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Bicyclic Compounds App 20220298102 - KONRADI; Andrei W. ;   et al. | 2022-09-22 |
Certain Chemical Compositions And Methods Of Use Thereof App 20220289725 - Konradi; Andrei W. ;   et al. | 2022-09-15 |
Bicyclic compounds Grant 11,420,935 - Konradi , et al. August 23, 2 | 2022-08-23 |
Bicyclic compounds Grant 11,384,049 - Konradi , et al. July 12, 2 | 2022-07-12 |
Arginine Gingipain Inhibitors App 20220204457 - Galemmo; Robert A. ;   et al. | 2022-06-30 |
Inhibitors of lysine gingipain Grant 11,332,464 - Konradi , et al. May 17, 2 | 2022-05-17 |
Ketone inhibitors of lysine gingipain Grant 11,325,884 - Konradi , et al. May 10, 2 | 2022-05-10 |
Inhibitors Of Jun N-terminal Kinase App 20220081427 - SHAM; Hing L. ;   et al. | 2022-03-17 |
Benzosulfonyl compounds Grant 11,192,865 - Konradi , et al. December 7, 2 | 2021-12-07 |
Non-fused tricyclic compounds Grant 11,186,554 - Konradi , et al. November 30, 2 | 2021-11-30 |
Aminopyridine Compounds And Methods For The Preparation And Use Thereof App 20210340105 - Konradi; Andrei W. ;   et al. | 2021-11-04 |
Pyridine Derivatives Substituted By Heterocyclic Ring And Amino Group App 20210275510 - KONRADI; Andrei W. ;   et al. | 2021-09-09 |
Oxadiazole Compounds App 20210238154 - KONRADI; Andrei W. ;   et al. | 2021-08-05 |
Aminopyridine compounds and methods for the preparation and use thereof Grant 11,059,786 - Konradi , et al. July 13, 2 | 2021-07-13 |
Ketone Inhibitors Of Lysine Gingipain App 20210053908 - Konradi; Andrei W. ;   et al. | 2021-02-25 |
Inhibitors Of Lysine Gingipain App 20210017167 - Konradi; Andrei W. ;   et al. | 2021-01-21 |
Prodrugs of phenolic TRPV1 agonists Grant 10,851,123 - Husfeld , et al. December 1, 2 | 2020-12-01 |
Benzosulfonyl Compounds App 20200354325 - KONRADI; Andrei W. ;   et al. | 2020-11-12 |
Bicyclic Compounds App 20200347009 - KONRADI; Andrei W. ;   et al. | 2020-11-05 |
Inhibitors Of Jun N-terminal Kinase App 20200277285 - SHAM; Hing L. ;   et al. | 2020-09-03 |
Ketone inhibitors of lysine gingipain Grant 10,730,826 - Konradi , et al. | 2020-08-04 |
Inhibitors of lysine gingipain Grant 10,676,470 - Konradi , et al. | 2020-06-09 |
Aminopyridine Compounds And Methods For The Preparation And Use Thereof App 20200148642 - Konradi; Andrei W. ;   et al. | 2020-05-14 |
Non-fused Tricyclic Compounds App 20200062721 - KONRADI; Andrei W. ;   et al. | 2020-02-27 |
Inhibitors Of Jun N-terminal Kinase App 20200039972 - SHAM; Hing L. ;   et al. | 2020-02-06 |
Inhibitors Of Lysine Gingipain App 20190322659 - Konradi; Andrei W. ;   et al. | 2019-10-24 |
Ketone Inhibitors Of Lysine Gingipain App 20190210960 - Konradi; Andrei W. ;   et al. | 2019-07-11 |
Inhibitors Of Jun N-terminal Kinase App 20190194176 - SHAM; Hing L. ;   et al. | 2019-06-27 |
Prodrugs Of Phenolic Trpv1 Agonists App 20190055272 - HUSFELD; Craig ;   et al. | 2019-02-21 |
Inhibitors Of Jun N-terminal Kinase App 20180037577 - SHAM; Hing L. ;   et al. | 2018-02-08 |
Inhibitors of Jun N-terminal kinase Grant 9,796,706 - Sham , et al. October 24, 2 | 2017-10-24 |
Inhibitors Of Jun N-terminal Kinase App 20170107209 - SHAM; Hing L. ;   et al. | 2017-04-20 |
Inhibitors Of Jun N-terminal Kinase App 20150259330 - SHAM; Hing L. ;   et al. | 2015-09-17 |
Inhibitors of Jun N-terminal kinase Grant 9,073,891 - Sham , et al. July 7, 2 | 2015-07-07 |
Preparation of Polymer Conjugates of Therapeutic, Agricultural, and Food Additive Compounds App 20140073788 - Konradi; Andrei W. ;   et al. | 2014-03-13 |
Multimeric VLA-4 Antagonists Comprising Polymers Moieties App 20130338164 - Konradi; Andrei W. ;   et al. | 2013-12-19 |
Preparation of polymer conjugates of therapeutic, agricultural, and food additive compounds Grant 8,569,426 - Konradi , et al. October 29, 2 | 2013-10-29 |
Inhibitors of Jun N-terminal kinase Grant 8,450,363 - Sham , et al. May 28, 2 | 2013-05-28 |
Inhibitors Of Jun N-terminal Kinase App 20130072494 - SHAM; Hing L. ;   et al. | 2013-03-21 |
Carbamate compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 8,367,688 - Semko , et al. February 5, 2 | 2013-02-05 |
Preparation of Polymer Conjugates of Therapeutic, Agricultural, and Food Additive Compounds App 20130018187 - Konradi; Andrei W. ;   et al. | 2013-01-17 |
N-sulfonamido polycyclic pyrazolyl compounds Grant 8,283,358 - Konradi , et al. October 9, 2 | 2012-10-09 |
Preparation of polymer conjugates of therapeutic, agricultural, and food additive compounds Grant 8,268,935 - Konradi , et al. September 18, 2 | 2012-09-18 |
Multimeric VLA-4 antagonists comprising polymer moieties Grant 8,263,063 - Konradi , et al. September 11, 2 | 2012-09-11 |
Carbamate compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 8,158,642 - Semko , et al. April 17, 2 | 2012-04-17 |
Preparation of polymer conjugates of therapeutic, agricultural, and food additive compounds Grant 8,138,272 - Konradi , et al. March 20, 2 | 2012-03-20 |
Bridged N-Bicyclic Sulfonamido Inhibitors of Gamma Secretase App 20110178119 - Konradi; Andrei W. ;   et al. | 2011-07-21 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,973,044 - Konradi , et al. July 5, 2 | 2011-07-05 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,968,547 - Konradi , et al. June 28, 2 | 2011-06-28 |
Multimeric VLA-4 Antagonists Comprising Polymer Moieties App 20110002876 - Konradi; Andrei W. ;   et al. | 2011-01-06 |
Bridged N-Cyclic Sulfonamido Inhibitors of Gamma Secretase App 20110003802 - Bowers; Simeon ;   et al. | 2011-01-06 |
Inhibitors of Jun N-Terminal Kinase App 20100331335 - Sham; Hing L. ;   et al. | 2010-12-30 |
Pyrimidinyl sulfonamide compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,820,687 - Smith , et al. October 26, 2 | 2010-10-26 |
5-(Arylsulfonyl)-Pyrazolopiperidines App 20100267747 - Ye; Xiaocong Michael ;   et al. | 2010-10-21 |
Carbamate Compounds Which Inhibit Leukocyte Adhesion Mediated By Vla-4 App 20100261715 - Semko; Christopher Michael ;   et al. | 2010-10-14 |
Pyrimidinyl amide compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,763,632 - Semko , et al. July 27, 2 | 2010-07-27 |
Bridged N-cyclic sulfonamido inhibitors of gamma secretase Grant 7,754,712 - Bowers , et al. July 13, 2 | 2010-07-13 |
Alpha amino acid derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 Grant 7,745,454 - Konradi , et al. June 29, 2 | 2010-06-29 |
Heteroaryl, Heterocyclic And Aryl Compounds Which Inhibit Leukocyte Adhesion Mediated By Vla-4 App 20100160343 - Konradi; Andrei W. ;   et al. | 2010-06-24 |
Heteroaryl, Heterocyclic And Aryl Compounds Which Inhibit Leukocyte Adhesion Mediated By Vla-4 App 20100160341 - Konradi; Andrei W. ;   et al. | 2010-06-24 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,741,328 - Konradi , et al. June 22, 2 | 2010-06-22 |
5-(arylsulfonyl)-pyrazolopiperidines Grant 7,732,609 - Ye , et al. June 8, 2 | 2010-06-08 |
Carbamate compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,727,996 - Semko , et al. June 1, 2 | 2010-06-01 |
Carbamate Compounds Which Inhibit Leukocyte Adhesion Mediated By Vla-4 App 20100113434 - Semko; Christopher Michael ;   et al. | 2010-05-06 |
N-sulfonamido Polycyclic Pyrazolyl Compounds App 20100081680 - Konradi; Andrei W. ;   et al. | 2010-04-01 |
Pyrimidinyl Sulfonamide Compounds Which Inhibit Leukocyte Adhesion Mediated By Vla-4 App 20100016345 - Smith; Jenifer ;   et al. | 2010-01-21 |
Methods and compositions for treating rheumatoid arthritis Grant 7,605,166 - Yednock , et al. October 20, 2 | 2009-10-20 |
Pyrimidinyl sulfonamide compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,579,466 - Smith , et al. August 25, 2 | 2009-08-25 |
Composition for and treatment of demyelinating diseases and paralysis by administration of remyelinating agents Grant 7,576,101 - Karlik , et al. August 18, 2 | 2009-08-18 |
Pyrimidinyl Amide Compounds Which Inhibit Leukocyte Adhesion Mediated By Vla-4 App 20090192181 - Semko; Christopher Michael ;   et al. | 2009-07-30 |
Compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,538,215 - Konradi , et al. May 26, 2 | 2009-05-26 |
Pyrimidinyl amide compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,511,052 - Semko , et al. March 31, 2 | 2009-03-31 |
Fused ring heteroaryl and heterocyclic compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,452,912 - Grant , et al. November 18, 2 | 2008-11-18 |
Heterocyclic compounds which inhibit leukocyte adhesion mediated by .alpha..sub.4 integrins Grant 7,427,628 - Konradi , et al. September 23, 2 | 2008-09-23 |
3-(heteroaryl)alanine Derivatives-inhibitors Of Leukocyte Adhesion Mediated By Vla-4 App 20080182850 - Konradi; Andrei W. ;   et al. | 2008-07-31 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,378,529 - Konradi , et al. May 27, 2 | 2008-05-27 |
3-(heteroaryl) alanine derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 Grant 7,365,073 - Konradi , et al. April 29, 2 | 2008-04-29 |
Bridged N-Cyclic Sulfonamido Inhibitors of Gamma Secretase App 20080090817 - Bowers; Simeon ;   et al. | 2008-04-17 |
Bridged N-cyclic sulfonamido inhibitors of gamma secretase Grant 7,345,056 - Bowers , et al. March 18, 2 | 2008-03-18 |
Pyrimidinyl Sulfonamide Compounds Which Inhibit Leukocyte Adhesion Mediated By Vla-4 App 20080058357 - Smith; Jenifer ;   et al. | 2008-03-06 |
Heteroaryl compounds which inhibit leukocyte adhesion mediated by .alpha..sub.4 integrins Grant 7,335,663 - Konradi , et al. February 26, 2 | 2008-02-26 |
Preparation of Polymer Conjugates of Therapeutic, Agricultural, and Food Additive Compounds App 20080031848 - Konradi; Andrei W. ;   et al. | 2008-02-07 |
Fused, Tricyclic Sulfonamide Inhibitors of Gamma Secretase App 20080021056 - Konradi; Andrei W. ;   et al. | 2008-01-24 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,320,960 - Thorsett , et al. January 22, 2 | 2008-01-22 |
Phenylalanine derivatives as alpha 4 integrin inhibitors Grant 7,291,645 - Konradi , et al. November 6, 2 | 2007-11-06 |
5-(Arylsulfonyl)-Pyrazolopiperidines App 20070155753 - Ye; Xiaocong Michael ;   et al. | 2007-07-05 |
Pyrimidinyl amide compounds with inhibit leukocyte adhesion mediated by VLA-4 App 20070142416 - Semko; Christopher Michael ;   et al. | 2007-06-21 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,229,970 - Thorsett , et al. June 12, 2 | 2007-06-12 |
Carbamate compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20070129390 - Semko; Christopher Michael ;   et al. | 2007-06-07 |
Beta-amino acid derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 Grant 7,223,762 - Konradi , et al. May 29, 2 | 2007-05-29 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20070099921 - Konradi; Andrei W. ;   et al. | 2007-05-03 |
Substituted n-phenyl sulfonamide bradykinin antagonists App 20070093485 - Farouz; Francine S. ;   et al. | 2007-04-26 |
Pyrimidine hydantoin analogues which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,205,310 - Konradi , et al. April 17, 2 | 2007-04-17 |
Bridged N-Cyclic Sulfonamido Inhibitors of Gamma Secretase App 20070049612 - Bowers; Simeon ;   et al. | 2007-03-01 |
Novel compounds useful for bradykinin B1 receptor antagonism App 20070032475 - Ye; Xiaocong Michael ;   et al. | 2007-02-08 |
Heterocyclic compounds which inhibit leukocyte adhesion mediated by alpha-4 integrins App 20070027131 - Konradi; Andrei W. ;   et al. | 2007-02-01 |
Preparation of polymer conjugates of therapeutic, agricultural, and food additive compounds App 20070021555 - Konradi; Andrei W. ;   et al. | 2007-01-25 |
Heterocyclic compounds which inhibit leukocyte adhesion mediated by .alpha..sub.4 integrins Grant 7,135,477 - Konradi , et al. November 14, 2 | 2006-11-14 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4. Grant 7,049,306 - Konradi , et al. May 23, 2 | 2006-05-23 |
Compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,030,114 - Thorsett , et al. April 18, 2 | 2006-04-18 |
Heterocyclic compounds which inhibit leukocyte adhesion mediated by .alpha..sub.4 integrins Grant 7,026,328 - Konradi , et al. April 11, 2 | 2006-04-11 |
Heteroaryl-.beta.-alanine derivatives as alpha 4 integrin inhibitors Grant 7,015,216 - Konradi , et al. March 21, 2 | 2006-03-21 |
Heterocyclic compounds which inhibit leukocyte adhesion mediated by .alpha..sub.4 integrins Grant 7,008,949 - Konradi , et al. March 7, 2 | 2006-03-07 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,005,433 - Konradi , et al. February 28, 2 | 2006-02-28 |
Multimeric VLA-4 antagonists comprising polymer moieties App 20060013799 - Konradi; Andrei W. ;   et al. | 2006-01-19 |
Compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20050261293 - Konradi, Andrei W. ;   et al. | 2005-11-24 |
Pyrimidine hydantoin analogues which inhibit leukocyte adhesion mediated by VLA-4 App 20050261324 - Konradi, Andrei W. ;   et al. | 2005-11-24 |
Beta-amino acid derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 Grant 6,953,802 - Konradi , et al. October 11, 2 | 2005-10-11 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20050222119 - Thorsett, Eugene D. ;   et al. | 2005-10-06 |
Composition for and treatment of demyelinating diseases and paralysis by administration of remyelinating agents App 20050215565 - Karlik, Stephen J. ;   et al. | 2005-09-29 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20050203093 - Konradi, Andrei W. ;   et al. | 2005-09-15 |
Beta-amino acid derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 App 20050192280 - Konradi, Andrei W. ;   et al. | 2005-09-01 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,911,439 - Konradi , et al. June 28, 2 | 2005-06-28 |
Heteroaryl compounds which inhibit leukocyte adhesion mediated by alpha-4 integrins App 20050130999 - Konradi, Andrei W. ;   et al. | 2005-06-16 |
Compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,903,088 - Konradi , et al. June 7, 2 | 2005-06-07 |
Heterocyclic compounds which inhibit leukocyte adhesion mediated by alpha4 integrins App 20050119290 - Konradi, Andrei W. ;   et al. | 2005-06-02 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,900,179 - Thorsett , et al. May 31, 2 | 2005-05-31 |
Alpha amino acid derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 App 20050085459 - Konradi, Andrei W. ;   et al. | 2005-04-21 |
Methods and compositions for treating rheumatoid arthritis App 20050074451 - Yednock, Theodore A. ;   et al. | 2005-04-07 |
Composition for and treatment of demyelinating diseases and paralysis by administration of remyelinating agents App 20050069541 - Karlik, Stephen J. ;   et al. | 2005-03-31 |
Methods and compositions for treating rheumatoid arthritis App 20050065192 - Yednock, Theodore A. ;   et al. | 2005-03-24 |
3-(heteroaryl) alanine derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 App 20040266763 - Konradi, Andrei W. ;   et al. | 2004-12-30 |
Alpha amino acid derivatives--inhibitors of leukocyte adhesion mediated by VLA-4 Grant 6,803,370 - Konradi , et al. October 12, 2 | 2004-10-12 |
3-(heteroaryl) alanine derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 Grant 6,794,506 - Konradi , et al. September 21, 2 | 2004-09-21 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20040147512 - Konradi, Andrei W. ;   et al. | 2004-07-29 |
Heteroaryl compounds which inhibit leukocyte adhesion mediated by alpha4 integrins App 20040142954 - Konradi, Andrei W. ;   et al. | 2004-07-22 |
Heterocyclic compounds which inhibit leukocyte adhesion mediated by alpha4integrins App 20040138243 - Konradi, Andrei W. ;   et al. | 2004-07-15 |
Phenylalanine derivatives as alpha 4 integrin inhibitors App 20040127486 - Konradi, Andrei W. ;   et al. | 2004-07-01 |
Fused ring heteroaryl and heterocyclic compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20040029873 - Grant, Francine S. ;   et al. | 2004-02-12 |
Phenylalanine derivatives as alpha 4 integrin inhibitors Grant 6,689,781 - Konradi , et al. February 10, 2 | 2004-02-10 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20040014677 - Thorsett, Eugene D. ;   et al. | 2004-01-22 |
Compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20040006093 - Thorsett, Eugene D. ;   et al. | 2004-01-08 |
Compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20030144328 - Konradi, Andrei W. ;   et al. | 2003-07-31 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated byVLA-4 App 20030139402 - Konradi, Andrei W. ;   et al. | 2003-07-24 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20030125324 - Konradi, Andrei W. ;   et al. | 2003-07-03 |
Benzyl compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,586,602 - Thorsett , et al. July 1, 2 | 2003-07-01 |
Compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,583,139 - Thorsett , et al. June 24, 2 | 2003-06-24 |
Fused ring heteroaryl and heterocyclic compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,545,003 - Grant , et al. April 8, 2 | 2003-04-08 |
Benzyl compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20030065193 - Thorsett, Eugene D. ;   et al. | 2003-04-03 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,525,026 - Thorsett , et al. February 25, 2 | 2003-02-25 |
Alpha-aminoacetic acid derivatives- alpha4beta7 receptor antagonists App 20030018195 - Konradi, Andrei W. ;   et al. | 2003-01-23 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20030017993 - Thorsett, Eugene D. ;   et al. | 2003-01-23 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20020193312 - Thorsett, Eugene D. ;   et al. | 2002-12-19 |
Substituted phenylalanine type compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,492,421 - Thorsett , et al. December 10, 2 | 2002-12-10 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,492,372 - Konradi , et al. December 10, 2 | 2002-12-10 |
Heteroaryl-beta-alanine derivatives as alpha 4 integrin inhibitors App 20020086882 - Konradi, Andrei W. ;   et al. | 2002-07-04 |
Beta-amino acid derivatives--inhibitors of leukocyte adhesion mediated by VLA-4 App 20020058664 - Konradi, Andrei W. ;   et al. | 2002-05-16 |
Phenylalanine derivatives as alpha 4 integrin inhibitors App 20020055509 - Konradi, Andrei W. ;   et al. | 2002-05-09 |
3-(Heteroaryal) alanine derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 App 20020052375 - Konradi, Andrei W. ;   et al. | 2002-05-02 |
Alpha amino acid derivatives--inhibitors of leukocyte adhesion mediated by VLA-4 App 20020052470 - Konradi, Andrei W. ;   et al. | 2002-05-02 |