Patent | Date |
---|
Pyrimidine derivatives Grant 11,446,298 - Boss , et al. September 20, 2 | 2022-09-20 |
N-substituted Indole Derivatives As Pge2 Receptor Modulators App 20220175775 - FRETZ; Heinz ;   et al. | 2022-06-09 |
Benzofurane and benzothiophene derivatives as PGE2 receptor modulators Grant 11,325,899 - Boss , et al. May 10, 2 | 2022-05-10 |
N-substituted indole derivatives as PGE2 receptor modulators Grant 11,241,431 - Fretz , et al. February 8, 2 | 2022-02-08 |
Benzimidazole-proline derivatives Grant 11,040,966 - Boss , et al. June 22, 2 | 2021-06-22 |
Benzofurane And Benzothiophene Derivatives As Pge2 Receptor Modulators App 20210115031 - BOSS; Christoph ;   et al. | 2021-04-22 |
Pyrimidine Derivatives As Pge2 Receptor Modulators App 20210113559 - BOSS; Christoph ;   et al. | 2021-04-22 |
N-substituted Indole Derivatives As Pge2 Receptor Modulators App 20200289507 - FRETZ; Heinz ;   et al. | 2020-09-17 |
Phenyl Derivatives As Pge2 Receptor Modulators App 20200179383 - BOSS; Christoph ;   et al. | 2020-06-11 |
Pyrimidine Derivatives App 20200108068 - BOSS; Christoph ;   et al. | 2020-04-09 |
N-substituted Indole Derivatives App 20200069686 - FRETZ; Heinz ;   et al. | 2020-03-05 |
Benzimidazole-proline Derivatives App 20190263797 - BOSS; Christoph ;   et al. | 2019-08-29 |
Benzimidazole-proline derivatives Grant 10,329,287 - Boss , et al. | 2019-06-25 |
Crystalline salt form of (S)-(2-(6 chloro-7-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-yl)(5-meth- oxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone as orexin receptor antagonist Grant 10,023,560 - Boss , et al. July 17, 2 | 2018-07-17 |
Crystalline form of (S)-(2-(6-chloro-7-methyl-1H-benzo[D]imidazol-2-yl)-2-methylpyrrolidin-1-- yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone and its use as orexin receptor antagonists Grant 9,914,720 - Boss , et al. March 13, 2 | 2018-03-13 |
Use of benzimidazole-proline derivatives Grant 9,914,721 - Boss , et al. March 13, 2 | 2018-03-13 |
Crystalline Salt Form Of (s)-(2-(6-chloro-7-methyl-1h-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-- Yl)(5-methoxy-2-(2h-1,2,3-triazol-2-yl)phenyl)methanone As Orexin Receptor Antagonist App 20180002317 - BOSS; Christoph ;   et al. | 2018-01-04 |
Benzimidazole-proline Derivatives App 20170305897 - BOSS; Christoph ;   et al. | 2017-10-26 |
Crystalline salt form of (S)-(2-(6-chloro-7-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-- yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone as orexin receptor antagonist Grant 9,790,208 - Boss , et al. October 17, 2 | 2017-10-17 |
Benzimidazole-proline derivatives Grant 9,732,075 - Boss , et al. August 15, 2 | 2017-08-15 |
Use Of Benzimidazole-proline Derivatives App 20170001985 - BOSS; Christoph ;   et al. | 2017-01-05 |
Crystalline Form Of (s)-(2-(6-chloro-7-methyl-1h-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1 -yl)(5-methoxy-2-(2h-1,2,3-triazol-2-yl)phenyl)methanone And Its Use As Orexin Receptor Antagonists App 20160368901 - BOSS; Christoph ;   et al. | 2016-12-22 |
Crystalline Salt Form Of (s)-(2-(6-chloro-7-methyl-1h-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-- Yl)(5-methoxy-2-(2h-1,2,3-triazol-2-yl)phenyl)methanone As Orexin Receptor Antagonist App 20160355506 - BOSS; Christoph ;   et al. | 2016-12-08 |
Orexin receptor antagonists which are [ortho bi-(hetero-)aryl]-[2-(meta bi-(hetero-)aryl)-pyrrolidin-1-yl]-methanone derivatives Grant 9,493,446 - Bolli , et al. November 15, 2 | 2016-11-15 |
Azetidine amide derivatives as orexin receptor antagonists Grant 9,403,813 - Bolli , et al. August 2, 2 | 2016-08-02 |
Pyrazole and imidazole derivatives useful as orexin antagonists Grant 9,303,023 - Bolli , et al. April 5, 2 | 2016-04-05 |
Azetidine Amide Derivatives As Orexin Receptor Antagonists App 20160024064 - BOLLI; Martin ;   et al. | 2016-01-28 |
Proline sulfonamide derivatives as orexin receptor antagonists Grant 9,211,279 - Boss , et al. December 15, 2 | 2015-12-15 |
2-(1,2,3-triazol-2-yl)benzamide and 3-(1,2,3-triazol-2-YL)picolinamide derivatives as orexin receptor antagonists Grant 9,150,566 - Bolli , et al. October 6, 2 | 2015-10-06 |
Orexin Receptor Antagonists Which Are [ortho Bi-(hetero-)aryl]-[2-(meta Bi-(hetero-)aryl)-pyrrolidin-1-yl]-methanone Derivatives App 20150252032 - Bolli; Martin ;   et al. | 2015-09-10 |
Proline Sulfonamide Derivatives As Orexin Receptor Antagonists App 20150246021 - BOSS; Christoph ;   et al. | 2015-09-03 |
Benzimidazole-proline Derivatives App 20150166527 - Boss; Christoph ;   et al. | 2015-06-18 |
2-(1,2,3-triazol-2-yl)benzamide And 3-(1,2,3-triazol-2-yl)picolinamide Derivatives As Orexin Receptor Antagonists App 20150158855 - Bolli; Martin ;   et al. | 2015-06-11 |
Proline sulfonamide derivatives as orexin receptor antagonists Grant 9,000,029 - Boss , et al. April 7, 2 | 2015-04-07 |
Proline Sulfonamide Derivatives As Orexin Receptor Antagonists App 20150057328 - BOSS; Christoph ;   et al. | 2015-02-26 |
Proline sulfonamide derivatives as orexin receptor antagonists Grant 8,895,606 - Boss , et al. November 25, 2 | 2014-11-25 |
Novel Pyrazole And Imidazole Derivatives Useful As Orexin Antagonists App 20130324579 - Bolli; Martin ;   et al. | 2013-12-05 |
Lactam Derivatives Useful As Orexin Receptor Antagonists App 20130237525 - Aissaoui; Hamed ;   et al. | 2013-09-12 |
Proline Sulfonamide Derivatives As Orexin Receptor Antagonists App 20130150424 - Boss; Christoph ;   et al. | 2013-06-13 |
Oxazolidinone derivatives Grant 8,329,706 - Aissaoui , et al. December 11, 2 | 2012-12-11 |
2-aza-bicyclo[3.3.0]octane derivatives Grant 8,288,429 - Aissaoui , et al. October 16, 2 | 2012-10-16 |
Pyrrolidines and piperidines as orexin receptor antagonists Grant 8,288,411 - Aissaoui , et al. October 16, 2 | 2012-10-16 |
2-aza-bicyclo[3.1.0]hexane derivatives as orexin receptor antagonists Grant 8,288,435 - Aissaoui , et al. October 16, 2 | 2012-10-16 |
2-aza-bicyclo[2.2.1]heptane derivatives Grant 8,236,801 - Aissaoui , et al. August 7, 2 | 2012-08-07 |
Thiazolidine derivatives as orexin receptor antagonists Grant 8,236,964 - Aissaoui , et al. August 7, 2 | 2012-08-07 |
Novel Oxazolidinone Deriviatives App 20120101111 - Aissaoui; Hamed ;   et al. | 2012-04-26 |
Thiazolidin-4-one And [1,3]-thiazinan-4-one Compounds As Orexin Receptor Antagonists App 20120088759 - Aissaoui; Hamed ;   et al. | 2012-04-12 |
Bicyclononene derivatives Grant 8,138,340 - Bezencon , et al. March 20, 2 | 2012-03-20 |
3-heteroaryl (amino or amido)-1-(biphenyl or phenylthiazolyl) carbonylpiperidine derivatives as orexin receptor inhibitors Grant 8,133,901 - Aissaoui , et al. March 13, 2 | 2012-03-13 |
3-aza-bicyclo[3.3.0]octane compounds Grant 8,106,215 - Aissaoui , et al. January 31, 2 | 2012-01-31 |
Trans-3-aza-bicyclo[3.1.0]hexane derivatives Grant 8,063,099 - Aissaoui , et al. November 22, 2 | 2011-11-22 |
1,2-diamido-ethylene Derivatives As Orexin Antagonists App 20110263662 - Aissaoui; Hamed ;   et al. | 2011-10-27 |
Phenethylamide Derivatives And Their Heterocyclic Analogues App 20110212968 - Aissaoui; Hamed ;   et al. | 2011-09-01 |
N-glycinsulfonamide derivatives and uses as orexin receptor antagonists Grant 8,003,654 - Aissaoui , et al. August 23, 2 | 2011-08-23 |
Azetidine compounds as orexin receptor antagonists Grant 7,994,336 - Aissaoui , et al. August 9, 2 | 2011-08-09 |
2-aza-bicyclo[3.1.0]hexane Derivatives As Orexin Receptor Antagonists App 20110124636 - Aissaoui; Hamed ;   et al. | 2011-05-26 |
Thiazolidine Compounds As Orexin Receptor Antagonists App 20110105491 - Aissaoui; Hamed ;   et al. | 2011-05-05 |
5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine Compounds App 20110105514 - Aissaoui; Hamed ;   et al. | 2011-05-05 |
Tetrazole Compounds As Orexin Receptor Antagonists App 20110086889 - Aissaoui; Hamed ;   et al. | 2011-04-14 |
Diazabicyclononene derivatives and use thereof Grant 7,915,259 - Bezencon , et al. March 29, 2 | 2011-03-29 |
Piperidine And Pyroolidine Compounds App 20110039857 - Aissaoui; Hamed ;   et al. | 2011-02-17 |
2-aza-bicyclo[3.3.0]octane Derivatives App 20110009461 - Aissaoui; Hamed ;   et al. | 2011-01-13 |
2-aza-bicyclo[2.2.1]heptane Derivatives App 20110009401 - Aissaoui; Hamed ;   et al. | 2011-01-13 |
Novel Piperidine Carboxylic Acid Amine Derivatives App 20100324052 - Bezencon; Olivier ;   et al. | 2010-12-23 |
Pyrazolo-tetrahydro pyridine derivatives as orexin receptor antagonists Grant 7,834,028 - Aissaoui , et al. November 16, 2 | 2010-11-16 |
Piperidine carboxylic acid amide derivatives Grant 7,799,805 - Bezencon , et al. September 21, 2 | 2010-09-21 |
2-cyclopropyl-thiazole Derivatives App 20100222328 - Aissaoui; Hamed ;   et al. | 2010-09-02 |
Azetidine Compounds As Orexin Receptor Antagonists App 20100222600 - Aissaoui; Hamed ;   et al. | 2010-09-02 |
Trans-3-aza-bicyclo[3.1.0]hexane Derivatives App 20100204285 - Aissaoui; Hamed ;   et al. | 2010-08-12 |
Pyrrolidines And Piperidines As Orexin Receptor Antagonists App 20100197733 - Aissaoui; Hamed ;   et al. | 2010-08-05 |
3-aza-bicyclo[3.3.0]octane Compounds App 20100184808 - Aissaoui; Hamed ;   et al. | 2010-07-22 |
Thiazolidine Derivatives As Orexin Receptor Antagonists App 20100113531 - Aissaoui; Hamed ;   et al. | 2010-05-06 |
5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine Derivatives App 20100093740 - Aissaoui; Hamed ;   et al. | 2010-04-15 |
3-heteroaryl (amino Or Amido)-1-(biphenyl Or Phenylthiazolyl) Carbonylpiperidine Derivatives As Orexin Receptor Inhibitors App 20100069418 - Aissaoui; Hamed ;   et al. | 2010-03-18 |
1,4,5,6,7,8-hexahydro-1,2,5-triaza-azulene Derivatives As Orexin Receptor Antagonists App 20100029617 - Aissaoui; Hamed ;   et al. | 2010-02-04 |
3-aza-bicyclo[3.1.0]hexane Derivatives App 20100016401 - Aissaoui; Hamed ;   et al. | 2010-01-21 |
Bicyclononene derivaties App 20090306123 - Bezencon; Olivier ;   et al. | 2009-12-10 |
Novel Sulfonamide Compounds App 20090275588 - Aissaoui; Hamed ;   et al. | 2009-11-05 |
Quinoxalin-3-one derivatives as orexin receptor antagonists Grant 7,538,109 - Aissaoui , et al. May 26, 2 | 2009-05-26 |
Pyrazolo-tetrahydro Pyridine Derivatives As Orexin Receptor Antagonists App 20090099228 - Aissaoui; Hamed ;   et al. | 2009-04-16 |
Sulfonylamino-acetic acid derivatives Grant 7,435,815 - Aissaoui , et al. October 14, 2 | 2008-10-14 |
Novel Tetrahydropyridine Derivatives App 20080234305 - Bezencon; Olivier ;   et al. | 2008-09-25 |
Novel Piperidine Carboxylic Acid Amide Derivatives App 20080214598 - Bezencon; Olivier ;   et al. | 2008-09-04 |
Diazabicyclononene Derivatives and Use Thereof App 20080161313 - Bezencon; Oliver ;   et al. | 2008-07-03 |
Novel Diazabicyclononene Derivative App 20080103152 - Bezencon; Olivier ;   et al. | 2008-05-01 |
Sulfonylamino-acetic Acid Derivatives App 20070244156 - Aissaoui; Hamed ;   et al. | 2007-10-18 |
Sulfonylamino-acetic acid derivatives Grant 7,279,578 - Aissaoui , et al. October 9, 2 | 2007-10-09 |
Novel diazabicyclonene derivatives and use thereof App 20070142363 - Bezencon; Olivier ;   et al. | 2007-06-21 |
Diazabicyclononene and tetrahydropyridine derivatives with a new side-chain App 20070135406 - Bezencon; Olivier ;   et al. | 2007-06-14 |
Novel diazabicyclononene and tetrahydropyridine derivatives with a new polar side-chain App 20070135405 - Bezencon; Olivier ;   et al. | 2007-06-14 |
Novel diazabicyclononene derivatives and use App 20070111989 - Bezencon; Olivier ;   et al. | 2007-05-17 |
Benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists Grant 7,192,950 - Aissaoui , et al. March 20, 2 | 2007-03-20 |
Quinoxalinone-3-one derivatives as orexin receptor antagonists App 20070027157 - Aissaoui; Hamed ;   et al. | 2007-02-01 |
9-Azabicyclo'3.3.1 inon-6-ee derivatives with a heteroatom at the 3-position as renin inhibitors App 20060258648 - Bezencon; Olivier ;   et al. | 2006-11-16 |
Novel diazabicyclononene derivatives App 20060223795 - Bezencon; Oliver ;   et al. | 2006-10-05 |
Tropane derivatives and their use as ace inhibitors App 20060205768 - Bezencon; Olivier ;   et al. | 2006-09-14 |
Tetrahydroisoquinolyl acetamide derivatives for use as orexin receptor antagonists App 20060178515 - Aissaoui; Hamed ;   et al. | 2006-08-10 |
7,8,9,10-tetrahydro-6H-azepino, 6,7,8,9-tetrahydro-pyrido and 2,3-dihydro-2H-pyrrolo[2,1-b]-quinazolinone derivatives Grant 7,067,519 - Aissaoui , et al. June 27, 2 | 2006-06-27 |
Sulfonylamino-acetic acid derivatives App 20060014783 - Aissaoui; Hamed ;   et al. | 2006-01-19 |
Novel benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists App 20040058912 - Aissaoui, Hamed ;   et al. | 2004-03-25 |