Patent | Date |
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Hpk1 Inhibitors App 20220177458 - MEVELLEC; Laurence Anne ;   et al. | 2022-06-09 |
Bicyclic Hpk1 Inhibitors App 20220169644 - MEVELLEC; Laurence Anne ;   et al. | 2022-06-02 |
Pyrazolyl Quinoxaline Kinase Inhibitors App 20220135544 - SAXTY; Gordon ;   et al. | 2022-05-05 |
Bicyclic pyridine, pyrazine, and pyrimidine derivatives as PI3K beta inhibitors Grant 10,894,793 - Berthelot , et al. January 19, 2 | 2021-01-19 |
Pyrazolyl Quinoxaline Kinase Inhibitors App 20200131153 - SAXTY; Gordon ;   et al. | 2020-04-30 |
Pyrazolyl quinoxaline kinase inhibitors Grant 10,519,137 - Saxty , et al. Dec | 2019-12-31 |
Azabenzimidazole Derivatives As Pi3k Beta Inhibitors App 20190263804 - Pilatte; Isabelle Noelle Constance ;   et al. | 2019-08-29 |
Substituted 4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyrimidine derivatives and 2,3-dihydro-1H-imidazo[1,2-b]pyrazole derivatives as ROS1 inhibitors Grant 10,342,795 - Mevellec , et al. July 9, 2 | 2019-07-09 |
Bicyclic Pyridine, Pyrazine, And Pyrimidine Derivatives As Pi3k Beta Inhibitors App 20190169199 - Berthelot; Didier Jean-Claude ;   et al. | 2019-06-06 |
Substituted 4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyrazine derivatives and 5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepine derivatives as Ros1 inhibitors Grant 10,280,170 - Mevellec , et al. | 2019-05-07 |
Heterocyclyl linked imidazopyridazine derivatives as PI3KB inhibitors Grant 10,202,387 - Mevellec , et al. Feb | 2019-02-12 |
Imidazopyridazine derivatives as PI3KB inhibitors Grant 10,087,187 - Mevellec , et al. October 2, 2 | 2018-10-02 |
Pyrazolyl Quinoxaline Kinase Inhibitors App 20180127397 - SAXTY; Gordon ;   et al. | 2018-05-10 |
Heterocyclyl Linked Imidazopyridazine Derivatives As Pi3kb Inhibitors App 20180057496 - Mevellec; Laurence Anne ;   et al. | 2018-03-01 |
Imidazopyridazine Derivatives As Pi3kb Inhibitors App 20180002336 - Mevellec; Laurence Anne ;   et al. | 2018-01-04 |
Pyrazolyl quinoxaline kinase inhibitors Grant 9,850,228 - Saxty , et al. December 26, 2 | 2017-12-26 |
SUBSTITUTED 4,5,6,7-TETRAHYDRO-PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND 2,3-DIHYDRO-1H-IMIDAZO[1,2-b]PYRAZOLE DERIVATIVES AS ROS1 INHIBITORS App 20170173014 - Mevellec; Laurence Anne ;   et al. | 2017-06-22 |
SUBSTITUTED 4,5,6,7-TETRAHYDRO-PYRAZOLO[1,5-a]PYRAZINE DERIVATIVES AND 5,6,7,8-TETRAHYDRO-4H-PYRAZOLO[1,5-a][1,4]DIAZEPINE DERIVATIVES AS ROS1 INHIBITORS App 20170174690 - Mevellec; Laurence Anne ;   et al. | 2017-06-22 |
Pyrazolyl Quinoxaline Kinase Inhibitors App 20160311800 - SAXTY; Gordon ;   et al. | 2016-10-27 |
Pyrazolyl quinoxaline kinase inhibitors Grant 9,464,071 - Saxty , et al. October 11, 2 | 2016-10-11 |
Tetrahydrophenanthridinones And Tetrahydrocyclopentaquinolinones As Parp And Tubulin Polymerization Inhibitors App 20150353526 - Angibaud; Patrick Rene ;   et al. | 2015-12-10 |
Tetrahydrophenanthridinones and tetrahydrocyclopentaquinolinones as parp and tubulin polymerization inhibitors Grant 9,150,540 - Angibaud , et al. October 6, 2 | 2015-10-06 |
Pyrazolyl Quinoxaline Kinase Inhibitors App 20150105368 - SAXTY; Gordon ;   et al. | 2015-04-16 |
Phthalazine Derivatives As Parp Inhibitors App 20150072972 - Mevellec; Laurence Anne ;   et al. | 2015-03-12 |
Tetrahydrophenanthridinones And Tetrahydrocyclopentaquinolinones As Parp And Tubulin Polymerization Inhibitors App 20150038521 - Angibaud; Patrick Rene ;   et al. | 2015-02-05 |
Phthalazine derivatives as PARP inhibitors Grant 8,946,221 - Mevellec , et al. February 3, 2 | 2015-02-03 |
Pyrazolyl quinoxaline kinase inhibitors Grant 8,895,601 - Saxty , et al. November 25, 2 | 2014-11-25 |
Tetrahydrophenanthridinones and tetrahydrocyclopentaquinolinones as PARP and tubulin polymerization inhibitors Grant 8,889,866 - Angibaud , et al. November 18, 2 | 2014-11-18 |
Quinolinone derivatives as PARP and tank inhibitors Grant 8,778,966 - Vialard , et al. July 15, 2 | 2014-07-15 |
MTKI quinazoline derivatives Grant 8,492,377 - Papanikos , et al. July 23, 2 | 2013-07-23 |
Quinolinone derivatives as PARP inhibitors Grant 8,404,713 - Angibaud , et al. March 26, 2 | 2013-03-26 |
Pyrazolyl Quinazoline Kinase Inhibitors App 20130072457 - Saxty; Gordon ;   et al. | 2013-03-21 |
Quinolinone Derivatives As Parp And Tank Inhibitors App 20130018017 - VIALARD; Jorge Eduardo ;   et al. | 2013-01-17 |
Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT.sub.4-antagonists Grant 8,334,304 - Bosmans , et al. December 18, 2 | 2012-12-18 |
Quinolinone derivatives as PARP and TANK inhibitors Grant 8,299,256 - Vialard , et al. October 30, 2 | 2012-10-30 |
Quinazolinone derivatives as tubulin polymerization inhibitors Grant 8,168,644 - Freyne , et al. May 1, 2 | 2012-05-01 |
Tetrahydrophenanthridinones And Tetrahydrocyclopentaquinolinones As Parp And Tubulin Polymerization Inhibitors App 20110263622 - Angibaud; Patrick Rene ;   et al. | 2011-10-27 |
Phthalazine Derivatives As Parp Inhibitors App 20110065684 - Mevellec; Laurence Anne ;   et al. | 2011-03-17 |
Quinazolinone Derivatives As Tubulin Polymerization Inhibitors App 20110028433 - Freyne; Eddy Jean Edgard ;   et al. | 2011-02-03 |
Phthalazine derivatives as parp inhibitors Grant 7,803,795 - Mevellec , et al. September 28, 2 | 2010-09-28 |
Quinolinone Derivatives As Parp Inhibitors App 20100222348 - Angibaud; Patrick Rene ;   et al. | 2010-09-02 |
Quinolinone Derivatives As Parp And Tank Inhibitors App 20100168065 - Vialard; Jorge Eduardo ;   et al. | 2010-07-01 |
Heterocyclic substituted 4-(aminomethyl)-piperidine benzamides as 5HT.sub.4-antagonists Grant 7,732,464 - Bosmans , et al. June 8, 2 | 2010-06-08 |
Aminosulfonyl Substituted 4-(Aminomethyl)-Piperidine Benzamides As 5HT 4-Antagonists App 20100087483 - BOSMANS; Jean-Paul Rene Marie Andre ;   et al. | 2010-04-08 |
Mtki Quinazoline Derivatives App 20100029627 - Papanikos; Alexandra ;   et al. | 2010-02-04 |
Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT.sub.4-antagonists Grant 7,652,040 - Bosmans , et al. January 26, 2 | 2010-01-26 |
4-(aminomethyl)-piperidine benzamides as 5HT.sub.4-antagonists Grant 7,638,535 - Bosmans , et al. December 29, 2 | 2009-12-29 |
5HT.sub.4-antagonistic 4-(aminomethyl)-piperidine benzamides Grant 7,635,706 - Bosmans , et al. December 22, 2 | 2009-12-22 |
Hydroxycarbonylphenyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT.sub.4 antagonists Grant 7,498,347 - Bosmans , et al. March 3, 2 | 2009-03-03 |
Phthalazine Derivatives as Parp Inhibitors App 20080139568 - Mevellec; Laurence Anne ;   et al. | 2008-06-12 |
Heterocyclic substituted 4-(aminomethyl)-piperidine benzamides as 5ht4-antagonists App 20070197600 - Bosmans; Jean-Paul Rene Marie Andre ;   et al. | 2007-08-23 |
Farnesyl transferase inhibiting 6-heterocyclylmethyl quinoline and quinazoline derivatives Grant 7,196,094 - Angibaud , et al. March 27, 2 | 2007-03-27 |
5Ht4-antagonistic 4-(aminomethyl)-piperidine benzamides App 20070032486 - Bosmans; Jean-Paul Rene Marie Andre ;   et al. | 2007-02-08 |
Farnesyl transferase inhibiting 6-[(substituted phenyl)methyl]-quinoline and quinazoline derinazoline derivatives Grant 7,173,040 - Angibaud , et al. February 6, 2 | 2007-02-06 |
4-(Aminomethyl)-piperidine benzamides as 5ht4 - antagonists App 20060281753 - Bosmans; Jean-Paul Rene Marie Andre ;   et al. | 2006-12-14 |
Hydroxycarbonylphenyl substituted 4-(aminomethyl)-piperidine benzamides as 5ht4 antagonists App 20060142340 - Bosmans; Jean-Paul Rene Marie Andre ;   et al. | 2006-06-29 |
Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5ht 4-antagonists App 20060142339 - Bosmans; Jean-Paul Rene Marie Andre ;   et al. | 2006-06-29 |
Farnesyl transferase inhibiting 6-heterocyclylmethyl quinolinone derivatives Grant 7,067,531 - Angibaud , et al. June 27, 2 | 2006-06-27 |
Farnesyl transferase inhibiting 6-(substituted phenyl) Methy)-quinoline and quinazoline derinazoline derivaties App 20040048882 - Angibaud, Patrick Rene ;   et al. | 2004-03-11 |
Farnesyl transferase inhibiting 6-heterocyclylmethyl quinoline and quinazoline derivatives App 20030207887 - Angibaud, Patrick Rene ;   et al. | 2003-11-06 |
Farnesyl transferase inhibiting 6-heterocyclylmethyl quinolinone derivatives App 20030199547 - Angibaud, Patrick Rene ;   et al. | 2003-10-23 |