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2,2-difluorodioxolo A.sub.2A receptor antagonists Grant 11,046,714 - Amjad , et al. June 29, 2 | 2021-06-29 |
Pyridinone- And Pyridazinone-based Compounds And Uses Thereof App 20200407339 - Hla; Timothy ;   et al. | 2020-12-31 |
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Spirocyclic Pyridotriazine Derivatives Useful As HIV Integrase Inhibitors App 20180325926 - Graham; Thomas H. ;   et al. | 2018-11-15 |
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Substituted quinolizine derivatives useful as HIV integrase inhibitors Grant 9,861,620 - Yu , et al. January 9, 2 | 2018-01-09 |
Processes For The Preparation Of A Bace Inhibitor App 20170233382 - Miller; Steven P. ;   et al. | 2017-08-17 |
Heterobicyclo-substituted [1,2,4]triazolo[1,5-c]quinazolin-5-amine Compounds With A2a Antagonist Properties App 20170197991 - Ali; Amjad ;   et al. | 2017-07-13 |
Compounds inhibiting leucine-rich repeat kinase enzyme activity Grant 9,688,654 - Miller , et al. June 27, 2 | 2017-06-27 |
Piperazine-substituted [1,2,4]triazolo[1,5-C]quinazolin-5-amine compounds with A.sub.2A antagonist properties Grant 9,676,780 - Ali , et al. June 13, 2 | 2017-06-13 |
Mineralocorticoid receptor antagonists Grant 9,511,052 - Cernak , et al. December 6, 2 | 2016-12-06 |
Substituted pyrido[1,2-a]pyrazines as HIV integrase inhibitors Grant 9,493,479 - Graham , et al. November 15, 2 | 2016-11-15 |
Compounds inhibiting leucine-rich repeat kinase enzyme activity Grant 9,493,440 - Miller , et al. November 15, 2 | 2016-11-15 |
Compounds Inhibiting Leucine-rich Repeat Kinase Enzyme Activity App 20160289207 - DeMong; Duane ;   et al. | 2016-10-06 |
Compounds inhibiting leucine-rich repeat kinase enzyme activity Grant 9,440,952 - Miller , et al. September 13, 2 | 2016-09-13 |
Compounds inhibiting leucine-rich repeat kinase enzyme activity Grant 9,416,126 - Miller , et al. August 16, 2 | 2016-08-16 |
Substituted Quinolizine Derivatives Useful As Hiv Integrase Inhibitors App 20160228419 - Yu; Tao ;   et al. | 2016-08-11 |
Bridged bicyclic piperidine derivatives and methods of use thereof Grant 9,409,918 - Harris , et al. August 9, 2 | 2016-08-09 |
2,2-difluorodioxolo A2a Receptor Antagonists App 20160214997 - Amjad; Ali ;   et al. | 2016-07-28 |
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4-pyridone Derivative Compounds And Uses Thereof As Hiv Integrase Inhibitors App 20160060272 - Graham; Thomas H. ;   et al. | 2016-03-03 |
Compounds Inhibiting Leucine-rich Repeat Kinase Enzyme Activity App 20160009696 - Miller; Michael ;   et al. | 2016-01-14 |
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Compounds Inhibiting Leucine-rich Repeat Kinase Enzyme Activity App 20160009682 - Miller; Michael ;   et al. | 2016-01-14 |
Compounds Inhibiting Leucine-rich Repeat Kinase Enzyme Activity App 20160009689 - Miller; Michael ;   et al. | 2016-01-14 |
Heterobicyclo-substituted [1,2,4]triazolo[1,5-c]quinazolin-5-amine Compounds With A2a Antagonist Properties App 20150361098 - Ali; Amjad ;   et al. | 2015-12-17 |
2'-azido substituted nucleoside derivatives and methods of use thereof for the treatment of viral diseases Grant 9,156,872 - Girijavallabhan , et al. October 13, 2 | 2015-10-13 |
2'-cyano substituted nucleoside derivatives and methods of use thereof useful for the treatment of viral diseases Grant 9,150,603 - Girijavallabhan , et al. October 6, 2 | 2015-10-06 |
Mineralocorticoid Receptor Antagonists App 20150182503 - Cernak; Timothy A. ;   et al. | 2015-07-02 |
Cyclic amide BACE-1 inhibitors having a benzamide substituent Grant 9,062,007 - Cumming , et al. June 23, 2 | 2015-06-23 |
2'-substituted nucleoside derivatives and methods of use thereof for the treatment of viral diseases Grant 9,061,041 - Girijavallabhan , et al. June 23, 2 | 2015-06-23 |
Substituted cyclopropyl compounds, compositions containing such compounds, and methods of treatment Grant 9,006,228 - Miller , et al. April 14, 2 | 2015-04-14 |
Pyrimidine ether derivatives and methods of use thereof Grant 8,912,206 - Neelamkavil , et al. December 16, 2 | 2014-12-16 |
2'-azido Substituted Nucleoside Derivatives And Methods Of Use Thereof For The Treatment Of Viral Diseases App 20140206640 - Girijavallabhan; Vinay ;   et al. | 2014-07-24 |
Heterocyclic aspartyl protease inhibitors Grant 8,778,980 - Zhu , et al. July 15, 2 | 2014-07-15 |
2'-cyano Substituted Nucleoside Derivatives And Methods Of Use Thereof Useful For The Treatment Of Viral Diseases App 20140161770 - Girijavallabhan; Vinay ;   et al. | 2014-06-12 |
2'-substituted Nucleoside Derivatives And Methods Of Use Thereof For The Treatment Of Viral Diseases App 20140154211 - Girijavallabhan; Vinay ;   et al. | 2014-06-05 |
Pyrimidine derivatives as GPCR modulators for use in the treatment of obesity and diabetes Grant 8,722,882 - Neustadt , et al. May 13, 2 | 2014-05-13 |
Substituted isoindolines as aspartyl protease inhibitors Grant 8,722,708 - Stamford , et al. May 13, 2 | 2014-05-13 |
Substituted Cyclopropyl Compounds, Compositions Containing Such Compounds, And Methods Of Treatment App 20140128368 - Miller; Michael ;   et al. | 2014-05-08 |
Cyclic Amide Bace-1 Inhibitors Having A Benzamide Substituent App 20140128361 - Cumming; Jared N. ;   et al. | 2014-05-08 |
Substituted imidazolones, compositions containing such compounds and methods of use Grant 8,633,231 - DeMong , et al. January 21, 2 | 2014-01-21 |
Aspartyl protease inhibitors Grant 8,629,155 - Wu , et al. January 14, 2 | 2014-01-14 |
Cyclic amine BACE-1 inhibitors having a benzamide substituent Grant 8,623,867 - Cumming , et al. January 7, 2 | 2014-01-07 |
Glucagon receptor antagonists, compositions, and methods for their use Grant 8,623,818 - Greenlee , et al. January 7, 2 | 2014-01-07 |
Substituted piperazines as CB1 antagonists Grant 8,623,873 - Gilbert , et al. January 7, 2 | 2014-01-07 |
Macrocyclic heterocyclic aspartyl protease inhibitors Grant 8,557,798 - Iserloh , et al. October 15, 2 | 2013-10-15 |
Thiophenyl-substituted 2-imino-3-methyl pyrrolo pyrimidinone compounds as BACE-1 inhibitors, compositions, and their use Grant 8,450,331 - Zhu , et al. May 28, 2 | 2013-05-28 |
Substituted Imidazolones, Compositions Containing Such Compounds And Methods Of Use App 20130123315 - DeMong; Duane ;   et al. | 2013-05-16 |
Bicyclic heterocycle derivatives and methods of use thereof Grant 8,410,122 - Harris , et al. April 2, 2 | 2013-04-02 |
Spiro-imidazolone derivatives as glucagon receptor antagonists Grant 8,361,959 - Stamford , et al. January 29, 2 | 2013-01-29 |
Heterocyclic Aspartyl Protease Inhibitors App 20130018066 - Zhu; Zhaoning ;   et al. | 2013-01-17 |
Cyclic Amine Bace-1 Inhibitors Having A Benzamide Substituent App 20130004518 - Cumming; Jared N. ;   et al. | 2013-01-03 |
Pyrimidine Ether Derivatives And Methods Of Use Thereof App 20120289525 - Neelamkavil; Santhosh Francis ;   et al. | 2012-11-15 |
Heterocyclic Aspartyl Protease Inhibitors App 20120276118 - Zhu; Zhaoning ;   et al. | 2012-11-01 |
Cyclic amine BACE-1 inhibitors having a benzamide substituent Grant 8,278,334 - Cumming , et al. October 2, 2 | 2012-10-02 |
Heterocyclic Aspartyl Protease Inhibitors App 20120231017 - ZHU; ZHAONING ;   et al. | 2012-09-13 |
Aspartyl Protease Inhibitors App 20120232064 - Wu; Yusheng ;   et al. | 2012-09-13 |
Heterocyclic Aspartyl Protease Inhibitors App 20120231018 - Zhu; Zhaoning ;   et al. | 2012-09-13 |
Fused Bicyclic Pyrimidine Derivatives And Methods Of Use Thereof App 20120232073 - Neelamkavil; Santhosh Francis ;   et al. | 2012-09-13 |
Bridged Bicyclic Piperidine Derivatives And Methods Of Use Thereof App 20120214805 - Harris; Joel M. ;   et al. | 2012-08-23 |
Heterocyclic aspartyl protease inhibitors Grant 8,183,252 - Zhu , et al. May 22, 2 | 2012-05-22 |
Aspartyl protease inhibitors Grant 8,168,641 - Wu , et al. May 1, 2 | 2012-05-01 |
Bridged Bicyclic Heterocycle Derivatives And Methods Of Use Thereof App 20120040975 - Neelamkavil; Santhosh Francis ;   et al. | 2012-02-16 |
Preparation and use of compounds as aspartyl protease inhibitors Grant 8,110,682 - McKittrick , et al. February 7, 2 | 2012-02-07 |
Aspartyl protease inhibitors Grant 8,093,254 - Zhu , et al. January 10, 2 | 2012-01-10 |
Pentafluorosulpholane-containing Antidiabetic Compounds App 20110313008 - Josien; Hubert B. ;   et al. | 2011-12-22 |
Pyrimidine Derivatives As Gpcr Modulators For Use In The Treatment Of Obesity And Diabetes App 20110263570 - Neustadt; Bernard R. ;   et al. | 2011-10-27 |
Bicyclic Heterocycle Derivatives And Methods Of Use Thereof App 20110263624 - Harris; Joel M. ;   et al. | 2011-10-27 |
Heterocyclic Aspartyl Protease Inhibitors App 20110218194 - Zhu; Zhaoning ;   et al. | 2011-09-08 |
Spiro-imidazolone Derivatives As Glucagon Receptor Antagonists App 20110178007 - Stamford; Andrew ;   et al. | 2011-07-21 |
Heterocyclic aspartyl protease inhibitors Grant 7,973,067 - Zhu , et al. July 5, 2 | 2011-07-05 |
Cyclic amine bace-1 inhibitors having a heterocyclic substituent Grant 7,910,590 - Huang , et al. March 22, 2 | 2011-03-22 |
Glucagon Receptor Antagonists, Compositions, And Methods For Their Use App 20110065634 - Greenlee; William J. ;   et al. | 2011-03-17 |
Aspartyl protease inhibitors Grant 7,868,000 - Zhu , et al. January 11, 2 | 2011-01-11 |
Heterocyclic Aspartyl Protease Inhibitors App 20100292203 - Zhu; Zhaoning ;   et al. | 2010-11-18 |
Macrocyclic heterocyclic aspartyl protease inhibitors Grant 7,812,013 - Iserloh , et al. October 12, 2 | 2010-10-12 |
Substituted Piperazines As Cb1 Antagonists App 20100249144 - Demong; Duane Eugene ;   et al. | 2010-09-30 |
Diaryl Morpholines As Cb1 Modulators App 20100197564 - Scott; Jack D. ;   et al. | 2010-08-05 |
Heterocyclic aspartyl protease inhibitors Grant 7,763,609 - Zhu , et al. July 27, 2 | 2010-07-27 |
Substituted spiro iminopyrimidinones as aspartyl protease inhibitors, compositions, and methods of treatment Grant 7,759,353 - Zhu , et al. July 20, 2 | 2010-07-20 |
Bicyclic guanidine derivatives as asparyl protease inhibitors, compositions, and uses thereof Grant 7,759,354 - Zhu , et al. July 20, 2 | 2010-07-20 |
Cyclic Amine Bace-1 Inhibitors Having A Benzamide Substituent App 20100152138 - Cumming; Jared N. ;   et al. | 2010-06-17 |
Adenosine A.sub.a2 receptor antagonists Grant 7,713,985 - Clasby , et al. May 11, 2 | 2010-05-11 |
Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A.sub.2a receptor antagonists Grant 7,709,492 - Neustadt , et al. May 4, 2 | 2010-05-04 |
Heterocyclic aspartyl protease inhibitors Grant 7,700,603 - Zhu , et al. April 20, 2 | 2010-04-20 |
Aspartyl Protease Inhibitors App 20100069406 - Zhu; Zhaoning ;   et al. | 2010-03-18 |
Macrocyclic Heterocyclic Aspartyl Protease Inhibitors App 20100063121 - Iserloh; Ulrich ;   et al. | 2010-03-11 |
Cyclic amine BACE-1 inhibitors having a benzamide substituent Grant 7,662,816 - Cumming , et al. February 16, 2 | 2010-02-16 |
Aspartyl Protease Inhibitors Containing A Tricyclic Ring System App 20100016341 - Zhu; Zhaoning ;   et al. | 2010-01-21 |
Cyclic Amine Bace-1 Inhibitors Having A Heterocyclic Substituent App 20090312341 - Cumming; Jared N. ;   et al. | 2009-12-17 |
Heterocyclic Aspartyl Protease Inhibitors App 20090306047 - Zhu; Zhaoning ;   et al. | 2009-12-10 |
Heterocyclic Aspartyl Protease Inhibitors App 20090258868 - Zhu; Zhaoning ;   et al. | 2009-10-15 |
Cyclic amine BACE-1 inhibitors having a heterocyclic substituent Grant 7,598,250 - Cumming , et al. October 6, 2 | 2009-10-06 |
Heterocyclic aspartyl protease inhibitors Grant 7,592,348 - Zhu , et al. September 22, 2 | 2009-09-22 |
Substituted Piperazines as CB1 Antagonists App 20090105208 - Gilbert; Eric J. ;   et al. | 2009-04-23 |
2-heteroaryl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists Grant 7,465,740 - Neustadt , et al. December 16, 2 | 2008-12-16 |
Neuropeptide receptor modulators Grant 7,459,450 - Zhu , et al. December 2, 2 | 2008-12-02 |
Adenosine A2a Receptor Antagonists App 20080255156 - Clasby; Martin C. ;   et al. | 2008-10-16 |
Heterocyclic aspartyl protease inhibitors App 20080200445 - Zhu; Zhaoning ;   et al. | 2008-08-21 |
Preparation and use of compounds as protease inhibitors App 20080176868 - Stamford; Andrew ;   et al. | 2008-07-24 |
Preparation and use of compounds as protease inhibitors App 20080113957 - McKittrick; Brian ;   et al. | 2008-05-15 |
2-alkynyl- and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A.sub.2a receptor antagonists Grant 7,368,449 - Neustadt , et al. May 6, 2 | 2008-05-06 |
Azetidinone Derivatives and Methods of Use Thereof App 20080076750 - Aslanian; Robert G. ;   et al. | 2008-03-27 |
Treating Pain, Diabetes, And Disorders Of Lipid Metabolism App 20080070892 - Harris; Joel M. ;   et al. | 2008-03-20 |
Metabolite of xanthine Phosphodiesterase 5 inhibitor and derivatives thereof useful for treatment of erectile dysfunction Grant 7,312,223 - Ghosal , et al. December 25, 2 | 2007-12-25 |
Heteroaryl urea neuropeptide Y Y5 receptor antagonists Grant 7,309,704 - Stamford , et al. December 18, 2 | 2007-12-18 |
Aspartyl Protease Inhibitors App 20070287692 - Wu; Yusheng ;   et al. | 2007-12-13 |
Xanthine phosphodiesterase V inhibitors Grant 7,268,141 - Chackalamannil , et al. September 11, 2 | 2007-09-11 |
Heterocyclic aspartyl protease inhibitors App 20070072852 - Zhu; Zhaoning ;   et al. | 2007-03-29 |
2-Heteroaryl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists App 20070066620 - Neustadt; Bernard R. ;   et al. | 2007-03-22 |
Aspartyl protease inhibitors App 20070060575 - Zhu; Zhaoning ;   et al. | 2007-03-15 |
Preparation and use of compounds as aspartyl protease inhibitors App 20070010667 - McKittrick; Brian ;   et al. | 2007-01-11 |
Aspartyl protease inhibitors App 20060287294 - Zhu; Zhaoning ;   et al. | 2006-12-21 |
Aspartyl protease inhibitors App 20060281730 - Zhu; Zhaoning ;   et al. | 2006-12-14 |
Macrocyclic heterocyclic aspartyl protease inhibitors App 20060281729 - Iserloh; Ulrich ;   et al. | 2006-12-14 |
Heterocyclic aspartyl protease inhibitors App 20060111370 - Zhu; Zhaoning ;   et al. | 2006-05-25 |
Neuropeptide receptor modulators App 20060089351 - Zhu; Zhaoning ;   et al. | 2006-04-27 |
Heteroaryl urea neuropeptide Y Y5 receptor antagonists App 20060030588 - Stamford; Andrew ;   et al. | 2006-02-09 |
Heteroaryl urea neuropeptide Y Y5 receptor antagonists Grant 6,982,267 - Stamford , et al. January 3, 2 | 2006-01-03 |
Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists App 20050239795 - Neustadt, Bernard R. ;   et al. | 2005-10-27 |
2-alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists App 20050222164 - Neustadt, Bernard R. ;   et al. | 2005-10-06 |
Heteroaryl urea neuropeptide Y Y5 receptor antagonists Grant 6,946,476 - Stamford , et al. September 20, 2 | 2005-09-20 |
Cyclic amine bace-1 inhibitors having a benzamide substituent App 20050119227 - Cumming, Jared N. ;   et al. | 2005-06-02 |
2-Alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists Grant 6,897,217 - Neustadt , et al. May 24, 2 | 2005-05-24 |
Cyclic amine BACE-1 inhibitors having a heterocyclic substituent App 20050043290 - Cumming, Jared N. ;   et al. | 2005-02-24 |
Substituted urea neuropeptide Y Y5 receptor antagonists App 20050038100 - Greenlee, William J. ;   et al. | 2005-02-17 |
Metabolite of xanthine phosphodiesterase 5 inhibitor and derivatives thereof useful for treatment of erectile dysfunction App 20050026939 - Ghosal, Anima ;   et al. | 2005-02-03 |
2-Alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists App 20040220194 - Neustadt, Bernard R. ;   et al. | 2004-11-04 |
Heteroaryl urea neuropeptide Y Y5 receptor antagonists App 20040006086 - Stamford, Andrew ;   et al. | 2004-01-08 |
Heteroaryl urea neuropeptide Y Y5 receptor antagonists App 20030055062 - Stamford, Andrew ;   et al. | 2003-03-20 |