Patent | Date |
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Substituted pyrrolidines as G-protein coupled receptor 43 agonists Grant 11,072,582 - Hoveyda , et al. July 27, 2 | 2021-07-27 |
NOVEL N-ACYL-[3-SUBSTITUTED]-[8-SUBSTITUTED]-5,6-DIHYDRO-[1,2,4]TRIAZOLO[4- ,3-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR-MEDIATED DISORDERS App 20210094959 - Hoveyda; Hamid R. ;   et al. | 2021-04-01 |
Chiral N-acyl-5,6,7(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazi- nes as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor mediated disorders and chiral synthesis thereof Grant 10,941,151 - Hoveyda , et al. March 9, 2 | 2021-03-09 |
Substituted Pyrrolidines As G-protein Coupled Receptor 43 Agonists App 20200347016 - Hoveyda; Hamid R. ;   et al. | 2020-11-05 |
Substituted pyrrolidines as G-protein coupled receptor 43 agonists Grant 10,781,171 - Hoveyda , et al. Sept | 2020-09-22 |
Novel Chiral N-acyl-5,6,7(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines As Selective Nk-3 Receptor Antagonists, Phar App 20200283447 - Hoveyda; Hamid R. ;   et al. | 2020-09-10 |
Chiral N-acyl-5,6,7(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-A]pyrazi- nes as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor mediated disorders and chiral synthesis thereof Grant 10,683,295 - Hoveyda , et al. | 2020-06-16 |
Pyrrolidine Or Thiazolidine Carboxylic Acid Derivatives, Pharmaceutical Composition And Methods For Use In Treating Metabolic Di App 20200148636 - Hoveyda; Hamid R. ;   et al. | 2020-05-14 |
Novel Nk-3 Receptor Selective Antagonist Compounds, Pharmaceutical Composition And Methods For Use In Nk-3 Receptors Mediated Di App 20200125564 - Hoveyda; Hamid R. ;   et al. | 2020-04-23 |
Substituted pyrrolidines as G-protein coupled receptor 43 agonists Grant 10,577,318 - Hoveyda , et al. | 2020-03-03 |
NK-3 receptor selective antagonist compounds, pharmaceutical composition and methods for use in NK-3 receptors mediated disorders Grant 10,544,150 - Hoveyda , et al. Ja | 2020-01-28 |
Substituted Pyrrolidines As G-protein Coupled Receptor 43 Agonists App 20190300478 - Hoveyda; Hamid R. ;   et al. | 2019-10-03 |
Substituted pyrrolidines as G-protein coupled receptor 43 agonists Grant 10,358,416 - Hoveyda , et al. July 23, 2 | 2019-07-23 |
Novel Chiral N-acyl-5,6,7(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines As Selective Nk-3 Receptor Antagonists, Pharmaceutical Composition, Methods For Use In Nk-3 Receptor Mediated Disorders And Chiral Synthesis Thereof App 20190023711 - Hoveyda; Hamid R. ;   et al. | 2019-01-24 |
Substituted Pyrrolidines As G-protein Coupled Receptor 43 Agonists App 20180297944 - Hoveyda; Hamid R. ;   et al. | 2018-10-18 |
Chiral N-acyl-5,6,7,(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyraz- ines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor mediated disorders and chiral synthesis thereof Grant 10,065,961 - Hoveyda , et al. September 4, 2 | 2018-09-04 |
NK-3 receptor selective antagonist compounds, pharmaceutical composition and methods for use in NK-3 receptors mediated disorders Grant 10,065,960 - Hoveyda , et al. September 4, 2 | 2018-09-04 |
Novel Nk-3 Receptor Selective Antagonist Compounds, Pharmaceutical Composition And Methods For Use In Nk-3 Receptors Mediated Disorders App 20180194772 - Hoveyda; Hamid R. ;   et al. | 2018-07-12 |
Substituted pyrrolidines as G-protein coupled receptor 43 agonists Grant 10,017,468 - Hoveyda , et al. July 10, 2 | 2018-07-10 |
Macrocyclic Modulators of the Ghrelin Receptor App 20180110824 - Hoveyda; Hamid R. ;   et al. | 2018-04-26 |
NK-3 receptor selective antagonist compounds, pharmaceutical composition and methods for use in NK-3 receptors mediated disorders Grant 9,926,325 - Hoveyda , et al. March 27, 2 | 2018-03-27 |
Substituted Pyrrolidines As G-protein Coupled Receptor 43 Agonists App 20170283376 - Hoveyda; Hamid R. ;   et al. | 2017-10-05 |
Substituted pyrrolidines as G-protein coupled receptor 43 agonists Grant 9,695,120 - Hoveyda , et al. July 4, 2 | 2017-07-04 |
Chiral N-acyl-5,6,7(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazi- nes as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor mediated disorders and chiral synthesis thereof Grant 9,475,814 - Hoveyda , et al. October 25, 2 | 2016-10-25 |
Novel Nk-3 Receptor Selective Antagonist Compounds, Pharmaceutical Composition And Methods For Use In Nk-3 Receptors Mediated Disorders App 20150315199 - Hoveyda; Hamid R. ;   et al. | 2015-11-05 |
Novel Nk-3 Receptor Selective Antagonist Compounds, Pharmaceutical Composition And Methods For Use In Nk-3 Receptors Mediated Disorders App 20140371218 - Hoveyda; Hamid R. ;   et al. | 2014-12-18 |
NK-3 receptor selective antagonist compounds, pharmaceutical composition and methods for use in NK-3 receptors mediated disorders Grant 8,871,761 - Hoveyda , et al. October 28, 2 | 2014-10-28 |
NOVEL CHIRAL N-ACYL-5,6,7(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF App 20140275097 - Hoveyda; Hamid R. ;   et al. | 2014-09-18 |
Spatially-defined macrocycles incorporating peptide bond surrogates Grant 8,557,765 - Deslongchamps , et al. October 15, 2 | 2013-10-15 |
Processes for intermediates for macrocyclic compounds Grant 8,497,242 - Marsault , et al. July 30, 2 | 2013-07-30 |
Methods of using macrocyclic modulators of the ghrelin receptor Grant 8,450,268 - Fraser , et al. May 28, 2 | 2013-05-28 |
Spatially-defined macrocyclic compounds useful for drug discovery Grant 8,440,851 - Marsault , et al. May 14, 2 | 2013-05-14 |
Pyrrolidine Or Thiazolidine Carboxylic Acid Derivatives, Pharmaceutical Composition And Methods For Use In Treating Metabolic Disorders As Agonists Of G-protein Coupled Receptor 43 (gpr43) App 20130023539 - Hoveyda; Hamid R. ;   et al. | 2013-01-24 |
Novel Nk-3 Receptor Selective Antagonist Compounds, Pharmaceutical Composition And Methods For Use In Nk-3 Receptors Mediated Disorders App 20130023530 - Hoveyda; Hamid R. ;   et al. | 2013-01-24 |
Methods of treating cachexia with macrocyclic modulators of the ghrelin receptor Grant 8,349,887 - Fraser , et al. January 8, 2 | 2013-01-08 |
Processes For Intermediates For Macrocyclic Compounds App 20120226067 - Marsault; Eric ;   et al. | 2012-09-06 |
Processes For Intermediates For Macrocyclic Compounds App 20120226072 - Marsault; Eric ;   et al. | 2012-09-06 |
Processes For Intermediates For Macrocyclic Compounds App 20120226066 - Marsault; Eric ;   et al. | 2012-09-06 |
Processes For Intermediates For Macrocyclic Compounds App 20120165566 - Marsault; Eric ;   et al. | 2012-06-28 |
Methods Of Using Macrocyclic Agonists Of The Ghrelin Receptor For Treatment Of Gastrointestinal Motility Disorders App 20120071412 - Fraser; Graeme L. ;   et al. | 2012-03-22 |
Processes for intermediates for macrocyclic compounds Grant 8,129,561 - Marsault , et al. March 6, 2 | 2012-03-06 |
Methods of using macrocyclic agonists of the ghrelin receptor for treatment of gastrointestinal motility disorders Grant 8,088,733 - Fraser , et al. January 3, 2 | 2012-01-03 |
Methods Of Using Macrocyclic Modulators Of The Ghrelin Receptor App 20110288163 - Fraser; Graeme L. ;   et al. | 2011-11-24 |
Salts, Solvates and Pharmaceutical Compositions of Macrocyclic Ghrelin Receptor Agonists and Methods of Using the Same App 20110245159 - Hoveyda; Hamid R. ;   et al. | 2011-10-06 |
Processes for Intermediates for Macrocyclic Compounds App 20110245459 - Marsault; Eric ;   et al. | 2011-10-06 |
Spatially-defined Macrocyclic Compounds Useful For Drug Discovery App 20110237785 - Marsault; Eric ;   et al. | 2011-09-29 |
Spatially-defined macrocyclic compounds useful for drug discovery Grant 8,022,252 - Deslongchamps , et al. September 20, 2 | 2011-09-20 |
Methods of using macrocyclic modulators of the ghrelin receptor Grant RE42,624 - Fraser , et al. August 16, 2 | 2011-08-16 |
Macrocyclic Ghrelin Receptor Antagonists and Inverse Agonists and Methods of Using the Same App 20110105389 - Hoveyda; Hamid R. ;   et al. | 2011-05-05 |
Spatially-defined Macrocycles Incorporating Peptide Bond Surrogates App 20090312540 - Deslongchamps; Pierre ;   et al. | 2009-12-17 |
Macrocyclic Ghrelin Receptor Antagonists And Inverse Agonists And Methods Of Using The Same App 20090275648 - Fraser; Graeme L. ;   et al. | 2009-11-05 |
Intermediates For Macrocyclic Compounds App 20090240027 - Marsault; Eric ;   et al. | 2009-09-24 |
Macrocyclic Modulators of the Ghrelin Receptor App 20090198050 - Marsault; Eric ;   et al. | 2009-08-06 |
Methods Of Using Macrocyclic Modulators Of The Ghrelin Receptor App 20090170757 - Fraser; Graeme L. ;   et al. | 2009-07-02 |
Spatially-defined macrocycles incorporating peptide bond surrogates Grant 7,550,431 - Deslongchamps , et al. June 23, 2 | 2009-06-23 |
Spatially-defined Macrocyclic Compounds Useful For Drug Discovery App 20090137817 - Deslongchamps; Pierre ;   et al. | 2009-05-28 |
Processes For Intermediates For Macrocyclic Compounds App 20090137835 - Marsault; Eric ;   et al. | 2009-05-28 |
Use of Piperidine Derivatives as Agonists of Chemokine Receptor Activity App 20090054451 - Huck; Jacques ;   et al. | 2009-02-26 |
Novel Piperidine-4-Acetic Acid Derivatives and Their Use App 20090048291 - Huck; Jacques ;   et al. | 2009-02-19 |
Methods of using macrocyclic modulators of the ghrelin receptor Grant 7,491,695 - Fraser , et al. February 17, 2 | 2009-02-17 |
Macrocyclic modulators of the ghrelin receptor Grant 7,476,653 - Hoveyda , et al. January 13, 2 | 2009-01-13 |
Methods Of Using Macrocyclic Agonists Of The Ghrelin Receptor For Treatment Of Gastrointestinal Motility Disorders App 20080051383 - Fraser; Graeme L. ;   et al. | 2008-02-28 |
Methods of using macrocyclic modulators of the ghrelin receptor App 20070021331 - Fraser; Graeme L. ;   et al. | 2007-01-25 |
Macrocyclic modulators of the ghrelin receptor App 20060025566 - Hoveyda; Hamid R. ;   et al. | 2006-02-02 |