Patent | Date |
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Diaza-spiro-{4,4}-nonane derivatives as neurokinin (NK.sub.1) antagonists Grant 8,604,200 - Janssens , et al. December 10, 2 | 2013-12-10 |
2-piperazin-1-yl-3H-imidazo[4,5-b]pyridine derivatives Grant 7,994,173 - Janssens , et al. August 9, 2 | 2011-08-09 |
Substituted 1-piperidin-4-yl-4-pyrrolidin-3-yl-piperazine derivatives and their use as neurokinin antagonists Grant 7,795,261 - Janssens , et al. September 14, 2 | 2010-09-14 |
Use of anti-histaminics for acute reduction of elevated intracranial pressure Grant 7,732,437 - Tegtmeier , et al. June 8, 2 | 2010-06-08 |
2-piperazin-1-yl-3h-imidazo[4,5-b]pyridine Derivatives App 20100004260 - Janssens; Frans Eduard | 2010-01-07 |
Substituted diaza-spiro-[4.5]-decane derivatives and their use as neurokinin antagonists Grant 7,612,056 - Janssens , et al. November 3, 2 | 2009-11-03 |
Diaza-spiro--nonane derivatives as neurokinin (nk1) antagonists App 20090221641 - Janssens; Frans Eduard ;   et al. | 2009-09-03 |
Substituted 1-piperidin-3-yl-4-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists Grant 7,572,786 - Janssens , et al. August 11, 2 | 2009-08-11 |
Substituted diaza-spiro-[5.5]-undecane derivatives and their use as neurokinin antagonists Grant 7,544,694 - Janssens , et al. June 9, 2 | 2009-06-09 |
Respiratory syncytial virus replication inhibitors Grant 7,528,149 - Janssens , et al. May 5, 2 | 2009-05-05 |
Substituted 4-(4-piperidin-4-yl-piperazin-1-yl)-azepane derivatives and their use as neurokinin antagonists Grant 7,514,424 - Janssens , et al. April 7, 2 | 2009-04-07 |
Amino-benzimidazoles Derivatives As Inhibitors Of Respiratory Syncytial Virus Replication App 20090036466 - Bonfanti; Jean-Francois ;   et al. | 2009-02-05 |
Substituted tetracyclic imidazole derivatives, processes for their preparation, pharmaceutical compositions comprising them and their use as a medicine Grant 7,476,662 - Janssens , et al. January 13, 2 | 2009-01-13 |
Substituted 1-piperidin-4-yl-4-azetidin-3-yl-piperazine derivatives and their use as neurokinin antagonists Grant 7,435,736 - Janssens , et al. October 14, 2 | 2008-10-14 |
Substituted 1,4,-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists Grant 7,410,970 - Janssens , et al. August 12, 2 | 2008-08-12 |
Respiratory syncytial virus replication inhibitors Grant 7,407,969 - Janssens , et al. August 5, 2 | 2008-08-05 |
Substituted 4-phenyl-4-[1H-imidazol-2-yl]-piperidine derivatives for reducing ischaemic damage Grant 7,390,822 - Janssens , et al. June 24, 2 | 2008-06-24 |
Respiratory syncytial virus replication inhibitors Grant 7,390,811 - Janssens , et al. June 24, 2 | 2008-06-24 |
Piperidine-amino-benzimidazole Derivatives As Inhibitors Of Respiratory Syncytial Virus Replication App 20080146613 - BONFANTI; Jean-Francois ;   et al. | 2008-06-19 |
Novel Substituted 4-Phenyl-4[H-Imidazol-2-YL]-Piperidine Derivatived And Their Use As Selective Non-Peptide Delta Opioid Agonists App 20080096925 - Janssens; Frans Eduard ;   et al. | 2008-04-24 |
Respiratory syncytial virus replication inhibitors Grant 7,361,657 - Janssens , et al. April 22, 2 | 2008-04-22 |
Piperdine-amino-benzimidazole derivatives as inhibitors of respiratory syncytial virus replication Grant 7,355,051 - Bonfanti , et al. April 8, 2 | 2008-04-08 |
Novel Formulations For Opioid-Based Treatments Of Pain Comprising 1-(1,2-Disubstituted Piperidinyl)-4-Substituted Piperazine Derivatives App 20080070924 - Janssens; Frans Eduard ;   et al. | 2008-03-20 |
Substituted homopiperidinyl benzimidazole analogues as fundic relaxants Grant 7,304,052 - Janssens , et al. December 4, 2 | 2007-12-04 |
Substituted Diaza-Spiro-[4.5]-Decane Derivatives and Their Use as Neurokinin Antagonists App 20070254904 - Janssens; Frans Eduard ;   et al. | 2007-11-01 |
Substituted 4-phenyl-4-(1H-imidazol-2-yl)-piperidine derivatives and their use as selective non-peptide delta opioid agonists Grant 7,282,508 - Janssens , et al. October 16, 2 | 2007-10-16 |
Substituted Diaza-Spiro-[5.5]-Undecane Derivaties and Their Use as Neurokinin Antagonists App 20070232636 - Janssens; Frans Eduard ;   et al. | 2007-10-04 |
Substituted 4-Alkyl-And 4-Alkanoyl-Piperidine Derivatives And Their Use As Neurokinin Antagonists App 20070213346 - Janssens; Frans Eduard ;   et al. | 2007-09-13 |
Respiratory Syncytial Virus Replication Inhibitors App 20070135404 - Janssens; Frans Eduard ;   et al. | 2007-06-14 |
Piperdine-amino-benzimidazole derivatives as inhibitors of respiratory syncytial virus replication App 20070093659 - Bonfanti; Jean-Francois ;   et al. | 2007-04-26 |
Respiratory syncytial virus replication inhibitors Grant 7,179,811 - Janssens , et al. February 20, 2 | 2007-02-20 |
Respiratory syncytial virus replication inhibitors Grant 7,173,034 - Janssens , et al. February 6, 2 | 2007-02-06 |
Respiratory syncytial virus replication inhibitors Grant 7,173,054 - Janssens , et al. February 6, 2 | 2007-02-06 |
Respiratory syncytial virus replication inhibitors App 20070021410 - Janssens; Frans Eduard ;   et al. | 2007-01-25 |
Respiratory Syncytial Virus Replication Inhibitors App 20070015747 - Janssens; Frans Eduard ;   et al. | 2007-01-18 |
Substituted 4-phenyl-4-[1h-imidazol-2-yl]-piperidine derivatives as selective non-peptide delta opiod agonists with antidepressant and anxiolytic activity App 20060287345 - Steckler; Thomas Horst Wolfgang ;   et al. | 2006-12-21 |
Antihistaminic spiro compounds Grant 7,148,214 - Janssens , et al. December 12, 2 | 2006-12-12 |
Antihistaminic spiro compounds Grant 7,087,595 - Janssens , et al. August 8, 2 | 2006-08-08 |
Substituted 1,4,-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists App 20060167008 - Janssens; Frans Eduard ;   et al. | 2006-07-27 |
Respiratory syncytial virus replication inhibitors App 20060154913 - Janssens; Frans Eduard ;   et al. | 2006-07-13 |
Respiratory syncytial virus replication inhibitors Grant 7,071,192 - Janssens , et al. July 4, 2 | 2006-07-04 |
Novel formulations of opioid-based treatments of pain comprising substituted 1,4-di-piperidin-4-yl-piperazine derivatives App 20060128721 - Janssens; Frans Eduard ;   et al. | 2006-06-15 |
Substituted 1-piperidin-4-yl-4-azetidin-3-yl-piperazine derivatives and their use as neurokinin antagonists App 20060074069 - Janssens; Frans Eduard ;   et al. | 2006-04-06 |
Respiratory syncytial virus replication inhibitors App 20060058309 - Janssens; Frans Eduard ;   et al. | 2006-03-16 |
Substituted 4-(4-piperidin-4-yl-piperazin-1-yl)-azepane derivatives and their use as neurokinin antagonists App 20060058285 - Janssens; Frans Eduard ;   et al. | 2006-03-16 |
Substituted 1-piperidin-4-yl-4-pyrrolidin-3-yl-piperazine derivatives and their use as neurokinin antagonists App 20060040950 - Janssens; Frans Eduard ;   et al. | 2006-02-23 |
Respiratory syncytial virus replication inhibitors App 20050239771 - Janssens, Frans Eduard ;   et al. | 2005-10-27 |
Respiratory syncytial virus replication inhibitors App 20050234047 - Janssens, Frans Eduard ;   et al. | 2005-10-20 |
Respiratory syncytial virus replication inhibitors Grant 6,924,287 - Janssens , et al. August 2, 2 | 2005-08-02 |
Use of anti-histaminics for acute reduction of elevated intracranial pressure App 20050070525 - Tegtmeier, Frank ;   et al. | 2005-03-31 |
Antihistaminic spiro compounds App 20050026901 - Janssens, Frans Eduard ;   et al. | 2005-02-03 |
Substituted 4-phenyl-4-[1h-imidazol-2-yl]-piperidine derivatives for reducing ischaemic damage App 20050004170 - Janssens, Frans Eduard ;   et al. | 2005-01-06 |
Novel substituted 4-phenyl-4-{1h-imidazol-2-yl}-piperidine derivatives and their use as selective non-peptide delta opioid agonists App 20040260096 - Janssens, Frans Eduard ;   et al. | 2004-12-23 |
Novel substituted tetracyclic imidazole derivatives, processes for their preparation, pharamaceutical compositions comprising them and their use as a medicine App 20040167138 - Janssens, Frans Eduard ;   et al. | 2004-08-26 |
Respiratory syncytial virus replication inhibitors Grant 6,747,028 - Janssens , et al. June 8, 2 | 2004-06-08 |
Substituted homopiperidinyl benzimidazole analogues as fundic relaxants App 20030139393 - Janssens, Frans Eduard ;   et al. | 2003-07-24 |
Fused imidazole derivatives as multidrug resistance modulators App 20030087895 - Janssens, Frans Eduard ;   et al. | 2003-05-08 |
1-(1,2-disubstituted piperidinyl)-4-substituted piperazine derivatives Grant 6,521,621 - Janssens , et al. February 18, 2 | 2003-02-18 |
1- (1,2-disubstituted piperidinyl) -4-substituted piperazine derivatives Grant 6,197,772 - Janssens , et al. March 6, 2 | 2001-03-06 |
1-(1,2-Disubstituted piperidinyl)-4-substituted piperidine derivatives Grant 6,169,097 - Janssens , et al. January 2, 2 | 2001-01-02 |
Triazolobenzazepine derivatives Grant 5,932,569 - Janssens , et al. August 3, 1 | 1999-08-03 |