Kruse; Cornelis G.

Patent Applications and Registrations

Patent applications and USPTO patent grants for Kruse; Cornelis G..The latest application filed is for "arylsulfonyl pyrazoline carboxamidine derivatives as 5-ht6 antagonists".

Company Profile

0.48.52

Kruse; Cornelis G. - CP Weesp NL
Kruse; Cornelis G. - Weesp NL
Kruse; Cornelis G. - Weep NL
Kruse; Cornelis G. - Weeps NL
Kruse; Cornelis G - Weesp NL

*profile and listings may contain filings by different individuals or companies with the same name. Review application materials to confirm ownership/assignment.

Patent Activity

Patent	Date
Arylsulfonyl pyrazoline carboxamidine derivatives as 5-HT.sub.6 antagonists Grant 9,126,942 - van Loevezijn , et al. September 8, 2	2015-09-08
Arylsulfonyl Pyrazoline Carboxamidine Derivatives As 5-ht6 Antagonists App 20150051239 - van Loevezijn; Arnold ; et al.	2015-02-19
Arylsulfonyl pyrazoline carboxamidine derivatives as 5-HT.sub.6 antagonists Grant 8,901,108 - Van Loevezijn , et al. December 2, 2	2014-12-02
Sulfonylpyrazole And Sulfonylpyrazoline Carboxamidine Derivatives As 5-ht6 Antagonists App 20140303372 - Van Loevezijn; Arnold ; et al.	2014-10-09
Heterocyclic compounds with affinity to muscarinic receptors Grant 8,735,388 - Stoit , et al. May 27, 2	2014-05-27
1H-imidazole derivative having CB.sub.1, agonistic, CB.sub.1 partial agonistic or CB.sub.1 antagnistic activity Grant 8,729,101 - Kruse , et al. May 20, 2	2014-05-20
Sulfonylpyrazole and sulfonylpyrazoline carboxamidine derivatives as 5-HT.sub.6 antagonists Grant 8,722,887 - Van Loevezijn , et al. May 13, 2	2014-05-13
Heterocyclic Compounds Iwth Affinity To Muscarinic Receptors App 20140080861 - Stoit; Axel ; et al.	2014-03-20
Arylsulfonyl Pyrazoline Carboxamidine Derivatives As 5-ht6 Antagonists App 20140011775 - van Loevezijn; Arnold ; et al.	2014-01-09
Heterocyclic compounds with affinity to muscarinic receptors Grant 8,586,606 - Stoit , et al. November 19, 2	2013-11-19
Arylsulfonyl pyrazoline carboxamidine derivatives as 5-HT.sub.6 antagonists Grant 8,563,723 - Van Loevezijn , et al. October 22, 2	2013-10-22
Sulphur containing pyrazole derivatives as selective cannabinoid CB.sub.1 receptor antagonists Grant 8,461,184 - Lange , et al. June 11, 2	2013-06-11
Azaindole derivatives with a combination of partial nicotinic acetyl-choline receptor agonism and dopamine reuptake inhibition Grant 8,252,930 - Stoit , et al. August 28, 2	2012-08-28
Heterocyclic Compounds With Affinity To Muscarinic Receptors App 20120095039 - Stoit; Axel ; et al.	2012-04-19
Compounds with a combination of cannabinoid CB.sub.1 antagonism and serotonin reuptake inhibition Grant 8,138,174 - Lange , et al. March 20, 2	2012-03-20
Phenylpiperazine derivatives with a combination of partial dopamine-D.sub.2 receptor agonism and serotonin reuptake inhibition Grant 8,101,619 - Feenstra , et al. January 24, 2	2012-01-24
Heterocyclic compounds with affinity to muscarinic receptors Grant 8,084,473 - Stoit , et al. December 27, 2	2011-12-27
Compounds with a combination of cannabinoid-CB.sub.1 antagonism and acetylcholinesterase inhibition Grant 8,063,062 - Lange , et al. November 22, 2	2011-11-22
Azaindole derivatives with a combination of partial nicotinic acetyl-choline receptor agonism and dopamine reuptake inhibition Grant 7,964,728 - Stoit , et al. June 21, 2	2011-06-21
Azaindole Derivatives With A Combination Of Partial Nicotinic Acetyl-choline Receptor Agonism And Dopamine Reuptake Inhibition App 20110053962 - Stoit; Axel ; et al.	2011-03-03
Arylsulfonyl Pyrazoline Carboxamidine Derivatives As 5-ht6 Antagonists App 20110046171 - Loevezijn; Arnold Van ; et al.	2011-02-24
Sulphur Containing Pyrazole Derivatives As Selective Cannabinoid Cb1 Receptor Antagonists App 20100292204 - Lange; Josephus H.M. ; et al.	2010-11-18
Sulphur containing pyrazole derivatives as selective cannabinoid CB.sub.1 receptor antagonists Grant 7,786,144 - Lange , et al. August 31, 2	2010-08-31
Piperazine and piperidine compounds Grant RE41,425 - Feenstra , et al. July 6, 2	2010-07-06
1,3,5-trisubstituted 4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity Grant 7,745,476 - Lange , et al. June 29, 2	2010-06-29
Sulfonylpyrazole And Sulfonylpyrazoline Carboxamidine Derivatives As 5-ht6 Antagonists App 20100145042 - Van Loevezijn; Arnold ; et al.	2010-06-10
Sulfonylpyrazole and sulfonylpyrazoline carboxamidine derivatives as 5-HT.sub.6 antagonists Grant 7,728,018 - Van Loevezijn , et al. June 1, 2	2010-06-01
Muscarinic Agonists To Treat Impulse Control Disorders App 20100120752 - De Bruin; Natasja M.W.J. ; et al.	2010-05-13
N-oxides of venlafaxine and o-desmethylvenlafaxine as prodrugs Grant 7,696,383 - Turski , et al. April 13, 2	2010-04-13
4,5-dihydro-1H-pyrazole derivatives having potent CB.sub.1-antagonistic activity Grant 7,608,718 - Lange , et al. October 27, 2	2009-10-27
Phenylpiperazine Grant 7,605,162 - Van Hes , et al. October 20, 2	2009-10-20
1h-imidazole Derivative Having Cb1, Agonistic, Cb1 Partial Agonistic Or Cb1 Antagnistic Activity App 20090181949 - KRUSE; Cornelis G. ; et al.	2009-07-16
New Phenylpiperazine App 20090143406 - Hes; Roelof Van ; et al.	2009-06-04
4,5-dihydro-1H-pyrazole derivatives having CB.sub.1-antagonistic activity Grant 7,528,162 - Kruse , et al. May 5, 2	2009-05-05
Tetrasubstituted imidazole derivatives as cannabinoid CB.sub.1 receptor modulators with a high CB.sub.1/CB.sub.2 receptor subtype selectivity Grant 7,524,867 - Lange , et al. April 28, 2	2009-04-28
1 H-imidazole derivatives as cannabinoid receptor modulators Grant 7,498,348 - Lange , et al. March 3, 2	2009-03-03
Imidazoline derivatives having CB.sub.1-antagonistic activity Grant 7,495,108 - Lange , et al. February 24, 2	2009-02-24
Heterocyclic Compounds with Affinity to Muscarinic Receptors App 20090018160 - Stoit; Axel ; et al.	2009-01-15
Sildenafil N-oxide As Prodrug App 20090005395 - Turski; Lechoslaw A. ; et al.	2009-01-01
N-oxides Of Venlafaxine And O-desmethylvenlafaxine As Prodrugs App 20090005455 - Turski; Lechoslaw A. ; et al.	2009-01-01
Sulfonylpyrazole And Sulfonylpyrazoline Carboxamidine Derivatives As 5-ht6 Antagonists App 20080311179 - Van Loevezijn; Arnold ; et al.	2008-12-18
Phenylpiperazines Grant 7,456,182 - Van Hes , et al. November 25, 2	2008-11-25
Compounds With A Combination Of Cannabinoid Cb1 Antagonism And Serotonin Reuptake Inhibition App 20080214559 - Lange; Josephus H.M. ; et al.	2008-09-04
Use Of 5-ht6 Antagonists To Prevent Relapse Into Addiction App 20080171779 - De Bruin; Natasja M.W.J. ; et al.	2008-07-17
Compounds With A Combination Of Cannabinoid-cb1 Antagonism And Acetylcholinesterase Inhibition App 20080153867 - Lange; Josephus H.M. ; et al.	2008-06-26
Selective inhibitors of neurotensin degrading enzymes App 20080146524 - Smid; Pieter ; et al.	2008-06-19
Tetrahydropyridin-4-yl indoles with a combination of affinity for dopamine-D.sub.2 receptors and serotonin reuptake sites Grant 7,371,769 - Hes , et al. May 13, 2	2008-05-13
Thiazole derivatives having CB.sub.1-antagonistic, agonistic or partial agonistic activity Grant 7,342,032 - Lange , et al. March 11, 2	2008-03-11
1H-1,2,4-triazole-3-carboxamide derivatives having cannabinoid-CB.sub.1 receptor agonistic, partial agonistic, inverse agonistic or antagonistic activity Grant 7,319,110 - Lange , et al. January 15, 2	2008-01-15
Azaindole Derivatives With A Combination Of Partial Nicotinic Acetyl-choline Receptor Agonism And Dopamine Reuptake Inhibition App 20080009514 - STOIT; Axel ; et al.	2008-01-10
1 H-imidazole Derivatives As Cannabinoid Receptor Modulators App 20070281974 - Lange; Josephus H.M. ; et al.	2007-12-06
Sulphur Containing Pyrazole Derivatives As Selective Cannabinoid Cb1 Receptor Antagonists App 20070281973 - Lange; Josephus H.M. ; et al.	2007-12-06
Piperazine and piperidine compounds Grant 7,297,699 - Feenstra , et al. November 20, 2	2007-11-20
Muscarinic Agonists To Treat Impulse Control Disorders App 20070259859 - De Bruin; Natasja M.W.J. ; et al.	2007-11-08
4,5-Dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activity App 20070259884 - Lange; Josephus H.M. ; et al.	2007-11-08
1H-imidazole derivatives as cannabinoid receptor modulators Grant 7,271,189 - Lange , et al. September 18, 2	2007-09-18
Phenypiperazine Derivatives With A Combination Of Partial Dopamine-d2 Receptor Agonism And Serotonin Reuptake Inhibition App 20070142397 - Feenstra; Roelof W. ; et al.	2007-06-21
Imidazoline derivatives having CB1-antagonistic activity App 20070135492 - Lange; Josephus H.M. ; et al.	2007-06-14
Neurotensin active 2,3,diaryl-pyrazolidine derivatives Grant 7,186,741 - Feenstra , et al. March 6, 2	2007-03-06
Imidazoline derivatives having CB.sub.1-antagonistic activity Grant 7,173,044 - Lange , et al. February 6, 2	2007-02-06
New phenylpiperazines App 20060293313 - Hes; Roelof Van ; et al.	2006-12-28
Phenylpiperazine derivatives with a combination of partial dopamine-D2 receptor agonism and serotonin reuptake inhibition App 20060247256 - Feenstra; Roelof W. ; et al.	2006-11-02
Imidazoline derivatives having CB1-antagonistic activity App 20060241152 - Lange; Josephus H.M. ; et al.	2006-10-26
1H-imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1-antagonistic activity Grant 7,109,216 - Kruse , et al. September 19, 2	2006-09-19
Phenylpiperazines Grant 7,067,513 - Van Hes , et al. June 27, 2	2006-06-27
Phenylpiperazine derivatives with a combination of partial dopamine-D2 receptor agonism and serotonin reuptake inhibition App 20060122190 - Feenstra; Roelof W. ; et al.	2006-06-08
Aryloxyethylamine and phenylpiperazine derivatives with a combination of partial dopamine-D2 receptor agonism and serotonin reuptake inhibition App 20060122247 - Feenstra; Roelof W. ; et al.	2006-06-08
Phenylpiperazine derivatives with a combination of partial dopamine-D2 receptor agonism and serotonin reuptake inhibition App 20060122189 - Feenstra; Roelof W. ; et al.	2006-06-08
Phenylpiperazines with a combination of affinity for dopamine-D2 receptors and serotonin reuptake sites App 20060122177 - Hes; Roelof van ; et al.	2006-06-08
Benzdioxane piperazine derivatives with a combination of affinity for dopamine-D2 receptors and serotonin reuptake sites App 20060122175 - Hes; Roelof van ; et al.	2006-06-08
Tetrahydropyridin-4-yl indoles with a combination of affinity for dopamine-D2 receptors and serotonin reuptake sites App 20060122206 - Hes; Roelof van ; et al.	2006-06-08
New piperazine and piperidine compounds App 20060089366 - Feenstra; Roelof W. ; et al.	2006-04-27
4,5-Dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activity Grant 6,974,810 - Lange , et al. December 13, 2	2005-12-13
Tetrasubstituted imidazole derivatives as cannabinoid CB1 receptor modulators with a high CB1/CB2 receptor subtype selectivity App 20050267161 - Lange, Josephus H.M. ; et al.	2005-12-01
Imidazoline derivatives having CB1-antagonistic activity App 20050187259 - Lange, Josephus H.M. ; et al.	2005-08-25
1,3,5-trisubstituted 4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity App 20050171179 - Lange, Josephus H.M. ; et al.	2005-08-04
Piperazine and piperidine compounds Grant 6,911,448 - Feenstra , et al. June 28, 2	2005-06-28
1H-imidazole derivatives as cannabinoid receptor modulators App 20050137197 - Lange, Josephus H.M. ; et al.	2005-06-23
Thiazole derivatives as cannabinoid receptor modulators App 20050065189 - Lange, Josephus H.M. ; et al.	2005-03-24
1 H-imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1-antagonistic activity App 20050054679 - Kruse, Cornelis G. ; et al.	2005-03-10
Thiazole derivatives having cb1-antagonistic, agonistic or partial agonistic activity App 20040266841 - Lange, Josephus H.M. ; et al.	2004-12-30
Novel 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic activity App 20040248944 - Kruse, Cornelis G ; et al.	2004-12-09
Phenylpiperazines Grant 6,828,325 - Feenstra , et al. December 7, 2	2004-12-07
Neurotensin active 2,3,diaryl-pyrazolidine derivatives App 20040242493 - Feenstra, Roelof W. ; et al.	2004-12-02
1H-imidazole derivatives having cb1 agonistic, cb1 partial agonistic or cb1 antagonistic activity App 20040235854 - Kruse, Cornelis G. ; et al.	2004-11-25
Piperazine and piperidine compounds Grant 6,780,864 - Feenstra , et al. August 24, 2	2004-08-24
1H-1,2,4-triazole-3-carboxamide derivatives having cannabinoid-CB1 receptor agonistic, partial agonistic, inverse agonistic or antagonistic activity App 20040106614 - Lange, Josephus H. M. ; et al.	2004-06-03
4,5-Dihydro-1h-pyrazole derivatives having potent cb1-antagonistic activity App 20040106800 - Lange, Josephus H.M. ; et al.	2004-06-03
Phenylpiperazines App 20030162791 - Feenstra, Roelof W ; et al.	2003-08-28
Piperazine and piperidine compounds App 20030119849 - Feenstra, Roelof W. ; et al.	2003-06-26
Benzisoxazole derivatives having d4-antagonistic activity Grant 6,335,326 - Den Hartog , et al. January 1, 2	2002-01-01
4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity App 20010053788 - Lange, Josephus H. M. ; et al.	2001-12-20
Bibyclic heteroacrylpiperazine derivatives having psychotropic activity, and pharmaceutical compositions containing these derivatives Grant 5,424,313 - Hartog , et al. June 13, 1	1995-06-13
Method of treating psychotropic conditions employing substituted piperazine compounds Grant 4,782,061 - Kruse , et al. November 1, 1	1988-11-01
Phenyl-substituted (N-piperazinyl) methylazoles for treating affections in the central nervous system Grant 4,772,604 - van Wijngaarden , et al. September 20, 1	1988-09-20