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Macrocycles as factor XIA inhibitors Grant 11,136,327 - Corte , et al. October 5, 2 | 2021-10-05 |
Lactam, cyclic urea and carbamate, and triazolone derivatives as potent and selective rock inhibitors Grant 10,730,858 - Hu , et al. | 2020-08-04 |
Macrocycles As Factor Xia Inhibitors App 20200087312 - Corte; James R. ;   et al. | 2020-03-19 |
Macrocycles as factor XIa inhibitors Grant 10,487,086 - Corte , et al. Nov | 2019-11-26 |
Lactam, Cyclic Urea And Carbamate, And Triazolone Derivatives As Potent And Selective Rock Inhibitors App 20190300510 - Hu; Zilun ;   et al. | 2019-10-03 |
Tied-back benzamide derivatives as potent rock inhibitors Grant 10,112,939 - Hu , et al. October 30, 2 | 2018-10-30 |
Diamide macrocycles that are FXIa inhibitors Grant 10,081,623 - Shi , et al. September 25, 2 | 2018-09-25 |
Spirocycloheptanes As Inhibitors Of Rock App 20180155296 - Ladziata; Vladimir ;   et al. | 2018-06-07 |
Tricyclic pyrido-carboxamide derivatives as rock inhibitors Grant 9,914,740 - Quan , et al. March 13, 2 | 2018-03-13 |
Spirocycloheptanes as inhibitors of rock Grant 9,902,702 - Ladziata , et al. February 27, 2 | 2018-02-27 |
Macrocycles As Factor Xia Inhibitors App 20180022753 - Corte; James R. ;   et al. | 2018-01-25 |
Phenylpyrazole derivatives as potent ROCK1 and ROCK2 inhibitors Grant 9,828,345 - Hu , et al. November 28, 2 | 2017-11-28 |
Macrocycles as factor XIa inhibitors Grant 9,802,939 - Corte , et al. October 31, 2 | 2017-10-31 |
Diamide Macrocycles That Are Fxia Inhibitors App 20170283403 - Shi; Jun ;   et al. | 2017-10-05 |
Tied-back Benzamide Derivatives As Potent Rock Inhibitors App 20170226105 - Hu; Zilun ;   et al. | 2017-08-10 |
Tricyclic pyrido-carboxamide derivatives as rock inhibitors Grant 9,663,529 - Quan , et al. May 30, 2 | 2017-05-30 |
Phenylpyrazole derivatives as potent ROCK1 and ROCK2 inhibitors Grant 9,458,110 - Quan , et al. October 4, 2 | 2016-10-04 |
Tricyclic Pyrido-carboxamide Derivatives As Rock Inhibitors App 20160152627 - Quan; Mimi L. ;   et al. | 2016-06-02 |
Tricyclic Pyrido-carboxamide Derivatives As Rock Inhibitors App 20160152628 - Quan; Mimi L. ;   et al. | 2016-06-02 |
Phenylpyrazole Derivatives As Potent Rock1 And Rock2 Inhibitors App 20160016910 - Quan; Mimi L. ;   et al. | 2016-01-21 |
Spirocycloheptanes As Inhibitors Of Rock App 20160016914 - Ladziata; Vladimir ;   et al. | 2016-01-21 |
Phenylpyrazole Derivatives As Potent Rock1 And Rock2 Inhibitors App 20160002172 - Hu; Zilun ;   et al. | 2016-01-07 |
Phenylpyrazole derivatives as potent ROCK1 and ROCK2 inhibitors Grant 9,126,944 - Quan , et al. September 8, 2 | 2015-09-08 |
Macrocycles As Factor Xia Inhibitors App 20150112058 - Corte; James R. ;   et al. | 2015-04-23 |
Macrocycles as factor XIa inhibitors Grant 8,940,720 - Corte , et al. January 27, 2 | 2015-01-27 |
Phenylpyrazole Derivatives As Potent Rock1 And Rock2 Inhibitors App 20140243338 - Quan; Mimi L. ;   et al. | 2014-08-28 |
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 8,604,056 - Pinto , et al. December 10, 2 | 2013-12-10 |
Pyridazine derivatives as factor xia inhibitors Grant 8,324,199 - Corte , et al. December 4, 2 | 2012-12-04 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20120270853 - Pinto; Donald J.P. ;   et al. | 2012-10-25 |
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 8,252,830 - Pinto , et al. August 28, 2 | 2012-08-28 |
Macrocycles As Factor Xia Inhibitors App 20120041190 - Corte; James R. ;   et al. | 2012-02-16 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20110028446 - Pinto; Donald J.P. ;   et al. | 2011-02-03 |
Pyridazine Derivatives As Factor Xia Inhibitors App 20110021492 - Corte; James R. ;   et al. | 2011-01-27 |
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 7,842,708 - Pinto , et al. November 30, 2 | 2010-11-30 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20100022506 - Pinto; Donald J.P. ;   et al. | 2010-01-28 |
Arylpropionamide, arylacrylamide, ayrlpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 7,626,039 - Pinto , et al. December 1, 2 | 2009-12-01 |
Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors Grant 7,524,863 - Smallheer , et al. April 28, 2 | 2009-04-28 |
Substituted pyrazolo[1,5-a]pyrimidines as potassium channel activators Grant 7,507,730 - Han , et al. March 24, 2 | 2009-03-24 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20080161373 - Pinto; Donald J.P. ;   et al. | 2008-07-03 |
Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors Grant 7,312,218 - Han , et al. December 25, 2 | 2007-12-25 |
Heterocyclic dihydropyrimidine compounds App 20070203157 - Han; Wei ;   et al. | 2007-08-30 |
Sulfonylaminovalerolactams And Derivatives Thereof As Factor Xa Inhibitors App 20070099922 - Han; Wei ;   et al. | 2007-05-03 |
Monocyclic and bicyclic lactams as factor Xa inhibitors Grant 7,199,149 - Han , et al. April 3, 2 | 2007-04-03 |
Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors Grant 7,169,795 - Han , et al. January 30, 2 | 2007-01-30 |
Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors Grant 7,157,470 - Smallheer , et al. January 2, 2 | 2007-01-02 |
Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors App 20060247243 - Smallheer; Joanne M. ;   et al. | 2006-11-02 |
Glycinamides as factor Xa inhibitors Grant 7,115,627 - Pinto , et al. October 3, 2 | 2006-10-03 |
Monocyclic and bicyclic lactams as factor Xa inhibitors App 20050107361 - Han, Wei ;   et al. | 2005-05-19 |
Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors App 20050096309 - Han, Wei ;   et al. | 2005-05-05 |
Quinazolinones and derivatives thereof as factor Xa inhibitors App 20040132732 - Han, Wei ;   et al. | 2004-07-08 |
Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors App 20040006062 - Smallheer, Joanne M. ;   et al. | 2004-01-08 |
Glycinamides as factor Xa inhibitors App 20030232804 - Pinto, Donald J.P. ;   et al. | 2003-12-18 |