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Triazolopyridazines as PAR1 inhibitors, production thereof, and use as medicaments Grant 9,079,906 - Heinelt , et al. July 14, 2 | 2015-07-14 |
Tricyclic pyridyl-vinyl pyrroles as PAR1 inhibitors Grant 8,871,798 - Schoenafinger , et al. October 28, 2 | 2014-10-28 |
Triazolium salts as PAR1 inhibitors, production thereof, and use as medicaments Grant 8,853,206 - Heinelt , et al. October 7, 2 | 2014-10-07 |
Imidazopyridazines as PAR1 inhibitors, production thereof, and use as medicaments Grant 8,598,177 - Heinelt , et al. December 3, 2 | 2013-12-03 |
SF.sub.5 derivatives as PAR1 inhibitors, production thereof, and use as medicaments Grant 8,466,169 - Heinelt , et al. June 18, 2 | 2013-06-18 |
Tricyclic Pyridyl-vinyl Pyrroles As Par1 Inhibitors App 20130040943 - SCHOENAFINGER; Karl ;   et al. | 2013-02-14 |
Cyclic pyridyl-N-[1,3,4]-thiadiazol-2-yl-benzene sulfonamides, processes for their preparation and their use as pharmaceuticals Grant 8,344,004 - Schoenafinger , et al. January 1, 2 | 2013-01-01 |
Urea- and urethane-substituted acylureas, process for their preparation and their use Grant 8,247,452 - DeFossa , et al. August 21, 2 | 2012-08-21 |
Triazolium Salts As Par1 Inhibitors, Production Thereof, And Use As Medicaments App 20120208805 - HEINELT; Uwe ;   et al. | 2012-08-16 |
Substituted 8-aminoalkylthioxanthines, and their use as inhibitors of dipeptidyl peptidase IV Grant 8,236,810 - Schoenafinger , et al. August 7, 2 | 2012-08-07 |
Triazolium salts as PAR1 inhibitors, production thereof, and use as medicaments Grant 8,198,272 - Heinelt , et al. June 12, 2 | 2012-06-12 |
Sulfonyl-phenyl-2H-[1,2,4]oxadiazol-5-one derivatives, processes for their preparation and their use as pharmaceuticals Grant 8,173,674 - Keil , et al. May 8, 2 | 2012-05-08 |
Amide-substituted 8-N-benzimidazoles, method for the production thereof, and use of the same as medicaments Grant 8,163,774 - DeFossa , et al. April 24, 2 | 2012-04-24 |
Aminocarbonyl-substituted 8-N-benzimidazoles, methods for their preparation and their use in pharmaceutical compositions Grant 8,138,207 - DeFossa , et al. March 20, 2 | 2012-03-20 |
Triazolopyridazines As Par1 Inhibitors, Production Thereof, And Use As Medicaments App 20120010203 - HEINELT; Uwe ;   et al. | 2012-01-12 |
Triazolopyridazines as PAR1 inhibitors, production thereof, and use as medicaments Grant 8,076,336 - Heinelt , et al. December 13, 2 | 2011-12-13 |
Cyclic pyridyl-N-[1,3,4]-thiadiazol-2-yl-benzene sulfonamides, processes for their preparation and their use as pharmaceuticals App 20110224263 - SCHOENAFINGER; Karl ;   et al. | 2011-09-15 |
Amino-substituted 8-N-benzimidazoles and methods for their use in blood sugar disorders Grant 8,003,668 - Defossa , et al. August 23, 2 | 2011-08-23 |
Pyridazinone kinase inhibitors Grant 7,968,546 - Hoelder , et al. June 28, 2 | 2011-06-28 |
4-oxy-N-[1,3,4]-thiadiazol-2-yl-benzene sulfonamides, pharmaceutical compositions and methods for their therapeutic use Grant 7,910,612 - Keil , et al. March 22, 2 | 2011-03-22 |
Substituted, bicyclic 8-pyrrolidinoxanthines, and methods for their use as inhibitors of dipeptidyl peptidase Grant 7,888,343 - Schoenafinger , et al. February 15, 2 | 2011-02-15 |
Triazolopyridazines As Par1 Inhibitors, Production Thereof, And Use As Medicaments App 20110034451 - HEINELT; Uwe ;   et al. | 2011-02-10 |
Sf5 Derivatives As Par1 Inhibitors, Production Thereof, And Use As Medicaments App 20110034461 - HEINELT; Uwe ;   et al. | 2011-02-10 |
Triazolium Salts As Par1 Inhibitors, Production Thereof, And Use As Medicaments App 20110034452 - HEINELT; Uwe ;   et al. | 2011-02-10 |
Imidazopyridazines As Par1 Inhibitors, Production Thereof, And Use As Medicaments App 20110034456 - HEINELT; Uwe ;   et al. | 2011-02-10 |
Substituted 8-aminoalkoxy-xanthine compounds and compositions useful in the treatment of hyperlipidemia and diabetes Grant 7,879,864 - Schoenafinger , et al. February 1, 2 | 2011-02-01 |
N-[1,3,4]-thiadiazol-2-yl-benzene sulfonamides, pharmaceutical compositions thereof and methods for their therapeutic use Grant 7,858,647 - Keil , et al. December 28, 2 | 2010-12-28 |
Substituted bicyclic 8-pyrrolidinoxanthines, methods for their production, pharmaceutical formulations and their use Grant 7,838,528 - Schoenafinger , et al. November 23, 2 | 2010-11-23 |
Substituted 2-aminoalkylthiobenzimidazole compounds, pharmaceutical compositions thereof and methods for their use Grant 7,795,445 - Defossa , et al. September 14, 2 | 2010-09-14 |
Substituted N-aminomethylene sulfonamides, production and use thereof as medicaments Grant 7,781,613 - Schoenafinger , et al. August 24, 2 | 2010-08-24 |
Carboxyalkoxy-substituted acyl-carboxyphenylurea derivatives and their use as medicaments Grant 7,781,459 - DeFossa , et al. August 24, 2 | 2010-08-24 |
Bicyclic aryl-sulfonic acid [1,3,4]-thiadiazol-2-yl-amides, processes for their preparation, pharmaceutical compositions and methods for their use Grant 7,772,257 - Schoenafinger , et al. August 10, 2 | 2010-08-10 |
4-benzimidazol-2-ylpyridazin-3-one derivatives Grant 7,754,713 - Hoelder , et al. July 13, 2 | 2010-07-13 |
Phenothiazin derivatives, method for the production thereof and use thereof as pharmaceuticals Grant 7,732,440 - Keil , et al. June 8, 2 | 2010-06-08 |
4-benzimidazol-2-yl-pyridazine-3-one-derivatives, production and use thereof in medicaments Grant 7,727,989 - Schoenafinger , et al. June 1, 2 | 2010-06-01 |
Acylated indanyl amines and their use as pharmaceuticals Grant 7,713,963 - Strobel , et al. May 11, 2 | 2010-05-11 |
Pyridazinone derivatives, methods for their production and their use as pharmaceuticals Grant 7,709,466 - Hoelder , et al. May 4, 2 | 2010-05-04 |
Cyclic N-[1,3,4]-thiadiazol-2-yl-benzene sulfonamides, pharmaceutical compositions and methods for the therapeutic use thereof Grant 7,683,181 - Schoenafinger , et al. March 23, 2 | 2010-03-23 |
Bicyclic Aryl-sulfonic Acid [1,3,4]-thiadiazol-2-yl-amides, Processes For Their Preparation, Pharmaceutical Compositions And Methods For Their Use App 20100022603 - SCHOENAFINGER; Karl ;   et al. | 2010-01-28 |
Phenothiazin Derivates, Method For The Production Thereof And Use Thereof As Pharmaceuticals App 20090325942 - KEIL; Stefanie ;   et al. | 2009-12-31 |
Sulfonyl-phenyl-2h-[1,2,4]oxadiazol-5-one Derivatives , Processes For Their Preparation And Their Use As Pharmaceuticals App 20090298871 - KEIL; Stefanie ;   et al. | 2009-12-03 |
Bicyclic aryl-sulfonic acid [1,3,4]-thiadiazol-2-yl-amides, processes for their preparation, pharmaceutical compositions and methods for their use Grant 7,612,104 - Schoenafinger , et al. November 3, 2 | 2009-11-03 |
Substituted, bicyclic 8-pyrrolidinobenzimidazoles, methods for their production and their use as medicaments Grant 7,569,700 - Defossa , et al. August 4, 2 | 2009-08-04 |
Novel Pyridazinone Derivatives App 20090130209 - HOELDER; Swen ;   et al. | 2009-05-21 |
Pyridazinone derivatives Grant 7,507,734 - Hoelder , et al. March 24, 2 | 2009-03-24 |
Substituted benzoylureidopyridylpiperidine-and-pyrrolidinecarboxylic acid derivatives, processes for preparing them and their use Grant 7,501,440 - Schoenafinger , et al. March 10, 2 | 2009-03-10 |
N-[1,3,4]-thiadiazol-2-yl-benzene Sulfonamides, Pharmaceutical Compositions Thereof And Methods For Their Therapeutic Use App 20090054494 - KEIL; Stefanie ;   et al. | 2009-02-26 |
Novel 4-benzimidazol-2-ylpyridazin-3-one Derivatives App 20090042880 - HOELDER; Swen ;   et al. | 2009-02-12 |
4-oxy-n-[1,3,4]-thiadiazol-2-yl-benzene Sulfonamides, Pharmaceutical Compositions And Methods For Their Therapeutic Use App 20090012131 - KEIL; Stefanie ;   et al. | 2009-01-08 |
4-benzimidazol-2-ylpyridazin-3-one derivatives Grant 7,470,689 - Hoelder , et al. December 30, 2 | 2008-12-30 |
Bicyclic Aryl-sulfonic Acid [1,3,4]-thiadiazol-2-yl-amides, Processes For Their Preparation, Pharmaceutical Compositions And Methods For Their Use App 20080293780 - SCHOENAFINGER; Karl ;   et al. | 2008-11-27 |
Cyclic N-[1,3,4]-thiadiazol-2-yl-benzene Sulfonamides, Pharmaceutical Compositions And Methods For The Therapeutic Use Thereof App 20080280959 - SCHOENAFINGER; Karl ;   et al. | 2008-11-13 |
Substituted benzoylureido-o-benzoylamides, process for their preparation and their use Grant 7,378,440 - Kadereit , et al. May 27, 2 | 2008-05-27 |
Amide-substituted 8 N Benzimidazoles, Method For The Production Thereof, And Use Of The Same As Medicaments App 20080090868 - DEFOSSA; Elisabeth ;   et al. | 2008-04-17 |
Substituted, Bicyclic 8-pyrrolidinobenzimidazoles, Methods For Their Production And Their Use As Medicaments App 20080090890 - DEFOSSA; Elisabeth ;   et al. | 2008-04-17 |
Amino-substituted 8-n-benzimidazoles And Methods For Their Use In Blood Sugar Disorders App 20080090870 - DEFOSSA; Elisabeth ;   et al. | 2008-04-17 |
Substituted 2-aminoalkylthiobenzimidazole Compounds, Pharmaceutical Compositions Thereof And Methods For Their Use App 20080090889 - DEFOSSA; Elisabeth ;   et al. | 2008-04-17 |
Aminocarbonyl-substituted 8-n-benzimidazoles, Methods For Their Preparation And Their Use In Pharmaceutical Compositions App 20080090869 - DEFOSSA; Elisabeth ;   et al. | 2008-04-17 |
Sulfonylamino carboxylic acid N-arylamides as guanylate cyclase activators Grant 7,351,703 - Schindler , et al. April 1, 2 | 2008-04-01 |
Substituted N-aminomethylene Sulfonamides, Production And Use Thereof As Medicaments App 20080069851 - SCHOENAFINGER; Karl ;   et al. | 2008-03-20 |
Urea-and Urethane-substituted Acylureas, Process For Their Preparation And Their Use App 20080033042 - Defossa; Elisabeth ;   et al. | 2008-02-07 |
Substituted 8-aminoalkoxy-xanthine Compounds And Compositions Useful In The Treatment Of Hyperlipidemia And Diabetes App 20070299090 - Schoenafinger; Karl ;   et al. | 2007-12-27 |
Substituted 8-aminoalkylthioxanthines, And Their Use As Inhibitors Of Dipeptidyl Peptidase Iv App 20070265284 - Schoenafinger; Karl ;   et al. | 2007-11-15 |
Novel Pyridazinone Derivatives App 20070259870 - HOELDER; Swen ;   et al. | 2007-11-08 |
Urea- and urethane-substituted acylureas, process for their preparation and their use Grant 7,262,220 - Defossa , et al. August 28, 2 | 2007-08-28 |
Substituted, Bicyclic 8-pyrrolidinoxanthines, And Methods For Their Use As Inhibitors Of Dipeptidyl Peptidase App 20070197563 - SCHOENAFINGER; Karl ;   et al. | 2007-08-23 |
Novel 4-benzimidazol-2-ylpyridazin-3-one derivatives App 20070173503 - Hoelder; Swen ;   et al. | 2007-07-26 |
Substituted Bicyclic 8-pyrr0lidinoxanthines, Methods For Their Production, Pharmaceutical Formulations And Their Use App 20070167468 - SCHOENAFINGER; Karl ;   et al. | 2007-07-19 |
Acyl-4-carboxyphenylurea derivatives, processes for preparing them and their use Grant 7,223,796 - Defossa , et al. May 29, 2 | 2007-05-29 |
Pyridazinone Derivatives, Methods For Their Production And Their Use As Pharmaceuticals App 20070088041 - Hoelder; Swen ;   et al. | 2007-04-19 |
Carboxyalkoxy-substituted Acyl-carboxyphenylurea Derivatives And Their Use As Medicaments App 20070088083 - DeFossa; Elisabeth ;   et al. | 2007-04-19 |
4-benzimidazol-2-yl-pyridazine-3-one-derivatives, Production And Use Thereof In Medicaments App 20070072866 - SCHOENAFINGER; Karl ;   et al. | 2007-03-29 |
Substituted 3-(benzoylureido) thiophene derivatives, processes for preparing them and their use Grant 7,196,114 - Schoenafinger , et al. March 27, 2 | 2007-03-27 |
Carbonylamino-substituted acyl phenyl urea derivatives, process for their preparation and their use Grant 7,179,941 - Defossa , et al. February 20, 2 | 2007-02-20 |
Heterocyclically Substituted Benzoylureas, Process For Their Preparation and Their Use as Pharmaceuticals App 20070021474 - Schoenafinger; Karl ;   et al. | 2007-01-25 |
Substituted 4-amino-2-arylcyclopenta[d]pyrimidines, their preparation, their use and pharmaceutical preparations comprising them Grant 7,138,398 - Schindler , et al. November 21, 2 | 2006-11-21 |
Heterocyclically substituted benzoylureas, process for their preparation and their use as pharmaceuticals Grant 7,138,414 - Schoenafinger , et al. November 21, 2 | 2006-11-21 |
Cyanopyrrolidides, process for their preparation and their use as medicaments Grant 7,094,800 - Schoenafinger , et al. August 22, 2 | 2006-08-22 |
Acyl-3-carboxyphenylurea derivatives, processes for preparing them and their use Grant 7,078,404 - Defossa , et al. July 18, 2 | 2006-07-18 |
N-benzoylureidocinnamic acid derivatives, processes for preparing them and their use Grant 7,049,341 - Schoenafinger , et al. May 23, 2 | 2006-05-23 |
Bicyclic cyanoheterocycles, process for their preparation and their use as medicaments Grant 7,008,957 - Wagner , et al. March 7, 2 | 2006-03-07 |
Substituted 3-phenyl-5-alkoxy-3H-(1,3,4)-oxadiazol-2-ones, pharmaceutical composition and method for treating obesity thereof Grant 6,900,233 - Schoenafinger , et al. May 31, 2 | 2005-05-31 |
Sulfonylaminocarboxiylic acid N-arylamides as guanylate cyclase activators App 20050080073 - Schindler, Ursula ;   et al. | 2005-04-14 |
Substituted benzoylureido-o-benzoylamides, process for their preparation and their use App 20050065142 - Kadereit, Dieter ;   et al. | 2005-03-24 |
Novel bicyclic cyanoheterocycles, process for their preparation and their use as medicaments App 20050059716 - Wagner, Holger ;   et al. | 2005-03-17 |
Novel cyanopyrrolidides, process for their preparation and their use as medicaments App 20050059724 - Schoenafinger, Karl ;   et al. | 2005-03-17 |
Carbonylamino-substituted acyl phenyl urea derivatives, process for their preparation and their use App 20050014822 - Defossa, Elisabeth ;   et al. | 2005-01-20 |
Substituted 4-amino-2aryl-pyrimidines, their production and use and pharmaceutical preparations containing same Grant 6,844,347 - Schnidler , et al. January 18, 2 | 2005-01-18 |
Substituted benzoylureidopyridylpiperidine-and-pyrrolidinecarboxylic acid derivatives, processes for preparing them and their use App 20040266768 - Schoenafinger, Karl ;   et al. | 2004-12-30 |
Sulfonylaminocarboxylic acid N-arylamides as guanylate cyclase activators Grant 6,809,089 - Schindler , et al. October 26, 2 | 2004-10-26 |
Substituted 3-(benzoylureido) thiophene derivatives, processes for preparing them and their use App 20040198742 - Schoenafinger, Karl ;   et al. | 2004-10-07 |
Carboxyalkoxy-substituted acyl-carboxyphenylurea derivatives and their use as medicaments App 20040157922 - Defossa, Elisabeth ;   et al. | 2004-08-12 |
Heterocyclically substituted benzoylureas, process for their preparation and their use as pharmaceuticals App 20040152743 - Schoenafinger, Karl ;   et al. | 2004-08-05 |
N-benzoylureidocinnamic acid derivatives, processes for preparing them and their use App 20040102518 - Schoenafinger, Karl ;   et al. | 2004-05-27 |
Urea- and urethane-substituted acylureas, process for their preparation and their use App 20040087659 - Defossa, Elisabeth ;   et al. | 2004-05-06 |
Acyl-4-carboxyphenylurea derivatives, processes for preparing them and their use App 20040077716 - Defossa, Elisabeth ;   et al. | 2004-04-22 |
Substituted 4-amino-2-arylcyclopenta[d]pyrimidines, their preparation, their use and pharmaceutical preparations comprising them App 20040048850 - Schindler, Ursula ;   et al. | 2004-03-11 |
Use of substituted 3-phenyl-5-alkoxy-3H-(1,3,4)-oxadizol-2-ones for inhibiting pancreatic lipase App 20030236288 - Schoenafinger, Karl ;   et al. | 2003-12-25 |
Acyl-3-carboxyphenylurea derivatives, processes for preparing them and their use App 20030216370 - Defossa, Elisabeth ;   et al. | 2003-11-20 |
Substituted 4-amino-2-aryl-cyclopenta[d]pyrimidines, their production and use and pharmaceutical preparations containing same Grant 6,627,628 - Schindler , et al. September 30, 2 | 2003-09-30 |
Substituted 3-phenyl-5-alkoxy-3H- (1,3,4)-oxadiazol-2-ones, pharmaceutical composition and method for treating obesity thereof App 20030181433 - Schoenafinger, Karl ;   et al. | 2003-09-25 |
Sulfonylaminocarboxylic acid N-arylamides as guanylate cyclase activators App 20030171352 - Schindler, Ursula ;   et al. | 2003-09-11 |
Substituted 3-phenyl-5-alkoxy-1,3,4-oxadiazol-2-ones, their preparation and their use in medicaments Grant 6,596,742 - Petry , et al. July 22, 2 | 2003-07-22 |
Sulfonylamino carboxylic acid N-arylamides as guanylate cyclase activators Grant 6,548,547 - Schindler , et al. April 15, 2 | 2003-04-15 |
Substituted isoindolones and their use as cyclic GMP modulators in medicaments Grant 6,344,468 - Schindler , et al. February 5, 2 | 2002-02-05 |
Substituted 3-phenyl-5-alkoxy-1,3,4-oxadiazol-2-ones, their preparation and their use as pharmaceuticals App 20010031772 - Schoenafinger, Karl ;   et al. | 2001-10-18 |