Patent | Date |
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Solid forms of n-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide Grant 11,291,662 - Hurter , et al. April 5, 2 | 2022-04-05 |
Solid Forms of (R)-1(2,2-Difluorobenzo[D][1,3]Dioxol-5-yl)-N-(1-(2,3-Dihydroxypropyl)-6-- Fluoro-2-(1-Hydroxy-2-Methylpropan-2-yl)-1H-Indol-5-yl)Cyclopropanecarboxa- mide App 20210340128 - Keshavarz-Shokri; Ali ;   et al. | 2021-11-04 |
Solid Forms Of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide App 20210251978 - Hurter; Patricia ;   et al. | 2021-08-19 |
Solid forms of (R)-1(2,2-difluorobenzo[d][1,3]dioxol-5-yl)-N-(1-(2,3-dihydroxypropyl)-6-- fluoro-2-(1-hydroxy-2-methylpropan-2-yl)-1H-indol-5-yl)cyclopropanecarboxa- mide Grant 10,906,891 - Keshavarz-Shokri , et al. February 2, 2 | 2021-02-02 |
Solid Forms Of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- Methylpyridin-2-yl) Benzoic Acid App 20200377484 - Keshavarz-Shokri; Ali ;   et al. | 2020-12-03 |
Solid Forms Of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide App 20200352930 - Hurter; Patricia ;   et al. | 2020-11-12 |
Solid forms of 3-(6-(1-(2,2-difluorobenzo[D][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- methylpyridin-2-yl) benzoic acid Grant 10,597,384 - Keshavarz-Shokri , et al. | 2020-03-24 |
Solid forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide Grant 10,537,565 - Hurter , et al. Ja | 2020-01-21 |
Solid Forms of (R)-1(2,2-Difluorobenzo[D][1,3]Dioxol-5-yl)-N-(1-(2,3-Dihydroxypropyl)-6-- Fluoro-2-(1-Hydroxy-2-Methylpropan-2-y App 20190270728 - Keshavarz-Shokri; Ali ;   et al. | 2019-09-05 |
Solid Forms Of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide App 20190070162 - Hurter; Patricia ;   et al. | 2019-03-07 |
Pharmaceutical Compositions And Administrations Thereof App 20190038615 - Van Goor; Fredrick F. ;   et al. | 2019-02-07 |
Solid forms of (R)-1(2,2-difluorobenzo[D][1,3]dioxol-5-yl)-N-(1-(2,3-dihydroxypropyl)-6-- fluoro-2-(1-hydroxy-2-methylpropan-2-yl)-1H-indol-5-yl)cyclopropanecarboxa- mide Grant 10,081,621 - Keshavarz-Shokri , et al. September 25, 2 | 2018-09-25 |
Pharmaceutical Compositions And Administrations Thereof App 20180153874 - Van Goor; Fredrick F. ;   et al. | 2018-06-07 |
Solid Forms Of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- Methylpyridin-2-yl) Benzoic Acid App 20180127398 - Keshavarz-Shokri; Ali ;   et al. | 2018-05-10 |
Solid forms of N[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline-- 3-carboxamide Grant 9,931,334 - Hurter , et al. April 3, 2 | 2018-04-03 |
Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- methylpyridin-2-yl) benzoic acid Grant 9,840,499 - Keshavarz-Shokri , et al. December 12, 2 | 2017-12-12 |
Solid Forms Of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide App 20170231970 - Hurter; Patricia ;   et al. | 2017-08-17 |
Solid forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide Grant 9,670,163 - Hurter , et al. June 6, 2 | 2017-06-06 |
Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- methylpyridin-2-yl) benzoic acid Grant 9,434,717 - Keshavarz-Shokri , et al. September 6, 2 | 2016-09-06 |
Solid Forms Of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide App 20160229806 - Hurter; Patricia ;   et al. | 2016-08-11 |
Solid Forms Of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- Methylpyridin-2-yl) Benzoic Acid App 20160221995 - Keshavarz-Shokri; Ali ;   et al. | 2016-08-04 |
Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- methylpyridin-2-yl)benzoic acid Grant 9,314,455 - Keshavarz-Shokri , et al. April 19, 2 | 2016-04-19 |
Pharmaceutical Compositions And Administrations Thereof App 20160067239 - Van Goor; Fredrick F. ;   et al. | 2016-03-10 |
Solid Forms Of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- Methylpyridin-2-yl) Benzoic Acid App 20160052916 - Keshavarz-Shokri; Ali ;   et al. | 2016-02-25 |
Pharmaceutical Compositions and Administrations Thereof App 20160022664 - Van Goor; Fredrick F. ;   et al. | 2016-01-28 |
Pharmaceutical Compositions and Administrations Thereof App 20160022665 - Van Goor; Fredrick F. ;   et al. | 2016-01-28 |
Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- methylpyridin-2-yl) benzoic acid Grant 9,150,552 - Keshavarz-Shokri , et al. October 6, 2 | 2015-10-06 |
Solid forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide Grant 9,139,530 - Hurter , et al. September 22, 2 | 2015-09-22 |
Solid Forms of (R)-1(2,2-Difluorobenzo[D][1,3]Dioxol-5-yl)-N-(1-(2,3-Dihydroxypropyl)-6-- Fluoro-2-(1-Hydroxy-2-Methylpropan-2-yl)-1H-Indol-5-yl)Cyclopropanecarboxa- mide App 20150203478 - Keshavarz-Shokri; Ali ;   et al. | 2015-07-23 |
Solid Forms of 3-(6-(1-(2,2-Difluorobenzo[D][1,3]Dioxol-5-yl)Cyclopropanecarboxamido)-3-- Methylpyridin-2-yl)Benzoic Acid App 20150196539 - Keshavarz-Shokri; Ali ;   et al. | 2015-07-16 |
Pharmaceutical Compositions And Administrations Thereof App 20150164883 - Van Goor; Fredrick F. ;   et al. | 2015-06-18 |
Pharmaceutical Compositions and Administrations Thereof App 20150164881 - Van Goor; Fredrick F. ;   et al. | 2015-06-18 |
Solid forms of (R)-1(2,2-difluorobenzo[D][1,3]dioxol-5-YL)-N-(1-(2,3-dihydroxypropyl-6-f- luoro-2-(1-hydroxy-2-methylpropan-2-YL)-1H-indol-5-YL)-cyclopropanecarboxa- mide Grant 9,051,303 - Keshavarz-Shokri , et al. June 9, 2 | 2015-06-09 |
Solid forms of gyrase inhibitor (R)-1-ethyl-3-[6-fluoro-5-[2-(1-hydroxy-1-methyl-ethyl)pryimidin-5-yl]-7-- (tetrahydrofuran-2-yl)-1H-benzimidazol-2-yl]urea Grant 9,040,542 - Shannon , et al. May 26, 2 | 2015-05-26 |
Pharmaceutical Compositions And Administrations Thereof App 20150141459 - Van Goor; Fredrick F. ;   et al. | 2015-05-21 |
Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- methylpyridin-2-yl)benzoic acid Grant 8,969,574 - Keshavarz-Shokri , et al. March 3, 2 | 2015-03-03 |
Solid Forms of (R)-1(2,2-Difluorobenzo[D][1,3]Dioxol-5-yl)-N-(1-(2,3-Dihydroxypropyl-6-F- luoro-2-(1-Hydroxy-2-Methylpropan-2-yl)-1H-lndol-5-yl)-Cyclopropanecarboxa- mide App 20150005344 - Keshavarz-Shokri; Ali ;   et al. | 2015-01-01 |
Solid Forms Of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- Methylpyridin-2-yl) Benzoic Acid App 20140371275 - Keshavarz-Shokri; Ali ;   et al. | 2014-12-18 |
Solid Forms Of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide App 20140329855 - Arekar; Sneha G. ;   et al. | 2014-11-06 |
Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxo1-5-yl) cyclopropanecarboxamido)-3-methylpyridin-2-yl) benzoic acid Grant 8,846,718 - Keshavarz-Shokri , et al. September 30, 2 | 2014-09-30 |
Solid Forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide App 20140242172 - Hurter; Patricia ;   et al. | 2014-08-28 |
Solid forms of (R)-1(2,2-difluorobenzo[D][1,3]dioxo1-5-yl)-N-(1-(2,3-dihydroxypropyl-6-f- luoro-2-(1-hydroxy-2-methylpropan2-yl)-1H-Indol-5-yl)-Cyclopropanecarboxam- ide Grant 8,802,868 - Keshavarz-Shokri , et al. August 12, 2 | 2014-08-12 |
Solid Forms of 3-(6-(1-(2,2-Difluorobenzo[D][1,3]Dioxol-5-yl)Cyclopropanecarboxamido)-3-- Methylpyridin-2-yl)Benzoic Acid App 20140221430 - KESHAVARZ-SHOKRI; Ali ;   et al. | 2014-08-07 |
Solid forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide Grant 8,785,476 - Arekar , et al. July 22, 2 | 2014-07-22 |
Solid forms of N-(4-(7-azabicyclo[2.2,1]heptan-7-yl)-2-trifluoromethyl)phenyl)-4-oxo-5-(- trifluoromethyl)-1,4-dihydroquinoline-3-carboxamide Grant 8,741,922 - Zhang , et al. June 3, 2 | 2014-06-03 |
Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- methylpyridin-2-yl)benzoic acid Grant 8,742,122 - Keshavarz-Shokri , et al. June 3, 2 | 2014-06-03 |
Solid Forms of N-(4-(7-azabicyclo[2.2.1]heptan-7-yl)-2-(trifluoromethyl)phenyl)-4-oxo-5-- (trifluoromethyl)-1,4-dihyroquinoline-3-carboxamide App 20140113933 - Zhang; Beili ;   et al. | 2014-04-24 |
Solid forms of 3-(6-(1-(2,2-difluorobenzo[D][1,3]dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic acid Grant 8,653,103 - Keshavarz-Shokri , et al. February 18, 2 | 2014-02-18 |
Solid Forms of 3-(6-(1-(2,2-Difluorobenzo[D][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- methylpyridin-2-yl) Benzoic Acid App 20140011846 - Keshavarz-Shokri; Ali ;   et al. | 2014-01-09 |
Pharmaceutical Compositions And Administrations Thereof App 20130338188 - Van Goor; Fredrick F. ;   et al. | 2013-12-19 |
Solid Forms Of Gyrase Inhibitor (r)-1-ethyl-3-[5-[2-(1-hydroxy-1-methyl-ethyl)pyrimidin-5-yl]-7-(tetrahyd- Rofuran-2-yl]-1h-benzimidazol-2-yl]urea App 20130317222 - Shannon; Dean ;   et al. | 2013-11-28 |
Solid Forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide App 20130317060 - Hurter; Patricia ;   et al. | 2013-11-28 |
Solid Forms of 3-(6-(1-(2,2-Difluorobenzo[D][1,3]Dioxol-5-yl)Cyclopropanecarboxamido)-3-- Methylpyridin-2-yl)Benzoic Acid App 20130296379 - Keshavarz-Shokri; Ali ;   et al. | 2013-11-07 |
Solid Forms Of Gyrase Inhibitor (r)-1-ethyl-3-[6-fluoro-5-[2-(1-hydroxy-1-methyl-ethyl)pyrimidin-5-yl]-7-- (tetrahydrofuran-2-yl)-1h-benzimidazol-2-yl]urea App 20130267540 - Shannon; Dean ;   et al. | 2013-10-10 |
Solid Forms of N-(4-(7-azabicyclo[2.2.1]heptan-7-yl)-2-(trifluorormethyl)phenyl)-4-oxo-5- -(trifluoromethyl)-1,4-dihyroquinoline-3-carboxamide App 20130231368 - Zhang; Beili ;   et al. | 2013-09-05 |
Solid forms of 3-(6-(1-(2,2-difluorobenzo[D][1,3]dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic acid Grant 8,507,687 - Keshavarz-Shokri , et al. August 13, 2 | 2013-08-13 |
Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic acid Grant 8,507,534 - Keshavarz-Shokri , et al. August 13, 2 | 2013-08-13 |
Solid forms of gyrase inhibitor (R)-1-ethyl-3-[5-[2-(1-hydroxy-1-methyl-ethyl)pyrimidin-5-YL]-7-(tetrahyd- rofuran-2-yl)-1H-benzimidazol-2-YL]urea Grant 8,481,552 - Shannon , et al. July 9, 2 | 2013-07-09 |
Solid forms of gyrase inhibitor (R)-1-ethyl-3-[6-fluoro-5-[2-(1-hydroxy-1-methyl-ethyl)pyrimidin-5-yl]-7-- (tetrahydrofuran-2-yl)-1H-benzimidazol-2-yl]urea Grant 8,476,281 - Shannon , et al. July 2, 2 | 2013-07-02 |
Solid forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide Grant 8,471,029 - Arekar , et al. June 25, 2 | 2013-06-25 |
Pharmaceutical Compositions And Administrations Thereof App 20130158071 - Van Goor; Fredrick F. ;   et al. | 2013-06-20 |
Solid Forms of (R)-1(2,2-Difluorobenzo[D][1,3]Dioxol-5-yl)-N-(1-(2,3-Dihydroxypropyl-6-F- luoro-2-(1-Hydroxy-2-Methylpropan-2-yl)-1H-Indol-5-yl)-Cyclopropanecarboxa- mide App 20130143918 - Keshavarz-Shokri; Ali ;   et al. | 2013-06-06 |
Pharmaceutical Compositions And Administrations Thereof App 20130143919 - Van Goor; Fredrick F. ;   et al. | 2013-06-06 |
Solid Forms Of N-(4-(7-azabicyclo[2.2.1]heptan-7-yl)-2-trifluoromethyl)phenyl)-4-oxo-5-(- Trifluoromethyl)-1,4-dihydroquinoline-3-carboxamide App 20130137722 - Zhang; Beili ;   et al. | 2013-05-30 |
Pharmaceutical Compositions And Administrations Thereof App 20130131107 - Van Goor; Fredrick F. ;   et al. | 2013-05-23 |
Solid forms of N-(4-(7-azabicyclo[2.2.1]heptan-7-yl)-2-(trifluorormethyl)phenyl)-4-oxo-5- -(trifluoromethyl)-1,4-dihyroquinoline-3-carboxamide Grant 8,436,014 - Zhang , et al. May 7, 2 | 2013-05-07 |
Solid Forms Of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl) Cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic Acid App 20130085158 - KESHAVARZ-SHOKRI; ALI ;   et al. | 2013-04-04 |
Solid forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide Grant 8,410,274 - Hurter , et al. April 2, 2 | 2013-04-02 |
Solid Forms Of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide App 20130079367 - Arekar; Sneha G. ;   et al. | 2013-03-28 |
Solid forms of N-(4-(7-Azabicyclo[2.2.1]Heptan-7-yl)-2-Trifluoromethyl)Phenyl)-4-Oxo-5-(- Trifluoromethyl)-1,4-Dihydroquinoline-3-Carboxamide Grant 8,389,727 - Zhang , et al. March 5, 2 | 2013-03-05 |
Solid Forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide App 20130018071 - Arekar; Sneha G. ;   et al. | 2013-01-17 |
Solid Forms Of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl) Cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic Acid App 20120277268 - Keshavarz-Shokri; Ali ;   et al. | 2012-11-01 |
Solid Forms Of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide App 20120214841 - Hurter; Patricia ;   et al. | 2012-08-23 |
Solid Forms Of Gyrase Inhibitor (r)-1-ethyl-3-[5-[2-(1-hydroxy-methyl-ethyl)pyrimidin-5-yl]-7-(tetrahydro- Furan-2-yl)-1h-benzimidazol-2-yl]urea App 20120184741 - Shannon; Dean ;   et al. | 2012-07-19 |
Solid Forms Of Gyrase Inhibitor (r)-1-ethyl-3-[6-fluoro-5-[2-(1-hydroxy-1-methyl-ethyl)pyrimidin-5-yl]-7-- (tetrahydrofuran-2-yl)-1h-benzimidazol-2-yl]urea App 20120184564 - Shannon; Dean ;   et al. | 2012-07-19 |
Solid Forms Of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl) Cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic Acid App 20110263654 - Keshavarz-Shokri; Ali ;   et al. | 2011-10-27 |
Solid Forms Of (r)-1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)-n-(1-(2,3-dihydroxypropyl)-6- -fluoro-2-(1-hydroxy-2-methylpropan-2-yl)-1h-indol-5-yl) Cyclopropanecarboxamide App 20110251253 - Keshavarz-Shokri; Ali ;   et al. | 2011-10-13 |
Solid Forms Of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide App 20110230519 - Arekar; Sneha G. ;   et al. | 2011-09-22 |
Solid Forms of N-(4-(7-Azabicyclo[2.2.1]Heptan-7-yl)-2-Trifluoromethyl)Phenyl)-4-Oxo-5-(- Trifluoromethyl)-1,4-Dihydroquinoline-3-Carboxamide App 20110123449 - Zhang; Beili ;   et al. | 2011-05-26 |
Solid forms of N-[2,4-BIS(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline- -3-carboxamide App 20110064811 - Hurter; Patricia ;   et al. | 2011-03-17 |
Solid Forms Of N-(4-(7-azabicyclo[2.2.1]heptan-7-yl)-2-(trifluorormethyl)phenyl)-4-oxo-5- -(trifluoromethyl)-1,4-dihyroquinoline-3-carboxamide App 20100130547 - Zhang; Beili ;   et al. | 2010-05-27 |
Solid Forms Of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl) Cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic Acid App 20090170905 - Keshavarz-Shokri; Ali ;   et al. | 2009-07-02 |