Sex Steroid Hormone Receptor Modulators App 20140066479 - Sui; Zhihua ;   et al. | 2014-03-06 |
Cyclopentylpyrazoles As N-type Calcium Channel Blockers App 20140051660 - WINTERS; Michael ;   et al. | 2014-02-20 |
Pyrrolopyrazoles As N-type Calcium Channel Blockers App 20140051688 - WINTERS; Michael ;   et al. | 2014-02-20 |
Octahydro-cyclopentapyrrolyl Antagonists Of Ccr2 App 20140024646 - Cai; Chaozhong ;   et al. | 2014-01-23 |
Fused Cyclopentyl Antagonists Of Ccr2 App 20140018356 - Winters; Michael P. ;   et al. | 2014-01-16 |
Cyclohexyl-azetidinyl Antagonists Of Ccr2 App 20130310365 - Lanter; James C. ;   et al. | 2013-11-21 |
Benzimidazole derivatives useful as selective androgen receptor modulators (SARMS) Grant 8,586,616 - Ng , et al. November 19, 2 | 2013-11-19 |
Tetracyclic heteroatom containing derivatives useful as sex steroid hormone receptor modulators Grant 8,580,840 - Sui , et al. November 12, 2 | 2013-11-12 |
Cyclohexyl-azetidinyl antagonists of CCR2 Grant 8,518,969 - Lanter , et al. August 27, 2 | 2013-08-27 |
4-Azetidinyl-1-phenyl-cyclohexane antagonists of CCR2 Grant 8,513,229 - Zhang , et al. August 20, 2 | 2013-08-20 |
4-azetidinyl-1-heteroaryl-cyclohexanol antagonists of CCR2 Grant 8,450,304 - Zhang , et al. May 28, 2 | 2013-05-28 |
Cyclohexyl-azetidinyl antagonists of CCR2 Grant 8,436,023 - Zhang , et al. May 7, 2 | 2013-05-07 |
Indole derivatives as selective androgen receptor modulators (SARMS) Grant 8,394,971 - Lanter , et al. March 12, 2 | 2013-03-12 |
4-azetidinyl-1-heteroatom linked-cyclohexane antagonists of CCR2 Grant 8,324,186 - Zhang , et al. December 4, 2 | 2012-12-04 |
Tetracyclic heteroatom containing derivatives useful as sex steroid hormone receptor modulators Grant 8,318,766 - Sui , et al. November 27, 2 | 2012-11-27 |
4-azetidinyl-1-heteroaryl-cyclohexane antagonists of CCR2 Grant 8,269,015 - Zhang , et al. September 18, 2 | 2012-09-18 |
4-substituted-cyclohexylamino-4-piperidinyl-acetamide Antagonists Of Ccr2 App 20120142733 - Lanter; James C. ;   et al. | 2012-06-07 |
Piperidyl acrylamide antagonists of CCR2 Grant 8,188,287 - Cai , et al. May 29, 2 | 2012-05-29 |
4-azetidinyl-1-phenyl-cyclohexane Antagonists Of Ccr2 App 20120040960 - Zhang; Xuqing ;   et al. | 2012-02-16 |
Bicyclic heterocycles useful as selective androgen receptor modulators Grant 8,097,730 - Zhang , et al. January 17, 2 | 2012-01-17 |
Heterocycle derivatives useful as selective androgen receptor modulators (SARMs) Grant 8,088,811 - Zhang , et al. January 3, 2 | 2012-01-03 |
Cyclohexyl-azetidinyl Antagonists Of Ccr2 App 20110312936 - Lanter; James C. ;   et al. | 2011-12-22 |
Cyclohexyl-azetidinyl Antagonists Of Ccr2 App 20110306592 - Zhang; Xuqing ;   et al. | 2011-12-15 |
Coumarin derivatives as ion channel openers Grant 8,067,619 - Jain , et al. November 29, 2 | 2011-11-29 |
Pyrazolylquinazolinones as potassium channel openers Grant 8,053,441 - Zhang , et al. November 8, 2 | 2011-11-08 |
Indazole Compounds Useful As Ketohexokinase Inhibitors App 20110263559 - ZHANG; Xuqing ;   et al. | 2011-10-27 |
Steroids derivatives as selective progesterone receptor modulators Grant 7,981,927 - Jain , et al. July 19, 2 | 2011-07-19 |
Imidazolidin-2-one derivatives as selective androgen receptor modulators (SARMS) Grant 7,968,580 - Lanter , et al. June 28, 2 | 2011-06-28 |
2-substituted benzimidazoles as selective androgen receptor modulators (SARMS) Grant 7,932,399 - Alford, Jr. , et al. April 26, 2 | 2011-04-26 |
Novel Benzimidazole Derivatives Useful As Selective Androgen Receptor Modulators (sarms) App 20110086883 - Ng; Raymond ;   et al. | 2011-04-14 |
Benzimidazole derivatives useful as selective androgen receptor modulators (SARMS) Grant 7,879,895 - Ng , et al. February 1, 2 | 2011-02-01 |
Novel Indole Derivatives As Selective Androgen Receptor Modulators (sarms) App 20110021785 - Lanter; James C. ;   et al. | 2011-01-27 |
Novel Benzimidazole Derivatives Useful As Selective Androgen Receptor Modulators (sarms) App 20100298383 - Ng; Raymond ;   et al. | 2010-11-25 |
Benzopyran derivatives as potassium channel openers Grant 7,838,553 - Zhang , et al. November 23, 2 | 2010-11-23 |
4-azetidinyl-1-heteroatom Linked-cyclohexane Antagonists Of Ccr2 App 20100267668 - Zhang; Xuqing ;   et al. | 2010-10-21 |
Novel Heterocycle Derivatives Useful As Selective Androgen Receptor Modulators (sarms) App 20100267670 - Zhang; Xuqing ;   et al. | 2010-10-21 |
4-azetidinyl-1-heteroaryl-cyclohexane Antagonists Of Ccr2 App 20100267688 - Zhang; Xuqing ;   et al. | 2010-10-21 |
4-azetidinyl-1-phenyl-cyclohexane Antagonists Of Ccr2 App 20100267689 - Zhang; Xuqing ;   et al. | 2010-10-21 |
Benzopyran derivatives as potassium channel openers Grant 7,812,183 - Zhang , et al. October 12, 2 | 2010-10-12 |
Benzimidazole derivatives useful as selective androgen receptor modulators (SARMS) Grant 7,795,446 - Ng , et al. September 14, 2 | 2010-09-14 |
Quinoline derivatives as potassium ion channel openers Grant 7,790,895 - Jain , et al. September 7, 2 | 2010-09-07 |
Heterocycle derivatives useful as selective androgen receptor modulators (SARMS) Grant 7,781,473 - Zhang , et al. August 24, 2 | 2010-08-24 |
Novel Tetracyclic Heteroatom Containing Derivatives Useful As Sex Steroid Hormone Receptor Modulators App 20100210658 - Sui; Zhihua ;   et al. | 2010-08-19 |
Novel Tetracyclic Heteroatom Containing Derivatives Useful As Sex Steroid Hormone Receptor Modulators App 20100204239 - Sui; Zhihua ;   et al. | 2010-08-12 |
Oxa-steroids derivatives as selective progesterone receptor modulators Grant 7,763,648 - Kang , et al. July 27, 2 | 2010-07-27 |
Tetracyclic heteroatom containing derivatives useful as sex steroid hormone receptor modulators Grant 7,759,498 - Sui , et al. July 20, 2 | 2010-07-20 |
Novel Bicyclic Heterocycles Useful As Selective Androgen Receptor Modulators App 20100160330 - Zhang; Xuqing ;   et al. | 2010-06-24 |
Novel Indole Derivatives As Selective Androgen Receptor Modulators (sarms) App 20100144823 - Lantar; James C. ;   et al. | 2010-06-10 |
4-azetidinyl-1-heteroaryl-cyclohexanol Antagonists Of Ccr2 App 20100144695 - Zhang; Xuqing ;   et al. | 2010-06-10 |
Indole derivatives as selective androgen receptor modulators (SARMS) Grant 7,705,147 - Lanter , et al. April 27, 2 | 2010-04-27 |
Tetracyclic heteroatom containing derivatives useful as sex steroid hormone receptor modulators Grant 7,696,239 - Sui , et al. April 13, 2 | 2010-04-13 |
Novel Coumarin Derivatives As Ion Channel Openers App 20100069474 - Jain; Nareshkumar F. ;   et al. | 2010-03-18 |
Indole derivatives as selective androgen receptor modulators (SARMS) Grant 7,678,926 - Lanter , et al. March 16, 2 | 2010-03-16 |
11-phosphorous steroid derivatives useful as progesterone receptor modulators Grant 7,678,781 - Fiordeliso , et al. March 16, 2 | 2010-03-16 |
Tricyclic dihydropyrazines as potassium channel openers Grant 7,674,793 - Zhang , et al. March 9, 2 | 2010-03-09 |
Pyridine derivatives as potassium ion channel openers Grant 7,671,065 - Jain , et al. March 2, 2 | 2010-03-02 |
17-phosphorous steroid derivatives useful as progesterone receptor modulators Grant 7,671,045 - Jiang , et al. March 2, 2 | 2010-03-02 |
Coumarin derivatives as ion channel openers Grant 7,662,975 - Jain , et al. February 16, 2 | 2010-02-16 |
Imidazolopyrazole derivatives useful as selective androgen receptor modulators Grant 7,655,683 - Zhang , et al. February 2, 2 | 2010-02-02 |
Pyridine Imidazoles and Aza-indoles as Progesterone Receptor Modulators App 20100016266 - Jiang; Weiqin ;   et al. | 2010-01-21 |
Trisubstituted thiophenes as progesterone receptor modulators Grant 7,638,525 - Jiang , et al. December 29, 2 | 2009-12-29 |
Piperidyl Acrylamide Antagonists Of Ccr2 App 20090318498 - Cai; Chaozhong ;   et al. | 2009-12-24 |
3,4-diamino-3-cyclobutene-1,2-dione Derivatives As Potassium Channel Openers App 20090312412 - Lanter; James C. ;   et al. | 2009-12-17 |
Trisubstituted Thiophenes as Progesterone Receptor Modulators App 20090306118 - Jiang; Weiqin ;   et al. | 2009-12-10 |
Bicyclic heterocycles useful as selective androgen receptor modulators Grant 7,626,036 - Zhang , et al. December 1, 2 | 2009-12-01 |
Pyridine imidazoles and aza-indoles as progesterone receptor modulators Grant 7,608,712 - Jiang , et al. October 27, 2 | 2009-10-27 |
Novel Benzimidazole Derivatives Useful as Selective Androgen Receptor Modulators (SARMS) App 20090258909 - Ng; Raymond ;   et al. | 2009-10-15 |
3,4-diamino-3-cyclobutene-1,2-dione derivatives as potassium channel openers Grant 7,595,409 - Lanter , et al. September 29, 2 | 2009-09-29 |
Novel Indole Derivatives As Selective Androgen Receptor Modulators (sarms) App 20090216023 - Lanter; James C. ;   et al. | 2009-08-27 |
Novel imidazolidIn-2-one derivatives as selective androgen receptor modulators (SARMS) App 20090215848 - Lanter; James C. ;   et al. | 2009-08-27 |
Benzimidazole derivatives useful as selective androgen receptor modulators (sarms) Grant 7,566,733 - Ng , et al. July 28, 2 | 2009-07-28 |
Novel Heterocycle Derivatives Useful As Selective Androgen Receptor Modulators (sarms) App 20090131365 - Zhang; Xuqing ;   et al. | 2009-05-21 |
Imidazolidin-2-one derivatives as selective androgen receptor modulators (SARMS) Grant 7,531,565 - Lanter , et al. May 12, 2 | 2009-05-12 |
Novel Spiro-benzo[c]chromene derivatives useful as modulators of the estrogen receptors App 20090069362 - Zhang; Xuqing ;   et al. | 2009-03-12 |
Heterocycle derivatives useful as selective androgen receptor modulators (SARMs) Grant 7,465,809 - Zhang , et al. December 16, 2 | 2008-12-16 |
Spiro-benzo[c]chromene derivatives useful as modulators of the estrogen receptors Grant 7,452,914 - Zhang , et al. November 18, 2 | 2008-11-18 |
Indole derivatives as selective androgen receptor modulators (SARMS) Grant 7,427,682 - Lanter , et al. September 23, 2 | 2008-09-23 |
Novel Heterocyclic Benzo[c]chromene Derivatives Useful As Modulators Of The Estrogen Receptors App 20080221125 - Zhang; Xuqing ;   et al. | 2008-09-11 |
Steroids Derivatives As Selective Progesterone Receptor Modulators App 20080221202 - Jain; Nareshkumar F. ;   et al. | 2008-09-11 |
Heterocyclic benzo[c]chromene derivatives useful as modulators of the estrogen receptors Grant 7,399,767 - Zhang , et al. July 15, 2 | 2008-07-15 |
Tetracyclic steroid derivatives useful as progesterone receptor modulators Grant 7,390,831 - Chen , et al. June 24, 2 | 2008-06-24 |
Novel Benzimidazole Derivatives Useful As Selective Androgen Receptor Modulators (sarms) App 20080119522 - Ng; Raymond ;   et al. | 2008-05-22 |
Pyridine Imidazoles And Aza-indoles As Progesterone Receptor Modulators App 20080119500 - Jiang; Weiqin ;   et al. | 2008-05-22 |
Novel Tetracyclic Heteroatom Containing Derivatives Useful As Sex Steroid Hormone Receptor Modulators App 20080114048 - SUI; Zhihua ;   et al. | 2008-05-15 |
Pyridine imidazoles and aza-indoles as progesterone receptor modulators Grant 7,348,432 - Jiang , et al. March 25, 2 | 2008-03-25 |
Benzimidazole derivatives useful as selective androgen receptor modulators (SARMS) Grant 7,348,438 - Ng , et al. March 25, 2 | 2008-03-25 |
Novel Indole Derivatives As Selective Androgen Receptor Modulators (sarms) App 20080070970 - Lanter; James C. ;   et al. | 2008-03-20 |
Indole derivatives useful as progesterone receptor modulators Grant 7,345,084 - Jiang , et al. March 18, 2 | 2008-03-18 |
Tetracyclic heteroatom containing derivatives useful as sex steroid hormone receptor modulators Grant 7,338,973 - Sui , et al. March 4, 2 | 2008-03-04 |
Heteroatom containing tetracyclic derivatives as selective estrogen receptor modulators Grant 7,329,654 - Kanojia , et al. February 12, 2 | 2008-02-12 |
Indole derivatives as selective androgen receptor modulator (SARMS) Grant 7,288,553 - Lanter , et al. October 30, 2 | 2007-10-30 |
Indole derivatives as selective androgen receptor modulators (SARMS) Grant 7,282,507 - Lanter , et al. October 16, 2 | 2007-10-16 |
3,4-diamino-3-cyclobutene-1,2-dione Derivatives As Potassium Channel Openers App 20070232689 - Lanter; James C. ;   et al. | 2007-10-04 |
11-phosphorous Steroid Derivatives Useful As Progesterone Receptor Modulators App 20070232570 - Fiordeliso; James J. ;   et al. | 2007-10-04 |
17-phosphorous Steroid Derivatives Useful As Progesterone Receptor Modulators App 20070207982 - Jiang; Weiqin ;   et al. | 2007-09-06 |
Novel Imidazolopyrazole Derivatives Useful As Selective Androgen Receptor Modulators App 20070197616 - Zhang; Xuqing ;   et al. | 2007-08-23 |
Novel Bicyclic Heterocycles Useful As Selective Androgen Receptor Modulators App 20070197521 - Zhang; Xuqing ;   et al. | 2007-08-23 |
Tetracyclic Steroid Derivatives Useful As Progesterone Receptor Modulators App 20070197634 - Chen; Ningyi ;   et al. | 2007-08-23 |
Novel Pyrazolylquinazolinones As Potassium Channel Openers App 20070197566 - Zhang; Xuqing ;   et al. | 2007-08-23 |
Oxa-steroids Derivatives As Selective Progesterone Receptor Modulators App 20070197635 - Kang; Fu-An ;   et al. | 2007-08-23 |
Novel Tricyclic Dihydropyrazines As Potassium Channel Openers App 20070191382 - Zhang; Xuqing ;   et al. | 2007-08-16 |
Cyclohexyl Derivatives As Selective Estrogen Receptor Modulators App 20070142379 - Jain; Nareshkumar F. ;   et al. | 2007-06-21 |
Indole Derivatives Useful As Progesterone Receptor Modulators App 20070135511 - Jiang; Weiqin ;   et al. | 2007-06-14 |
Novel Benzopyran Derivatives As Potassium Channel Openers App 20070072832 - Zhang; Xuqing ;   et al. | 2007-03-29 |
Novel pyridine derivatives as potassium ion channel openers App 20070054935 - Jain; Nareshkumar ;   et al. | 2007-03-08 |
Novel quinoline derivatives as potassium ion channel openers App 20070054936 - Jain; Nareshkumar ;   et al. | 2007-03-08 |
Novel Benzopyran Derivatives As Potassium Channel Openers App 20070049556 - Zhang; Xuqing ;   et al. | 2007-03-01 |
Indole derivatives useful as progesterone receptor modulators Grant 7,183,309 - Jiang , et al. February 27, 2 | 2007-02-27 |
Cyclohexyl derivatives as selective estrogen receptor modulators Grant 7,183,445 - Jain , et al. February 27, 2 | 2007-02-27 |
Novel coumarin derivatives as ion channel openers App 20070037877 - Jain; Nareshkumar F. ;   et al. | 2007-02-15 |
Novel heterocycle derivatives useful as selective androgen receptor modulators (SARMs) App 20060211756 - Zhang; Xuqing ;   et al. | 2006-09-21 |
Novel heterocyclic benzo[c]chromene derivatives useful as modulators of the estrogen receptors App 20060205741 - Zhang; Xuqing ;   et al. | 2006-09-14 |
Heteroatom containing tetracyclic derivatives as selective estrogen receptor modulators Grant 7,105,679 - Kanojia , et al. September 12, 2 | 2006-09-12 |
N-heterocyclyl hydrazides as neurotrophic agents Grant 7,087,628 - Sui , et al. August 8, 2 | 2006-08-08 |
Novel 2H-chromene derivatives as selective estrogen receptor modulators App 20060166933 - Jain; Nareshkumar F. ;   et al. | 2006-07-27 |
Estrieno[3,2-b]/[3,4-c]pyrrole derivatives useful as modulators of the estrogen receptors Grant 7,074,779 - Sui , et al. July 11, 2 | 2006-07-11 |
Novel tetracyclic heteroatom containing derivatives useful as sex steroid hormone receptor modulators App 20060116415 - Sui; Zhihua ;   et al. | 2006-06-01 |
Novel tetracyclic heteroatom containing derivatives useful as sex steroid hormone receptor modulators App 20060116513 - Sui; Zhihua ;   et al. | 2006-06-01 |
Novel benzimidazole derivatives useful as selective androgen receptor modulators (sarms) App 20060116412 - Ng; Raymond ;   et al. | 2006-06-01 |
Indole derivatives useful as progesterone receptor modulators App 20060111427 - Jiang; Weiqin ;   et al. | 2006-05-25 |
Novel benzimidazole derivatives useful as selective androgen receptor modulators (SARMS) App 20060111402 - Ng; Raymond ;   et al. | 2006-05-25 |
Pyridine imidazoles and aza-indoles as progesterone receptor modulators App 20060111391 - Jiang; Weiqin ;   et al. | 2006-05-25 |
Trisubstituted thiophenes as progesterone receptor modulators App 20060106047 - Jiang; Weiqin ;   et al. | 2006-05-18 |
Novel imidazolidin-2-one derivatives as selective androgen receptor modulators (SARMS) App 20060063819 - Lanter; James C. ;   et al. | 2006-03-23 |
Benzoxazepine derivatives as selective estrogen receptor modulators App 20060040917 - Lanter; James C. ;   et al. | 2006-02-23 |
Novel spiro-benzo[c]chromene derivatives useful as modulators of the estrogen receptors App 20060020018 - Zhang; Xuqing ;   et al. | 2006-01-26 |
Novel indole derivatives as selective androgen receptor modulator (SARMS) App 20050250740 - Lanter, James C. ;   et al. | 2005-11-10 |
Novel indole derivatives as selective androgen receptor modulators (SARMS) App 20050250741 - Lanter, James C. ;   et al. | 2005-11-10 |
Novel indole derivatives as selective androgen receptor modulators (SARMS) App 20050245485 - Lanter, James C. ;   et al. | 2005-11-03 |
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors App 20050113402 - Sui, Zhihua ;   et al. | 2005-05-26 |
2-(Quinolonyl)-fused heterocycles as androgen receptor modulators App 20050107372 - Lanter, James C. ;   et al. | 2005-05-19 |
Benzo[4,5]thieno[2,3-c]pyridine and Benzo[4,5]furo[2,3-c]pyridine Derivatives Useful as Inhibitors of Phosphodiesterase Grant 6,864,253 - Sui , et al. March 8, 2 | 2005-03-08 |
2-(quinolonyl)-fused heterocycles as androgen receptor modulators Grant 6,858,621 - Lanter , et al. February 22, 2 | 2005-02-22 |
Novel thiazoline derivatives as selective androgen receptor modulators (SARMS) App 20050014952 - Ng, Raymond A. ;   et al. | 2005-01-20 |
Cyclohexyl derivatives as selective estrogen receptor modulators App 20050009799 - Jain, Nareshkumar F. ;   et al. | 2005-01-13 |
Novel estrieno[3,2-b]/[3,4-c]pyrrole derivatives useful as modulators of the estrogen receptors App 20050004090 - Sui, Zhihua ;   et al. | 2005-01-06 |
Novel heteroatom containing tetracyclic derivatives as selective estrogen receptor modulators App 20040259915 - Kanojia, Ramesh M. ;   et al. | 2004-12-23 |
Triazepine derivatives as neurotrophic agents Grant 6,821,993 - Sui , et al. November 23, 2 | 2004-11-23 |
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors Grant 6,818,646 - Sui , et al. November 16, 2 | 2004-11-16 |
Substituted 2,4-dihydro-pyrrolo[3,4-b]quinolin-9-one derivatives useful as phosphodiesterase inhibitors Grant 6,800,625 - Jiang , et al. October 5, 2 | 2004-10-05 |
7-heterocyclyl quinoline and thieno[2,3-b]pyridine derivatives useful as antagonists of gonadotropin releasing hormone Grant 6,765,011 - Sui , et al. July 20, 2 | 2004-07-20 |
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors App 20040044021 - Sui, Zhihua ;   et al. | 2004-03-04 |
Substituted tetracyclic pyrroloquinolone derivatives useful as phosphodiesterase inhibitors Grant 6,686,349 - Jiang , et al. February 3, 2 | 2004-02-03 |
2-(Quinolonyl)-fused heterocycles as androgen receptor modulators App 20040014743 - Lanter, James C. ;   et al. | 2004-01-22 |
Substituted 2,4-dihydro-pyrrolo[3,4-b]quinolin-9-one Derivatives Useful As Phosphodiesterase Inhibitors App 20040006079 - Jiang, Weiqin ;   et al. | 2004-01-08 |
7-Heterocyclyl quinoline and thieno[2,3-b]pyridine derivatives useful as antagonists of gonadotropin releasing hormone App 20030216429 - Sui, Zhihua ;   et al. | 2003-11-20 |
Novel heteroatom containing tetracyclic derivatives as selective estrogen receptor modulators App 20030216463 - Kanojia, Ramesh M. ;   et al. | 2003-11-20 |
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors Grant 6,635,638 - Sui , et al. October 21, 2 | 2003-10-21 |
Beta-carboline derivatives useful as inhibitors of phosphodiesterase App 20030166641 - Sui, Zhihua ;   et al. | 2003-09-04 |
N-heterocyclyl hydrazides as neurotrophic agents App 20030144262 - Sui, Zhihua ;   et al. | 2003-07-31 |
Substituted tetracyclic pyrroloquinolone derivatives useful as phosphodiesterase inhibitors App 20030144268 - Jiang, Weiqin ;   et al. | 2003-07-31 |
.beta.-carboline derivatives useful as inhibitors of phosphodiesterase Grant 6,492,358 - Sui , et al. December 10, 2 | 2002-12-10 |
7-Heterocyclyl quinoline and thieno(2,3-b)pyridine derivatives useful as antagonists of gonadotropin releasing hormone App 20020123506 - Sui, Zhihua ;   et al. | 2002-09-05 |
beta-carboline derivatives useful as inhibitors of phosphodiesterase App 20020010189 - Sui, Zhihua ;   et al. | 2002-01-24 |
Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors App 20020010183 - Sui, Zhihua ;   et al. | 2002-01-24 |
Neurotrophic tetrahydroisoquinolines and tetrahydrothienopyridines, and related compositions and methods Grant 6,323,215 - Macielag , et al. November 27, 2 | 2001-11-27 |
1,3- and 2,3-diarylcycloalkano and cycloalkeno pyrazoles as selective inhibitors of cyclooxygenase-2 and antiinflammatory agents Grant 6,083,969 - Ferro , et al. July 4, 2 | 2000-07-04 |
5-heterocyclyl pyrazolo[4,3-d]pyrimidin-7-ones for the treatment of male erectile dysfunction Grant 6,077,841 - Sui , et al. June 20, 2 | 2000-06-20 |
Aryl phenylhydrazides as selective COX-2 inhibitors for treatment of inflammation Grant 6,077,869 - Sui , et al. June 20, 2 | 2000-06-20 |