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N-(4-(azaindazol-6-yl)-phenyl)-sulfonamides and their use as pharmaceuticals Grant 9,718,825 - Nazare , et al. August 1, 2 | 2017-08-01 |
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Acylamino-substituted cyclic carboxylic acid derivatives and their use as pharmaceuticals Grant 9,018,383 - Pernerstorfer , et al. April 28, 2 | 2015-04-28 |
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Substituted isoquinolines and isoquinolinones as Rho kinase inhibitors Grant 8,541,449 - Plettenburg , et al. September 24, 2 | 2013-09-24 |
Use of norgestimate as a selective inhibitor of TRPC3, TRPC6 and TRPC7 ion channels Grant 8,455,469 - Miehe , et al. June 4, 2 | 2013-06-04 |
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6-Substituted isoquinolines and isoquinolinones App 20130109715 - PLETTENBURG; Oliver ;   et al. | 2013-05-02 |
Pentafluorosulfanylbenzoylguanidines, processes for their preparation, their use as medicaments or diagnostic aids, and medicaments comprising them Grant 8,404,893 - Kleemann March 26, 2 | 2013-03-26 |
6-substituted isoquinolines and isoquinolinones Grant 8,399,482 - Plettenburg , et al. March 19, 2 | 2013-03-19 |
Heteroarylacrylamides and their use as pharmaceuticals Grant 8,304,438 - Strobel , et al. November 6, 2 | 2012-11-06 |
Acylamino-substituted Cyclic Carboxylic Acid Derivatives And Their Use As Pharmaceuticals App 20120264790 - PERNERSTORFER; Josef ;   et al. | 2012-10-18 |
Process for preparing (3-oxo-2,3-dihydro-1H-isoindol-1-yl) acetylguanidine derivatives Grant 8,283,374 - Schubert , et al. October 9, 2 | 2012-10-09 |
Heteroaryl-substituted carboxamides and their use as pharmaceuticals Grant 8,188,291 - Strobel , et al. May 29, 2 | 2012-05-29 |
Pentafluorosulfanylbenzoylguanidines, Processes For Their Preparation, Their Use As Medicaments Or Diagnostic Aids, And Medicaments Comprising Them App 20110306670 - KLEEMANN; Heinz-Werner | 2011-12-15 |
Di(hetero)arylcyclohexane derivatives, their preparation, their use and pharmaceutical compositions comprising them Grant 8,076,324 - Bohme , et al. December 13, 2 | 2011-12-13 |
Pentafluorosulfanylbenzoylguanidines, processes for their preparation, their use as medicaments or diagnostic aids, and medicaments comprising them Grant 8,008,352 - Kleemann August 30, 2 | 2011-08-30 |
Substituted Isoquinolines And Isoquinolinones As Rho Kinase Inhibitors App 20110190341 - Plettenburg; Oliver ;   et al. | 2011-08-04 |
6-substituted Isoquinolines And Isoquinolinones App 20110190339 - PLETTENBURG; Oliver ;   et al. | 2011-08-04 |
Ortho-substituted pentafluorosulfanylbenzenes, process for their preparation and their use as valuable synthetic intermediates Grant 7,932,416 - Kleemann , et al. April 26, 2 | 2011-04-26 |
Use Of Norgestimate As A Selective Inhibitor Of Trpc3, Trpc6 And Trpc7 Ion Channels App 20110015167 - Miehe; Susanne ;   et al. | 2011-01-20 |
Di(hetero)arylcyclohexane derivatives, their preparation, their use and pharmaceutical compositions comprising them App 20100204206 - BOHME; Thomas ;   et al. | 2010-08-12 |
Substituted benzoylguanidines, method for production and use thereof as medicament or diagnostic and medicament comprising the same Grant 7,772,262 - Kleemann August 10, 2 | 2010-08-10 |
Ortho-substituted pentafluorosulfanyl benzenes, method for the production thereof and their use as synthesis intermediates Grant 7,763,661 - Kleemann , et al. July 27, 2 | 2010-07-27 |
Process for preparing 4-pentafluorosulfanylbenzoylguanidines Grant 7,659,429 - Schubert , et al. February 9, 2 | 2010-02-09 |
Heteroarylacrylamides And Their Use As Pharmaceuticals App 20100016272 - STROBEL; Hartmut ;   et al. | 2010-01-21 |
Heteroaryl-substituted Carboxamides And Their Use As Pharmaceuticals App 20100016337 - STROBEL; Hartmut ;   et al. | 2010-01-21 |
3-guanidinocarbonyl-1-heteroaryl-indole derivatives, preparation process, their use as medicaments, and pharmaceutical compositions comprising them Grant 7,638,521 - Kleemann , et al. December 29, 2 | 2009-12-29 |
Pentafluorosulfanylbenzoylguanidines, process for their preparation, use as a medicament or diagnostic aid, and medicament comprising same Grant 7,622,611 - Kleemann November 24, 2 | 2009-11-24 |
Isoindolone derivatives, preparation process and intermediates of this process, their use as medicaments, and pharmaceutical compositions comprising them Grant 7,589,117 - Kleemann , et al. September 15, 2 | 2009-09-15 |
Process For Preparing (3-oxo-2,3-dihydro-1h-isoindol-1-yl) Acetylguanidine Derivatives App 20090203761 - SCHUBERT; Gerrit ;   et al. | 2009-08-13 |
Use Of Inhibitors Of The Cellular Na+/h+ Exchanger (nhe) For Preparing A Medicament For Normalizing Serum Lipids App 20090143473 - LANG; Hans Jochen ;   et al. | 2009-06-04 |
3-guanidinocarbonyl-1-heteroaryl-indole derivatives, preparation process, their use as medicaments, and pharmaceutical compositions comprising them Grant 7,531,663 - Kleemann , et al. May 12, 2 | 2009-05-12 |
Process for preparing (3-oxo-2,3-dihydro-1H-isoindol-1-yl) acetylguanidine derivatives Grant 7,531,569 - Schubert , et al. May 12, 2 | 2009-05-12 |
Process for Preparing 4-Pentafluorosulfanylbenzoylguanidines App 20090036704 - Schubert; Gerrit ;   et al. | 2009-02-05 |
Process for preparing 4-pentafluorosulfanylbenzoylguanidines Grant 7,449,594 - Schubert , et al. November 11, 2 | 2008-11-11 |
Methods For The Improvement Of Memory And Neurological Function Comprising The Administration Of Compositions That Act As Inhibitors Of The Sodium Proton (na+ /h+ ) Exchanger, Subtype 5 (nhe-5) App 20080234317 - KLEEMANN; Heinz-Werner ;   et al. | 2008-09-25 |
Pentafluorosulfanylbenzoylguanidines, Processes For Their Preparation, Their Use As Medicaments Or Diagnostic Aids, And Medicaments Comprising Them App 20080200553 - KLEEMANN; Heinz-Werner | 2008-08-21 |
Pentafluorosulfanylbenzoylguanidines, Process For Their Preparation, Use As A Medicament Or Diagnostic Aid, And Medicament Comprising Same App 20080146673 - KLEEMANN; Heinz-Werner | 2008-06-19 |
Pentafluorosulfanylphenyl-substituted benzoylguanidines, processes for their preparation, their use as medicament or diagnostic aid, and medicament comprising them Grant 7,381,841 - Kleemann June 3, 2 | 2008-06-03 |
Pentafluorosulfanylbenzoylguanidines, processes for their preparation, their use as medicaments or diagnostic aids, and medicaments comprising them Grant 7,375,138 - Kleemann May 20, 2 | 2008-05-20 |
Ortho-substituted pentafluorosulfanylbenzenes, process for their preparation and their use as valuable synthetic intermediates App 20080091031 - KLEEMANN; Heinz-Werner ;   et al. | 2008-04-17 |
Anthranilamides and methods of their use Grant 7,332,608 - Brendel , et al. February 19, 2 | 2008-02-19 |
Ortho-substituted pentafluorosulfanylbenzenes, process for their preparation and their use as valuable synthetic intermediates Grant 7,317,124 - Kleemann , et al. January 8, 2 | 2008-01-08 |
Substituted Benzoylguanidines, Method For Production And Use Thereof As Medicament Or Diagnostic And Medicament Comprising The Same App 20070270414 - Kleemann; Heinz-Werner | 2007-11-22 |
Pentafluorosulfanylphenyl-substituted benzoylguanidines, method for the production thereof, their use as a medicament or diagnostic agent, and a medicament containing these compounds App 20070259963 - KLEEMANN; Heinz-Werner | 2007-11-08 |
Ortho-substituted Pentafluorosulfanyl Benzenes, Method For The Production Thereof And Their Use As Synthesis Intermediates App 20070259943 - KLEEMANN; Heinz-Werner ;   et al. | 2007-11-08 |
Anthranilamides with heteroarylsulfonyl side chain, process of preparation, and use Grant 7,235,664 - Brendel , et al. June 26, 2 | 2007-06-26 |
Anthranilamides and methods of their use Grant 7,235,690 - Brendel , et al. June 26, 2 | 2007-06-26 |
Derivatives of 3-(Guanidinocarbonyl) heterocycle, methods of preparation and intermediates thereof, their use as medicaments, and pharmaceutical compositions therefrom Grant 7,230,007 - Carry , et al. June 12, 2 | 2007-06-12 |
Anthranilamides And Methods Of Their Use App 20070117807 - Brendel; Joachim ;   et al. | 2007-05-24 |
Process For Preparing 4-Pentafluorosulfanylbenzoylguanidines App 20070106094 - Schubert; Gerrit ;   et al. | 2007-05-10 |
Process for preparing 4-pentafluorosulfanylbenzoylguanidines Grant 7,126,026 - Schubert , et al. October 24, 2 | 2006-10-24 |
Isoindolone derivatives, preparation process and intermediates of this process, their use as medicaments, and pharmaceutical compositions comprising them Grant 7,078,428 - Kleemann , et al. July 18, 2 | 2006-07-18 |
Derivatives of 3-guanidinocarbonyl-1-heteroaryl-pyrrole, preparation process and intermediates of this process, their use as medicaments, and pharmaceutical compositions comprising them Grant 7,078,414 - Kleemann , et al. July 18, 2 | 2006-07-18 |
Isoindolone derivatives, preparation process and intermediates of this process, their use as medicaments, and pharmaceutical compositions comprising them App 20060148880 - Kleemann; Heinz-Werner ;   et al. | 2006-07-06 |
Use of inhibitors of the sodium-dependent chloride/bicarbonate exchanger for the treatment of thrombotic and inflammatory disorders App 20060025401 - Lang; Hans-Jochen ;   et al. | 2006-02-02 |
Arylated furan- and thiophenecarboxamides, processes for their preparation, their use as medicaments, and pharmaceutical preparations comprising them Grant 6,982,279 - Peukert , et al. January 3, 2 | 2006-01-03 |
Ortho, meta-substituted bisaryl compounds, processes for their preparation, their use as medicaments, and pharmaceutical preparations comprising them Grant 6,924,392 - Peukert , et al. August 2, 2 | 2005-08-02 |
Ortho-substituted pentafluorosulfanylbenzenes, process for their preparation and their use as valuable synthetic intermediates App 20050148652 - Kleemann, Heinz-Werner ;   et al. | 2005-07-07 |
Anthranilamides with heteroarylsulfonyl side chain, process of preparation, and use App 20050137200 - Brendel, Joachim ;   et al. | 2005-06-23 |
Process for preparing 4-pentafluorosulfanylbenzoylguanidines App 20050131070 - Schubert, Gerrit ;   et al. | 2005-06-16 |
Process for preparing (3-oxo-2,3-dihydro-1H-isoindol-1-yl) acetylguanidine derivatives App 20050124681 - Schubert, Gerrit ;   et al. | 2005-06-09 |
Pentafluorosulfanylbenzoylguanidines, process for their preparation, use as a medicament or diagnostic aid, and medicament comprising same App 20050124666 - Kleemann, Heinz-Werner | 2005-06-09 |
Anthranilamides with heteroarylsulfonyl side chain, process of preparation, and use Grant 6,903,216 - Brendel , et al. June 7, 2 | 2005-06-07 |
Fluorinated cycloalkyl-derivatized benzoylguanidines, process for their preparation, their uses as medicament, and medicament containing them Grant 6,878,748 - Kleemann April 12, 2 | 2005-04-12 |
Pentafluorosulfanylphenyl-substituted benzoylguanidines, processes for their preparation, their use as medicament or diagnostic aid, and medicament comprising them App 20050043401 - Kleemann, Heinz-Werner | 2005-02-24 |
3-Guanidinocarbonyl-1-heteroaryl-indole derivatives, preparation process, their use as medicaments, and pharmaceutical compositions comprising them App 20050026989 - Kleemann, Heinz-Werner ;   et al. | 2005-02-03 |
Derivatives of 3-(guanidinocarbonyl) heterocycle, methods of preparation and intermediates thereof, their use as medicaments, and pharmaceutical compositions therefrom App 20050014758 - Carry, Jean-Christophe ;   et al. | 2005-01-20 |
Derivatives of 3-guanidinocarbonyl-1-heteroaryl-pyrrole, preparation process and intermediates of this process, their use as medicaments, and pharmaceutical compositions comprising them App 20040266775 - Kleemann, Heinz-Werner ;   et al. | 2004-12-30 |
Substituted norbornylamino derivatives, processes for their preparation, their use as medicaments or diagnostics, and a medicament comprising them Grant 6,825,231 - Heinelt , et al. November 30, 2 | 2004-11-30 |
3-guanidinocarbonyl-1-heteroaryl-indole derivatives, preparation process, their use as medicaments, and pharmaceutical compositions comprising them App 20040214820 - Kleemann, Heinz-Werner ;   et al. | 2004-10-28 |
Ortho, ortho-substituted nitrogen-containing bisaryl compounds, processes for their preparation, their use as medicaments, and pharmaceutical preparation comprising them Grant 6,794,377 - Peukert , et al. September 21, 2 | 2004-09-21 |
Use of inhibitors of the cellular Na+/H+ exchanger (NHE) for preparing a medicament for normalizing serum lipids App 20040122096 - Lang, Hans Jochen ;   et al. | 2004-06-24 |
Dihydrothiaphenanthrenecarbonylguanidines: composition, process of making, and use as medicament or diagnostic aid Grant 6,730,697 - Kleemann , et al. May 4, 2 | 2004-05-04 |
Arylated furan- and thiophenecarboxamides, processes for their preparation, their use as medicaments, and pharmaceutical preparations comprising them App 20040068120 - Peukert, Stefan ;   et al. | 2004-04-08 |
Isoindolone derivatives, preparation process and intermediates of this process, their use as medicaments, and pharmaceutical compositions comprising them App 20040048916 - Kleemann, Heinz-Werner ;   et al. | 2004-03-11 |
Substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament containing them Grant 6,703,411 - Weichert , et al. March 9, 2 | 2004-03-09 |
Diacyl-substituted guanidines, a process for their preparation, their use as medicament or diagnostic aid, and medicament containing them App 20040044081 - Kleemann, Heinz-Werner ;   et al. | 2004-03-04 |
Ortho, meta-substituted bisaryl compounds, processes for their preparation, their use as medicaments, and pharmaceutical preparations comprising them App 20030225099 - Peukert, Stefan ;   et al. | 2003-12-04 |
Use of inhibitors of the sodium-dependent chloride/bicarbonate exchanger for the treatment of thrombotic and inflammatory disorders App 20030220383 - Lang, Hans-Jochen ;   et al. | 2003-11-27 |
Pentafluorosulfanylbenzoylguanidines, processes for their preparation, their use as medicaments or diagnostic aids, and medicaments comprising them App 20030216476 - Kleemann, Heinz-Werner | 2003-11-20 |
Monoacyl-substituted guanidines, a process for their preparation, their use as a medicament or diagnostic aid, and pharmaceutical compositions containing them Grant 6,632,840 - Kleemann , et al. October 14, 2 | 2003-10-14 |
Anthranilamides and methods of their use App 20030187033 - Brendel, Joachim ;   et al. | 2003-10-02 |
Dihydrothiaphenanthrenecarbonylguanidines: composition, process of making, and use as medicament or diagnostic aid App 20030181511 - Kleemann, Heinz-Werner ;   et al. | 2003-09-25 |
Heterocyclically substituted benzoylguanidines, process for their preparation, their use as medicaments or diagnostics, and medicaments comprising them Grant 6,617,344 - Weichert , et al. September 9, 2 | 2003-09-09 |
Ortho, meta-substituted bisaryl compounds, processes for their preparation, their use as medicaments, and pharmaceutical preparations comprising them Grant 6,605,625 - Peukert , et al. August 12, 2 | 2003-08-12 |
Mercaptoacetylamide derivatives, a process for their preparation and their use Grant 6,602,866 - Flynn , et al. August 5, 2 | 2003-08-05 |
Heterocyclically Substituted Benzoylguanidines, Process For Their Preparation, Their Use As Medicaments Or Diagnostics, And Medicaments Comprising Them App 20030139607 - Weichert, Andreas ;   et al. | 2003-07-24 |
Substituted anthranilic acids, their use as a medicament or diagnostic, and medicament comprising them, and a pharmaceutical combination preparation containing a sodium/hydrogen exchange (NHE) blocker Grant 6,593,352 - Weichert , et al. July 15, 2 | 2003-07-15 |
Anthranilamides with heteroarylsulfonyl side chain, process of preparation, and use App 20030114499 - Brendel, Joachim ;   et al. | 2003-06-19 |
Ortho, ortho-substituted nitrogen-containing bisaryl compounds, processes for their preparation, their use as medicaments, and pharmaceutical preparation comprising them App 20030060470 - Peukert, Stefan ;   et al. | 2003-03-27 |
Substituted 1-naphthoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament containing them App 20030013760 - Brendel, Joachim ;   et al. | 2003-01-16 |
Mercaptoacetylamide derivatives, a process for their preparation and their use App 20020193589 - Flynn, Gary A. ;   et al. | 2002-12-19 |
Substituted acylguanidines, process for their preparation, their use as medicaments or diagnostics, and medicaments comprising them Grant 6,451,781 - Kleemann , et al. September 17, 2 | 2002-09-17 |
Fluorophenyl-substituted alkenylcarboxylic acid guanidides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them App 20020123529 - Schwark, Jan-Robert ;   et al. | 2002-09-05 |
Substituted anthranilic acids, their use as a medicament or diagnostic, and medicament comprising them, and a pharmaceutical combination preparation containing a sodium/hydrogen exchange (NHE) blocker App 20020123632 - Weichert, Andreas ;   et al. | 2002-09-05 |
Heterocyclically substituted benzoylguanidines, process for their preparation, their use as medicaments or diagnostics, and medicaments comprising them App 20020099222 - Weichert, Andreas ;   et al. | 2002-07-25 |
Five-membered heterocycles having biphenylsulfonyl substitution, process for their preparation, their use as a medicament or diagnostic, and medicament comprising them App 20020045761 - Kleemann, Heinz-Werner ;   et al. | 2002-04-18 |
Substituted 4-benzylaminoquinolines and their hetero analogs, process for their preparation, pharmaceuticals containing these compounds and use thereof Grant 6,339,077 - Hofmeister , et al. January 15, 2 | 2002-01-15 |
Heterocyclically substituted benzoylguanidines, process for their preparation, their use as medicaments or diagnostics, and medicaments comprising them App 20010049446 - Weichert, Andreas ;   et al. | 2001-12-06 |
Substituted norbornylamino derivatives, processes for their preparation, their use as medicaments or diagnostics, and a medicament comprising them App 20010023257 - Heinelt, Uwe ;   et al. | 2001-09-20 |
Fluorophenyl-substituted alkenylcarboxylic acid guanidides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them App 20010020042 - Schwark, Jan-Robert ;   et al. | 2001-09-06 |
Substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament containing them App 20010016596 - Weichert, Andreas ;   et al. | 2001-08-23 |
Phenyl.-substituted alkenylcarboguanidides carrying perfluoroalkyl groups, a process for their preparation, their use as a medicament or diagnostic agent, and also a medicament containing them Grant 6,025,349 - Schwark , et al. February 15, 2 | 2000-02-15 |
Substituted benzoylguanidines, process for their preparation, their use as a pharmaceutical as inhibitors of the cellular NA+/H+ exchange or as a diagnostic, and pharmaceutical containing them Grant 5,866,610 - Lang , et al. February 2, 1 | 1999-02-02 |
Substituted benzyloxycarbonylguanidines, a process for their preparation, their use as a medicament or diagnostic, and a medicament containing them Grant 5,753,710 - Kleemann , et al. May 19, 1 | 1998-05-19 |
Substituted sulfonimidamides, processes for their preparation, their use as a medicament or diagnostic, and medicament comprising them Grant 5,708,034 - Kleemann , et al. January 13, 1 | 1998-01-13 |
Substituted N-heteroaroylguanidines, a process for their preparation, their use as a medicament or diagnostic agent, and a medicament containing them Grant 5,698,581 - Kleemann , et al. December 16, 1 | 1997-12-16 |
Benzoylguanidines, pharmaceutical composition containing them and treatment of arrthythmias therewith Grant 5,591,754 - Lang , et al. January 7, 1 | 1997-01-07 |