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Bicyclic heterocycle derivatives and methods of use thereof Grant 8,815,876 - Neelamkavil , et al. August 26, 2 | 2014-08-26 |
Pyrimidine derivatives as GPCR modulators for use in the treatment of obesity and diabetes Grant 8,722,882 - Neustadt , et al. May 13, 2 | 2014-05-13 |
Adenosine A.sub.2a receptor antagonists Grant RE44,205 - Neustadt , et al. May 7, 2 | 2013-05-07 |
Substituted [1,2,4]triazolo[4,3-alpha]quinoxalines as adenosine A2a receptor antagonists Grant 8,435,994 - Harris , et al. May 7, 2 | 2013-05-07 |
Bicyclic Heterocycle Derivatives And Methods Of Use Thereof App 20130096141 - Neustadt; Bernard R. ;   et al. | 2013-04-18 |
Amino-quinoxaline and amino-quinoline compounds for use as adenosine A.sub.2a receptor antagonists Grant 8,415,353 - Harris , et al. April 9, 2 | 2013-04-09 |
Bicyclic heterocycle derivatives and methods of use thereof Grant 8,410,122 - Harris , et al. April 2, 2 | 2013-04-02 |
Pyrimidinone derivatives and methods of use thereof Grant 8,318,751 - Boyle , et al. November 27, 2 | 2012-11-27 |
FUSED TRICYCLIC COMPOUNDS WITH ADENOSINE A2a RECEPTOR ANTAGONIST ACTIVITY App 20120232086 - Harris; Joel M. ;   et al. | 2012-09-13 |
Fused Bicyclic Pyrimidine Derivatives And Methods Of Use Thereof App 20120232073 - Neelamkavil; Santhosh Francis ;   et al. | 2012-09-13 |
1,2,4-triazolo[4,3-c]pyrimidin-3-one and pyrazolo[4,3-e]-1,2,4-triazolo[4,3-c]pyrimidin-3-one compounds for use as adenosine A.sub.2a receptor antagonists Grant 8,222,259 - Harris , et al. July 17, 2 | 2012-07-17 |
Bridged Bicyclic Heterocycle Derivatives And Methods Of Use Thereof App 20120040975 - Neelamkavil; Santhosh Francis ;   et al. | 2012-02-16 |
Piperazine derivatives useful as CCR5 antagonists Grant 8,114,879 - Baroudy , et al. February 14, 2 | 2012-02-14 |
Bicyclic Heterocycle Derivatives And Methods Of Use Thereof App 20110263624 - Harris; Joel M. ;   et al. | 2011-10-27 |
Pyrimidine Derivatives As Gpcr Modulators For Use In The Treatment Of Obesity And Diabetes App 20110263570 - Neustadt; Bernard R. ;   et al. | 2011-10-27 |
Bicyclic Heterocycle Derivatives And Methods Of Use Thereof App 20110166167 - Neelamkavil; Santhosh Francis ;   et al. | 2011-07-07 |
Bicyclic Heterocycle Derivatives And Use Thereof As Gpr119 Modulators App 20110166165 - Neelamkavil; Santhosh Francis ;   et al. | 2011-07-07 |
1,2,4-TRIAZOLO[4,3-c]PYRIMIDIN-3-ONE AND PYRAZOLO[4,3-e]-1,2,4-TRIAZOLO[4,3-c]PYRIMIDIN-3-ONE COMPOUNDS FOR USE AS ADENOSINE A2a RECEPTOR ANTAGONISTS App 20110152256 - Harris; Joel M. ;   et al. | 2011-06-23 |
Bicyclic Heterocycle Derivatives And Their Use As Gpcr Modulators App 20110118286 - Neelamkavil; Santhosh Francis ;   et al. | 2011-05-19 |
AMINO-QUINOXALINE AND AMINO-QUINOLINE COMPOUNDS FOR USE AS ADENOSINE A2a RECEPTOR ANTAGONISTS App 20110105513 - Harris; Joel M. ;   et al. | 2011-05-05 |
Bicyclic Heterocycle Derivatives And Use Thereof As Gpr119 Modulators App 20110065671 - Harris; Joel M. ;   et al. | 2011-03-17 |
p53 modulators Grant 7,790,474 - Dasmahapatra , et al. September 7, 2 | 2010-09-07 |
Pyrimidinone Derivatives And Methods Of Use Thereof App 20100190687 - Boyle; Craig D. ;   et al. | 2010-07-29 |
Pyrazolo [1,5-A]pyrimidine adenosine A.sub.2a receptor antagonists Grant 7,741,318 - Clasby , et al. June 22, 2 | 2010-06-22 |
Pyrimidinone Derivatives And Methods Of Use Thereof App 20100113487 - Boyle; Craig D ;   et al. | 2010-05-06 |
Tetrahydropyrido[4,3-d]pyrimidinone Derivatives And Methods Of Use Thereof App 20100113330 - Boyle; Craig D. ;   et al. | 2010-05-06 |
Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A.sub.2a receptor antagonists Grant 7,709,492 - Neustadt , et al. May 4, 2 | 2010-05-04 |
2-heteroaryl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists Grant 7,465,740 - Neustadt , et al. December 16, 2 | 2008-12-16 |
Piperidine Derivatives Useful As Ccr5 Antagonists App 20080188485 - Baroudy; Bahige M. ;   et al. | 2008-08-07 |
Piperazine derivatives useful as CCR5 antagonists Grant 7,384,944 - Baroudy , et al. June 10, 2 | 2008-06-10 |
2-alkynyl- and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A.sub.2a receptor antagonists Grant 7,368,449 - Neustadt , et al. May 6, 2 | 2008-05-06 |
Azetidinone Derivatives and Methods of Use Thereof App 20080076750 - Aslanian; Robert G. ;   et al. | 2008-03-27 |
Treating Pain, Diabetes, And Disorders Of Lipid Metabolism App 20080070892 - Harris; Joel M. ;   et al. | 2008-03-20 |
2-Heteroaryl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists App 20070066620 - Neustadt; Bernard R. ;   et al. | 2007-03-22 |
Quinazoline derivatives useful in cancer treatment App 20070032502 - Mallams; Alan K. ;   et al. | 2007-02-08 |
Quinazoline derivatives useful in cancer treatment App 20070015774 - Mallams; Alan K. ;   et al. | 2007-01-18 |
[1,2,4]-Triazole bicyclic adenosine A2a receptor antagonists Grant 7,078,408 - Neustadt , et al. July 18, 2 | 2006-07-18 |
Adenosine A2a receptor antagonists Grant 7,067,655 - Neustadt , et al. June 27, 2 | 2006-06-27 |
Pyrazolo [1,5-A] pyrimidine adenosine A2a receptor antagonists App 20060135526 - Clasby; Martin C. ;   et al. | 2006-06-22 |
Adenosine A2a receptor antagonists Grant 7,041,666 - Matasi , et al. May 9, 2 | 2006-05-09 |
Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists App 20050239795 - Neustadt, Bernard R. ;   et al. | 2005-10-27 |
2-alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists App 20050222164 - Neustadt, Bernard R. ;   et al. | 2005-10-06 |
[1,2,4]-Triazole bicyclic adenosine A2a receptor antagonists App 20050113380 - Neustadt, Bernard R. ;   et al. | 2005-05-26 |
Adenosine A2a receptor antagonists Grant 6,897,216 - Neustadt , et al. May 24, 2 | 2005-05-24 |
2-Alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists Grant 6,897,217 - Neustadt , et al. May 24, 2 | 2005-05-24 |
[1,2,4]-Triazole bicyclic adeonsine A2a receptor antagonists Grant 6,875,772 - Neustadt , et al. April 5, 2 | 2005-04-05 |
Adenosine A2a receptor antagonists App 20050026932 - Neustadt, Bernard R. ;   et al. | 2005-02-03 |
2-Alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists App 20040220194 - Neustadt, Bernard R. ;   et al. | 2004-11-04 |
Piperazine derivatives useful as CCR5 antagonists App 20040067961 - Baroudy, Bahige M. ;   et al. | 2004-04-08 |
Piperazine derivatives useful as CCR5 antagonists Grant 6,689,765 - Baroudy , et al. February 10, 2 | 2004-02-10 |
Adenosine A2a receptor antagonists App 20040023997 - Neustadt, Bernard R. ;   et al. | 2004-02-05 |
Adenosine A2a receptor antagonists App 20030212080 - Matasi, Julius J. ;   et al. | 2003-11-13 |
[1,2,4]-Triazole bicyclic adenosine A2a receptor antagonists App 20030191130 - Neustadt, Bernard R. ;   et al. | 2003-10-09 |
Adenosine A2a receptor antagonists Grant 6,630,475 - Neustadt , et al. October 7, 2 | 2003-10-07 |
Piperidine derivatives useful as CCR5 antagonists Grant 6,602,885 - Baroudy , et al. August 5, 2 | 2003-08-05 |
Piperazine derivatives useful as CCR5 antagonists App 20030069252 - Baroudy, Bahige M. ;   et al. | 2003-04-10 |
Piperidine derivatives useful as CCR5 antagonists App 20030004185 - Baroudy, Bahige M. ;   et al. | 2003-01-02 |
Adenosine A2a receptor antagonists App 20020099061 - Neustadt, Bernard R. ;   et al. | 2002-07-25 |
Piperazine derivatives useful as CCR5 antagonists Grant 6,391,865 - Baroudy , et al. May 21, 2 | 2002-05-21 |
Piperidine derivatives useful as CCR5 antagonists Grant 6,387,930 - Baroudy , et al. May 14, 2 | 2002-05-14 |
Neuropeptide Y5 receptor antagonists Grant 6,329,395 - Dugar , et al. December 11, 2 | 2001-12-11 |
Derivatives of aminobenzoic and aminobiphenylcarboxylic acids useful as anti-cancer agents Grant 6,228,985 - Blood , et al. May 8, 2 | 2001-05-08 |
Polycyclic guanine derivatives Grant 5,393,755 - Neustadt , et al. February 28, 1 | 1995-02-28 |
N-(mercaptoalkyl)ureas and carbamates Grant 5,356,925 - Neustadt , et al. October 18, 1 | 1994-10-18 |
N-(acylaminomethyl)glutaryl amino acids and use Grant 5,208,236 - Neustadt May 4, 1 | 1993-05-04 |
Mercaptoacyl aminolactam endopeptidase inhibitors Grant 5,075,302 - Neustadt December 24, 1 | 1991-12-24 |
Carboxyalkyl dipeptides as antiglaucoma agents Grant 5,017,567 - Neustadt , et al. May 21, 1 | 1991-05-21 |
Mercapto-acylamino acid antihypertensives Grant 4,929,641 - Haslanger , et al. May 29, 1 | 1990-05-29 |
Mercapto-acylamino acids as antihypertensives Grant 4,879,309 - Doll , et al. November 7, 1 | 1989-11-07 |
Preparation of angiotensin-converting enzyme inhibitors Grant 4,831,157 - Gold , et al. May 16, 1 | 1989-05-16 |
Carboxyalkyl dipeptides and medical use thereof in treating hypertension and congestive heart failure Grant 4,818,749 - Gold , et al. April 4, 1 | 1989-04-04 |
Carboxyalkyl dipeptides and anti-hypertensive use thereof Grant 4,808,573 - Gold , et al. February 28, 1 | 1989-02-28 |
Mercapto-acylamino acid antihypertensives Grant 4,801,609 - Haslanger , et al. January 31, 1 | 1989-01-31 |
Antiglaucoma compositions and methods Grant 4,783,444 - Watkins , et al. November 8, 1 | 1988-11-08 |
Angiotensin-converting enzyme inhibitors Grant 4,587,258 - Gold , et al. May 6, 1 | 1986-05-06 |
Antihypertensive agents Grant 4,559,340 - Neustadt , et al. December 17, 1 | 1985-12-17 |
Arylmethoxy-, arylmethylthio-, heteroarylmethoxy-, and heteroarylmethylthio-alkylaminoalcohols Grant 4,379,166 - Neustadt , et al. April 5, 1 | 1983-04-05 |
Anti-hypertensive 5-[2-(substituted anilinoalkylamino)-1-hydroxyalkyl]salicylamides Grant 4,163,053 - Neustadt , et al. July 31, 1 | 1979-07-31 |
Anti-hypertensive polyhaloisopropyl-substituted arylureas Grant 4,093,742 - Neustadt June 6, 1 | 1978-06-06 |