Patent | Date |
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Synthesis of substituted pyrazoline carboxamidine derivatives Grant 9,422,244 - van Loevezijn , et al. August 23, 2 | 2016-08-23 |
1H-imidazole derivatives as cannabinoid CB2 receptor modulators Grant 8,937,184 - Lange , et al. January 20, 2 | 2015-01-20 |
1H-imidazole derivative having CB.sub.1, agonistic, CB.sub.1 partial agonistic or CB.sub.1 antagnistic activity Grant 8,729,101 - Kruse , et al. May 20, 2 | 2014-05-20 |
Spiro azepane-oxazolidinones as Kv1.3 potassium channel blockers Grant 8,575,148 - Smid , et al. November 5, 2 | 2013-11-05 |
Sulphur containing pyrazole derivatives as selective cannabinoid CB.sub.1 receptor antagonists Grant 8,461,184 - Lange , et al. June 11, 2 | 2013-06-11 |
4,5 dihydro-(1H)-pyrazole derivatives as cannabinoid CB.sub.1 receptor modulators Grant 8,410,135 - Lange , et al. April 2, 2 | 2013-04-02 |
Synthesis Of Substituted Pyrazoline Carboxamidine Derivatives App 20130060041 - van Loevezijn; Arnold ;   et al. | 2013-03-07 |
Compounds with a combination of cannabinoid CB.sub.1 antagonism and serotonin reuptake inhibition Grant 8,138,174 - Lange , et al. March 20, 2 | 2012-03-20 |
Compounds with a combination of cannabinoid-CB.sub.1 antagonism and acetylcholinesterase inhibition Grant 8,063,062 - Lange , et al. November 22, 2 | 2011-11-22 |
SPIRO AZEPANE-OXAZOLIDINONES AS Kv1.3 POTASSIUM CHANNEL BLOCKERS App 20110237569 - Smid; Pieter ;   et al. | 2011-09-29 |
Fluoro-substituted 3,4-diaryl-4,5-dihydro-1h-pyrazole-1-carboxamidine Derivatives Having Cb1-antagonistic Activity App 20110172274 - Lange; Josephus H.M. ;   et al. | 2011-07-14 |
5-aryl-4,5-dihydro-(1h)-pyrazolines As Cannabinoid Cb1 Receptor Agonists App 20110160459 - LANGE; Josephus H.M. ;   et al. | 2011-06-30 |
Synthesis Of 3,4-diaryl-4,5-dihydro-(h)-pyrazole-1-carboxamidine Derivatives App 20110137040 - Lange; Josephus H.M. ;   et al. | 2011-06-09 |
5-aryl-4,5-dihydro-(1H)-pyrazolines as cannabinoid CB1 receptor agonists Grant 7,928,134 - Lange , et al. April 19, 2 | 2011-04-19 |
(5r)-1,5-diaryl-4,5-dihydro-1h-pyrazole-3-carboxamidine Derivatives Having Cb1-antagonistic Activity App 20110053983 - Lange; Josephus H.M. ;   et al. | 2011-03-03 |
Sulphur Containing Pyrazole Derivatives As Selective Cannabinoid Cb1 Receptor Antagonists App 20100292204 - Lange; Josephus H.M. ;   et al. | 2010-11-18 |
Sulphur containing pyrazole derivatives as selective cannabinoid CB.sub.1 receptor antagonists Grant 7,786,144 - Lange , et al. August 31, 2 | 2010-08-31 |
1,3,5-trisubstituted 4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity Grant 7,745,476 - Lange , et al. June 29, 2 | 2010-06-29 |
4,5-dihydro-1H-pyrazole derivatives having potent CB.sub.1-antagonistic activity Grant 7,608,718 - Lange , et al. October 27, 2 | 2009-10-27 |
1h-imidazole Derivative Having Cb1, Agonistic, Cb1 Partial Agonistic Or Cb1 Antagnistic Activity App 20090181949 - KRUSE; Cornelis G. ;   et al. | 2009-07-16 |
4,5-dihydro-1H-pyrazole derivatives having CB.sub.1-antagonistic activity Grant 7,528,162 - Kruse , et al. May 5, 2 | 2009-05-05 |
Tetrasubstituted imidazole derivatives as cannabinoid CB.sub.1 receptor modulators with a high CB.sub.1/CB.sub.2 receptor subtype selectivity Grant 7,524,867 - Lange , et al. April 28, 2 | 2009-04-28 |
5-aryl-4,5-dihydro-(1h)-pyrazolines As Cannabinoid Cb1 Receptor Agonists App 20090082396 - Lange; Josephus H.M. ;   et al. | 2009-03-26 |
1 H-imidazole derivatives as cannabinoid receptor modulators Grant 7,498,348 - Lange , et al. March 3, 2 | 2009-03-03 |
Imidazoline derivatives having CB.sub.1-antagonistic activity Grant 7,495,108 - Lange , et al. February 24, 2 | 2009-02-24 |
4,5 Dihydro-(1H)-Pyrazole Derivatives as Cannabinoid CB1 Receptor Modulators App 20080312276 - Lange; Josephus H.M. ;   et al. | 2008-12-18 |
Compounds With A Combination Of Cannabinoid Cb1 Antagonism And Serotonin Reuptake Inhibition App 20080214559 - Lange; Josephus H.M. ;   et al. | 2008-09-04 |
Compounds With A Combination Of Cannabinoid-cb1 Antagonism And Acetylcholinesterase Inhibition App 20080153867 - Lange; Josephus H.M. ;   et al. | 2008-06-26 |
Thiazole derivatives having CB.sub.1-antagonistic, agonistic or partial agonistic activity Grant 7,342,032 - Lange , et al. March 11, 2 | 2008-03-11 |
1H-1,2,4-triazole-3-carboxamide derivatives having cannabinoid-CB.sub.1 receptor agonistic, partial agonistic, inverse agonistic or antagonistic activity Grant 7,319,110 - Lange , et al. January 15, 2 | 2008-01-15 |
Sulphur Containing Pyrazole Derivatives As Selective Cannabinoid Cb1 Receptor Antagonists App 20070281973 - Lange; Josephus H.M. ;   et al. | 2007-12-06 |
1 H-imidazole Derivatives As Cannabinoid Receptor Modulators App 20070281974 - Lange; Josephus H.M. ;   et al. | 2007-12-06 |
4,5-Dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activity App 20070259884 - Lange; Josephus H.M. ;   et al. | 2007-11-08 |
1H-imidazole derivatives as cannabinoid receptor modulators Grant 7,271,189 - Lange , et al. September 18, 2 | 2007-09-18 |
4,5-Dihydro-(1H)-pyrazole derivatives as cannabinoid CB1 receptor modulators App 20070142362 - Lange; Josephus H.M. ;   et al. | 2007-06-21 |
Imidazoline derivatives having CB1-antagonistic activity App 20070135492 - Lange; Josephus H.M. ;   et al. | 2007-06-14 |
Neurotensin active 2,3,diaryl-pyrazolidine derivatives Grant 7,186,741 - Feenstra , et al. March 6, 2 | 2007-03-06 |
Imidazoline derivatives having CB.sub.1-antagonistic activity Grant 7,173,044 - Lange , et al. February 6, 2 | 2007-02-06 |
Imidazoline derivatives having CB1-antagonistic activity App 20060241152 - Lange; Josephus H.M. ;   et al. | 2006-10-26 |
1H-imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1-antagonistic activity Grant 7,109,216 - Kruse , et al. September 19, 2 | 2006-09-19 |
1H-imidazole derivatives as cannabinoid CB2 receptor modulators App 20060194779 - Lange; Josephus H.M. ;   et al. | 2006-08-31 |
4,5-Dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activity Grant 6,974,810 - Lange , et al. December 13, 2 | 2005-12-13 |
Tetrasubstituted imidazole derivatives as cannabinoid CB1 receptor modulators with a high CB1/CB2 receptor subtype selectivity App 20050267161 - Lange, Josephus H.M. ;   et al. | 2005-12-01 |
Imidazoline derivatives having CB1-antagonistic activity App 20050187259 - Lange, Josephus H.M. ;   et al. | 2005-08-25 |
1,3,5-trisubstituted 4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity App 20050171179 - Lange, Josephus H.M. ;   et al. | 2005-08-04 |
1H-imidazole derivatives as cannabinoid receptor modulators App 20050137197 - Lange, Josephus H.M. ;   et al. | 2005-06-23 |
Thiazole derivatives as cannabinoid receptor modulators App 20050065189 - Lange, Josephus H.M. ;   et al. | 2005-03-24 |
1 H-imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1-antagonistic activity App 20050054679 - Kruse, Cornelis G. ;   et al. | 2005-03-10 |
Thiazole derivatives having cb1-antagonistic, agonistic or partial agonistic activity App 20040266841 - Lange, Josephus H.M. ;   et al. | 2004-12-30 |
Novel 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic activity App 20040248944 - Kruse, Cornelis G ;   et al. | 2004-12-09 |
Neurotensin active 2,3,diaryl-pyrazolidine derivatives App 20040242493 - Feenstra, Roelof W. ;   et al. | 2004-12-02 |
1H-imidazole derivatives having cb1 agonistic, cb1 partial agonistic or cb1 antagonistic activity App 20040235854 - Kruse, Cornelis G. ;   et al. | 2004-11-25 |
1H-1,2,4-triazole-3-carboxamide derivatives having cannabinoid-CB1 receptor agonistic, partial agonistic, inverse agonistic or antagonistic activity App 20040106614 - Lange, Josephus H. M. ;   et al. | 2004-06-03 |
4,5-Dihydro-1h-pyrazole derivatives having potent cb1-antagonistic activity App 20040106800 - Lange, Josephus H.M. ;   et al. | 2004-06-03 |
Benzisoxazole derivatives having d4-antagonistic activity Grant 6,335,326 - Den Hartog , et al. January 1, 2 | 2002-01-01 |
4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity App 20010053788 - Lange, Josephus H. M. ;   et al. | 2001-12-20 |