Patent | Date |
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(R)-chiral halogenated substituted fused heterocyclic amino compounds useful for inhibiting cholesterol ester transfer protein activity Grant 7,700,658 - Sikorsky , et al. April 20, 2 | 2010-04-20 |
Pyridinone Pyrazole Urea and Pyrimidinone Pyrazole Urea Derivatives App 20090270350 - Devadas; Balekudru ;   et al. | 2009-10-29 |
(r)-chiral Halogenated Substituted Fused Heterocyclic Amino Compounds Useful For Inhibiting Cholesterol Ester Transfer Protein Activity App 20090156685 - Sikorski; James A. ;   et al. | 2009-06-18 |
(R)-Chiral Halogenated Substituted Fused Heterocyclic Amino Compounds Useful for Inhibiting Cholesterol Ester Transfer Protein Activity App 20070219274 - Sikorski; James A. ;   et al. | 2007-09-20 |
(R)-chiral halogenated substituted fused heterocyclic amino compounds useful for inhibiting cholesterol ester transfer protein activity Grant 7,253,211 - Sikorski , et al. August 7, 2 | 2007-08-07 |
(R)-chiral halogenated substituted fused heterocyclic amino compounds useful for inhibiting cholesterol ester transfer protein activity Grant 7,122,536 - Sikorski , et al. October 17, 2 | 2006-10-17 |
(R)-chiral halogenated substituted fused heterocyclic amino compounds useful for inhibiting cholesterol ester transfer protein activity App 20060229304 - Sikorski; James A. ;   et al. | 2006-10-12 |
Piperidinyl- and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors Grant 7,119,203 - Barta , et al. October 10, 2 | 2006-10-10 |
Aromatic sulfone hydroxamic acids and their use as protease inhibitors App 20050101641 - Freskos, John N. ;   et al. | 2005-05-12 |
Aromatic sulfone hydroxamic acids and their use as protease inhibitors Grant 6,890,928 - Freskos , et al. May 10, 2 | 2005-05-10 |
(R)-chiral halogenated substituted fused heterocyclic amino compounds useful for inhibiting cholesterol ester transfer protein activity App 20050043294 - Sikorski, James A. ;   et al. | 2005-02-24 |
Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors App 20050009838 - Barta, Thomas E. ;   et al. | 2005-01-13 |
(R)-Chiral halogenated substituted n,n-bis-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,803,388 - Sikorski , et al. October 12, 2 | 2004-10-12 |
Substituted biphenyl compounds for the treatment of inflammation App 20040158074 - Reitz, David B. ;   et al. | 2004-08-12 |
Use of substituted N, N-disubstituted reverse aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,765,023 - Sikorski , et al. July 20, 2 | 2004-07-20 |
Aromatic sulfone hydroxamic acids and their use as protease inhibitors App 20040110805 - Freskos, John N. ;   et al. | 2004-06-10 |
Substituted n-benzyl-n-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,723,753 - Sikorski , et al. April 20, 2 | 2004-04-20 |
(R)-chiral halogenated substituted n-benzyl-n-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,723,752 - Sikorski , et al. April 20, 2 | 2004-04-20 |
Substituted N-fused-phenyl-N-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,710,089 - Sikorski , et al. March 23, 2 | 2004-03-23 |
(R)-chiral halogenated 1-substitutedamino-(n+1)-alkanols useful for inhibiting cholesteryl ester transfer protein activity App 20040044048 - Sikorski, James A. ;   et al. | 2004-03-04 |
Substituted N,N-disubstituted non-fused heterocyclo amino compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,699,898 - Sikorski , et al. March 2, 2 | 2004-03-02 |
Substituted N,N-disubstituted fused-heterocyclo amino compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,696,435 - Sikorski , et al. February 24, 2 | 2004-02-24 |
Substituted N-phenoxy-N-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,696,472 - Sikorski , et al. February 24, 2 | 2004-02-24 |
Aromatic sulfone hydroxamates and their use as protease inhibitors Grant 6,689,794 - Freskos , et al. February 10, 2 | 2004-02-10 |
Aromatic sulfone hydroxamates and their use as protease inhibitors App 20040024024 - Freskos, John N. ;   et al. | 2004-02-05 |
(R)-chiral halogenated substituted N,N-Bis-benzyl aminioalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,683,113 - Sikorski , et al. January 27, 2 | 2004-01-27 |
Substituted N,N-disubstituted cycloalkyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,683,099 - Sikorski , et al. January 27, 2 | 2004-01-27 |
Aromatic sulfone hydroxamates and their use as protease inhibitors App 20040010019 - Freskos, John N. ;   et al. | 2004-01-15 |
Substituted biphenyl compounds for the treatment of inflammation Grant 6,677,488 - Reitz , et al. January 13, 2 | 2004-01-13 |
(R)-Chiral halogenated substituted heteroaryl benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,677,341 - Sikorski , et al. January 13, 2 | 2004-01-13 |
Substituted N, N-disubstituted mercapto amino compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,677,380 - Sikorski , et al. January 13, 2 | 2004-01-13 |
Substituted N-phenyl-N-heteroaralkyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,677,353 - Sikorski , et al. January 13, 2 | 2004-01-13 |
Substituted N,N-bis-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,677,375 - Sikorski , et al. January 13, 2 | 2004-01-13 |
Substituted N,N-bis-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,677,382 - Sikorski , et al. January 13, 2 | 2004-01-13 |
Substituted N,N-disubstituted diamino compounds useful for inhibiting cholesteryl ester transfer protein activity Grant 6,677,379 - Sikorski , et al. January 13, 2 | 2004-01-13 |
Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity App 20030125328 - Sikorski, James A. ;   et al. | 2003-07-03 |
Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity App 20030125329 - Sikorski, James A. ;   et al. | 2003-07-03 |
Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity App 20030119833 - Sikorski, James A. ;   et al. | 2003-06-26 |
Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity App 20030114454 - Sikorski, James A. ;   et al. | 2003-06-19 |
Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity App 20030109528 - Sikorski, James A. ;   et al. | 2003-06-12 |
Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity App 20030105100 - Sikorski, James A. ;   et al. | 2003-06-05 |
Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity App 20030100559 - Sikorski, James A. ;   et al. | 2003-05-29 |
Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity App 20030096818 - Sikorski, James A. ;   et al. | 2003-05-22 |
Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity App 20030087905 - Sikorski, James A. ;   et al. | 2003-05-08 |
Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity App 20030083331 - Sikorski, James A. ;   et al. | 2003-05-01 |
(R)-chiral halogenated substituted N,N-bis-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity App 20030078264 - Sikorski, James A. ;   et al. | 2003-04-24 |
(R)-chiral halogenated substituted n,n-bis-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity App 20030050317 - Sikorski, James A. ;   et al. | 2003-03-13 |
(R)-Chiral halogenated substituted fused heterocyclic amino compounds useful for inhibiting cholesteryl ester transfer protein activity App 20030040545 - Sikorski, James A. ;   et al. | 2003-02-27 |
Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity App 20030032644 - Sikorski, James A. ;   et al. | 2003-02-13 |
(R)-Chiral halogenated substituted heteroaryl benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity App 20030027826 - Sikorski, James A. ;   et al. | 2003-02-06 |
Substituted n-phenyl-n-fused-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity App 20020183397 - Sikorski, James A. ;   et al. | 2002-12-05 |
(R)-chiral halogenated substituted N-benzyl-N-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity App 20020177708 - Sikorski, James A. ;   et al. | 2002-11-28 |
Substituted N-heteroaryl-N-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity App 20020165231 - Sikorski, James A. ;   et al. | 2002-11-07 |
Substituted N, N-disubstituted cycloalkyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity App 20020165232 - Sikorski, James A. ;   et al. | 2002-11-07 |
Use of substituted N, N-bis-benzyl aminoalcohol compounds inhibiting cholesteryl ester transfer protein activity Grant 6,476,075 - Sikorski , et al. November 5, 2 | 2002-11-05 |
Substituted N-phenyl-N-heteroaralkyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity Grant 6,458,803 - Sikorski , et al. October 1, 2 | 2002-10-01 |
Substituted N, N-disubstituted diamino compounds useful for inhibiting cholesteryl ester transfer protein activity App 20020120011 - Sikorski, James A. ;   et al. | 2002-08-29 |
Substituted terphenyl compounds for the treatment of inflammation Grant 5,739,166 - Reitz , et al. April 14, 1 | 1998-04-14 |