Patent | Date |
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Novel Ptefb Inhibiting Macrocyclic Compounds App 20220281892 - LUCKING; Ulrich ;   et al. | 2022-09-08 |
Ptefb Inhibiting Macrocyclic Compounds App 20220267353 - LUCKING; Ulrich ;   et al. | 2022-08-25 |
PTEFb inhibiting macrocyclic compounds Grant 11,254,690 - Lucking , et al. February 22, 2 | 2022-02-22 |
PTEFb inhibiting macrocyclic compounds Grant 11,242,356 - Lucking , et al. February 8, 2 | 2022-02-08 |
2-(morpholin-4-yl)-1,7-naphthyridines App 20200383991 - WORTMANN; Lars ;   et al. | 2020-12-10 |
Novel Ptefb Inhibiting Macrocyclic Compounds App 20200347079 - LUCKING; Ulrich ;   et al. | 2020-11-05 |
2-(morpholin-4-yl)-1,7-naphthyridines Grant 10,772,893 - Wortmann , et al. Sept | 2020-09-15 |
5-substituted 2-(morpholin-4-yl)-1,7-naphthyridines Grant 10,729,680 - Lucking , et al. | 2020-08-04 |
Macrocyclic sulfondiimine compounds Grant 10,717,749 - Lucking , et al. | 2020-07-21 |
Novel Ptefb Inhibiting Macrocyclic Compounds App 20200123174 - Lucking; Ulrich ;   et al. | 2020-04-23 |
5-substituted 2-(morpholin-4-yl)-1,7-naphthyridines App 20190142812 - LUCKING; Ulrich ;   et al. | 2019-05-16 |
Modified macrocyclic compounds Grant 10,214,542 - Lucking , et al. Feb | 2019-02-26 |
Novel Modified Macrocyclic Compounds App 20180282346 - LUCKING; Ulrich ;   et al. | 2018-10-04 |
Novel Macrocyclic Sulfondiimine Compounds App 20180273548 - LUCKING; Ulrich ;   et al. | 2018-09-27 |
2-(morpholin-4-yl)-1,7-naphthyridines App 20180256591 - WORTMANN; Lars ;   et al. | 2018-09-13 |
2-(morpholin-4-yl)-1,7-naphthyridines Grant 9,993,484 - Wortmann , et al. June 12, 2 | 2018-06-12 |
4-aryl-N-phenyl-1,3,5-triazin-2-amines containing a sulfoximine group Grant 9,962,389 - Lucking , et al. May 8, 2 | 2018-05-08 |
Macrocyclic compounds Grant 9,963,464 - Lucking , et al. May 8, 2 | 2018-05-08 |
Fluorinated benzofuranyl-pyrimidine derivatives containing a sulfone group Grant 9,902,716 - Kosemund , et al. February 27, 2 | 2018-02-27 |
Fluorinated benzofuranyl-pyrimidine derivatives containing a sulfoximine group Grant 9,884,849 - Kosemund , et al. February 6, 2 | 2018-02-06 |
5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfoximine group Grant 9,877,954 - Lucking , et al. January 30, 2 | 2018-01-30 |
5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfone group Grant 9,856,242 - Kosemund , et al. January 2, 2 | 2018-01-02 |
Compounds For The Treatment Of Cancer App 20170342064 - SCHULZE; Volker ;   et al. | 2017-11-30 |
Disubstituted 5-fluoro pyrimidine derivatives containing a sulfondiimine group Grant 9,790,189 - Lucking , et al. October 17, 2 | 2017-10-17 |
Sulfoximine substituted 5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives and their use as CDK9 kinase inhibitors Grant 9,770,445 - Kosemund , et al. September 26, 2 | 2017-09-26 |
Fluorinated Benzofuranyl-pyrimidine Derivatives Containing A Suflone Group App 20170226092 - KOSEMUND; Dirk ;   et al. | 2017-08-10 |
Fluorinated Benzofuranyl-pyrimidine Derivatives Containing A Sulfoximine Group App 20170217938 - KOSEMUND; Dirk ;   et al. | 2017-08-03 |
4-aryl-n-phenyl-1,3,5-triazin-2-amines Containing A Sulfoximine Group App 20170217949 - LUCKING; Ulrich ;   et al. | 2017-08-03 |
2-(morpholin-4-yl)-1,7-naphthyridines App 20170216304 - WORTMANN; Lars ;   et al. | 2017-08-03 |
5-fluoro-n-(pyridin-2-yl)pyridin-2-amine Derivatives Containing A Sulfoximine Group App 20170202815 - LUCKING; Ulrich ;   et al. | 2017-07-20 |
N-(pyridin-2-yl)pyrimidin-4-amine derivatives containing a sulfone group Grant 9,708,293 - Lucking , et al. July 18, 2 | 2017-07-18 |
4-aryl-N-phenyl-1,3,5-triazin-2-amines containing a sulfoximine group Grant 9,669,034 - Lucking , et al. June 6, 2 | 2017-06-06 |
5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfone group Grant 9,670,161 - Lucking , et al. June 6, 2 | 2017-06-06 |
N-(pyridin-2-yl)pyrimidin-4-amine derivatives containing a sulfoximine group Grant 9,650,361 - Lucking , et al. May 16, 2 | 2017-05-16 |
5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfoximine group Grant 9,650,340 - Lucking , et al. May 16, 2 | 2017-05-16 |
Prodrug derivatives of substituted triazolopyridines Grant 9,586,958 - Schulze , et al. March 7, 2 | 2017-03-07 |
Novel Macrocyclic Compounds App 20170029439 - LUCKING; Ulrich ;   et al. | 2017-02-02 |
2-(morpholin-4-yl)-1,7-naphthyridines Grant 9,549,932 - Wortmann , et al. January 24, 2 | 2017-01-24 |
Disubstituted 5-fluoro Pyrimidine Derivatives Containing A Sulfondiimine Group App 20170015634 - LUCKING; Ulrich ;   et al. | 2017-01-19 |
5-fluoro-n-(pyridin-2-yl)pyridin-2-amine Derivatives Containing A Sulfone Group App 20170001989 - KOSEMUND; Dirk ;   et al. | 2017-01-05 |
4-(ortho)-fluorophenyl-5-fluoropyrimidin-2-yl amines containing a sulfoximine group Grant 9,499,492 - Lucking , et al. November 22, 2 | 2016-11-22 |
2-(morpholin-4-yl)-1,7-naphthyridines App 20160287604 - Wortmann; Lars ;   et al. | 2016-10-06 |
Prodrug Derivatives Of Substituted Triazolopyridines App 20160207915 - Schulze; Volker ;   et al. | 2016-07-21 |
Novel Compounds For The Treatment Of Cancer App 20160207928 - SCHULZE; Volker ;   et al. | 2016-07-21 |
Substituted Benzylpyrazoles App 20160151370 - HITCHCOCK; Marion ;   et al. | 2016-06-02 |
Sulfoximine Substituted 5-fluoro-n-(pyridin-2-yl)pyridin-2-amine Derivatives And Their Use As Cdk9 Kinase Inhibitors App 20160143893 - KOSEMUND; Dirk ;   et al. | 2016-05-26 |
5-fluoro-n-(pyridin-2-yl)pyridin-2-amine Derivatives Containing A Sulfoximine Group App 20150291528 - Lucking; Ulrich ;   et al. | 2015-10-15 |
4-(ortho)-fluorophenyl-5-fluoropyrimidin-2-yl Amines Containing A Sulfoximine Group App 20150291537 - Lucking; Ulrich ;   et al. | 2015-10-15 |
N-(pyridin-2-yl)pyrimidin-4-amine Derivatives Containing A Sulfoximine Group App 20150291559 - Lucking; Ulrich ;   et al. | 2015-10-15 |
N-(pyridin-2-yl)pyrimidin-4-amine Derivatives Containing A Sulfone Group App 20150274695 - Lucking; Ulrich ;   et al. | 2015-10-01 |
5-fluoro-n-(pyridin-2-yl)pyridin-2-amine Derivatives Containing A Sulfone Group App 20150274666 - Lucking; Ulrich ;   et al. | 2015-10-01 |
4-(ortho)-fluorophenyl-5-fluoropyrimidin-2-yl Amines Containing A Sulfone Group App 20150259300 - Lucking; Ulrich ;   et al. | 2015-09-17 |
Disubstituted 5-fluoro pyrimidine derivatives containing a sulfoximine group Grant 9,133,171 - Lucking , et al. September 15, 2 | 2015-09-15 |
Disubstituted 5-fluoro-pyrimidines Grant 9,108,926 - Lucking , et al. August 18, 2 | 2015-08-18 |
Disubstituted 5-fluoro Pyrimidine Derivatives Containing A Sulfoximine Group App 20150005329 - Lucking; Ulrich ;   et al. | 2015-01-01 |
Substituted 4-Aryl-N-phenyl-1,3,5-triazin-2-amines Grant 8,916,557 - Lucking , et al. December 23, 2 | 2014-12-23 |
4-aryl-n-phenyl-1,3,5-triazin-2-amines Containing A Sulfoximine Group App 20140315906 - Lucking; Ulrich ;   et al. | 2014-10-23 |
Disubstituted 5-fluoro-pyrimidines App 20140228387 - Lucking; Ulrich ;   et al. | 2014-08-14 |
Sulfone-substituted anilinopyrimidine derivatives as CDK inhibitors, the production thereof, and use as a medicine Grant 8,802,686 - Lucking , et al. August 12, 2 | 2014-08-12 |
Sulfoximine-substituted anilinopyrimidine derivatives as CDK inhibitors, the production thereof, and use as medicine Grant 8,735,412 - Lucking , et al. May 27, 2 | 2014-05-27 |
Substituted 4-aryl-n-phenyl-1,3,5-triazin-2-amines App 20140045852 - Lucking; Ulrich ;   et al. | 2014-02-13 |
Use Of Novel Pan-cdk Inhibitors For Treating Tumors App 20130210846 - Lucking; Ulrich ;   et al. | 2013-08-15 |
Sulfoximine-substituted pyrimidines as CDK- and/or VEGF inhibitors, their production and use as pharmaceutical agents Grant 8,507,510 - Lucking , et al. August 13, 2 | 2013-08-13 |
Pharmaceutically Active Disubstituted Triazine Derivatives App 20130079345 - Eickhoff; Jan ;   et al. | 2013-03-28 |
Substituted (Heteroarylmethyl)thiohydantoins App 20120251551 - Lucking; Ulrich ;   et al. | 2012-10-04 |
(Heteroarylmethyl) Thiohydantoins as anticancer drugs App 20120238533 - Cleve; Arwed ;   et al. | 2012-09-20 |
Sulfoximine-substituted Anilinopyrimidine Derivatives As Cdk Inhibitors, The Production Thereof, And Use As Medicine App 20110294838 - Lucking; Ulrich ;   et al. | 2011-12-01 |
Sulfone-substituted Anilinopyrimidine Derivatives As Cdk Inhibitors, The Production Thereof, And Use As A Medicine App 20110251222 - Lucking; Ulrich ;   et al. | 2011-10-13 |
Sulphoximine-substituted quinoline and quinazoline derivatives as kinase inhibitors Grant 8,003,787 - Eis , et al. August 23, 2 | 2011-08-23 |
Sulfoximine-substituted pyrimidines, processes for production thereof and use thereof as drugs Grant 7,825,128 - Lucking , et al. November 2, 2 | 2010-11-02 |
Substituted imidazo[1,2b]pyridazines as kinase inhibitors, their preparation and use as medicaments Grant 7,750,000 - Prien , et al. July 6, 2 | 2010-07-06 |
Sulfoximine-substituted Pyrimidines As Cdk- And/or Vegf Inhibitors, Their Production And Use As Pharmaceutical Agents App 20100076000 - Lucking; Ulrich ;   et al. | 2010-03-25 |
CDK-inhibitory pyrimidines, their production and use as pharmaceutical agents Grant 7,598,260 - Brumby , et al. October 6, 2 | 2009-10-06 |
Novel Sulphoximine-substituted Quinoline And Quinazoline Derivatives As Kinase Inhibitors App 20090226377 - EIS; Knut ;   et al. | 2009-09-10 |
Substituted Sulfonamido-macrocycles As Tie2 Inhibitors And Salts Thereof, Pharmaceutical Compositions Comprising Same, Methods Of Preparing Same And Uses Of Same App 20090005373 - Hartung; Ingo ;   et al. | 2009-01-01 |
CDK-Inhibitory pyrimidines, their production and use as pharmaceutical agents App 20080039447 - Brumby; Thomas ;   et al. | 2008-02-14 |
CDK-inhibitory pyrimidines, their production and use as pharmaceutical agents Grant 7,291,624 - Brumby , et al. November 6, 2 | 2007-11-06 |
CDK-inhibitory 2-heteroaryl-pyrimidines, their production and use as pharmaceutical agents Grant 7,288,547 - Lucking , et al. October 30, 2 | 2007-10-30 |
Sulfoximine-substituted pyrimidines, processes for production thereof and use thereof as drugs App 20070232632 - Lucking; Ulrich ;   et al. | 2007-10-04 |
Macrocyclic anilinopyrimidines with substituted sulphoximine as selective inhibitors of cell cycle kinases App 20070191393 - Lucking; Ulrich ;   et al. | 2007-08-16 |
Compound and a composition including such a compound Grant 7,235,561 - Brumby , et al. June 26, 2 | 2007-06-26 |
Substituted imidazo[1,2b]pyridazines as kinase inhibitors, their preparation and use as medicaments App 20070093490 - Prien; Olaf ;   et al. | 2007-04-26 |
Substituted 2-anilinopyrimidines as cell-cycle-kinase or receptor-tyrosine-kinase inhibitors, their production and use as pharmaceutical agents App 20060111378 - Cleve; Arwed ;   et al. | 2006-05-25 |
CDK-inhibitory pyrimidines, their production and use as pharmaceutical agents App 20040224966 - Brumby, Thomas ;   et al. | 2004-11-11 |
CDK-inhibitory pyrimidines, their production and use as pharmaceutical agents App 20040102630 - Brumby, Thomas ;   et al. | 2004-05-27 |
CDK-inhibitory 2-heteroaryl-pyrimidines, their production and use as pharmaceutical agents App 20040063737 - Lucking, Ulrich ;   et al. | 2004-04-01 |