Patent | Date |
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Novel intermediates useful for the preparation of antihistaminic piperidine derivatives App 20020077482 - Krauss, Richard C. ;   et al. | 2002-06-20 |
Novel intermediates useful for the preparation of antihistaminic piperidine derivatives App 20010031895 - Krauss, Richard C. ;   et al. | 2001-10-18 |
2-substituted indane-2-mercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace Grant 5,529,996 - Warshawsky , et al. June 25, 1 | 1996-06-25 |
.alpha.-glucosidase inhibitors Grant 5,504,078 - Ducep , et al. April 2, 1 | 1996-04-02 |
Sulfonic stilbene derivatives in the treatment of viral disease Grant 5,494,932 - Cardin , et al. February 27, 1 | 1996-02-27 |
2-substituted indane-2-mercaptoacetylamide tricyclic derivatives useful as inhibitors of enkephalinase Grant 5,491,142 - Warshawsky , et al. February 13, 1 | 1996-02-13 |
2-substituted indane-2-mercaptoacetylamide tricyclic derivatives useful as inhibitors of enkephalinase Grant 5,491,141 - Warshawsky , et al. February 13, 1 | 1996-02-13 |
4-amino-17.beta.-(cyclopropyloxy)androst-4-en-3-one, 4-amino-17.beta.-(cyclopropylamino)androst-4-en-3-one and related compounds as C.sub.17-20 lyase and 5.alpha.-reductase Grant 5,486,511 - Weintraub , et al. January 23, 1 | 1996-01-23 |
2-substituted indane-2-mercaptoacetylamide derivatives useful as inhibitors or enkephalinase and ace Grant 5,486,513 - Warshawsky , et al. January 23, 1 | 1996-01-23 |
Tissue protective tocopherol analogs Grant 5,484,810 - Grisar , et al. January 16, 1 | 1996-01-16 |
Hypocholesterolemic, antiatherosclerotic and hypotriglyceridemic mercaptoacetylamide and benzazapine derivatives Grant 5,484,783 - Flynn , et al. January 16, 1 | 1996-01-16 |
NMDA antagonists Grant 5,470,870 - Palfreyman , et al. November 28, 1 | 1995-11-28 |
2-substituted indane-2-carboxyalkyl derivatives useful as inhibitors of enkephalinase and ACE Grant 5,457,196 - Warshawsky , et al. October 10, 1 | 1995-10-10 |
Carboxyalkyl tricyclic derivatives useful as inhibitors of enkephalinase and ace Grant 5,455,242 - Warshawsky , et al. October 3, 1 | 1995-10-03 |
5-aryl-3H-1,2,4-triazol-3-ones and their use in the treatment of neurodegenerative disorders Grant 5,436,252 - Sorensen , et al. July 25, 1 | 1995-07-25 |
Serotonin receptor agents Grant 5,436,246 - Bernotas , et al. | 1995-07-25 |
Mercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace Grant 5,430,145 - Flynn , et al. July 4, 1 | 1995-07-04 |
2-substituted indane-2-mercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace Grant 5,428,158 - Warshawsky , et al. June 27, 1 | 1995-06-27 |
Narrow poly- and mono-dispersed anionic oligomers, and their uses, formulations and process Grant 5,424,063 - Cardin , et al. | 1995-06-13 |
2-substituted indane-2-mercaptoacetylamide tricyclic derivatives useful as inhibitors of enkephalinase Grant 5,420,271 - Warshawsky , et al. May 30, 1 | 1995-05-30 |
Process for preparing 2,6-di-tertiarybutyl-4-mercaptophenol and 4,4'-isopropylidenedithio-bis-(2,6-di-tertiarybutylphenol) Grant 5,401,883 - Laskovics , et al. March 28, 1 | 1995-03-28 |
Anti-herpes castanospermine esters Grant 5,385,911 - Sunkara , et al. January 31, 1 | 1995-01-31 |
2'-halomethylidene cytidine, uridine and guanosine compounds and their pharmaceutical compositions Grant 5,378,693 - McCarthy , et al. January 3, 1 | 1995-01-03 |
Despiramine in the treatment of drug-resistant malarial infections Grant 5,373,005 - McCann , et al. December 13, 1 | 1994-12-13 |
Mercaptoacetylamido pyridazo [1,2]pyridazine, pyrazolo[1,2]pyridazine pyrazolo[1,2]pyridazine, pyridazol[1,2-a][1,2]diazepine and pyrazolol[1,2-a][1,2]diazepine Grant 5,366,973 - Flynn , et al. November 22, 1 | 1994-11-22 |
5-aryl-4-alkyl-3H-1,2,4-triazole-3-thiones useful as memory enhancers Grant 5,331,002 - Miller July 19, 1 | 1994-07-19 |
Pharmaceutical lozenges Grant 5,322,694 - Sixsmith June 21, 1 | 1994-06-21 |
Controlled release formulation for pharmaceutical compounds Grant 5,320,853 - Noda , et al. June 14, 1 | 1994-06-14 |
Inhibitors of nitric oxide biosynthesis Grant 5,318,992 - Whitten , et al. June 7, 1 | 1994-06-07 |
5'-amine substituted adenosine analogs as immunosuppressants Grant 5,308,837 - Bowlin May 3, 1 | 1994-05-03 |
Superior tasting composition having porous particles and the process of preparing such pharmaceutical composition Grant 5,302,396 - Phadke , et al. April 12, 1 | 1994-04-12 |
Cyclic nitrones, pharmaceutical compositions thereof and their use in treating shock Grant 5,292,746 - Carr , et al. March 8, 1 | 1994-03-08 |
Difluoroglutamic acid conjugates with folates and anti-folates for the treatment of neoplastic diseases Grant 5,286,726 - Bey , et al. February 15, 1 | 1994-02-15 |
Piperidinyl compounds Grant 5,286,866 - Carr , et al. February 15, 1 | 1994-02-15 |
bis[4-(2,6-di-alkyl)phenol]silane derivatives as antiatherosclerotic agents Grant 5,281,738 - Parker , et al. January 25, 1 | 1994-01-25 |
Selective adenosine receptor agents Grant 5,256,650 - Peet , et al. October 26, 1 | 1993-10-26 |
Inhibitors of lysyl oxidase Grant 5,252,608 - Palfreyman , et al. October 12, 1 | 1993-10-12 |
Cyclic anticoagulant peptides Grant 5,236,898 - Krstenansky , et al. August 17, 1 | 1993-08-17 |
Polyamine thiols as radioprotective agents Grant 5,217,964 - Edwards , et al. June 8, 1 | 1993-06-08 |
Alkoxyimino ether derivatives of 5-acyl-2(1H)-pyridinones Grant 5,212,315 - Jones , et al. May 18, 1 | 1993-05-18 |
8-substituted purines as selective adenosine receptor agents Grant 5,208,240 - Peet , et al. May 4, 1 | 1993-05-04 |
Inhibitors of lysyl oxidase Grant 5,182,297 - Palfreyman , et al. January 26, 1 | 1993-01-26 |
Treatment of multi-drug resistant tumors with pyridyloxazole-2-ones Grant 5,182,293 - Sunkara , et al. January 26, 1 | 1993-01-26 |
.alpha.-glucosidase inhibitors Grant 5,157,116 - Ducep , et al. October 20, 1 | 1992-10-20 |
2,6-di-alkyl-4-silyl-phenols as antiatheroscerotic agents Grant 5,155,250 - Parker , et al. October 13, 1 | 1992-10-13 |
Antidepressants Grant 5,149,714 - Freedman September 22, 1 | 1992-09-22 |
Cholesterol-lowering tocopherol analogs Grant 5,135,945 - Robinson , et al. August 4, 1 | 1992-08-04 |
(+)-.alpha.-(2,3-dimethoxyphenyl)-1-[ 2-(4-fluorophenyl)ethyl]-4-piperidinemethanol Grant 5,134,149 - Carr , et al. July 28, 1 | 1992-07-28 |
Inhibitors of lysyl oxidase Grant 5,120,764 - McCarthy , et al. June 9, 1 | 1992-06-09 |
Analog of peptidase substrates Grant 5,114,927 - Schirlin May 19, 1 | 1992-05-19 |
Allenyl amines Grant 5,112,852 - McCarthy , et al. May 12, 1 | 1992-05-12 |
Polyamine derivatives as antineoplastic agents Grant 5,109,024 - Prakash , et al. April 28, 1 | 1992-04-28 |
Excitatory amino acid antagonists, compositions and use Grant 5,106,847 - Salituro , et al. April 21, 1 | 1992-04-21 |
Cyclopropyl squalene derivatives and their use as inhibitors of cholesterol synthesis Grant 5,102,915 - Angelastro , et al. April 7, 1 | 1992-04-07 |
Novel A-nor-steroid-3-carboxylic acid derivatives Grant 5,100,917 - Flynn , et al. March 31, 1 | 1992-03-31 |
.alpha.-glucosidase inhibitors Grant 5,097,023 - Ducep , et al. March 17, 1 | 1992-03-17 |
NMDA antagonists Grant 5,095,009 - Whitten , et al. March 10, 1 | 1992-03-10 |
N-aralkyl piperidine derivatives useful as antithrombolytic agents Grant 5,093,341 - Carr , et al. March 3, 1 | 1992-03-03 |
Tricyclic fused adenine derivatives Grant 5,086,176 - Peet , et al. February 4, 1 | 1992-02-04 |
17.beta.-(cyclopropylamino)androstene derivatives Grant 5,075,464 - Blohm , et al. December 24, 1 | 1991-12-24 |
Difluoroglutamic acid conjugates with folates and anti-folates for the treatment of neoplastic diseases Grant 5,066,828 - Bey , et al. November 19, 1 | 1991-11-19 |
Selective adenosine reseptor compounds Grant 5,064,947 - Peet , et al. November 12, 1 | 1991-11-12 |
Bis(alkyl-substituted-4-hydroxyphenylthio)alkane analogs as inhibitors of cataractogenesis Grant 5,061,734 - Mao , et al. October 29, 1 | 1991-10-29 |
Inhibitors of lysyl oxidase Grant 5,059,714 - Palfreyman , et al. October 22, 1 | 1991-10-22 |
3-indolyl thioacetate derivatives and NMDA receptor antagonistic use thereof Grant 5,051,442 - Salituro , et al. September 24, 1 | 1991-09-24 |
Liquid pharmaceutical composition for piperidinoalkanol derivatives Grant 5,049,568 - Kristof , et al. September 17, 1 | 1991-09-17 |
Selective adenosine receptor agents Grant 5,047,534 - Peet , et al. September 10, 1 | 1991-09-10 |
Method of preventing AIDS transmission resulting from blood transfusions Grant 5,039,688 - Lewis August 13, 1 | 1991-08-13 |
Hydroxymethyl-indolizidines and quinolizidines and their use as .alpha.-glucosidase I inhibitors Grant 5,028,614 - Liu , et al. July 2, 1 | 1991-07-02 |
Novel chemical compounds for the prophylactic treatment of migraine Grant 5,021,428 - Carr , et al. June 4, 1 | 1991-06-04 |
Inhibitors of lysyl oxidase Grant 5,021,456 - Palfreyman , et al. June 4, 1 | 1991-06-04 |
Tablet Grant D316,914 - Withington May 14, 1 | 1991-05-14 |
Method of effecting immunosuppression Grant 5,013,719 - Bowlin May 7, 1 | 1991-05-07 |
Medicament compositions derived from quinolizine and quinolizinone and methods of use thereof Grant 5,011,846 - Gittos , et al. April 30, 1 | 1991-04-30 |
Anti-retroviral castanospermine esters Grant 5,004,746 - Liu , et al. April 2, 1 | 1991-04-02 |
Pharmaceutical compositions for piperidinoalkanol-ibuprofen combination Grant 4,999,226 - Schock , et al. March 12, 1 | 1991-03-12 |
5'-deoxy-4',5'-unsaturated-5'-substituted adenosines Grant 4,997,924 - Jarvi , et al. March 5, 1 | 1991-03-05 |
Pharmaceutical composition for piperidinoalkanol-decongestant combination Grant 4,996,061 - Webb , et al. February 26, 1 | 1991-02-26 |
Phosphonoalkylpurine derivatives Grant 4,988,680 - Halazy , et al. January 29, 1 | 1991-01-29 |
Method of inhibiting interleukin-1 release and alleviating interleukin-1 mediated conditions Grant 4,975,467 - Ku , et al. December 4, 1 | 1990-12-04 |
Process for the preparation of castanospermine esters Grant 4,970,317 - Margolin , et al. November 13, 1 | 1990-11-13 |
4-substituted 17.beta.-(cyclopropyloxy)androst-5-en-3.beta.-ol and related compounds useful as C17-20 lyase inhibitors Grant 4,966,897 - Angelastro , et al. October 30, 1 | 1990-10-30 |
Inhibitors of lysyl oxidase Grant 4,965,288 - Palfreyman , et al. October 23, 1 | 1990-10-23 |
Excitatory amino acid antagonists Grant 4,960,786 - Salituro , et al. October 2, 1 | 1990-10-02 |
Inhibitors of lysyl oxidase Grant 4,943,593 - Palfreyman , et al. July 24, 1 | 1990-07-24 |
N-2,3-butadienyl tri- and tetraaminoalkane derivatives Grant 4,935,449 - Bey , et al. June 19, 1 | 1990-06-19 |
Pharmaceutical composition for piperidinoalkanol derivatives Grant 4,929,605 - Domet , et al. May 29, 1 | 1990-05-29 |
Method of treating parkinson's syndrome Grant 4,916,151 - Bey , et al. April 10, 1 | 1990-04-10 |
Use of 1,4-disubstituted-piperidinyl compounds in the manufacture of a medicament for the treatment of insomnia Grant 4,908,369 - Schechter , et al. March 13, 1 | 1990-03-13 |
Antihistaminic piperidinyl benzimidazoles Grant 4,908,372 - Carr , et al. March 13, 1 | 1990-03-13 |
Esters of hexahydro-8-hydroxy-2,6-methano-2H-quinolizin-3-(4H)-one and related compounds Grant 4,906,755 - Gittos March 6, 1 | 1990-03-06 |
Controlling the growth of certain tumor tissue with chalcone derivatives Grant 4,904,697 - Sunkara , et al. February 27, 1 | 1990-02-27 |
Method of inhibiting interleukin-1 release Grant 4,870,101 - Ku , et al. September 26, 1 | 1989-09-26 |
Reducing reperfusion injury with 1,3-dihydro-4-methyl-5-(4-methylthio)benzoyl)-2H-imidazol-2-thione Grant 4,868,197 - Schnettler , et al. September 19, 1 | 1989-09-19 |
Enhancement of prazosin Grant 4,868,182 - Dage September 19, 1 | 1989-09-19 |
Methods of treating gout with chalcone derivatives Grant 4,863,968 - Edwards , et al. September 5, 1 | 1989-09-05 |
Process for preparing 4,4'-isopropylidenedithio-bis-(2,6-di-tertiarybutylphenol) by electrocatalysis Grant 4,861,443 - Van Effen August 29, 1 | 1989-08-29 |
Certain 3-carboxylate or 3-carbamyl-5-acyl-2-(1H)-pyridinones having cardiotonic properties Grant 4,853,395 - Jones , et al. August 1, 1 | 1989-08-01 |
Treatment of thromobocytosis with 5-(4-chlorophenyl)-2,4-diemthyl-3H-1,2,4-triazole-3-thione Grant 4,847,276 - Yarrington July 11, 1 | 1989-07-11 |
Sulfhydryl containing tricyclic lactams and their pharmacological methods of use Grant 4,824,832 - Flynn , et al. April 25, 1 | 1989-04-25 |
Novel imidazole dopamine beta hydroxylase inhibitors Grant 4,810,800 - Matthews , et al. March 7, 1 | 1989-03-07 |
Antifungal 2-anilinothiazolines Grant 4,788,209 - Baumann , et al. November 29, 1 | 1988-11-29 |
N-aralkyl piperidine methanol derivatives and the uses thereof Grant 4,783,471 - Carr , et al. November 8, 1 | 1988-11-08 |
Gem-dihalo and tetrahalo-1,12-diamino-4,9-diaza-dodecanes Grant 4,778,926 - Gerhart , et al. October 18, 1 | 1988-10-18 |
Process for preparing 2,6-di-tertiarybutyl-4-mercaptophenol by electrocatalysis Grant 4,772,363 - Van Effen September 20, 1 | 1988-09-20 |
Method of treating multiple sclerosis with chalcone derivatives Grant 4,753,965 - Stemerick , et al. June 28, 1 | 1988-06-28 |
Preparation of polymorphically pure terfenadine Grant 4,742,175 - Fawcett , et al. May 3, 1 | 1988-05-03 |
Antirhinovirus agents Grant 4,738,984 - Parker April 19, 1 | 1988-04-19 |
Process for preparing 2,6-di-tertiarybutyl-4-mercaptophenol Grant 4,734,527 - Krauss March 29, 1 | 1988-03-29 |
Derivatives of 2,6-diamino-3-haloheptanedioic acid Grant 4,730,006 - Bohme , et al. March 8, 1 | 1988-03-08 |
Cardiac antiarrythmic method employing probucol Grant 4,719,237 - McCaughan January 12, 1 | 1988-01-12 |
Fluoroallylamine derivatives Grant 4,699,928 - McDonald October 13, 1 | 1987-10-13 |
Medroxalol intermediates Grant 4,697,024 - Donaldson , et al. September 29, 1 | 1987-09-29 |
Method of alleviating withdrawal symptoms Grant 4,670,459 - Sjoerdsma June 2, 1 | 1987-06-02 |
Cardiotonic thiazolones Grant 4,670,450 - Schenttler , et al. June 2, 1 | 1987-06-02 |
Nonaromatic fluoroallylamine MAO inhibitors Grant 4,650,907 - Bey , et al. March 17, 1 | 1987-03-17 |
Process for the preparation of 4(3H)-quinazolinones Grant 4,644,065 - Vinogradoff February 17, 1 | 1987-02-17 |
Homodisaccharide hypoglycemic agents Grant 4,634,765 - Liu January 6, 1 | 1987-01-06 |
Process for preparing sucrose encrusted methylcellulose particles for use in bulk laxative compositions Grant 4,626,287 - Shah , et al. December 2, 1 | 1986-12-02 |
Process for preparing 5-vinyl-2-pyrrolidinone and intermediates therefor Grant 4,621,145 - Frieben , et al. November 4, 1 | 1986-11-04 |
Antirhinovirus agents Grant 4,602,099 - Parker July 22, 1 | 1986-07-22 |
Treatment of migraine with substituted tropyl benzoate derivatives Grant 4,585,866 - Fozard , et al. April 29, 1 | 1986-04-29 |
Isoquinoline thromboxane synthetase inhibitors Grant 4,584,379 - Wagner April 22, 1 | 1986-04-22 |
Method of alleviating withdrawal symptoms Grant 4,575,510 - Sjoerdsma March 11, 1 | 1986-03-11 |
Pyrrole-3-carboxylate cardiotonic agents Grant 4,560,700 - Schnettler , et al. December 24, 1 | 1985-12-24 |
N-2,3-Butadienyl-1,4-butanediamine derivatives Grant 4,551,550 - Bey November 5, 1 | 1985-11-05 |
Process for treating diseases with ODC inhibitors Grant 4,499,072 - Sunkara , et al. February 12, 1 | 1985-02-12 |
4-Alkanoylimidazol-2-ones Grant 4,447,619 - Grisar , et al. | 1984-05-08 |
Method of inhibiting algae Grant 4,437,873 - Sjoerdsma | 1984-03-20 |
Cardiotonic 4-aroylimidazolidin-2-ones Grant 4,410,540 - Schnettler , et al. October 18, 1 | 1983-10-18 |
Controlled release suppositories consisting essentially of a linear polymer particularly, polyvinyl pyrrolidones Grant 4,406,883 - Byrne , et al. September 27, 1 | 1983-09-27 |
4-Aroylimidazol-2-ones and their use as pharmaceuticals Grant 4,405,635 - Schnettler , et al. September 20, 1 | 1983-09-20 |
Antiviral 1-aryl-5-amino-1-penten-3-ones Grant 4,400,380 - Ritter , et al. August 23, 1 | 1983-08-23 |
Method of inhibiting the growth of protozoa Grant 4,399,151 - Sjoerdsma , et al. August 16, 1 | 1983-08-16 |
Method of alleviating withdrawal symptoms Grant 4,382,946 - Sjoerdsma May 10, 1 | 1983-05-10 |
10-Alkynyl steroids Grant 4,322,416 - Metcalf , et al. March 30, 1 | 1982-03-30 |
10-(1,2-Propadienyl) steroids as irreversible aromatase inhibitors Grant 4,289,762 - Metcalf , et al. September 15, 1 | 1981-09-15 |