Patent | Date |
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Isoindolinone compounds as GPR119 modulators for the treatment of diabetes, obesity, dyslipidemia and related disorders Grant 9,908,868 - Schwink , et al. March 6, 2 | 2018-03-06 |
Substituted indanone compounds as GPR119 modulators for the treatment of diabetes, obesity, dyslipidemia and related disorders Grant 9,896,434 - Schwink , et al. February 20, 2 | 2018-02-20 |
Substituted fused heterocycles as GPR119 modulators for the treatment of diabetes, obesity, dyslipidemia and related disorders Grant 9,758,520 - Schwink , et al. September 12, 2 | 2017-09-12 |
Substituted Indanone Compounds As Gpr119 Modulators For The Treatment Of Diabetes, Obesity, Dyslipidemia And Related Disorders App 20170029405 - SCHWINK; Lothar ;   et al. | 2017-02-02 |
Substituted Fused Heterocycles As Gpr119 Modulators For The Treatment Of Diabetes, Obesity, Dyslipidemia And Related Disorders App 20170022198 - SCHWINK; Lothar ;   et al. | 2017-01-26 |
Isoindolinone Compounds As Gpr119 Modulators For The Treatment Of Diabetes, Obesity, Dyslipidemia And Related Disorders App 20170022182 - SCHWINK; Lothar ;   et al. | 2017-01-26 |
Amino alcohol-substituted arylthienopyrimidinones, process for their preparation and their use as medicaments Grant 8,853,208 - Schwink , et al. October 7, 2 | 2014-10-07 |
Pyrrolidinone derivatives as GPR119 modulators for the treatment of diabetes, obesity, dyslipidemia and related disorders Grant 8,853,412 - Schwink , et al. October 7, 2 | 2014-10-07 |
Substituted tetrahydronaphthalenes, method for the production thereof, and use thereof as drugs Grant 8,841,290 - Schwink , et al. September 23, 2 | 2014-09-23 |
Azacyclyl-substituted arylthienopyrimidinones, process for their preparation and their use as medicaments Grant 8,828,991 - Schwink , et al. September 9, 2 | 2014-09-09 |
Azacyclyl-substituted aryldihydroisoquinolinones, process for their preparation and their use as medicaments Grant 8,822,495 - Schwink , et al. September 2, 2 | 2014-09-02 |
Pyrrolidinone Derivatives As Gpr119 Modulators For The Treatment Of Diabetes, Obesity, Dyslipidemia And Related Disorders App 20140099333 - SCHWINK; Lothar ;   et al. | 2014-04-10 |
Novel Substituted Tetrahydronaphthalenes, Process For The Preparation Thereof And The Use Thereof As Medicaments App 20140088077 - Schwink; Lothar ;   et al. | 2014-03-27 |
Substituted tetrahydronaphthalenes, process for the preparation thereof and the use thereof as medicaments Grant 8,609,731 - Schwink , et al. December 17, 2 | 2013-12-17 |
Aryl-substituted polycyclic amines, method for the production thereof, and use thereof as a medicament Grant 8,586,609 - Schwink , et al. November 19, 2 | 2013-11-19 |
Substituted indanes, method for the production thereof, and use thereof as drugs Grant 8,552,199 - Schwink , et al. October 8, 2 | 2013-10-08 |
Aminoalcohol-substituted aryldihydroisoquinolinones, process for their preparation and their use as medicaments Grant 8,501,771 - Schwink , et al. August 6, 2 | 2013-08-06 |
Aryl-substituted polycyclic amines, method for the production thereof, and use thereof as a medicament Grant 8,357,686 - Schwink , et al. January 22, 2 | 2013-01-22 |
Medicinal Targeted Local Lipolysis App 20120329765 - Boderke; Peter ;   et al. | 2012-12-27 |
Aryl-substituted heterocycles, process for their preparation and their use as medicaments Grant 8,299,104 - Schwink , et al. October 30, 2 | 2012-10-30 |
Use of aryl-substituted polycyclic amines as medicaments Grant 8,163,741 - Schwink , et al. April 24, 2 | 2012-04-24 |
Novel Substituted Indanes, Method For The Production Thereof, And Use Thereof As Drugs App 20120022039 - Schwink; Lothar ;   et al. | 2012-01-26 |
Substituted Tetrahydronaphthalenes, Method For The Production Thereof, And Use Thereof As Drugs App 20120015936 - Schwink; Lothar ;   et al. | 2012-01-19 |
Hexahydro-pyrazino[1,2-A]pyrimidine-4,7-dione derivatives substituted with amino acids Grant 7,994,168 - Lennig , et al. August 9, 2 | 2011-08-09 |
Novel phenyl-substituted imidazolidines, process for preparation thereof, medicaments comprising said compounds and use thereof App 20110178134 - JAEHNE; Gerhard ;   et al. | 2011-07-21 |
Substituted N-aryl heterocycles, process for their preparation and their use as medicaments Grant 7,968,550 - Schwink , et al. June 28, 2 | 2011-06-28 |
Substituted imidazoline-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof App 20110112097 - Jaehne; Gerhard ;   et al. | 2011-05-12 |
Arylchalcogenoarylalkyl-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof App 20110053947 - JAEHNE; Gerhard ;   et al. | 2011-03-03 |
Arylchalcogenoarylalkyl-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof App 20110046185 - JAEHNE; Gerhard ;   et al. | 2011-02-24 |
Heterocycle-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising them and use thereof App 20110046105 - Jaehne; Gerhard ;   et al. | 2011-02-24 |
Aryl-substituted Polycyclic Amines, Method For The Production Thereof, And Use Thereof As A Medicament App 20100298378 - SCHWINK; Lothar ;   et al. | 2010-11-25 |
Aryl-substituted polycyclic amines, method for the production thereof, and use thereof as a medicament Grant 7,838,547 - Schwink , et al. November 23, 2 | 2010-11-23 |
Novel Substituted Tetrahydronaphthalenes, Process For The Preparation Thereof And The Use Thereof As Medicaments App 20100249097 - SCHWINK; Lothar ;   et al. | 2010-09-30 |
Use of C2-substituted indan-1-ol systems for preparing medicaments for the prophylaxis or treatment of obesity Grant 7,763,662 - Jaehne , et al. July 27, 2 | 2010-07-27 |
Arylaminoaryl-alkyl-substituted imidazolidine-2,4-diones, process for preparing them, medicaments comprising these compounds, and their use Grant 7,759,366 - Jaehne , et al. July 20, 2 | 2010-07-20 |
Substituted hexahydropyrazino [1,2-A] pyrimidine-4,7-dione derivatives, process for their preparation and their use as medicaments Grant 7,750,005 - Flohr , et al. July 6, 2 | 2010-07-06 |
Nitrogen-substituted hexahydropyrazino[1,2-A]pyrimidine-4,7-dione derivatives, processes for their preparation and their use as medicaments Grant 7,652,007 - Flohr , et al. January 26, 2 | 2010-01-26 |
Medicinal lipolysis of accumulation of fat App 20100004216 - Boderke; Peter ;   et al. | 2010-01-07 |
Medicinal targeted local lipolysis App 20090275545 - Boderke; Peter ;   et al. | 2009-11-05 |
Novel Azacyclyl-substituted Aryldihydroisoquinolinones, Process For Their Preparation And Their Use As Medicaments App 20090264403 - SCHWINK; Lothar ;   et al. | 2009-10-22 |
Use Of Aryl-substituted Polycyclic Amines As Medicaments App 20090258872 - SCHWINK; Lothar ;   et al. | 2009-10-15 |
Aryl-substituted Polycyclic Amines, Method For The Production Thereof, And Use Thereof As A Medicament App 20090258881 - SCHWINK; Lothar ;   et al. | 2009-10-15 |
Arylaminoaryl-alkyl-substituted imidazolidine-2,4-diones, process for preparing them, medicaments comprising these compounds, and their use App 20090215728 - JAEHNE; Gerhard ;   et al. | 2009-08-27 |
Aryl-substituted polycyclic amines, method for the production thereof, and use thereof as a medicament Grant 7,569,583 - Schwink , et al. August 4, 2 | 2009-08-04 |
Novel Azacyclyl-substituted Arylthienopyrimidinones, Process For Their Preparation And Their Use As Medicaments App 20090082339 - SCHWINK; Lothar ;   et al. | 2009-03-26 |
Novel Aminoalcohol-substituted Aryldihydroisoquinolinones, Process For Their Preparation And Their Use As Medicaments App 20090082391 - SCHWINK; Lothar ;   et al. | 2009-03-26 |
Novel Amino Alcohol-substituted Arylthienopyrimidinones, Process For Their Preparation And Their Use As Medicaments App 20090076002 - SCHWINK; Lothar ;   et al. | 2009-03-19 |
Substituted Hexahydropyrazino [1,2-a] Pyrimidine-4,7-dione Derivatives, Process For Their Preparation And Their Use As Medicaments App 20080221113 - Flohr; Stefanie ;   et al. | 2008-09-11 |
Aryl-substituted Heterocycles, Process For Their Preparation And Their Use As Medicaments App 20080207707 - Schwink; Lothar ;   et al. | 2008-08-28 |
Substituted hexahydropyrazino [1,2-a] pyrimidine-4,7-dione derivatives, process for their preparation and their use as medicaments Grant 7,390,814 - Flohr , et al. June 24, 2 | 2008-06-24 |
Aryl-substituted heterocycles, process for their preparation and their use as medicaments Grant 7,319,108 - Schwink , et al. January 15, 2 | 2008-01-15 |
Aryl-substituted Polycyclic Amines, Method For The Production Thereof, And Use Thereof As A Medicament App 20070299077 - SCHWINK; Lothar ;   et al. | 2007-12-27 |
Substituted N-aryl Heterocycles, Process For Their Preparation and Their Use As Medicaments App 20070207991 - Schwink; Lothar ;   et al. | 2007-09-06 |
Hexahydro-pyrazino[1,2-a]pyrimidine-4,7-dione Derivatives Substituted With Amino Acids App 20070197539 - Lennig; Petra ;   et al. | 2007-08-23 |
Aryl-substituted Polycyclic Amines, Method For The Production Thereof, And Use Thereof As A Medicament App 20070197584 - SCHWINK; Lothar ;   et al. | 2007-08-23 |
Substituted N-cycloexylimidazolinones, process for their preparation and their use as medicaments Grant 7,241,787 - Schwink , et al. July 10, 2 | 2007-07-10 |
Substituted N-aryl heterocycles, process for their preparation and their use as medicaments Grant 7,223,788 - Schwink , et al. May 29, 2 | 2007-05-29 |
Substituted diaryl heterocycles, process for their preparation and their use as medicaments Grant 7,141,561 - Schwink , et al. November 28, 2 | 2006-11-28 |
C2-disubstituted indan-1-ones and their derivatives, processes for their preparation and their use as pharmaceuticals Grant 7,081,467 - Jaehne , et al. July 25, 2 | 2006-07-25 |
C2-substituted idan-1-ols and their derivatives, processes for their preparation and their use as pharmaceuticals Grant 7,045,649 - Jaehne , et al. May 16, 2 | 2006-05-16 |
C2-substituted indan-1-ols and their derivatives, processes for their preparation and their use as pharmaceuticals Grant 7,015,208 - Jaehne , et al. March 21, 2 | 2006-03-21 |
Use of C2-substituted indan-1-one systems for preparing medicaments for the treatment of obesity Grant 6,946,492 - Jaehne , et al. September 20, 2 | 2005-09-20 |
Substituted N-cycloexylimidazolinones, process for their preparation and their use as medicaments App 20050176795 - Schwink, Lothar ;   et al. | 2005-08-11 |
Aryl-substituted heterocycles, process for their preparation and their use as medicaments App 20050176710 - Schwink, Lothar ;   et al. | 2005-08-11 |
Derivatives of C2-substituted indan-1-ol systems for the prophylaxis or treatment of obesity Grant 6,919,380 - Jaehne , et al. July 19, 2 | 2005-07-19 |
Medicinal lipolysis of accumulations of fat App 20050143347 - Boderke, Peter ;   et al. | 2005-06-30 |
C2-substituted idan-1-ols and their derivatives, processes for their preparation and their use as pharmaceuticals App 20050113595 - Jaehne, Gerhard ;   et al. | 2005-05-26 |
C2-substituted idan-1-ols and their derivatives, processes for their preparation and their use as pharmaceuticals App 20050101798 - Jaehne, Gerhard ;   et al. | 2005-05-12 |
Medicinal targeted local lipolysis App 20050089555 - Boderke, Peter ;   et al. | 2005-04-28 |
Nitrogen-substituted hexahydropyrazino[1,2-a]pyrimidine-4,7-dione derivatives, processes for their preparation and their use as medicaments App 20050085483 - Flohr, Stefanie ;   et al. | 2005-04-21 |
Use of C2-substituted indan-1-ol systems for preparing medicaments for the prophylaxis or treatment of obesity App 20050080057 - Jaehne, Gerhard ;   et al. | 2005-04-14 |
Substituted hexahydropyrazino (1,2-a) pyrimidine-4,7-dione derivatives, processes for their preparation and their use as medicaments App 20050004131 - Flohr, Stefanie ;   et al. | 2005-01-06 |
Substituted N-aryl heterocycles, process for their preparation and their use as medicaments App 20040220191 - Schwink, Lothar ;   et al. | 2004-11-04 |
Polysubstituted indan-1-ol systems for the prophylaxis or treatment of obesity Grant 6,812,256 - Jaehne , et al. November 2, 2 | 2004-11-02 |
Polysubstituted indan-1-ol systems for the prophylaxis or treatment of obesity Grant 6,812,257 - Jaehne , et al. November 2, 2 | 2004-11-02 |
Aminoalkyl-substituted aromatic bicyclic compounds, methods for their preparation and their use as pharmaceuticals App 20040198733 - Schwink, Lothar ;   et al. | 2004-10-07 |
Aminoalkyl-substituted aromatic bicyclic compounds, methods for their preparation and their use as pharmaceuticals App 20040198731 - Schwink, Lothar ;   et al. | 2004-10-07 |
Aminoalkyl-substituted aromatic bicyclic compounds, methods for their preparation and their use as pharmaceuticals App 20040198732 - Schwink, Lothar ;   et al. | 2004-10-07 |
Aminoalkyl-substituted aromatic bicyclic compounds, methods for their preparation and their use as pharmaceuticals App 20040192693 - Schwink, Lothar ;   et al. | 2004-09-30 |
C2-substituted idan-1-ones and their derivatives, processes for their preparation and their use as pharmaceuticals Grant 6,762,326 - Jaehne , et al. July 13, 2 | 2004-07-13 |
Substituted diaryl heterocycles, process for their preparation and their use as medicaments App 20040132752 - Schwink, Lothar ;   et al. | 2004-07-08 |
Polysubstituted indan-1-ol systems for the prophylaxis or treatment of obesity App 20040106583 - Jaehne, Gerhard ;   et al. | 2004-06-03 |
Polysubstituted indan-1-ol compounds, and methods for their preparation and use App 20040092489 - Jaehne, Gerhard ;   et al. | 2004-05-13 |
Derivatives of C2-substituted indan-1-ol systems for the prophylaxis or treatment of obesity App 20040092748 - Jaehne, Gerhard ;   et al. | 2004-05-13 |
Polysubstituted idan-1-ol compounds, and methods for their preparation and use App 20040092749 - Jaehne, Gerhard ;   et al. | 2004-05-13 |
Polysubstituted indan-1-ol systems for the prophylaxis or treatment of obesity App 20040092488 - Jaehne, Gerhard ;   et al. | 2004-05-13 |
C2-substituted idan-1-ols and their derivatives, processes for their preparation and their use as pharmaceuticals App 20040068016 - Jaehne, Gerhard ;   et al. | 2004-04-08 |
Derivatives of C2-substituted indan-1-ol compounds, methods for their preparation and use Grant 6,717,008 - Jaehne , et al. April 6, 2 | 2004-04-06 |
Polysubstituted indan-1-ol systems for the prophylaxis or treatment of obesity Grant 6,686,397 - Jaehne , et al. February 3, 2 | 2004-02-03 |
Polysubstituted indan-1-ol compounds, and methods for their preparation and use Grant 6,670,401 - Jaehne , et al. December 30, 2 | 2003-12-30 |
Derivatives of C2-substituted indan-1-ol systems for the prophylaxis or treatment of obesity Grant 6,667,345 - Jaehne , et al. December 23, 2 | 2003-12-23 |
C2-substituted indan-1-ols and their derivatives, processes for their preparation and their use as pharmaceuticals Grant 6,657,086 - Jaehne , et al. December 2, 2 | 2003-12-02 |
Aminoalkyl-substituted aromatic bicyclic compounds, methods for their preparation and their use as pharmaceuticals App 20030212070 - Schwink, Lothar ;   et al. | 2003-11-13 |
C2-disubstituted indan-1-ol compounds, their derivatives, processes for their preparation, and their use as pharmaceuticals App 20030181491 - Jaehne, Gerhard ;   et al. | 2003-09-25 |
C2-disubstituted indan-1-ones and their derivatives, processes for their preparation and their use as pharmaceuticals App 20030153609 - Jaehne, Gerhard ;   et al. | 2003-08-14 |
Use of C2-substituted indan-1-one systems for preparing medicaments for the prophylaxis or treatment of obesity App 20030134882 - Jaehne, Gerhard ;   et al. | 2003-07-17 |
Use of C2-substituted indan-1-ol systems for preparing medicaments for the prophylaxis or treatment of obesity App 20030134879 - Jaehne, Gerhard ;   et al. | 2003-07-17 |
Derivatives of C2-substituted indan-1 ol systems for the prophylaxis or treatment of obesity App 20030134881 - Jaehne, Gerhard ;   et al. | 2003-07-17 |
C2-substituted idan-1-ones and their derivatives, processes for their preparation and their use as pharmaceuticals App 20030130345 - Jaehne, Gerhard ;   et al. | 2003-07-10 |
Polysubstituted indan-1-ol- systems for the prophylaxis or treatment of obesity App 20030130323 - Jaehne, Gerhard ;   et al. | 2003-07-10 |
C2-substituted indan-1-ols and their derivatives, processes for their preparation and their use as pharmaceuticals App 20030114681 - Jaehne, Gerhard ;   et al. | 2003-06-19 |
Polysubstituted indan-1-ol compounds, and methods for their preparation and use App 20030105145 - Jaehne, Gerhard ;   et al. | 2003-06-05 |
Derivatives of C2-substituted indan-1-ol compounds, methods for their preparation and use App 20030105331 - Jaehne, Gerhard ;   et al. | 2003-06-05 |
8,8a-dihydroindeno[1,2-d]thiazole derivatives which carry in the 2-position a substituent having a sulfonamide structure or sulfone structure; processes for their preparation and their use as medicaments App 20020103231 - Jaehne, Gerhard ;   et al. | 2002-08-01 |
8,8A-dihydroindeno[1,2-D] thiazole derivatives which are substituted in the 8A-position; processes for their preparation and their use as medicaments App 20020058658 - Jaehne, Gerhard ;   et al. | 2002-05-16 |
8,8a-dihydroindeno[1,2-d]thiazole derivatives which carry in the 2-position a substituent having a sulfonamide structure or sulfone structure; processes for their preparation and their use as medicaments App 20010039278 - Jaehne, Gerhard ;   et al. | 2001-11-08 |
Substituted 8,8a-dihydro-3ah-indeno[1,2-d]thiazoles, processes for their preparation and their use as medicaments App 20010031752 - Jaehne, Gerhard ;   et al. | 2001-10-18 |