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Antimalarial Hexahydropyrimidine Analogues App 20220289685 - De Haro Garcia; Teresa ;   et al. | 2022-09-15 |
Aminopyrimidine Compound App 20220112184 - MATSUNAGA; Nobuyuki ;   et al. | 2022-04-14 |
Fused Heteroaryl Compounds And Their Use As Camkii Inhibitors App 20220098207 - MATSUNAGA; Nobuyuki ;   et al. | 2022-03-31 |
Iminotetrahydropyrimidinone derivatives as plasmepsin V inhibitors Grant 11,136,310 - Charlton , et al. October 5, 2 | 2021-10-05 |
Aminopyrimidine compound Grant 11,130,752 - Matsunaga , et al. September 28, 2 | 2021-09-28 |
Fused Pentacyclic Imidazole Derivatives as Modulators of TNF Activity App 20210252012 - Brookings; Daniel Christopher ;   et al. | 2021-08-19 |
Alkoxy bis-heteroaryl derivatives as modulators of protein aggregation Grant 11,091,474 - Hall , et al. August 17, 2 | 2021-08-17 |
Fused pentacyclic imidazole derivatives as modulators of TNF activity Grant 10,980,814 - Brookings , et al. April 20, 2 | 2021-04-20 |
Bis-heteroaryl derivatives as modulators of protein aggregation Grant 10,975,066 - Wrasidlo , et al. April 13, 2 | 2021-04-13 |
Antimalarial Hexahydropyrimidine Analogues App 20210094941 - De Haro Garcia; Teresa ;   et al. | 2021-04-01 |
Bicyclic bis-heteroaryl derivatives as modulators of protein aggregation Grant 10,889,584 - Hall , et al. January 12, 2 | 2021-01-12 |
Alkoxy Bis-heteroaryl Derivatives As Modulators Of Protein Aggregation App 20200291013 - HALL; Adrian ;   et al. | 2020-09-17 |
Iminotetrahydropyrimidinone Derivatives As Plasmepsin V Inhibitors App 20200283416 - Charlton; Rebecca Louise ;   et al. | 2020-09-10 |
Beta-amino Heterocyclic Dipeptidyl Peptidase Inhibitors For The Treatment Or Prevention Of Diabetes App 20200206221 - Edmondson; Scott D. ;   et al. | 2020-07-02 |
Aminopyrimidine Compound App 20200095240 - MATSUNAGA; Nobuyuki ;   et al. | 2020-03-26 |
Fused Pentacyclic Imidazole Derivatives as Modulators of TNF Activity App 20200046723 - Brookings; Daniel Christopher ;   et al. | 2020-02-13 |
Bicyclic Bis-heteroaryl Derivatives As Modulators Of Protein Aggregation App 20190367513 - HALL; Adrian ;   et al. | 2019-12-05 |
Iminothiadiazinane dioxide derivatives as plasmepsin V inhibitors Grant 10,464,932 - De Haro Garcia , et al. No | 2019-11-05 |
Iminothiadiazinane Dioxide Derivatives as Plasmepsin V Inhibitors App 20190040053 - De Haro Garcia; Teresa ;   et al. | 2019-02-07 |
Fused tricyclic imidazole derivatives as modulators of TNF activity Grant 10,087,179 - Alexander , et al. October 2, 2 | 2018-10-02 |
Bis-heteroaryl Derivatives As Modulators Of Protein Aggregation App 20180222899 - WRASIDLO; Wolfgang ;   et al. | 2018-08-09 |
Beta-amino Heterocyclic Dipeptidyl Peptidase Inhibitors For The Treatment Or Prevention Of Diabetes App 20170348309 - Edmondson; Scott D. ;   et al. | 2017-12-07 |
Nucleoside Derivatives As Inhibitors Of Rna-dependent Rna Viral Polyermase App 20170183373 - Bhat; Balkrishen ;   et al. | 2017-06-29 |
Compounds and methods for antiviral treatment Grant 9,593,108 - Maccoss , et al. March 14, 2 | 2017-03-14 |
Substituted pyridine and pyrimidine derivatives and their use in treating viral infections Grant 9,433,621 - Arasappan , et al. September 6, 2 | 2016-09-06 |
Beta-amino Heterocyclic Dipeptidyl Peptidase Inhibitors For The Treatment Or Prevention Of Diabetes App 20150359793 - Edmondson; Scott D. ;   et al. | 2015-12-17 |
SUBSTITUTED PIPERIDINES THAT INCREASE p53 ACTIVITY AND THE USES THEREOF App 20140336222 - Bogen; Stephane L. ;   et al. | 2014-11-13 |
Substituted piperidines that increase p53 activity and the uses thereof Grant 8,859,776 - Bogen , et al. October 14, 2 | 2014-10-14 |
Substituted Pyridine And Pyrimidine Derivatives And Their Use In Treating Viral Infections App 20140242027 - Arasappan; Ashok ;   et al. | 2014-08-28 |
Gamma secretase modulators Grant 8,809,318 - Zhu , et al. August 19, 2 | 2014-08-19 |
Indole derivatives and methods for antiviral treatment Grant 8,735,414 - MacCoss , et al. May 27, 2 | 2014-05-27 |
Beta-amino Heterocyclic Dipeptidyl Peptidase Inhibitors For The Treatment Or Prevention Of Diabetes App 20130217695 - Edmondson; Scott D. ;   et al. | 2013-08-22 |
Beta-amino heterocyclic dipeptidyl peptidase inhibitors for the treatment of type 2 diabetes Grant 8,440,668 - Edmondson , et al. May 14, 2 | 2013-05-14 |
Substituted Piperidines That Increase P53 Activity And The Uses Thereof App 20120208844 - Bogen; Stephane L. ;   et al. | 2012-08-16 |
Indole Derivatives And Methods For Antiviral Treatment App 20120184574 - Maccoss; Malcolm ;   et al. | 2012-07-19 |
Compounds And Methods For Antiviral Treatment App 20120135999 - Maccoss; Malcolm ;   et al. | 2012-05-31 |
Beta-amino heterocyclic dipeptidyl peptidase inhibitors for the treatment of diabetes Grant 8,168,637 - Edmondson , et al. May 1, 2 | 2012-05-01 |
Gamma Secretase Modulators App 20110306593 - Zhu; Zhaoning ;   et al. | 2011-12-15 |
Deuterated Compounds As Hepatitis C Virus (hcv) Inhibitors App 20110286969 - MacCoss; Malcolm ;   et al. | 2011-11-24 |
Novel Cyclic Azabenzimidazole Derivatives Useful As Anti-diabetic Agents App 20110190308 - Edmondson; Scott D. ;   et al. | 2011-08-04 |
Nucleoside aryl phosphoramidates for the treatment of RNA-dependent RNA viral infection Grant 7,879,815 - MacCoss , et al. February 1, 2 | 2011-02-01 |
Nucleoside Aryl Phosphoramidates for the Treatment of RNA-Dependent RNA Viral Infection App 20100234316 - MacCoss; Malcolm ;   et al. | 2010-09-16 |
Beta-amino Heterocyclic Dipeptidyl Peptidase Inhibitors For The Treatment Or Prevention Of Diabetes App 20100130504 - Edmondson; Scott D. ;   et al. | 2010-05-27 |
Ribonucleoside cyclic acetal derivatives for the treatment of RNA-dependent RNA viral infection Grant 7,632,821 - Butora , et al. December 15, 2 | 2009-12-15 |
C-purine nucleoside analogs as inhibitors of RNA-dependent RNA viral polymerase Grant 7,534,767 - Butora , et al. May 19, 2 | 2009-05-19 |
Novel 2'-c-methyl and 4'c-methyl nucleoside derivatives App 20090118223 - Erion; Mark D. ;   et al. | 2009-05-07 |
Ribonucleoside Cyclic Acetal Derivatives for the Treatment of RNA-Dependent RNA Viral Infection App 20090099126 - Butora; Gabor ;   et al. | 2009-04-16 |
Fluorinated Pyrrolo[2,3-D]Pyrimidine Nucleosides for the Treatment of Rna-Dependent Rna Viral Infection App 20080280842 - MacCoss; Malcolm ;   et al. | 2008-11-13 |
Compositions and Methods For the Treatment Of Obesity and Sexual Dysfunction App 20080200376 - MacCoss; Malcolm ;   et al. | 2008-08-21 |
C-Purine Nucleoside Analogs As Inhibitors Of Rna-Dependent Rna Viral Polymerase App 20080021047 - Butora; Gabor ;   et al. | 2008-01-24 |
Nucleoside Aryl Phosphoramidates for the Treatment of Rna-Dependent Rna Viral Infection App 20070265222 - MacCoss; Malcolm ;   et al. | 2007-11-15 |
Novel 2'-C methyl nucleoside derivatives App 20070179114 - Erion; Mark D. ;   et al. | 2007-08-02 |
Aminocyclopentyl pyridopyrazinone modulators of chemokine receptor activity App 20070155731 - Butora; Gabor ;   et al. | 2007-07-05 |
Anti-hypercholesterolemic compounds App 20070135357 - Sings; Heather L. ;   et al. | 2007-06-14 |
Beta-amino heterocyclic dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes App 20060270679 - Edmondson; Scott D. ;   et al. | 2006-11-30 |
Nucleoside derivatives as inhibitors of rna-dependent rna viral polymerase App 20060264389 - Bhat; Balkrishen ;   et al. | 2006-11-23 |
Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase Grant 7,125,855 - Bhat , et al. October 24, 2 | 2006-10-24 |
Pyrrolidine modulators of CCR5 chemokine receptor activity Grant 7,125,887 - Hale , et al. October 24, 2 | 2006-10-24 |
Beta-amino tetrahydroimidazo (1, 2-a) pyrazines and tetrahydrotrioazolo (4, 3-a) pyrazines as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes Grant 7,125,873 - Edmondson , et al. October 24, 2 | 2006-10-24 |
Nucleoside derivatives as inhibitors of rna-dependent rna viral polymerase App 20060234962 - Olsen; David B. ;   et al. | 2006-10-19 |
Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase App 20060205686 - Bhat; Balkrishen ;   et al. | 2006-09-14 |
Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase Grant 7,105,499 - Carroll , et al. September 12, 2 | 2006-09-12 |
Heterocyclic amide compounds as cell adhesion inhibitors Grant 6,903,075 - Durette , et al. June 7, 2 | 2005-06-07 |
Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase App 20040229840 - Bhat, Balkrishen ;   et al. | 2004-11-18 |
Beta-amino tetrahydroimidazo (1, 2-a) pyrazines and tetrahydrotrioazolo (4,3-a) pyrazines as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes App 20040167133 - Edmondson, Scott D. ;   et al. | 2004-08-26 |
Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase of hepatitis C virus Grant 6,777,395 - Bhat , et al. August 17, 2 | 2004-08-17 |
Nucleoside derivatives as inhibitors of rna-dependent rna viral polymerase App 20040110717 - Carroll, Steven S. ;   et al. | 2004-06-10 |
Substituted amidine derivatives as inhibitors of cell adhesion Grant 6,734,311 - Hagmann , et al. May 11, 2 | 2004-05-11 |
Pyrrolidine modulators of ccr5 chemokine receptor activity App 20040087552 - Hale, Jeffrey J ;   et al. | 2004-05-06 |
Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase App 20040067901 - Bhat, Balkrishen ;   et al. | 2004-04-08 |
Beta-amino heterocyclic dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes Grant 6,699,871 - Edmondson , et al. March 2, 2 | 2004-03-02 |
Substituted .beta.-alanine derivatives as cell adhesion inhibitors Grant 6,645,939 - Durette , et al. November 11, 2 | 2003-11-11 |
Morpholine and thiomorpholine tachykinin receptor antagonists Grant 6,638,930 - Dorn , et al. October 28, 2 | 2003-10-28 |
Beta-amino heterocyclic dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes App 20030100563 - Edmondson, Scott D. ;   et al. | 2003-05-29 |
Substituted amidine derivatives as inhibitors of cell adhesion App 20030092746 - Hagmann, William K. ;   et al. | 2003-05-15 |
Pyrrolidine modulators of chemokine receptor activity Grant 6,498,161 - Caldwell , et al. December 24, 2 | 2002-12-24 |
Cyclic amine modulators of chemokine receptor activity Grant 6,476,054 - Caldwell , et al. November 5, 2 | 2002-11-05 |
Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase App 20020147160 - Bhat, Balkrishen ;   et al. | 2002-10-10 |
N-cyclopentyl modulators of chemokine receptor activity App 20020120146 - Finke, Paul E. ;   et al. | 2002-08-29 |
Phosphate derivatives as immunoregulatory agents Grant 6,437,165 - Mandala , et al. August 20, 2 | 2002-08-20 |
Pyrrolidine modulators of CCR5 chemokine receptor activity App 20020094989 - Hale, Jeffrey J. ;   et al. | 2002-07-18 |
Phosphate derivatives as immunoregulatory agents App 20020091105 - Mandala, Suzanne ;   et al. | 2002-07-11 |
Pyrrolidine modulators of chemokine receptor activity Grant 6,399,619 - Berk , et al. June 4, 2 | 2002-06-04 |
Zwitterionic tachykinin receptor antagonists App 20020042431 - Finke, Paul E. ;   et al. | 2002-04-11 |
N-cyclopentyl modulators of chemokine receptor activity Grant 6,358,979 - Finke , et al. March 19, 2 | 2002-03-19 |
Morpholine and thiomorpholine tachykinin receptor antagonists App 20020002164 - Dorn, Conrad P. ;   et al. | 2002-01-03 |
Biarylalkanoic acids as cell adhesion inhibitors Grant 6,291,511 - Durette , et al. September 18, 2 | 2001-09-18 |
Sulfonamides as cell adhesion inhibitors Grant 6,221,888 - Durette , et al. April 24, 2 | 2001-04-24 |
Pyrrolidine and piperidine modulators of chemokine receptor activity Grant 6,166,037 - Budhu , et al. December 26, 2 | 2000-12-26 |
Cyclic amine modulators of chemokine receptor activity Grant 6,140,349 - Caldwell , et al. October 31, 2 | 2000-10-31 |
Cyclic amine modulations of chemokine receptor activity Grant 6,136,827 - Caldwell , et al. October 24, 2 | 2000-10-24 |
3,3-disubstituted piperidines as modulators of chemokine receptor activity Grant 6,124,319 - MacCoss , et al. September 26, 2 | 2000-09-26 |
Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases Grant 6,043,358 - Caldwell , et al. March 28, 2 | 2000-03-28 |
Spiro-substituted azacycles as neurokinin antagonists Grant 6,013,652 - Maccoss , et al. January 11, 2 | 2000-01-11 |
Spiro-substituted azacycles as modulators of chemokine receptor activity Grant 6,013,644 - Mills , et al. January 11, 2 | 2000-01-11 |
Spiro-substituted azacycles as modulators of chemokine receptor activity Grant 5,962,462 - Mills , et al. October 5, 1 | 1999-10-05 |
Phenyl spiroethercycloalkyl tachykinin receptor antagonists Grant 5,877,191 - Caldwell , et al. March 2, 1 | 1999-03-02 |
Morpholine and thiomorpholine tachykinin receptor antagonists Grant 5,872,116 - Dorn , et al. February 16, 1 | 1999-02-16 |
Trypthophan ureas as neurokinnin antagonists Grant 5,869,489 - Shah , et al. February 9, 1 | 1999-02-09 |
Morpholine compounds are prodrugs useful as tachykinin receptor antagonists Grant 5,780,467 - Dorn , et al. July 14, 1 | 1998-07-14 |
Cycloalkyl tachykinin receptor antagonists Grant 5,750,549 - Caldwell , et al. May 12, 1 | 1998-05-12 |
Morpholine and thiomorpholine tachykinin receptor antagonists Grant 5,719,147 - Dorn , et al. February 17, 1 | 1998-02-17 |
Morpholine compounds are prodrugs useful as tachykinin receptor antagonists Grant 5,691,336 - Dorn , et al. November 25, 1 | 1997-11-25 |
Process for preparing morpholine tachykinin receptor antagonists Grant 5,637,699 - Dorn , et al. June 10, 1 | 1997-06-10 |
Cyclic amidine analogs as inhibitors of nitric oxide synthase Grant 5,629,322 - Guthikonda , et al. May 13, 1 | 1997-05-13 |
Substituted aryl piperazines as neurokinin antagonists Grant 5,607,936 - Chiang , et al. March 4, 1 | 1997-03-04 |
Substituted azetidinones as anti-inflammatory and antidegenerative agents Grant 5,591,737 - Doherty , et al. January 7, 1 | 1997-01-07 |
Treatment of emesis with morpholine tachykinin receptor antagonists Grant 5,512,570 - Dorn , et al. April 30, 1 | 1996-04-30 |
Peptidyl derivatives as inhibitors of interleukin-1.beta. converting enzyme Grant 5,434,248 - Chapman , et al. July 18, 1 | 1995-07-18 |
Peptidyl derivatives as inhibitors of interleukin-1.beta. converting enzyme Grant 5,430,128 - Chapman , et al. July 4, 1 | 1995-07-04 |
Substituted triazolinones, triazolinethiones, and triazolinimines as angiotensin II antagonists Grant 5,411,980 - Ashton , et al. May 2, 1 | 1995-05-02 |
Substituted imidazo-fused 5-membered ring heterocycles as angiotensin II antagonists Grant 5,389,660 - Greenlee , et al. February 14, 1 | 1995-02-14 |
N,N-diacylpiperazines Grant 5,292,726 - Ashton , et al. March 8, 1 | 1994-03-08 |
Substituted pyrazolopyrimidines as angiotensin II antagonists Grant 5,250,521 - Allen , et al. October 5, 1 | 1993-10-05 |
Substituted azetidinones as anti-inflammatory and antidegenerative agents Grant 5,229,381 - Doherty , et al. July 20, 1 | 1993-07-20 |
Angiotensin II antagonists incorporating a substituted benzyl element Grant 5,162,325 - Chakravarty , et al. November 10, 1 | 1992-11-10 |
Novel betalactam elastase inhibitors containing phosphorous acid derivatives at the 4-position of the 2-azetidinone Grant 5,100,880 - Durette , et al. March 31, 1 | 1992-03-31 |
Piperazinyl derivatives of purines and isosteres thereof as hypoglycemic agents Grant 5,057,517 - Johnston , et al. October 15, 1 | 1991-10-15 |
Piperazinylalkylpyrimidines as hypoglycemic agents Grant 4,980,350 - MacCoss , et al. December 25, 1 | 1990-12-25 |
Regioselective synthesis of 9-substituted purine acyclonucleoside derivatives Grant 4,801,710 - MacCoss , et al. January 31, 1 | 1989-01-31 |
Cyclic pyrophosphates of purine and pyrimidine acyclonucleosides Grant 4,670,424 - MacCoss , et al. June 2, 1 | 1987-06-02 |
N-alkylguanine acyclonucleosides as antiviral agents Grant 4,579,849 - MacCoss , et al. April 1, 1 | 1986-04-01 |
Prodrugs based on phospholipid-nucleoside conjugates Grant 4,471,113 - MacCoss September 11, 1 | 1984-09-11 |