Patent | Date |
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Cyclopropyl urea formyl peptide 2 receptor and formyl peptide 1 receptor agonists Grant 11,180,490 - Smallheer , et al. November 23, 2 | 2021-11-23 |
Macrocycles as factor XIA inhibitors Grant 11,136,327 - Corte , et al. October 5, 2 | 2021-10-05 |
Triazolopyridine inhibitors of myeloperoxidase Grant 11,059,818 - Smallheer , et al. July 13, 2 | 2021-07-13 |
Triazolopyridine inhibitors of myeloperoxidase and/or EPX Grant 11,008,317 - Kick , et al. May 18, 2 | 2021-05-18 |
Triazolopyridine Inhibitors Of Myeloperoxidase App 20200291015 - Smallheer; Joanne M. ;   et al. | 2020-09-17 |
Cyclopropyl Urea Formyl Peptide 2 Receptor And Formyl Peptide 1 Receptor Agonists App 20200199113 - Smallheer; Joanne M. ;   et al. | 2020-06-25 |
Macrocycles As Factor Xia Inhibitors App 20200087312 - Corte; James R. ;   et al. | 2020-03-19 |
Macrocyclic inhibitors of myeloperoxidase Grant 10,577,383 - Smallheer , et al. | 2020-03-03 |
Macrocycles as factor XIa inhibitors Grant 10,487,086 - Corte , et al. Nov | 2019-11-26 |
Triazolopyridine inhibitors of myeloperoxidase Grant 10,407,422 - Smallheer , et al. Sept | 2019-09-10 |
Macrocyclic Inhibitors Of Myeloperoxidase App 20190177340 - Smallheer; Joanne M. ;   et al. | 2019-06-13 |
Triazolopyridine inhibitors of myeloperoxidase Grant 10,214,527 - Shaw , et al. Feb | 2019-02-26 |
Triazolopyridine Inhibitors Of Myeloperoxidase App 20190023701 - Smallheer; Joanne M. ;   et al. | 2019-01-24 |
Five-membered heterocycles useful as serine protease inhibitors Grant 10,112,936 - Hangeland , et al. October 30, 2 | 2018-10-30 |
Triazolopyridine Inhibitors Of Myeloperoxidase App 20180282320 - Shaw; Scott A. ;   et al. | 2018-10-04 |
Macrocycles As Factor Xia Inhibitors App 20180022753 - Corte; James R. ;   et al. | 2018-01-25 |
Macrocycles as factor XIa inhibitors Grant 9,802,939 - Corte , et al. October 31, 2 | 2017-10-31 |
Five-membered Heterocycles Useful As Serine Protease Inhibitors App 20170166560 - Hangeland; Jon J. ;   et al. | 2017-06-15 |
Five-membered heterocycles useful as serine protease inhibitors Grant 9,617,224 - Hangeland , et al. April 11, 2 | 2017-04-11 |
Five-membered Heterocycles Useful As Serine Protease Inhibitors App 20150259297 - Hangeland; Jon J. ;   et al. | 2015-09-17 |
Five-membered heterocycles useful as serine protease inhibitors Grant 9,079,860 - Hangeland , et al. July 14, 2 | 2015-07-14 |
Macrocycles As Factor Xia Inhibitors App 20150112058 - Corte; James R. ;   et al. | 2015-04-23 |
Macrocycles as factor XIa inhibitors Grant 8,940,720 - Corte , et al. January 27, 2 | 2015-01-27 |
Five-membered Heterocycles Useful As Serine Protease Inhibitors App 20140206706 - Hangeland; Jon J. ;   et al. | 2014-07-24 |
Five-membered heterocycles useful as serine protease inhibitors Grant 8,716,492 - Hangeland , et al. May 6, 2 | 2014-05-06 |
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 8,604,056 - Pinto , et al. December 10, 2 | 2013-12-10 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20120270853 - Pinto; Donald J.P. ;   et al. | 2012-10-25 |
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 8,252,830 - Pinto , et al. August 28, 2 | 2012-08-28 |
Five-membered Heterocycles Useful As Serine Protease Inhibitors App 20120088758 - Hangeland; Jon J. ;   et al. | 2012-04-12 |
Macrocycles As Factor Xia Inhibitors App 20120041190 - Corte; James R. ;   et al. | 2012-02-16 |
Five-membered heterocycles useful as serine protease inhibitors Grant 8,101,778 - Hangeland , et al. January 24, 2 | 2012-01-24 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20110028446 - Pinto; Donald J.P. ;   et al. | 2011-02-03 |
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 7,842,708 - Pinto , et al. November 30, 2 | 2010-11-30 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20100022506 - Pinto; Donald J.P. ;   et al. | 2010-01-28 |
Substituted biaryl compounds as factor XIa inhibitors Grant 7,645,799 - Corte , et al. January 12, 2 | 2010-01-12 |
Arylpropionamide, arylacrylamide, ayrlpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 7,626,039 - Pinto , et al. December 1, 2 | 2009-12-01 |
Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors Grant 7,524,863 - Smallheer , et al. April 28, 2 | 2009-04-28 |
Substituted Biaryl Compounds As Factor Xia Inhibitors App 20090062287 - Corte; James R. ;   et al. | 2009-03-05 |
Five-membered Heterocycles Useful As Serine Protease Inhibitors App 20090036438 - Hangeland; Jon J. ;   et al. | 2009-02-05 |
Substituted biaryl compounds as factor XIa inhibitors Grant 7,459,564 - Corte , et al. December 2, 2 | 2008-12-02 |
Five-membered heterocycles useful as serine protease inhibitors Grant 7,453,002 - Hangeland , et al. November 18, 2 | 2008-11-18 |
Six-membered heterocycles useful as serine protease inhibitors Grant 7,429,604 - Corte , et al. September 30, 2 | 2008-09-30 |
Bicyclic heterocycles useful as serine protease inhibitors Grant 7,417,063 - Smallheer , et al. August 26, 2 | 2008-08-26 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20080161373 - Pinto; Donald J.P. ;   et al. | 2008-07-03 |
Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors Grant 7,157,470 - Smallheer , et al. January 2, 2 | 2007-01-02 |
Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors App 20060247243 - Smallheer; Joanne M. ;   et al. | 2006-11-02 |
Biarylmethyl indolines and indoles as antithromboembolic agents Grant 7,129,264 - Smallheer , et al. October 31, 2 | 2006-10-31 |
Substituted biaryl compounds as factor XIa inhibitors App 20060154915 - Corte; James R. ;   et al. | 2006-07-13 |
Six-membered heterocycles useful as serine protease inhibitors App 20060009455 - Corte; James R. ;   et al. | 2006-01-12 |
Five-membered heterocycles useful as serine protease inhibitors App 20050282805 - Hangeland, Jon J. ;   et al. | 2005-12-22 |
Bicyclic heterocycles useful as serine protease inhibitors App 20050228000 - Smallheer, Joanne M. ;   et al. | 2005-10-13 |
Monocyclic or bicyclic carbocycles and heterocycles as factor Xa inhibitors Grant 6,951,872 - Jacobson , et al. October 4, 2 | 2005-10-04 |
Biarylmethyl indolines, indoles and tetrahydroquinolines, useful as serine protease inhibitors App 20040220206 - Smallheer, Joanne M. ;   et al. | 2004-11-04 |
Monocyclic or bicyclic carbocycles and heterocycles as factor Xa inhibitors App 20040132718 - Jacobson, Irina C. ;   et al. | 2004-07-08 |
Monocyclic or bicyclic carbocycles and heterocycles as factor Xa inhibitors Grant 6,710,058 - Jacobson , et al. March 23, 2 | 2004-03-23 |
Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors App 20040006062 - Smallheer, Joanne M. ;   et al. | 2004-01-08 |
Monocyclic or bicyclic carbocycles and heterocycles as factor Xa inhibitors App 20020183324 - Jacobson, Irina C. ;   et al. | 2002-12-05 |
Novel isoxazoline fibrinogen receptor antagonists App 20020094978 - Smallheer, Joanne M. ;   et al. | 2002-07-18 |