Patent | Date |
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Substituted N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase Grant 11,078,168 - Steeneck , et al. August 3, 2 | 2021-08-03 |
Novel Lxr Modulators With Bicyclic Core Moiety App 20210147398 - Gege; Christian ;   et al. | 2021-05-20 |
Spirocyclic Compounds As Modulators Of Indoleamine 2,3-dioxygenase App 20210122757 - KINZEL; Olaf ;   et al. | 2021-04-29 |
Oxalamides As Modulators Of Indoleamine 2,3-dioxygenase App 20200352931 - Steeneck; Christoph ;   et al. | 2020-11-12 |
FXR (NR1H4) binding and activity modulating compounds Grant 10,485,795 - Kinzel , et al. Nov | 2019-11-26 |
Substituted N-hydroxyamidinoheterocycles As Modulators Of Indoleamine 2,3-dioxygenase App 20190292160 - Steeneck; Christoph ;   et al. | 2019-09-26 |
Carboxamide or sulfonamide substituted thiazoles and related derivatives as modulators for the orphan nuclear receptor ROR[.gamma.] Grant 10,301,272 - Gege , et al. | 2019-05-28 |
Novel FXR (NR1H4) binding and activity modulating compounds App 20190142814 - Kinzel; Olaf ;   et al. | 2019-05-16 |
FXR (NR1H4) binding and activity modulating compounds Grant 10,220,027 - Kinzel , et al. | 2019-03-05 |
Trifluoromethyl alcohols as modulators of ROR.gamma.t Grant 10,150,762 - Goldberg , et al. Dec | 2018-12-11 |
Thiazoles as modulators of ROR.gamma.t Grant 10,080,744 - Goldberg , et al. September 25, 2 | 2018-09-25 |
Novel FXR (NR1H4) binding and activity modulating compounds App 20180200243 - Kinzel; Olaf ;   et al. | 2018-07-19 |
FXR (NR1H4) modulating compounds Grant 9,938,278 - Gege , et al. April 10, 2 | 2018-04-10 |
THIAZOLES AS MODULATORS OF RORyt App 20180064690 - Goldberg; Steven ;   et al. | 2018-03-08 |
Thiazoles as modulators of ROR.gamma.t Grant 9,861,618 - Goldberg , et al. January 9, 2 | 2018-01-09 |
Trifluoromethyl alcohols as modulators of ROR.gamma.t Grant 9,850,236 - Goldberg , et al. December 26, 2 | 2017-12-26 |
Amide substituted thiazoles as modulators of RORyt Grant 9,845,319 - Goldberg , et al. December 19, 2 | 2017-12-19 |
FXR (NR1H4) binding and activity modulating compounds Grant 9,820,979 - Kinzel , et al. November 21, 2 | 2017-11-21 |
TRIFLUOROMETHYL ALCOHOLS AS MODULATORS OF RORyt App 20170327492 - Goldberg; Steven ;   et al. | 2017-11-16 |
Pyrrolo carboxamides as modulators of orphan nuclear receptor RAR-related orphan receptor-gamma (ROR.gamma., NR1F3) activity and for the treatment of chronic inflammatory and autoimmune diseases Grant 9,815,851 - Steeneck , et al. November 14, 2 | 2017-11-14 |
Novel Fxr (nr1h4) Modulating Compounds App 20170298068 - GEGE; CHRISTIAN ;   et al. | 2017-10-19 |
Hydroxy containing FXR (NR1H4) modulating compounds Grant 9,751,874 - Gege , et al. September 5, 2 | 2017-09-05 |
Novel Fxr (nr1h4) Binding And Activity Modulating Compounds App 20170143684 - Kinzel; Olaf ;   et al. | 2017-05-25 |
FXR (NR1H4) binding and activity modulating compounds Grant 9,539,244 - Kinzel , et al. January 10, 2 | 2017-01-10 |
Carboxamide or sulfonamide substituted nitrogen-containing 5-membered heterocycles as modulators for the orphan nuclear receptor ROR.gamma. Grant 9,458,104 - Gege , et al. October 4, 2 | 2016-10-04 |
Hydroxy Containing Fxr (nr1h4) Modulating Compounds App 20160176861 - Gege; Christian ;   et al. | 2016-06-23 |
TRIFLUOROMETHYL ALCOHOLS AS MODULATORS OF RORyt App 20160122336 - Goldberg; Steven ;   et al. | 2016-05-05 |
THIAZOLES AS MODULATORS OF RORyt App 20160120850 - Goldberg; Steven ;   et al. | 2016-05-05 |
AMIDE SUBSTITUTED THIAZOLES AS MODULATORS OF RORyt App 20160122335 - Goldberg; Steven ;   et al. | 2016-05-05 |
Novel Fxr (nr1h4) Binding And Activity Modulating Compounds App 20150342930 - Kinzel; Olaf ;   et al. | 2015-12-03 |
Carboxamide Or Sulfonamide Substituted Nitrogen-containing 5-membered Heterocycles As Modulators For The Orphan Nuclear Receptor Ror Gamma App 20150344423 - GEGE; Christian ;   et al. | 2015-12-03 |
FXR (NR1H4) binding and activity modulating compounds Grant 9,139,539 - Kinzel , et al. September 22, 2 | 2015-09-22 |
Carboxamide Or Sulfonamide Substituted Thiazoles And Related Derivatives As Modulators For The Orphan Nuclear Receptor Ror[gamma] App 20150175562 - Gege; Christian ;   et al. | 2015-06-25 |
FXR (NR1H4) binding and activity modulating compounds Grant 8,952,042 - Kremoser , et al. February 10, 2 | 2015-02-10 |
Pyrrolo sulfonamide compounds for modulation of orphan nuclear receptor RAR-related orphan receptor-.gamma. (ROR-.gamma., NR1F3) activity and for the treatment of chronic inflammatory and autoimmune diseases Grant 8,946,446 - Steeneck , et al. February 3, 2 | 2015-02-03 |
Compounds for modulation of orphan nuclear receptor RAR-related orphan receptor-gamma (ROR.gamma., NR1F3) activity and for the treatment of chronic inflammatory and autoimmune disease Grant 8,940,722 - Kinzel , et al. January 27, 2 | 2015-01-27 |
PYRROLO CARBOXAMIDES AS MODULATORS OF ORPHAN NUCLEAR RECEPTOR RAR-RELATED ORPHAN RECEPTOR-GAMMA (RORy, NR1F3) ACTIVITY AND FOR THE TREATMENT OF CHRONIC INFLAMMATORY AND AUTOIMMUNE DISEASES App 20140349987 - Steeneck; Christoph ;   et al. | 2014-11-27 |
Novel Fxr (nr1h4) Binding And Activity Modulating Compounds App 20140221659 - Kinzel; Olaf ;   et al. | 2014-08-07 |
Pyrrolo Sulfonamide Compounds For Modulation Of Orphan Nuclear Receptor Rar-related Orphan Receptor-gamma (ror-gamma, Nr1f3) Activity And For The Treatment Of Chronic Inflammatory And Autoimmune Diseases App 20140142082 - Steeneck; Christoph ;   et al. | 2014-05-22 |
Saturated bicyclic heterocyclic derivatives as SMO antagonists Grant 8,470,823 - Branca , et al. June 25, 2 | 2013-06-25 |
Novel compounds for modulation of orphan nuclear receptor RAR-related orphan receptor-gamma (RORgamma, NR1F3) activity and for the treatment of chronic inflammatory and autoimmune disease App 20130053380 - Kinzel; Olaf ;   et al. | 2013-02-28 |
Quinolin-4-one and 4-oxodihydrocinnoline derivatives as inhibitors of poly(ADP-ribose) polymerase (PARP) Grant 8,354,413 - Jones , et al. January 15, 2 | 2013-01-15 |
Pyridazinone derivatives as PARP inhibitors Grant 8,268,827 - Branca , et al. September 18, 2 | 2012-09-18 |
Novel Fxr (nr1h4) Binding And Activity Modulating Compounds App 20120232116 - Kremoser; Claus ;   et al. | 2012-09-13 |
Pyridinone and pyridazinone derivatives as inhibitors of poly (ADP-ribose) polymerase (PARP) Grant 8,188,084 - Jones , et al. May 29, 2 | 2012-05-29 |
Quinolin-4-one And 4-oxodihyrdocinnoline Derivatives As Inhibitors Of Poly(adp-ribose) Polymerase (parp) App 20110207720 - Jones; Philip ;   et al. | 2011-08-25 |
Saturated Bicyclic Heterocyclic Derivatives As Smo Antagonists App 20110183989 - Branca; Danila ;   et al. | 2011-07-28 |
Tetrahydro-4H-pyrido[1,2-a] pyrimidines useful as HIV integrase inhibitors Grant 7,968,553 - Crescenzi , et al. June 28, 2 | 2011-06-28 |
HIV integrase inhibitors Grant 7,939,537 - Summa , et al. May 10, 2 | 2011-05-10 |
Heterocycle derivatives as histone deacetylase (HDAC) inhibitors Grant 7,863,294 - Attenni , et al. January 4, 2 | 2011-01-04 |
Pyrrolo[1,2-a] pyrazin-1(2H)-one and pyrrolo[1,2-d][1,2,4]triazin-1(2H)-one derivatives as inhibitors of poly(ADP-ribose)polymerase (PARP) Grant 7,834,015 - Jones , et al. November 16, 2 | 2010-11-16 |
Pyridazinone Derivatives As Parp Inhibitors App 20100261709 - Branca; Danila ;   et al. | 2010-10-14 |
Imidazolopyrimidines And Imidazolotriazine Derivatives As Inhibitors Of Poly(adp-ribose)polymerase(parp) App 20100173895 - Jones; Philip ;   et al. | 2010-07-08 |
Hiv Integrase Inhibitors App 20090221571 - Summa; Vincenzo ;   et al. | 2009-09-03 |
Pyrrolo[1,2-A] Pyrazin-1(2H)-One and Pyrrolo[1,2-D][1,2,4]Triazin-1(2H)-One Derivatives as Inhibitors of Poly(Adp-Ribose)Polymerase (Parp) App 20090209523 - Jones; Philip ;   et al. | 2009-08-20 |
Pyridinone and Pyridazinone Derivatives as Inhibitors of Poly (Adp-Ribose) Polymerase (Parp) App 20090176765 - Jones; Philip ;   et al. | 2009-07-09 |
Heterocycle Derivatives As Histone Deacetylase (Hdac) Inhibitors App 20090048228 - Attenni; Barbara ;   et al. | 2009-02-19 |
Substituted pyrimido[1,2-a]azepines useful as HIV integrase inhibitors Grant 7,414,045 - Crescenzi , et al. August 19, 2 | 2008-08-19 |
Tetrahydro-4H-pyrido[1,2-a] pyrimidines useful as HIV integrase inhibitors App 20080176869 - Crescenzi; Benedetta ;   et al. | 2008-07-24 |
Tetrahydro--4h-pyrido[1,2-a}pyrimidines and related compounds useful as hiv integrase inhibitors App 20060046985 - Crescenzi; Benedetta ;   et al. | 2006-03-02 |
Vectors for dna delivery App 20030207400 - Bianchi, Elisabetta ;   et al. | 2003-11-06 |