Patent applications and USPTO patent grants for Heptares Therapeutics Limited.The latest application filed is for "cgrp antagonist compounds".
Patent | Date |
---|---|
Cgrp Antagonist Compounds App 20220306651 - Brown; Giles Albert ;   et al. | 2022-09-29 |
Oxime Compounds As Agonists Of The Muscarinic M1 And/or M4 Receptor App 20220298133 - Brown; Giles Albert ;   et al. | 2022-09-22 |
Cgrp Antagonist Compounds App 20220251110 - Brown; Giles Albert ;   et al. | 2022-08-11 |
Substituted Cyclohexanes As Muscarinic M1 Receptor And/or M4 Receptor Agonists App 20220213034 - Brown; Giles Albert ;   et al. | 2022-07-07 |
Pharmaceutical compounds Grant 11,352,342 - Brown , et al. June 7, 2 | 2022-06-07 |
G proteins Grant 11,339,383 - Carpenter , et al. May 24, 2 | 2022-05-24 |
Muscarinic agonists Grant 11,324,738 - Brown , et al. May 10, 2 | 2022-05-10 |
Pharmaceutical compounds Grant 11,319,312 - Brown , et al. May 3, 2 | 2022-05-03 |
Oxexin 1 Receptor Antagonists App 20220098165 - Brown; Giles Albert ;   et al. | 2022-03-31 |
4-(3-cyanophenyl)-6-pyridinylpyrimidine Mglu5 Modulators App 20220056009 - CHRISTOPHER; John Andrew ;   et al. | 2022-02-24 |
Muscarinic agonists Grant 11,254,656 - Brown , et al. February 22, 2 | 2022-02-22 |
Muscarinic Receptor Agonists App 20220048928 - Congreve; Miles Stuart ;   et al. | 2022-02-17 |
Orexin 1 Receptor Antagonists App 20220041573 - Brown; Giles Albert ;   et al. | 2022-02-10 |
Oxime compounds as agonists of the muscarinic M1 and/or M4 receptor Grant 11,208,396 - Brown , et al. December 28, 2 | 2021-12-28 |
Bicyclic Aza Compounds As Muscarinic M1 And/or M4 Receptor Agonists App 20210387969 - Brown; Giles Albert ;   et al. | 2021-12-16 |
Cyclohexapeptides As Selective Somatostatin Sst5 Receptor Agonists App 20210363188 - Brown; Giles Albert ;   et al. | 2021-11-25 |
Muscarinic M1 Receptor Agonists App 20210353637 - Congreve; Miles Stuart ;   et al. | 2021-11-18 |
Glp-1 Receptor Antagonists App 20210355186 - Brown; Giles Albert ;   et al. | 2021-11-18 |
4-(3-cyanophenyl)-6-pyridinylpyrimidine Mglu5 Modulators App 20210309632 - Christopher; John Andrew ;   et al. | 2021-10-07 |
Pyrazole Derivatives As H4 Antagonist Compounds App 20210300906 - Brown; Giles Albert ;   et al. | 2021-09-30 |
Muscarinic agonists Grant 11,091,456 - Brown , et al. August 17, 2 | 2021-08-17 |
Cgrp Receptor Antagonists App 20210213011 - Christopher; John Andrew ;   et al. | 2021-07-15 |
Ox1 Antagonists App 20210179578 - Christopher; John Andrew ;   et al. | 2021-06-17 |
Muscarinic receptor agonists Grant 11,034,704 - Congreve , et al. June 15, 2 | 2021-06-15 |
Substituted cyclohexanes as muscarinic M1 receptor and/or M4 receptor agonists Grant 11,014,880 - Brown , et al. May 25, 2 | 2021-05-25 |
Methods For Screening For Binding Partners Of G-protein Coupled Receptors App 20210148939 - Weir; Malcolm Peter ;   et al. | 2021-05-20 |
Inhibitors of protease-activated receptor-2 Grant 10,995,072 - Cumming , et al. May 4, 2 | 2021-05-04 |
1,2,4-triazine-4-amine derivatives Grant 10,988,455 - Congreve , et al. April 27, 2 | 2021-04-27 |
4-(3-cyanophenyl)-6-pyridinylpyrimidine mGlu5 modulators Grant 10,981,889 - Christopher , et al. April 20, 2 | 2021-04-20 |
Muscarinic M1 receptor agonists Grant 10,973,832 - Congreve , et al. April 13, 2 | 2021-04-13 |
Pharmaceutical Compounds App 20210101893 - Brown; Giles Albert ;   et al. | 2021-04-08 |
Bicyclic AZA compounds as muscarinic M1 receptor and/or M4 receptor Grant 10,961,225 - Brown , et al. March 30, 2 | 2021-03-30 |
Mutant G-protein Coupled Receptors And Methods For Selecting Them App 20210061882 - Henderson; Richard ;   et al. | 2021-03-04 |
Pharmaceutical Compounds App 20210040067 - Brown; Giles Albert ;   et al. | 2021-02-11 |
CGRP receptor antagonists Grant 10,888,561 - Christopher , et al. January 12, 2 | 2021-01-12 |
Pharmaceutical Compounds App 20210002271 - Brown; Giles Albert ;   et al. | 2021-01-07 |
Pharmaceutical compounds Grant 10,858,352 - Brown , et al. December 8, 2 | 2020-12-08 |
Muscarinic Agonists App 20200354339 - Brown; Giles Albert ;   et al. | 2020-11-12 |
Bicyclic Aza Compounds As Muscarinic M1 Receptor And/or M4 Receptor App 20200325118 - Brown; Giles Albert ;   et al. | 2020-10-15 |
Pharmaceutical compounds Grant 10,787,447 - Brown , et al. September 29, 2 | 2020-09-29 |
Substituted Cyclohexanes As Muscarinic M1 Receptor And/or M4 Receptor Agonists App 20200290963 - Brown; Giles Albert ;   et al. | 2020-09-17 |
Stable proteins Grant 10,766,945 - Jazayeri-Dezfuly , et al. Sep | 2020-09-08 |
Substituted spirocyclohexanes as muscarinic M.sub.1 receptor and/or M.sub.4 receptor agonists Grant 10,759,751 - Brown , et al. Sep | 2020-09-01 |
Pharmaceutical compounds Grant 10,752,610 - Brown , et al. A | 2020-08-25 |
Muscarinic M1 Receptor Agonists App 20200253982 - Kind Code | 2020-08-13 |
Muscarinic agonists Grant 10,738,029 - Brown , et al. A | 2020-08-11 |
G proteins Grant 10,738,287 - Carpenter , et al. A | 2020-08-11 |
G Proteins App 20200231949 - Carpenter; Byron ;   et al. | 2020-07-23 |
Use of glycopyrrolate for treating tachycardia Grant 10,695,321 - Snape , et al. | 2020-06-30 |
Bicyclic aza compounds as muscarinic M1 receptor and/or M4 receptor Grant 10,689,368 - Brown , et al. | 2020-06-23 |
4-(3-cyanophenyl)-6-pyridinylpyrimidine Mglu5 Modulators App 20200172505 - Christopher; John Andrew ;   et al. | 2020-06-04 |
Oxime Compounds As Agonists Of The Muscarinic M1 And/or M4 Receptor App 20200165220 - Brown; Giles Albert ;   et al. | 2020-05-28 |
Inhibitors Of Protease-activated Receptor-2 App 20200140392 - Cumming; John Graham ;   et al. | 2020-05-07 |
Muscarinic Agonists App 20200129496 - Brown; Giles Albert ;   et al. | 2020-04-30 |
4-(3-cyanophenyl)-6-pyridinylpyrimidine mGlu5 modulators Grant 10,584,111 - Christopher , et al. | 2020-03-10 |
Muscarinic agonists Grant 10,548,884 - Brown , et al. Fe | 2020-02-04 |
Inhibitors of protease-activated receptor-2 Grant 10,550,089 - Cumming , et al. Fe | 2020-02-04 |
Muscarinic Receptor Agonists App 20200017530 - Congreve; Miles Stuart ;   et al. | 2020-01-16 |
Pharmaceutical Compounds App 20200002328 - Brown; Giles Albert ;   et al. | 2020-01-02 |
Pharmaceutical Compounds App 20190389849 - Brown; Giles Albert ;   et al. | 2019-12-26 |
Bicyclic Aza Compounds As Muscarinic M1 Receptor And/or M4 Receptor App 20190337925 - Brown; Giles Albert ;   et al. | 2019-11-07 |
Assay for assessing conformational stability of membrane protein Grant 10,458,993 - Marshall , et al. Oc | 2019-10-29 |
Muscarinic receptor agonists Grant 10,428,088 - Congreve , et al. October 1, 2 | 2019-10-01 |
Muscarinic M1 receptor agonists Grant 10,413,553 - Congreve , et al. Sept | 2019-09-17 |
Pharmaceutical Compounds App 20190276437 - Brown; Giles Albert ;   et al. | 2019-09-12 |
Muscarinic Agonists App 20190270718 - Brown; Giles Albert ;   et al. | 2019-09-05 |
Bicyclic aza compounds as muscarnic M1 receptor and/or M4 receptor antagonists Grant 10,385,039 - Brown , et al. A | 2019-08-20 |
Mutant G-protein Coupled Receptors And Methods For Selecting Them App 20190241644 - Henderson; Richard ;   et al. | 2019-08-08 |
Cgrp Receptor Antagonists App 20190231773 - Christopher; John Andrew ;   et al. | 2019-08-01 |
Muscarinic agonists Grant 10,351,545 - Brown , et al. July 16, 2 | 2019-07-16 |
Substituted Cyclohexanes As Muscarinic M1 Receptor And/or M4 Receptor Agonists App 20190202783 - Brown; Giles Albert ;   et al. | 2019-07-04 |
Pharmaceutical compounds Grant 10,329,278 - Brown , et al. | 2019-06-25 |
4-(3-cyanophenyl)-6-pyridinylpyrimidine Mglu5 Modulators App 20190177297 - Christopher; John Andrew ;   et al. | 2019-06-13 |
Orexin receptor antagonists Grant 10,316,028 - Congreve , et al. | 2019-06-11 |
CGRP receptor antagonists Grant 10,300,056 - Christopher , et al. | 2019-05-28 |
Inhibitors Of Protease-activated Receptor-2 App 20190144394 - Cumming; John Graham ;   et al. | 2019-05-16 |
Bicyclic Aza Compounds As Muscarnic M1 Receptor And/or M4 Receptor Antagonists App 20190112294 - Brown; Giles Albert ;   et al. | 2019-04-18 |
Stable Proteins App 20190112355 - Jazayeri-Dezfuly; Seyed Ali ;   et al. | 2019-04-18 |
Substituted cyclohexanes as muscarinic M1 receptor and/or M4 receptor agonists Grant 10,259,787 - Brown , et al. | 2019-04-16 |
Bicyclic aza compounds as muscarinic M1 receptor antagonists Grant 10,259,802 - Brown , et al. | 2019-04-16 |
CGRP receptor antagonists Grant 10,259,812 - Christopher , et al. | 2019-04-16 |
4-(3-cyanophenyl)-6-pyridinylpyrimidine mGlu5 modulators Grant 10,246,432 - Christopher , et al. | 2019-04-02 |
Methods For Screening For Binding Partners Of G-protein Coupled Receptors App 20190094247 - Weir; Malcolm Peter ;   et al. | 2019-03-28 |
1,2,4-triazine-4-amine Derivatives App 20190047978 - Congreve; Miles Stuart ;   et al. | 2019-02-14 |
Bicyclic aza compounds as muscarinic M1 receptor and/or M4 receptor agonists Grant 10,196,380 - Brown , et al. Fe | 2019-02-05 |
G Proteins App 20190032033 - Carpenter; Byron ;   et al. | 2019-01-31 |
Stable proteins Grant 10,174,101 - Jazayeri-Dezfuly , et al. J | 2019-01-08 |
CGRP receptor antagonists Grant 10,166,226 - Christopher , et al. J | 2019-01-01 |
Muscarinic agonists Grant 10,167,272 - Brown , et al. J | 2019-01-01 |
Spirocyclic compounds as agonists of the muscarinic M.sub.1 receptor and/or M.sub.4 receptor Grant 10,167,284 - Congreve , et al. J | 2019-01-01 |
Orexin Receptor Antagonists App 20180370961 - Congreve; Miles Stuart ;   et al. | 2018-12-27 |
Pharmaceutical Compounds App 20180362507 - Brown; Giles Albert ;   et al. | 2018-12-20 |
Muscarinic Receptor Agonists App 20180327426 - Congreve; Miles Stuart ;   et al. | 2018-11-15 |
Methods for screening for binding partners of G-protein coupled receptors Grant 10,126,313 - Weir , et al. November 13, 2 | 2018-11-13 |
1,2,4-triazine-4-amine derivatives Grant 10,112,923 - Congreve , et al. October 30, 2 | 2018-10-30 |
Bicyclic Aza Compounds As Muscarinic M1 Receptor Antagonists App 20180258085 - Brown; Giles Albert ;   et al. | 2018-09-13 |
Muscarinic Agonists App 20180228791 - Brown; Giles Albert ;   et al. | 2018-08-16 |
Muscarinic Agonists App 20180222885 - Brown; Giles Albert ;   et al. | 2018-08-09 |
Piperidin-1-yl and azepin-1-yl carboxylates as muscarinic M4 receptor agonists Grant 10,030,012 - Livermore , et al. July 24, 2 | 2018-07-24 |
Muscarinic receptor agonists Grant 10,030,035 - Congreve , et al. July 24, 2 | 2018-07-24 |
Bicyclic Aza Compounds As Muscarinic M1 Receptor And/or M4 Receptor Agonists App 20180179184 - Brown; Giles Albert ;   et al. | 2018-06-28 |
Muscarinic Agonists App 20180155315 - Brown; Giles Albert ;   et al. | 2018-06-07 |
Muscarinic M1 Receptor Agonists App 20180153900 - Congreve; Miles Stuart ;   et al. | 2018-06-07 |
CGRP Receptor Antagonists App 20180153876 - Christopher; John Andrew ;   et al. | 2018-06-07 |
Bicyclic AZA compounds as muscarinic M1 receptor antagonists Grant 9,975,890 - Brown , et al. May 22, 2 | 2018-05-22 |
Pharmaceutical Compounds App 20180105491 - Brown; Giles Albert ;   et al. | 2018-04-19 |
Mutant G-protein Coupled Receptors And Methods For Selecting Them App 20180086814 - Henderson; Richard ;   et al. | 2018-03-29 |
CGRP receptor antagonists Grant 9,925,178 - Christopher , et al. March 27, 2 | 2018-03-27 |
Bicyclic AZA compounds as muscarinic M1 receptor and/or M4 receptor agonists Grant 9,926,297 - Brown , et al. March 27, 2 | 2018-03-27 |
Spirocyclic Compounds As Agonists Of The Muscarinic M1 Receptor And/or M4 Receptor App 20180072727 - Congreve; Miles Stuart ;   et al. | 2018-03-15 |
Muscarinic M1 receptor agonists Grant 9,907,805 - Congreve , et al. March 6, 2 | 2018-03-06 |
Muscarinic Agonists App 20180022726 - Brown; Giles Albert ;   et al. | 2018-01-25 |
CGRP Receptor Antagonists App 20180015085 - Christopher; John Andrew ;   et al. | 2018-01-18 |
CGRP Receptor Antagonists App 20180009808 - Christopher; John Andrew ;   et al. | 2018-01-11 |
Orexin receptor antagonists Grant 9,850,237 - Congreve , et al. December 26, 2 | 2017-12-26 |
CGRP receptor antagonists Grant 9,808,457 - Christopher , et al. November 7, 2 | 2017-11-07 |
CGRP receptor antagonists Grant 9,802,935 - Christopher , et al. October 31, 2 | 2017-10-31 |
1,2,4-triazine-4-amine Derivatives App 20170291888 - Congreve; Miles Stuart ;   et al. | 2017-10-12 |
4-(3-cyanophenyl)-6-pyridinylpyrimidine Mglu5 Modulators App 20170275265 - Christopher; John Andrew ;   et al. | 2017-09-28 |
Muscarinic agonists Grant 9,758,506 - Brown , et al. September 12, 2 | 2017-09-12 |
Bicyclic Aza Compounds As Muscarinic M1 Receptor Antagonists App 20170247369 - Brown; Giles Albert ;   et al. | 2017-08-31 |
CGRP Receptor Antagonists App 20170239236 - Christopher; John Andrew ;   et al. | 2017-08-24 |
Bicyclic Aza Compounds As Muscarinic M1 Receptor And/or M4 Receptor Agonists App 20170240530 - Brown; Giles Albert ;   et al. | 2017-08-24 |
Piperidin-1 -yl And Azepin-1 -yl Carboxylates As Muscarinic M4 Receptor Agonists App 20170183338 - Livermore; David ;   et al. | 2017-06-29 |
CGRP receptor antagonists Grant 9,688,660 - Christopher , et al. June 27, 2 | 2017-06-27 |
4-(3-cyanophenyl)-6-pyridinylpyrimidine mGlu5 modulators Grant 9,676,745 - Christopher , et al. June 13, 2 | 2017-06-13 |
Muscarinic M1 Receptor Agonists App 20170157139 - Congreve; Miles Stuart ;   et al. | 2017-06-08 |
Bicyclic AZA compounds as muscarinic M1 receptor and/or M4 receptor agonists Grant 9,670,183 - Brown , et al. June 6, 2 | 2017-06-06 |
Bicyclic aza compounds as muscarinic M1 receptor agonists Grant 9,669,013 - Brown , et al. June 6, 2 | 2017-06-06 |
Mutant G-protein Coupled Receptor Proteins And Methods For Producing Them App 20170145075 - Robertson; Nathan Jacob ;   et al. | 2017-05-25 |
Orexin Receptor Antagonists App 20170121320 - Congreve; Miles Stuart ;   et al. | 2017-05-04 |
CGRP Receptor Antagonists App 20170121331 - Christopher; John Andrew ;   et al. | 2017-05-04 |
Cgrp Receptor Antagonists App 20170121311 - Christopher; John Andrew ;   et al. | 2017-05-04 |
CGRP Receptor Antagonists App 20170121348 - Christopher; John Andrew ;   et al. | 2017-05-04 |
Muscarinic Receptor Agonists App 20170096437 - Congreve; Miles Stuart ;   et al. | 2017-04-06 |
Piperidin-1-yl and azepin-1-yl carboxylates as muscarinic M4 receptor agonists Grant 9,593,106 - Livermore , et al. March 14, 2 | 2017-03-14 |
Muscarinic M1 receptor agonists Grant 9,573,929 - Congreve , et al. February 21, 2 | 2017-02-21 |
Muscarinic Agonists App 20170037025 - Brown; Giles Albert ;   et al. | 2017-02-09 |
Orexin receptor antagonists Grant 9,555,044 - Congreve , et al. January 31, 2 | 2017-01-31 |
Bicyclic Aza Compounds As Muscarinic M1 Receptor And/or M4 Receptor Agonists App 20170015650 - Brown; Giles Albert ;   et al. | 2017-01-19 |
Methods For Screening For Binding Partners Of G-protein Coupled Receptors App 20160327576 - Weir; Malcolm Peter ;   et al. | 2016-11-10 |
Orexin Receptor Antagonists App 20160213678 - Congreve; Miles Stuart ;   et al. | 2016-07-28 |
1,2,4-triazine-4-amine Derivatives App 20160175314 - Congreve; Miles Stuart ;   et al. | 2016-06-23 |
4-(3-cyanophenyl)-6-pyridinylpyrimidine Mglu5 Modulators App 20160145236 - Christopher; John Andrew ;   et al. | 2016-05-26 |
Bicyclic Aza Compounds As Muscarinic M1 Receptor Agonists App 20160128996 - Brown; Giles Albert ;   et al. | 2016-05-12 |
Muscarinic M1 Receptor Agonists App 20160068508 - Congreve; Miles Stuart ;   et al. | 2016-03-10 |
Mutant G-protein Coupled Receptors And Methods For Selecting Them App 20160052991 - Henderson; Richard ;   et al. | 2016-02-25 |
Bicyclic AZA compounds as muscarinic M1 receptor agonists Grant 9,266,857 - Brown , et al. February 23, 2 | 2016-02-23 |
Methods for screening for binding partners of G-protein coupled receptors Grant 9,260,505 - Weir , et al. February 16, 2 | 2016-02-16 |
1,2,4-triazine-4-amine derivatives Grant 9,249,130 - Congreve , et al. February 2, 2 | 2016-02-02 |
Orexin receptor antagonists Grant 9,249,160 - Congreve , et al. February 2, 2 | 2016-02-02 |
Muscarinic M1 receptor agonists Grant 9,187,451 - Congreve , et al. November 17, 2 | 2015-11-17 |
Crystal Structure App 20150261911 - Bortolato; Andrea ;   et al. | 2015-09-17 |
Bicyclic Aza Compounds As Muscarinic M1 Receptor Agonists App 20150232443 - Brown; Giles Albert ;   et al. | 2015-08-20 |
Mutant proteins and methods for selecting them Grant 9,081,020 - Weir , et al. July 14, 2 | 2015-07-14 |
Assays App 20150147822 - Marshall; Fiona Hamilton ;   et al. | 2015-05-28 |
Orexin Receptor Antagonists App 20150126498 - Congreve; Miles Stuart ;   et al. | 2015-05-07 |
1,2,4-triazine-4-amine Derivatives App 20150005276 - Congreve; Miles Stuart ;   et al. | 2015-01-01 |
Vaccines comprising mutant GPCRs with increased conformational stability relative to parent receptors Grant 8,900,591 - Hutchings , et al. December 2, 2 | 2014-12-02 |
Muscarinic M1 Receptor Agonists App 20140329803 - Congreve; Miles ;   et al. | 2014-11-06 |
Stable Proteins App 20140315299 - Jazayeri-Dezfuly; Seyed Ali ;   et al. | 2014-10-23 |
Methods For Screening For Binding Partners Of G-protein Coupled Receptors App 20140316116 - Weir; Malcolm Peter ;   et al. | 2014-10-23 |
1,2,4-triazine-4-amine derivatives Grant 8,809,525 - Congreve , et al. August 19, 2 | 2014-08-19 |
Screening Grant 8,790,933 - Weir , et al. July 29, 2 | 2014-07-29 |
Mutant G-protein coupled receptors and methods for selecting them Grant 8,785,135 - Henderson , et al. July 22, 2 | 2014-07-22 |
Mutant proteins and methods for producing them Grant 8,748,182 - Heal , et al. June 10, 2 | 2014-06-10 |
Mutant proteins and methods for producing them Grant 8,703,915 - Jazayeri-Dezfuly , et al. April 22, 2 | 2014-04-22 |
Mutant G-protein Coupled Receptor Proteins And Methods For Producing Them App 20140031525 - Robertson; Nathan Jacob ;   et al. | 2014-01-30 |
Gpcr As Vaccines Or For Removing/inhibiting Autoantibodies, Toxins Or Ligands Binding To The Gpcr App 20130224238 - Hutchings; Catherine Jane ;   et al. | 2013-08-29 |
1,2,4-triazine-4-amine Derivatives App 20130029963 - Congreve; Miles Stuart ;   et al. | 2013-01-31 |
Mutant G-protein Coupled Receptors And Methods For Selecting Them App 20120270230 - Henderson; Richard ;   et al. | 2012-10-25 |
Mutant Proteins And Methods For Producing Them App 20120165507 - Jazayeri-Dezfuly; Seyed Ali ;   et al. | 2012-06-28 |
Crystal structure .beta..sub.2 adrenoreceptor Grant 7,912,654 - Kobilka , et al. March 22, 2 | 2011-03-22 |
Mutant Proteins And Methods For Selecting Them App 20110046351 - Weir; Malcolm Peter ;   et al. | 2011-02-24 |
Mutant Proteins And Methods For Producing Them App 20110028700 - Heal; Jonathan Richard | 2011-02-03 |
Mutant G-protein Coupled Receptors And Methods For Selecting Them App 20100190188 - Henderson; Richard ;   et al. | 2010-07-29 |
NCAGE Code | U0RW3 | HEPTARES THERAPEUTICS LIMITED |
CAGE Code | U0RW3 | HEPTARES THERAPEUTICS LIMITED |
S.A.M. Registration | U0RW3 [210011328] | HEPTARES THERAPEUTICS LIMITED |
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