Patent | Date |
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Spirocyclic Lactams As Jak2 V617f Inhibitors App 20220281887 - Shepard; Stacey ;   et al. | 2022-09-08 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20220251087 - Buesking; Andrew W. ;   et al. | 2022-08-11 |
Substituted heterocyclic derivatives as PI3K inhibitors Grant 11,396,502 - Shepard , et al. July 26, 2 | 2022-07-26 |
Pyridine And Pyridimine Compounds As Pi3k-gamma Inhibitors App 20220227736 - Sparks; Richard B. ;   et al. | 2022-07-21 |
TERTIARY ALCOHOLS AS PI3K-y INHIBITORS App 20220213107 - Douty; Brent ;   et al. | 2022-07-07 |
AMINOPYRAZINE DIOL COMPOUNDS AS PI3K-y INHIBITORS App 20220213065 - Shepard; Stacey ;   et al. | 2022-07-07 |
Pyridine and pyridimine compounds as PI3K-gamma inhibitors Grant 11,352,340 - Sparks , et al. June 7, 2 | 2022-06-07 |
Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors Grant 11,331,320 - Rodgers , et al. May 17, 2 | 2022-05-17 |
3-(5-amino-pyrazin-2-yl)-benzenesulfonamide derivatives and related compounds as PI3K-gamma kinase inhibitors Grant 11,306,079 - Shvartsbart , et al. April 19, 2 | 2022-04-19 |
Tertiary alcohols as PI3K-.gamma. inhibitors Grant 11,225,486 - Douty , et al. January 18, 2 | 2022-01-18 |
Heterocyclic Derivatives As Pi3k Inhibitors App 20210395258 - Shepard; Stacey ;   et al. | 2021-12-23 |
Naphthyridinone Compounds As Jak2 V617f Inhibitors App 20210395251 - Shepard; Stacey ;   et al. | 2021-12-23 |
Heterocyclic derivatives as PI3K inhibitors Grant 11,161,838 - Shepard , et al. November 2, 2 | 2021-11-02 |
Tricyclic heterocycles as BET protein inhibitors Grant 11,091,484 - Rodgers , et al. August 17, 2 | 2021-08-17 |
Heterocyclic compounds as PI3K-y inhibitors Grant 11,091,491 - Shvartsbart , et al. August 17, 2 | 2021-08-17 |
Heterocyclic derivatives as PI3K inhibitors Grant 11,078,204 - Shepard , et al. August 3, 2 | 2021-08-03 |
Aminopyrazine derivatives as PI3K-.gamma. inhibitors Grant 11,046,658 - Douty , et al. June 29, 2 | 2021-06-29 |
Imidazo[2,1-f][1,2,4]triazine compounds as pi3k-y inhibitors Grant 10,975,088 - Buesking , et al. April 13, 2 | 2021-04-13 |
TERTIARY ALCOHOLS AS PI3K-y INHIBITORS App 20200385392 - Douty; Brent ;   et al. | 2020-12-10 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20200338077 - Rodgers; James D. ;   et al. | 2020-10-29 |
AMINOPYRAZINE DIOL COMPOUNDS AS PI3K-y INHIBITORS App 20200339542 - Shepard; Stacey ;   et al. | 2020-10-29 |
3-(5-amino-pyrazin-2-yl)-benzenesulfonamide Derivatives And Related Compounds As Pi3k-gamma Kinase Inhibitors For Treating E.g. Cancer App 20200331903 - SHVARTSBART; Artem ;   et al. | 2020-10-22 |
Tertiary alcohols as PI3K-.gamma. inhibitors Grant 10,738,057 - Douty , et al. A | 2020-08-11 |
Aminopyrazine diol compounds as PI3K-.gamma. inhibitors Grant 10,669,262 - Shepard , et al. | 2020-06-02 |
Heterocyclic Derivatives As Pi3k Inhibitors App 20200148689 - Shepard; Stacey ;   et al. | 2020-05-14 |
Substituted Heterocyclic Derivatives As Pi3k Inhibitors App 20200148667 - Shepard; Stacey ;   et al. | 2020-05-14 |
Heterocyclic Derivatives As Pi3k Inhibitors App 20200148671 - Shepard; Stacey ;   et al. | 2020-05-14 |
Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors Grant 10,639,310 - Rodgers , et al. | 2020-05-05 |
Cyclobutyl substituted pyrrolopyridine and pyrrolopyrimidines derivatives as JAK inhibitors Grant 10,640,506 - Rodgers , et al. | 2020-05-05 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20200102315 - Buesking; Andrew W. ;   et al. | 2020-04-02 |
METABOLITES OF THE JANUS KINASE INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYL- PROPANENITR App 20200038404 - Rodgers; James D. ;   et al. | 2020-02-06 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20200031837 - Shvartsbart; Artem ;   et al. | 2020-01-30 |
Tricyclic Heterocycles As Bet Protein Inhibitors App 20200017497 - Rodgers; James D. ;   et al. | 2020-01-16 |
AMINOPYRAZINE DERIVATIVES AS PI3K-y INHIBITORS App 20200002295 - Douty; Brent ;   et al. | 2020-01-02 |
Pyridine And Pyridimine Compounds As Pi3k-gamma Inhibitors App 20190359592 - Sparks; Richard B. ;   et al. | 2019-11-28 |
Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines and substituted imidazo[1,2-b]pyridazines as PI3K-gamma inhibitors Grant 10,479,795 - Buesking , et al. Nov | 2019-11-19 |
Heterocyclic compounds as PI3K-.gamma. inhibitors Grant 10,472,368 - Shvartsbart , et al. Nov | 2019-11-12 |
Metabolites of the janus kinase inhibitor (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentyl- propanenitrile Grant 10,463,667 - Rodgers , et al. No | 2019-11-05 |
Tricyclic heterocycles as bet protein inhibitors Grant 10,442,803 - Rodgers , et al. Oc | 2019-10-15 |
AMINOPYRAZINE DIOL COMPOUNDS AS PI3K-y INHIBITORS App 20190276435 - Shepard; Stacey ;   et al. | 2019-09-12 |
Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as janus kinase inhibitors Grant 10,398,699 - Rodgers , et al. Sep | 2019-09-03 |
TERTIARY ALCOHOLS AS PI3K-y INHIBITORS App 20190152975 - Douty; Brent ;   et al. | 2019-05-23 |
Cyclobutyl Substituted Pyrrolopyridine And Pyrrolopyrimidines Derivatives As Jak Inhibitors App 20190135813 - Rodgers; James D. ;   et al. | 2019-05-09 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20190125750 - Rodgers; James D. ;   et al. | 2019-05-02 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20190119287 - Buesking; Andrew W. ;   et al. | 2019-04-25 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20190062336 - Shvartsbart; Artem ;   et al. | 2019-02-28 |
Piperidin-4-yl Azetidine Derivatives As Jak1 Inhibitors App 20180353499 - Huang; Taisheng ;   et al. | 2018-12-13 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20180338978 - Rodgers; James D. ;   et al. | 2018-11-29 |
Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines, substituted imidazo[1,2-b]pyridazines and substituted imidazo[1,2-a]pyrazines as PI3K-.gamma. inhibitors Grant 10,138,248 - Buesking , et al. Nov | 2018-11-27 |
Heterocyclic compounds as PI3K-.gamma. inhibitors Grant 10,065,963 - Shvartsbart , et al. September 4, 2 | 2018-09-04 |
Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as janus kinase inhibitors Grant 9,974,790 - Rodgers , et al. May 22, 2 | 2018-05-22 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20180009816 - Buesking; Andrew W. ;   et al. | 2018-01-11 |
Tricyclic Heterocycles As Bet Protein Inhibitors App 20180002334 - Rodgers; James D. ;   et al. | 2018-01-04 |
METABOLITES OF THE JANUS KINASE INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYL- PROPANENITRILE App 20170326144 - Rodgers; James D. ;   et al. | 2017-11-16 |
Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as janus kinase inhibitors Grant 9,814,722 - Rodgers , et al. November 14, 2 | 2017-11-14 |
Tricyclic heterocycles as bet protein inhibitors Grant 9,777,003 - Shepard , et al. October 3, 2 | 2017-10-03 |
Piperidin-4-yl Azetidine Derivatives As Jak1 Inhibitors App 20170246157 - Huang; Taisheng ;   et al. | 2017-08-31 |
Pyridine And Pyridimine Compounds As Pi3k-gamma Inhibitors App 20170190689 - Sparks; Richard B. ;   et al. | 2017-07-06 |
Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as janus kinase inhibitors Grant 9,662,335 - Rodgers , et al. May 30, 2 | 2017-05-30 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20170129899 - Shvartsbart; Artem ;   et al. | 2017-05-11 |
Heteroaryl Substituted Pyrrolo[2,3-B] Pyridines And Pyrrolo[2,3-B] Pyrimidines As Janus Kinase Inhibitors App 20170071947 - Rodgers; James D. ;   et al. | 2017-03-16 |
Hydroxyl, keto, and glucuronide derivatives of 3-(4-(7H-pyrrolo[2,3-D]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylprop- anenitrile Grant 9,512,161 - Rodgers , et al. December 6, 2 | 2016-12-06 |
Heteroaryl Substituted Pyrrolo[2,3-B] Pyridines And Pyrrolo[2,3-B] Pyrimidines As Janus Kinase Inhibitors App 20160346286 - Rodgers; James D. ;   et al. | 2016-12-01 |
Heteroaryl Substituted Pyrrolo[2,3-B] Pyridines And Pyrrolo[2,3-B] Pyrimidines As Janus Kinase Inhibitors App 20160272648 - Rodgers; James D. ;   et al. | 2016-09-22 |
Tricyclic Heterocycles As Bet Protein Inhibitors App 20160168148 - Shepard; Stacey | 2016-06-16 |
N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors Grant 9,334,274 - Rodgers , et al. May 10, 2 | 2016-05-10 |
Tricyclic heterocycles as BET protein inhibitors Grant 9,309,246 - Rodgers , et al. April 12, 2 | 2016-04-12 |
Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors Grant 9,249,145 - Rodgers , et al. February 2, 2 | 2016-02-02 |
Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as Janus kinase Grant 9,206,187 - Rodgers , et al. December 8, 2 | 2015-12-08 |
Piperidinylcyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as JAK inhibitors Grant 9,193,733 - Rodgers , et al. November 24, 2 | 2015-11-24 |
Heteroaryl Substituted Pyrrolo[2,3-B] Pyridines And Pyrrolo[2,3-B] Pyrimidines As Janus Kinase Inhibitors App 20150238492 - Rodgers; James D. ;   et al. | 2015-08-27 |
Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as Janus kinase inhibitors Grant 9,079,912 - Rodgers , et al. July 14, 2 | 2015-07-14 |
Tricyclic Heterocycles As Bet Protein Inhibitors App 20150175604 - Rodgers; James D. ;   et al. | 2015-06-25 |
METABOLITES OF THE JANUS KINASE INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYL- PROPANENITRILE App 20150164900 - Rodgers; James D. ;   et al. | 2015-06-18 |
Cyclobutyl Substituted Pyrrolopyridine And Pyrrolopyrimidines Derivatives As Jak Inhibitors App 20150087632 - Rodgers; James D. ;   et al. | 2015-03-26 |
Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors Grant 8,946,245 - Rodgers , et al. February 3, 2 | 2015-02-03 |
Cyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as JAK inhibitors Grant 8,933,085 - Rodgers , et al. January 13, 2 | 2015-01-13 |
Heteroaryl substituted pyrrolo[2,3-B]pyridines and pyrrolo[2,3-B]pyrimidines as Janus kinase inhibitors Grant 8,933,086 - Rodgers , et al. January 13, 2 | 2015-01-13 |
HYDROXYL, KETO, AND GLUCURONIDE DERIVATIVES OF 3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROP- ANENITRILE App 20140378400 - Rodgers; James D. ;   et al. | 2014-12-25 |
Metabolites of the janus kinase inhibitor (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentyl- propanenitrile Grant 8,889,697 - Rodgers , et al. November 18, 2 | 2014-11-18 |
Piperidin-4-yl Azetidine Derivatives As Jak1 Inhibitors App 20140275031 - Huang; Taisheng ;   et al. | 2014-09-18 |
Heteroaryl Substituted Pyrrolo[2,3-B] Pyridines And Pyrrolo[2,3-B] Pyrimidines As Janus Kinase Inhibitors App 20140243360 - Rodgers; James D. ;   et al. | 2014-08-28 |
N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-d]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20140221379 - Rodgers; James D ;   et al. | 2014-08-07 |
Hydroxyl, keto, and glucuronide derivatives of 3-(4-(7H pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitril- e Grant 8,748,401 - Rodgers , et al. June 10, 2 | 2014-06-10 |
N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors Grant 8,716,303 - Rodgers , et al. May 6, 2 | 2014-05-06 |
Heteroaryl Substituted Pyrrolo[2,3-B]Pyridines And Pyrrolo[2,3-B]Pyrimidines As Janus Kinase Inhibitors App 20140018374 - Rodgers; James D. ;   et al. | 2014-01-16 |
Piperidinylcyclobutyl Substituted Pyrrolopyridine And Pyrrolopyrimidine Derivatives As Jak Inhibitors App 20140005166 - RODGERS; JAMES D. ;   et al. | 2014-01-02 |
Heteroaryl Substituted Pyrrolo[2,3-B] Pyridines And Pyrrolo[2,3-B] Pyrimidines As Janus Kinase Inhibitors App 20140005210 - Rodgers; James D. ;   et al. | 2014-01-02 |
HYDROXYL, KETO, AND GLUCURONIDE DERIVATIVES OF 3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROP- ANENITRILE App 20130345157 - Rodgers; James D. ;   et al. | 2013-12-26 |
Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors Grant 8,541,425 - Rodgers , et al. September 24, 2 | 2013-09-24 |
Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors Grant 8,530,485 - Rodgers , et al. September 10, 2 | 2013-09-10 |
Azetidine And Cyclobutane Derivatives As Jak Inhibitors App 20130225556 - RODGERS; James D. ;   et al. | 2013-08-29 |
Hydroxyl, keto, and glucuronide derivatives of 3-(4-(7H-pyrrolo[2,3-d] pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile Grant 8,486,902 - Rodgers , et al. July 16, 2 | 2013-07-16 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20130137681 - Rodgers; James D. ;   et al. | 2013-05-30 |
Azetidine and cyclobutane derivatives as JAK inhibitors Grant 8,420,629 - Rodgers , et al. April 16, 2 | 2013-04-16 |
Pyrazolyl substituted pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors Grant 8,415,362 - Rodgers , et al. April 9, 2 | 2013-04-09 |
Cyclobutyl Substituted Pyrrolopyridine And Pyrrolopyrimidine Derivatives As Jak Inhibitors App 20120149681 - RODGERS; JAMES D. ;   et al. | 2012-06-14 |
Azetidine and cyclobutane derivatives as JAK inhibitors Grant 8,158,616 - Rodgers , et al. April 17, 2 | 2012-04-17 |
Azetidine And Cyclobutane Derivatives As Jak Inhibitors App 20120077798 - RODGERS; James D. ;   et al. | 2012-03-29 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20110224157 - Rodgers; James D. ;   et al. | 2011-09-15 |
Piperidin-4-yl Azetidine Derivatives As Jak1 Inhibitors App 20110224190 - Huang; Taisheng ;   et al. | 2011-09-15 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20110223210 - Rodgers; James D. ;   et al. | 2011-09-15 |
HYDROXYL, KETO, AND GLUCURONIDE DERIVATIVES OF 3-(4-(7H-PYRROLO[2,3-d] PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROPANENITRILE App 20110086810 - RODGERS; James D. ;   et al. | 2011-04-14 |
METABOLITES OF THE JANUS KINASE INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYL- PROPANENITRILE App 20110082159 - RODGERS; James D. ;   et al. | 2011-04-07 |
HETEROCYCLIC DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20110059951 - Rodgers; James D. ;   et al. | 2011-03-10 |
N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-d]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20100298334 - Rodgers; James D. ;   et al. | 2010-11-25 |
Metabolites of the Janus kinase inhibitor (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentyl- propanenitrile Grant 7,834,022 - Rodgers , et al. November 16, 2 | 2010-11-16 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20100022522 - Rodgers; James D. ;   et al. | 2010-01-28 |
Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as janus kinase inhibitors Grant 7,598,257 - Rodgers , et al. October 6, 2 | 2009-10-06 |
Azetidine And Cyclobutane Derivatives As Jak Inhibitors App 20090233903 - Rodgers; James D. ;   et al. | 2009-09-17 |
Tetracyclic Inhibitors Of Janus Kinases App 20090215766 - Rodgers; James D. ;   et al. | 2009-08-27 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20090181959 - Rodgers; James D. ;   et al. | 2009-07-16 |
Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as janus kinase inhibitors App 20070135461 - Rodgers; James D. ;   et al. | 2007-06-14 |
Tetracyclic inhibitors of Janus kinases App 20060106020 - Rodgers; James D. ;   et al. | 2006-05-18 |