Patent | Date |
---|
N3-cyclically Substituted Thienouracils And Use Thereof App 20200016159 - HAERTER; Michael ;   et al. | 2020-01-16 |
Heterocyclylmethyl-thienouracile as antagonists of the adenosine-A2B-receptor Grant 10,428,083 - Harter , et al. October 1, 2 | 2019-10-01 |
4-aryl-N-phenyl-1,3,5-triazin-2-amines containing a sulfoximine group Grant 9,962,389 - Lucking , et al. May 8, 2 | 2018-05-08 |
Heterocyclylmethyl-thienouracile As Antagonists Of The Adenosine-a2b-receptor App 20180065981 - HARTER; Michael ;   et al. | 2018-03-08 |
Fluorinated benzofuranyl-pyrimidine derivatives containing a sulfone group Grant 9,902,716 - Kosemund , et al. February 27, 2 | 2018-02-27 |
Fluorinated benzofuranyl-pyrimidine derivatives containing a sulfoximine group Grant 9,884,849 - Kosemund , et al. February 6, 2 | 2018-02-06 |
5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfoximine group Grant 9,877,954 - Lucking , et al. January 30, 2 | 2018-01-30 |
5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfone group Grant 9,856,242 - Kosemund , et al. January 2, 2 | 2018-01-02 |
Sulfoximine substituted 5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives and their use as CDK9 kinase inhibitors Grant 9,770,445 - Kosemund , et al. September 26, 2 | 2017-09-26 |
Fluorinated Benzofuranyl-pyrimidine Derivatives Containing A Suflone Group App 20170226092 - KOSEMUND; Dirk ;   et al. | 2017-08-10 |
Fluorinated Benzofuranyl-pyrimidine Derivatives Containing A Sulfoximine Group App 20170217938 - KOSEMUND; Dirk ;   et al. | 2017-08-03 |
4-aryl-n-phenyl-1,3,5-triazin-2-amines Containing A Sulfoximine Group App 20170217949 - LUCKING; Ulrich ;   et al. | 2017-08-03 |
5-fluoro-n-(pyridin-2-yl)pyridin-2-amine Derivatives Containing A Sulfoximine Group App 20170202815 - LUCKING; Ulrich ;   et al. | 2017-07-20 |
N-(pyridin-2-yl)pyrimidin-4-amine derivatives containing a sulfone group Grant 9,708,293 - Lucking , et al. July 18, 2 | 2017-07-18 |
Triazolopyridines Grant 9,676,766 - Schulze , et al. June 13, 2 | 2017-06-13 |
Substituted triazolopyridines Grant 9,670,202 - Schirok , et al. June 6, 2 | 2017-06-06 |
4-aryl-N-phenyl-1,3,5-triazin-2-amines containing a sulfoximine group Grant 9,669,034 - Lucking , et al. June 6, 2 | 2017-06-06 |
5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfone group Grant 9,670,161 - Lucking , et al. June 6, 2 | 2017-06-06 |
Substituted triazolopyridines and their use as TTK inhibitors Grant 9,663,510 - Schulze , et al. May 30, 2 | 2017-05-30 |
N-(pyridin-2-yl)pyrimidin-4-amine derivatives containing a sulfoximine group Grant 9,650,361 - Lucking , et al. May 16, 2 | 2017-05-16 |
5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfoximine group Grant 9,650,340 - Lucking , et al. May 16, 2 | 2017-05-16 |
Prodrug derivatives of substituted triazolopyridines Grant 9,586,958 - Schulze , et al. March 7, 2 | 2017-03-07 |
Substituted triazolopyridines Grant 9,555,022 - Schulze , et al. January 31, 2 | 2017-01-31 |
Thienopyrimidines Grant 9,540,392 - Kettschau , et al. January 10, 2 | 2017-01-10 |
5-fluoro-n-(pyridin-2-yl)pyridin-2-amine Derivatives Containing A Sulfone Group App 20170001989 - KOSEMUND; Dirk ;   et al. | 2017-01-05 |
4-(ortho)-fluorophenyl-5-fluoropyrimidin-2-yl amines containing a sulfoximine group Grant 9,499,492 - Lucking , et al. November 22, 2 | 2016-11-22 |
Imidazopyrazines Grant 9,468,642 - Klar , et al. October 18, 2 | 2016-10-18 |
Substituted Triazolopyridines App 20160297811 - SCHIROK; Hartmut ;   et al. | 2016-10-13 |
Prodrug Derivatives Of Substituted Triazolopyridines App 20160207915 - Schulze; Volker ;   et al. | 2016-07-21 |
Novel Compounds For The Treatment Of Cancer App 20160207928 - SCHULZE; Volker ;   et al. | 2016-07-21 |
Substituted benzimidazoles Grant 9,388,140 - Klar , et al. July 12, 2 | 2016-07-12 |
Substituted Thienopyrimidines And Pharmaceutical Use Thereof App 20160159816 - KETTSCHAU; Georg ;   et al. | 2016-06-09 |
Sulfoximine Substituted 5-fluoro-n-(pyridin-2-yl)pyridin-2-amine Derivatives And Their Use As Cdk9 Kinase Inhibitors App 20160143893 - KOSEMUND; Dirk ;   et al. | 2016-05-26 |
Substituted benzothienopyrimidines Grant 9,296,757 - Klar , et al. March 29, 2 | 2016-03-29 |
Substituted imidazo[1,2-a]pyrazines as MPS-1 inhibitors Grant 9,284,317 - Koppitz , et al. March 15, 2 | 2016-03-15 |
Substituted imidazopyridazines Grant 9,255,100 - Klar , et al. February 9, 2 | 2016-02-09 |
6-thio-substituted imidazo[1,2-a]pyrazines as Mps-1 inhibitors Grant 9,212,184 - Koppitz , et al. December 15, 2 | 2015-12-15 |
Substituted imidazopyrazines Grant 9,199,999 - Klar , et al. December 1, 2 | 2015-12-01 |
4-(ortho)-fluorophenyl-5-fluoropyrimidin-2-yl Amines Containing A Sulfoximine Group App 20150291537 - Lucking; Ulrich ;   et al. | 2015-10-15 |
N-(pyridin-2-yl)pyrimidin-4-amine Derivatives Containing A Sulfoximine Group App 20150291559 - Lucking; Ulrich ;   et al. | 2015-10-15 |
5-fluoro-n-(pyridin-2-yl)pyridin-2-amine Derivatives Containing A Sulfoximine Group App 20150291528 - Lucking; Ulrich ;   et al. | 2015-10-15 |
N-(pyridin-2-yl)pyrimidin-4-amine Derivatives Containing A Sulfone Group App 20150274695 - Lucking; Ulrich ;   et al. | 2015-10-01 |
5-fluoro-n-(pyridin-2-yl)pyridin-2-amine Derivatives Containing A Sulfone Group App 20150274666 - Lucking; Ulrich ;   et al. | 2015-10-01 |
4-(ortho)-fluorophenyl-5-fluoropyrimidin-2-yl Amines Containing A Sulfone Group App 20150259300 - Lucking; Ulrich ;   et al. | 2015-09-17 |
Disubstituted 5-fluoro pyrimidine derivatives containing a sulfoximine group Grant 9,133,171 - Lucking , et al. September 15, 2 | 2015-09-15 |
Disubstituted 5-fluoro-pyrimidines Grant 9,108,926 - Lucking , et al. August 18, 2 | 2015-08-18 |
Substituted Triazolopyridines And Their Use As Ttk Inhibitors App 20150210683 - Schulze; Volker ;   et al. | 2015-07-30 |
Substituted Benzothienopyrimidines App 20150152121 - Klar; Ulrich ;   et al. | 2015-06-04 |
Thienopyrimidines App 20150133425 - Kettschau; Georg ;   et al. | 2015-05-14 |
Substituted Pyrrolopyrimidines App 20150133426 - Klar; Ulrich ;   et al. | 2015-05-14 |
Disubstituted 5-fluoro Pyrimidine Derivatives Containing A Sulfoximine Group App 20150005329 - Lucking; Ulrich ;   et al. | 2015-01-01 |
Substituted 4-Aryl-N-phenyl-1,3,5-triazin-2-amines Grant 8,916,557 - Lucking , et al. December 23, 2 | 2014-12-23 |
4-aryl-n-phenyl-1,3,5-triazin-2-amines Containing A Sulfoximine Group App 20140315906 - Lucking; Ulrich ;   et al. | 2014-10-23 |
Substituted Benzimidazoles App 20140302010 - Klar; Ulrich ;   et al. | 2014-10-09 |
Sulphone-substituted quinazoline derivatives as immuno-modulators, their preparation and use as medicaments Grant 8,841,311 - Buchmann , et al. September 23, 2 | 2014-09-23 |
Disubstituted 5-fluoro-pyrimidines App 20140228387 - Lucking; Ulrich ;   et al. | 2014-08-14 |
6 Substituted Imidazopyrazines For Use As Mps-1 And Tkk Inhibitors In The Treatment Of Hyperproliferative Disorders App 20140187548 - Koppitz; Marcus ;   et al. | 2014-07-03 |
6-substituted Imidazopyrazines For Use As Mps-1 And Tkk Inhibitors In The Treatment Of Hyperproliferative Disorders App 20140135319 - Koppitz; Marcus ;   et al. | 2014-05-15 |
Triazolopyridines App 20140120087 - Schulze; Volker ;   et al. | 2014-05-01 |
Substituted 4-aryl-n-phenyl-1,3,5-triazin-2-amines App 20140045852 - Lucking; Ulrich ;   et al. | 2014-02-13 |
Substituted Imidazopyridazines App 20130338133 - Klar; Ulrich ;   et al. | 2013-12-19 |
Imidazopyrazines For Use As Mps-1 And Tkk Inhibitors In The Treatment Hyperproliferative Disorders App 20130303532 - Koppitz; Marcus ;   et al. | 2013-11-14 |
6-thio-substituted Imidazopyrazines For Use As Mps-1 And Tkk Inhibitors In The Treatment Of Hyperproliferative Disorders App 20130281460 - Koppitz; Marcus ;   et al. | 2013-10-24 |
Substituted 6-imidazopyrazines For Use As Mps-1 And Tkk Inhibitors In The Treatment Of Hyperproliferative Disorders App 20130267527 - Koppitz; Marcus ;   et al. | 2013-10-10 |
Substituted triazolopyridines Grant 8,551,980 - Schulze , et al. October 8, 2 | 2013-10-08 |
6,7-dihydro-5h-benzo[7]annulene Derivatives, Process For Preparation Thereof, Pharmaceutical Preparations Comprising Them, And The Use Thereof For Production Of Medicaments App 20130252890 - Wintermantel; Tim ;   et al. | 2013-09-26 |
Substituted Imidazopyrazines App 20130210815 - Klar; Ulrich ;   et al. | 2013-08-15 |
Imidazopyrazines App 20130195848 - Klar; Ulrich ;   et al. | 2013-08-01 |
2-substituted estra-1,3,5(10)-triene-3-yl sulfamate with an anti-tumor action Grant 8,492,570 - Hillisch , et al. July 23, 2 | 2013-07-23 |
Substituted Triazolopyridines App 20130156756 - Schulze; Volker ;   et al. | 2013-06-20 |
Triazolopyridine Derivatives App 20130121994 - Koppitz; Marcus ;   et al. | 2013-05-16 |
Triazolopyridines App 20120328610 - Schulze; Volker ;   et al. | 2012-12-27 |
Substituted Triazolopyridines App 20120328611 - Schulze; Volker ;   et al. | 2012-12-27 |
Sulphone-substituted quinazoline derivatives as immuno-modulators, their preparation and use as medicaments App 20110166168 - Buchmann; Bernd ;   et al. | 2011-07-07 |
Metasubstituted Thiazolidinones, Their Manufacture And Use As A Drug App 20100048891 - SCHULZE; Klause ;   et al. | 2010-02-25 |
2-substituted Estra-1,3,5(10)-triene-3-yl Sulfamate With An Anti-tumour Action App 20090221841 - HILLISCH; Alexander ;   et al. | 2009-09-03 |
Azaindoles As Inhibitors Of Soluble Adenylate Cyclase App 20090098189 - BUCHMANN; Bernd ;   et al. | 2009-04-16 |
Thiazolidinones, their production and use as pharmaceutical agents Grant 7,511,059 - Schulze , et al. March 31, 2 | 2009-03-31 |
Arylmethylene Substituted N-Acyl-Beta-Amino Alcohols App 20090082372 - WORTMANN; Lars ;   et al. | 2009-03-26 |
Chk-, Pdk- and Akt-inhibitory pyrimidines, their production and use as pharmaceutical agents Grant 7,504,410 - Bryant , et al. March 17, 2 | 2009-03-17 |
Arylmethylen Substituted N-acyl-y-aminoalcohols App 20080287493 - Wortmann; Lars ;   et al. | 2008-11-20 |
Inhibitors of soluble adenylate cyclase Grant 7,449,459 - Buchmann , et al. November 11, 2 | 2008-11-11 |
Sulfonyltryptophanols App 20080255117 - WORTMANN; Lars ;   et al. | 2008-10-16 |
2-substituted estra-1,3,5(10)-triene-3-yl sulfamate with an anti-tumour action Grant 7,427,610 - Hillisch , et al. September 23, 2 | 2008-09-23 |
1,2-diarylacetylene Derivatives Of Acyltryptophanols App 20080221195 - Wortmann; Lars ;   et al. | 2008-09-11 |
Bicyclic Acyltryptophanols App 20080207728 - Wortmann; Lars ;   et al. | 2008-08-28 |
9-.alpha.-substituted estratrienes as selectively active estrogens Grant 7,414,043 - Kosemund , et al. August 19, 2 | 2008-08-19 |
Substituted Estratrienes As Selectively Active Estrogens App 20080132476 - KOSEMUND; Dirk ;   et al. | 2008-06-05 |
Inhibitors of soluble adenylate cyclase App 20070259872 - Buchmann; Bernd ;   et al. | 2007-11-08 |
Inhibitors of soluble adenylate cyclase App 20070232605 - Buchmann; Bernd ;   et al. | 2007-10-04 |
Inhibitors of soluble adenylate cyclase App 20070225284 - Buchmann; Bernd ;   et al. | 2007-09-27 |
Prodrugs of ERbeta-selective substances, processes for their preparation and pharmaceutical compositions comprising these compounds App 20070123500 - Mueller; Gerd ;   et al. | 2007-05-31 |
Acyltryptophanols App 20070060573 - Wortmann; Lars ;   et al. | 2007-03-15 |
Metasubstituted thiazolidinones, their manufacture and use as a drug App 20070015759 - Schulze; Volker Klaus ;   et al. | 2007-01-18 |
Thiazolidinones without basic nitrogen, their production and use as pharmaceutical agents App 20070010566 - Prien; Olaf ;   et al. | 2007-01-11 |
New thiazolidinones without basic nitrogen, their production and use as pharmaceutical agents App 20070010565 - Prien; Olaf ;   et al. | 2007-01-11 |
16-Hydroxyestratrienes as selectively active estrogens App 20060270845 - Kuenzer; Hermann ;   et al. | 2006-11-30 |
Thiazolidinones, their production and use as pharmaceutical agents App 20060223833 - Schulze; Volker ;   et al. | 2006-10-05 |
16-hydroxyestratrienes as selectively active estrogens Grant 7,109,360 - Kuenzer , et al. September 19, 2 | 2006-09-19 |
2-Substituted estra-1,3,5(10)-triene-3-yl sulfamate with an anti-tumour action App 20060160782 - Hillisch; Alexander ;   et al. | 2006-07-20 |
Use of ERbeta-selective ligands for regulating fertility and compounds useful therefor App 20050020695 - Hegele-Hartung, Christa ;   et al. | 2005-01-27 |
Chk-, Pdk- and Akt-inhibitory pyrimidines, their production and use as pharmaceutical agents App 20040186118 - Bryant, Judi ;   et al. | 2004-09-23 |
Use of ER.beta.-selective ligands for regulating fertility and compounds useful therefor Grant 6,794,409 - Hegele-Hartung , et al. September 21, 2 | 2004-09-21 |
9-alpha-substituted estratrienes as selectively active estrogens App 20040087565 - Kosemund, Dirk ;   et al. | 2004-05-06 |
19-nor-17.alpha.-pregna-1,3,5(10)-trien-17.beta.-ols with a 21,16.alpha.-lactone ring Grant 6,670,347 - Muller , et al. December 30, 2 | 2003-12-30 |
Therapeutic use of estrogen receptor (ER)beta-selective agonists for triggering somatotropic, organotropic and anticatabolic effects (somatotropic therapy) App 20030130249 - Elger, Walter ;   et al. | 2003-07-10 |
C13-substituted estra-1,3,5,(10)-trien-3-yl sulfamates, methods of preparing same, and pharmaceutical compositions containing these compounds Grant 6,583,130 - Schwarz , et al. June 24, 2 | 2003-06-24 |
Use of ERbeta-selective ligands for regulating fertility and compounds useful therefor App 20030083377 - Hegele-Hartung, Christa ;   et al. | 2003-05-01 |
19-nor-17alpha-pregna-1,3,5 (10) -trien-17beta-ols with a 21, 16alpha-lactone ring App 20020156271 - Muller, Gerd ;   et al. | 2002-10-24 |