Patent | Date |
---|
Anilinopiperazine derivatives and methods of use thereof Grant 9,206,142 - Shipps, Jr. , et al. December 8, 2 | 2015-12-08 |
Substituted piperidines as HDM2 inhibitors Grant 9,062,071 - Ma , et al. June 23, 2 | 2015-06-23 |
Modulators of cell cycle checkpoints and their use in combination with checkpoint kinase inhibitors Grant 8,993,535 - Popovici-Muller , et al. March 31, 2 | 2015-03-31 |
SUBSTITUTED PIPERIDINES THAT INCREASE p53 ACTIVITY AND THE USES THEREOF App 20140336222 - Bogen; Stephane L. ;   et al. | 2014-11-13 |
Substituted Piperidines As Hdm2 Inhibitors App 20140323482 - Ma; Yao ;   et al. | 2014-10-30 |
Substituted piperidines that increase p53 activity and the uses thereof Grant 8,859,776 - Bogen , et al. October 14, 2 | 2014-10-14 |
Substituted pyrazolo[1,5-a]pyrimidines as cyclin dependent kinase inhibitors Grant 8,673,924 - Guzi , et al. March 18, 2 | 2014-03-18 |
Modulators of cell cycle checkpoints and their use in combination with checkpoint kinase inhibitors Grant 8,603,998 - Guzi , et al. December 10, 2 | 2013-12-10 |
Substituted pyrazolo[1,5-a]pyrimidines as cyclin dependent kinase inhibitors Grant 8,586,576 - Guzi , et al. November 19, 2 | 2013-11-19 |
Substituted pyrazolo[1,5-a]pyrimidines as cyclin dependent kinase inhibitors Grant 8,580,782 - Guzi , et al. November 12, 2 | 2013-11-12 |
Thiazole Derivatives as protein kinase inhibitors Grant 8,476,278 - Reddy , et al. July 2, 2 | 2013-07-02 |
Anilinopiperazine Derivatives And Methods Of Use Thereof App 20120328691 - Shipps, JR.; Gerald W. ;   et al. | 2012-12-27 |
2-aminothiazole-4-carboxylic amides as protein kinase inhibitors Grant 8,318,735 - Shipps, Jr. , et al. November 27, 2 | 2012-11-27 |
Heterocyclic amide compounds as protein kinase inhibitors Grant 8,293,747 - Reddy , et al. October 23, 2 | 2012-10-23 |
Substituted Piperidines That Increase P53 Activity And The Uses Thereof App 20120208844 - Bogen; Stephane L. ;   et al. | 2012-08-16 |
Modulators Of Cell Cycle Checkpoints And Their Use In Combination With Checkpoint Kinase Inhibitors App 20120184505 - Popovici-Muller; Janeta ;   et al. | 2012-07-19 |
Methods for inhibiting protein kinases Grant 8,211,854 - Guzi , et al. July 3, 2 | 2012-07-03 |
Synthesis Of Substituted-3-aminopyrazoles App 20120029204 - Alvarez; Carmen S. ;   et al. | 2012-02-02 |
Novel Modulators Of Cell Cycle Checkpoints And Their Use In Combination With Checkpoint Kinase Inhibitors App 20110183933 - Guzi; Timothy J. ;   et al. | 2011-07-28 |
Heterocyclic Urea and Thiourea Derivatives and Methods of Use Thereof App 20110129440 - Tadikonda; Praveen K. ;   et al. | 2011-06-02 |
Thiazole Derivatives as Protein Kinase Inhibitors App 20100331313 - Reddy; Panduranga Adulla P. ;   et al. | 2010-12-30 |
Heterocyclic Amide Compounds As Protein Kinase Inhibitors App 20100286135 - Reddy; Panduranga Adulla P. ;   et al. | 2010-11-11 |
N-heteroaryl pyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,807,683 - Guzi , et al. October 5, 2 | 2010-10-05 |
Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors Grant 7,776,865 - Paruch , et al. August 17, 2 | 2010-08-17 |
2-aminothiazole-4-carboxylic Amides As Protein Kinase Inhibitors App 20100130465 - Shipps, JR.; Gerald W. ;   et al. | 2010-05-27 |
Methods For Inhibiting Protein Kinases App 20100125068 - Guzi; Timothy J. ;   et al. | 2010-05-20 |
Substituted pyrazolo[1,5-a] pyrimidines as protein kinase inhibitors Grant 7,645,762 - Paruch , et al. January 12, 2 | 2010-01-12 |
Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors Grant 7,642,266 - Guzi , et al. January 5, 2 | 2010-01-05 |
Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors Grant 7,605,155 - Guzi , et al. October 20, 2 | 2009-10-20 |
Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors Grant 7,601,724 - Guzi , et al. October 13, 2 | 2009-10-13 |
Imidazopyrazines as cyclin dependent kinase inhibitors Grant 7,576,085 - Guzi , et al. August 18, 2 | 2009-08-18 |
Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors Grant 7,563,798 - Guzi , et al. July 21, 2 | 2009-07-21 |
Imidazopyrazines as protein kinase inhibitors Grant 7,557,104 - Zhao , et al. July 7, 2 | 2009-07-07 |
Trisubstituted 4-aminopyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,514,442 - Guzi , et al. April 7, 2 | 2009-04-07 |
Pyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,511,049 - Guzi , et al. March 31, 2 | 2009-03-31 |
Imidazopyrazines as protein kinase inhibitors Grant 7,511,040 - Belanger , et al. March 31, 2 | 2009-03-31 |
17.beta.-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases Grant 7,485,645 - Guzi , et al. February 3, 2 | 2009-02-03 |
17.beta.-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases Grant 7,476,681 - Paruch , et al. January 13, 2 | 2009-01-13 |
N-heteroaryl pyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,470,695 - Guzi , et al. December 30, 2 | 2008-12-30 |
Trisubstituted 4-aminopyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,468,372 - Guzi , et al. December 23, 2 | 2008-12-23 |
Imidazopyridines as cyclin dependent kinase inhibitors Grant 7,452,902 - Dwyer , et al. November 18, 2 | 2008-11-18 |
Pyrazolopyrimidines as protein kinase inhibitors Grant 7,449,488 - Paruch , et al. November 11, 2 | 2008-11-11 |
Imidazopyrazines as cyclin dependent kinase inhibitors Grant 7,432,265 - Paruch , et al. October 7, 2 | 2008-10-07 |
Imidazopyrazines As Protein Kinase Inhibitors App 20080139571 - Belanger; David B. ;   et al. | 2008-06-12 |
Pyrazolotriazines as kinase inhibitors Grant 7,354,921 - Guzi , et al. April 8, 2 | 2008-04-08 |
Farnesyl protein transferase inhibitors as antitumor agents Grant 7,342,016 - Zhu , et al. March 11, 2 | 2008-03-11 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20080050384 - Guzi; Timothy J. ;   et al. | 2008-02-28 |
Imidazopyrazines As Protein Kinase Inhibitors App 20080027063 - Zhao; Lianyun ;   et al. | 2008-01-31 |
17beta-hydroxysteroid Dehydrogenase Type 3 Inhibitors For The Treatment Of Androgen Dependent Diseases App 20080004248 - Guzi; Timothy J. ;   et al. | 2008-01-03 |
Pyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,309,705 - Guzi , et al. December 18, 2 | 2007-12-18 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20070281951 - Guzi; Timothy J. ;   et al. | 2007-12-06 |
Novel Pyrazolopyrimidines As Cyclin Dependent Kinase Inhibitors App 20070275983 - Guzi; Timothy J. ;   et al. | 2007-11-29 |
PYRAZOLO[1,5-a]PYRIMIDINES App 20070275963 - Guzi; Timothy J. ;   et al. | 2007-11-29 |
Pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20070225270 - Guzi; Timothy J. ;   et al. | 2007-09-27 |
17.beta.-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases Grant 7,271,175 - Guzi , et al. September 18, 2 | 2007-09-18 |
Novel Imidazopyrazines As Cyclin Dependent Kinase Inhibitors App 20070155751 - PARUCH; KAMIL ;   et al. | 2007-07-05 |
Imidazopyrazines as protein kinase inhibitors App 20070117804 - Zhao; Lianyun ;   et al. | 2007-05-24 |
Methods for inhibiting protein kinases App 20070105864 - Guzi; Timothy J. ;   et al. | 2007-05-10 |
Trisubstituted 7-aminopyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,205,308 - Guzi , et al. April 17, 2 | 2007-04-17 |
Pyrazolopyrimidines as protein kinase inhibitors App 20070082901 - Guzi; Timothy J. ;   et al. | 2007-04-12 |
Pyrazolopyrimidines as protein kinase inhibitors App 20070082902 - Paruch; Kamil ;   et al. | 2007-04-12 |
Methods for inhibiting protein kinases App 20070082900 - Guzi; Timothy J. ;   et al. | 2007-04-12 |
Pyrazolopyrimidines as protein kinase inhibitors App 20070083044 - Paruch; Kamil ;   et al. | 2007-04-12 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20070072880 - Guzi; Timothy J. ;   et al. | 2007-03-29 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20070072881 - Guzi; Timothy J. ;   et al. | 2007-03-29 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20070072882 - Guzi; Timothy J. ;   et al. | 2007-03-29 |
N-heteroaryl pyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,196,092 - Guzi , et al. March 27, 2 | 2007-03-27 |
Trisubstituted and tetrasubstituted pyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,196,078 - Guzi , et al. March 27, 2 | 2007-03-27 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20070054925 - Guzi; Timothy J. ;   et al. | 2007-03-08 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20070054906 - Guzi; Timothy J. ;   et al. | 2007-03-08 |
Imidazopyrazines as cyclin dependent kinase inhibitors Grant 7,186,740 - Paruch , et al. March 6, 2 | 2007-03-06 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20070037824 - Guzi; Timothy J. ;   et al. | 2007-02-15 |
Pyrazolotriazines as kinase inhibitors App 20070032495 - Guzi; Timothy J. ;   et al. | 2007-02-08 |
Pyrazolotriazines as kinase inhibitors Grant 7,166,602 - Guzi , et al. January 23, 2 | 2007-01-23 |
Pyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,161,003 - Guzi , et al. January 9, 2 | 2007-01-09 |
Pyrazolopyridines as cyclin dependent kinase inhibitors Grant 7,151,104 - Dwyer , et al. December 19, 2 | 2006-12-19 |
Compounds for inhibiting KSP Kinesin activity App 20060281778 - Tagat; Jayaram R. ;   et al. | 2006-12-14 |
17 .beta.-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases Grant 7,138,396 - Guzi , et al. November 21, 2 | 2006-11-21 |
Compounds for inhibiting KSP kinesin activity App 20060247320 - Tagat; Jayaram R. ;   et al. | 2006-11-02 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20060235025 - Guzi; Timothy J. ;   et al. | 2006-10-19 |
Pyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,119,200 - Guzi , et al. October 10, 2 | 2006-10-10 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20060178371 - Guzi; Timothy J. ;   et al. | 2006-08-10 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20060173016 - Guzi; Timothy J. ;   et al. | 2006-08-03 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20060173017 - Guzi; Timothy J. ;   et al. | 2006-08-03 |
Pyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,084,271 - Guzi , et al. August 1, 2 | 2006-08-01 |
Pyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,078,525 - Guzi , et al. July 18, 2 | 2006-07-18 |
17.beta.-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases Grant 7,074,795 - Paruch , et al. July 11, 2 | 2006-07-11 |
Pyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,074,924 - Guzi , et al. July 11, 2 | 2006-07-11 |
17Beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases App 20060148816 - Paruch; Kamil ;   et al. | 2006-07-06 |
17beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases App 20060142338 - Guzi; Timothy J. ;   et al. | 2006-06-29 |
Pyrazolopyrimidines as cyclin dependent kinase inhibitors Grant 7,067,661 - Guzi , et al. June 27, 2 | 2006-06-27 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20060128725 - Guzi; Timothy J. ;   et al. | 2006-06-15 |
Pyrazolotriazines as kinase inhibitors App 20060122389 - Guzi; Timothy J. ;   et al. | 2006-06-08 |
17 .beta.-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases Grant 7,053,091 - Guzi , et al. May 30, 2 | 2006-05-30 |
Novel imidazopyrazines as cyclin dependent kinase inhibitors App 20060106023 - Guzi; Timothy J. ;   et al. | 2006-05-18 |
Pyrazolopyrimidines as protein kinase inhibitors App 20060094706 - Paruch; Kamil ;   et al. | 2006-05-04 |
Pyrazolotriazines as kinase inhibitors Grant 7,038,045 - Guzi , et al. May 2, 2 | 2006-05-02 |
17 Beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases App 20060069103 - Guzi; Timothy J. ;   et al. | 2006-03-30 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20060040958 - Guzi; Timothy J. ;   et al. | 2006-02-23 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20060041131 - Guzi; Timothy J. ;   et al. | 2006-02-23 |
Novel imidazopyridines as cyclin dependent kinase inhibitors App 20060030555 - Dwyer; Michael P. ;   et al. | 2006-02-09 |
Imidazopyridines as cyclin dependent kinase inhibitors Grant 6,992,080 - Dwyer , et al. January 31, 2 | 2006-01-31 |
17 Beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases App 20060014755 - Guzi; Timothy J. ;   et al. | 2006-01-19 |
17-.beta. hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases Grant 6,969,718 - Guzi , et al. November 29, 2 | 2005-11-29 |
Pyrazolotriazines as kinase inhibitors App 20050187219 - Guzi, Timothy J. ;   et al. | 2005-08-25 |
Imidazopyrazines as cyclin dependent kinase inhibitors Grant 6,919,341 - Paruch , et al. July 19, 2 | 2005-07-19 |
Novel imidazopyrazines as cyclin dependent kinase inhibitors App 20050130980 - Paruch, Kamil ;   et al. | 2005-06-16 |
17.beta.-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases Grant 6,903,102 - Guzi , et al. June 7, 2 | 2005-06-07 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20040209878 - Guzi, Timothy J. ;   et al. | 2004-10-21 |
17 Beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases App 20040138226 - Guzi, Timothy J. ;   et al. | 2004-07-15 |
17 Beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases App 20040132736 - Guzi, Timothy J. ;   et al. | 2004-07-08 |
17Beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases App 20040127503 - Paruch, Kamil ;   et al. | 2004-07-01 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20040116442 - Guzi, Timothy J. ;   et al. | 2004-06-17 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20040106624 - Guzi, Timothy J. ;   et al. | 2004-06-03 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20040102452 - Guzi, Timothy J. ;   et al. | 2004-05-27 |
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors App 20040102451 - Guzi, Timothy J. ;   et al. | 2004-05-27 |
Novel pyrazolopyridines as cyclin dependent kinase inhibitors App 20040097516 - Dwyer, Michael P. ;   et al. | 2004-05-20 |
Novel imidazopyridines as cyclin dependent kinase inhibitors App 20040097517 - Dwyer, Michael P. ;   et al. | 2004-05-20 |
Treatment of malaria with farnesyl protein transferase inhibitors App 20040087592 - Windsor, William T. ;   et al. | 2004-05-06 |
Novel imidazopyrazines as cyclin dependent kinase inhibitors App 20040072835 - Paruch, Kamil ;   et al. | 2004-04-15 |
Novel imidazopyrazines as cyclin dependent kinase inhibitors App 20040063715 - Paruch, Kamil ;   et al. | 2004-04-01 |
17-Beta hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases App 20030232837 - Guzi, Timothy J. ;   et al. | 2003-12-18 |
Treatment of malaria with farnesyl protein transferase inhibitors App 20030092705 - Windsor, William T. ;   et al. | 2003-05-15 |
Farnesyl protein transferase inhibitors Grant 6,399,615 - Guzi , et al. June 4, 2 | 2002-06-04 |