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Purine derivatives and the use thereof as medicament Grant 11,376,258 - Giovannini , et al. July 5, 2 | 2022-07-05 |
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4-Pyrazin-2-ylmethyl-morpholine derivatives and the use thereof as medicament App 20210393644 - GIOVANNINI; Riccardo ;   et al. | 2021-12-23 |
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4-pyrazin-2-ylmethyl-morpholine derivatives and the use thereof as medicament Grant 11,166,958 - Giovannini , et al. November 9, 2 | 2021-11-09 |
4-pyridinylmethyl-morpholine derivatives and the use thereof as medicament Grant 11,155,539 - Giovannini , et al. October 26, 2 | 2021-10-26 |
4-pyrimidin-5-ylmethyl-morpholine derivatives and the use thereof as medicament Grant 11,104,670 - Giovannini , et al. August 31, 2 | 2021-08-31 |
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Medical Use Of Compound Iii App 20210130362 - SAND; Michael Steven ;   et al. | 2021-05-06 |
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Cyclic Ether Derivatives Of Pyrazolo[1,5-a]pyrimidine-3-carboxyamide App 20210032259 - HOENKE; Christoph ;   et al. | 2021-02-04 |
Cyclic ether derivatives of pyrazolo[1,5-a]pyrimidine-3-carboxyamide Grant 10,875,867 - Hoenke , et al. December 29, 2 | 2020-12-29 |
Imidazopyridine derivatives and the use thereof as medicament Grant 10,849,907 - Giovannini , et al. December 1, 2 | 2020-12-01 |
Somatostatin receptor subtype 4 (SSTR4) agonists Grant 10,675,268 - Giovannini , et al. | 2020-06-09 |
Heteroarylcarboxamide derivatives as plasma kallikrein inhibitors Grant 10,640,486 - Frattini , et al. | 2020-05-05 |
4-Pyridinylmethyl-Morpholine Derivatives and the use thereof as Medicament App 20200123141 - GIOVANNINI; Riccardo ;   et al. | 2020-04-23 |
4-Pyrimidin-5-ylmethyl-morpholine derivatives and the use thereof as medicament App 20200123140 - GIOVANNINI; Riccardo ;   et al. | 2020-04-23 |
4-Pyrazin-2-ylmethyl-morpholine derivatives and the use thereof as medicament App 20200121691 - GIOVANNINI; Riccardo ;   et al. | 2020-04-23 |
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Cyclic Ether Derivatives Of Pyrazolo[1,5-a]pyrimidine-3-carboxyamide App 20200039991 - HOENKE; Christoph ;   et al. | 2020-02-06 |
Cyclic ether derivatives of pyrazolo[1,5-a]pyrimidine-3-carboxyamide Grant 10,479,794 - Hoenke , et al. Nov | 2019-11-19 |
Ccr2 Receptor Antagonists And Uses Thereof App 20190300541 - Ebel; Heiner ;   et al. | 2019-10-03 |
New Somatostatin Receptor Subtype 4 (sstr4) Agonists App 20190269650 - Giovannini; Riccardo ;   et al. | 2019-09-05 |
Heteroarylcarboxamide derivatives as plasma kallikrein inhibitors Grant 10,399,961 - Frattini , et al. Sep | 2019-09-03 |
Imidazopyridine derivatives and the use thereof as medicament App 20190175605 - GIOVANNINI; Riccardo ;   et al. | 2019-06-13 |
CCR2 receptor antagonists and uses thereof Grant 10,196,402 - Ebel , et al. Fe | 2019-02-05 |
Aryl and heteroaryl-fused tetrahydro-1,4-oxazepine amides as somatostatin receptor subtype 4 (SSTR4) agonists Grant 10,183,940 - Mazzaferro , et al. Ja | 2019-01-22 |
Somatostatin receptor subtype 4 (SSTR4) agonists Grant 10,166,214 - Giovannini , et al. J | 2019-01-01 |
Morpholine And 1,4-oxazepane Amides As Somatostatin Receptor Subtype 4 (sstr4) Agonists App 20180339971 - MAZZAFERRO; Rocco ;   et al. | 2018-11-29 |
Heteroarylcarboxamide Derivatives As Plasma Kallikrein Inhibitors App 20180319771 - FRATTINI; Sara ;   et al. | 2018-11-08 |
Heteroarylcarboxamide Derivatives As Plasma Kallikrein Inhibitors App 20180305338 - FRATTINI; Sara ;   et al. | 2018-10-25 |
Aryl And Heteroaryl-fused Tetrahydro-1,4-oxazepine Amides As Somatostatin Receptor Subtype 4 (sstr4) Agonists App 20180291018 - MAZZAFERRO; Rocco ;   et al. | 2018-10-11 |
Morpholine and 1,4-oxazepane amides as somatostatin receptor subtype 4 (SSTR4) agonists Grant 10,071,974 - Mazzaferro , et al. September 11, 2 | 2018-09-11 |
Medical Use of Compound III App 20180237445 - SAND; Michael Steven ;   et al. | 2018-08-23 |
Cyclic ether derivatives of pyrazolo[1,5-a]pyrimidine-3-carboxyamide Grant 10,023,575 - Hoenke , et al. July 17, 2 | 2018-07-17 |
Cyclic Ether Derivatives Of Pyrazolo[1,5-a]pyrimidine-3-carboxyamide App 20180134720 - HOENKE; Christoph ;   et al. | 2018-05-17 |
Somatostatin Receptor Subtype 4 (sstr4) Agonists App 20180092880 - Giovannini; Riccardo ;   et al. | 2018-04-05 |
New Ccr2 Receptor Antagonists And Uses Thereof App 20170362249 - Ebel; Heiner ;   et al. | 2017-12-21 |
Morpholine And 1,4-oxazepane Amides As Somatostatin Receptor Subtype 4 (sstr4) Agonists App 20170320838 - MAZZAFERRO; Rocco ;   et al. | 2017-11-09 |
Somatostatin receptor subtype 4 (SSTR4) agonists Grant 9,789,082 - Giovannini , et al. October 17, 2 | 2017-10-17 |
CCR2 receptor antagonists and uses thereof Grant 9,670,222 - Ebel , et al. June 6, 2 | 2017-06-06 |
Cyclic Ether Derivatives Of Pyrazolo[1,5-a]pyrimidine-3-carboxyamide App 20170101411 - HOENKE; Christoph ;   et al. | 2017-04-13 |
New Somatostatin Receptor Subtype 4 (sstr4) Agonists App 20170014381 - Giovannini; Riccardo ;   et al. | 2017-01-19 |
Somatostatin receptor subtype 4 (SSTR4) agonists Grant 9,371,282 - Giovannini , et al. June 21, 2 | 2016-06-21 |
6-cycloalkyl-pyrazolopyrimidinones for the treatment of CNS disorders Grant 9,328,120 - Heine , et al. May 3, 2 | 2016-05-03 |
Derivatives of 4-(piperazinylcarbonyl)thiane-1, 1-dione which inhibit GlyT1 Grant 9,233,953 - Hoenke , et al. January 12, 2 | 2016-01-12 |
Selective CCR2 antagonists Grant 9,108,958 - Ebel , et al. August 18, 2 | 2015-08-18 |
Compounds for the treatment of CNS disorders Grant 9,102,679 - Giovannini , et al. August 11, 2 | 2015-08-11 |
1-heterocyclyl-1,5-dihydro-pyrazolo[3,4-D] pyrimidin-4-one derivatives and their use as PDE9A modulators Grant 9,096,603 - Giovannini , et al. August 4, 2 | 2015-08-04 |
Substituted pyrido[3,2-E][1,2,4]-triazolo[4,3-A]pyrazines for the treatment of central nervous system disorders Grant 9,085,584 - Giovannini , et al. July 21, 2 | 2015-07-21 |
Compounds for the treatment of CNS disorders Grant 9,079,905 - Fuchs , et al. July 14, 2 | 2015-07-14 |
Process and intermediates for the production of CCR2 antagonists Grant 9,067,951 - Ebel , et al. June 30, 2 | 2015-06-30 |
Tricyclic pyridine derivatives, medicaments containing such compounds, their use and process for their preparation Grant 9,029,544 - Wagner , et al. May 12, 2 | 2015-05-12 |
Pyridazine carboxamides as CCR2 receptor antagonists Grant 9,018,212 - Ebel , et al. April 28, 2 | 2015-04-28 |
Phenyl-3-aza-bicyclo[3.1.0]hex-3-yl-methanones and the use thereof as medicament Grant 9,012,489 - Giovannini , et al. April 21, 2 | 2015-04-21 |
Piperazine derivatives and the use thereof as medicament App 20150105397 - HOENKE; Christoph ;   et al. | 2015-04-16 |
CCR2 antagonists Grant 8,962,656 - Ebel , et al. February 24, 2 | 2015-02-24 |
CCR2 receptor antagonists, method for producing the same, and use thereof as medicaments Grant 8,946,218 - Ebel , et al. February 3, 2 | 2015-02-03 |
6-cycloalkyl-pyrazolopyrimidinones For The Treatment Of Cns Disorders App 20150025088 - HEINE; Niklas ;   et al. | 2015-01-22 |
Substituted piperidines as CCR3 antagonists Grant RE45,323 - Grundl , et al. January 6, 2 | 2015-01-06 |
6-cycloalkyl-pyrazolopyrimidinones for the treatment of CNS disorders Grant 8,912,201 - Heine , et al. December 16, 2 | 2014-12-16 |
Compounds For The Treatment Of Cns Disorders App 20140350025 - GIOVANNINI; Riccardo ;   et al. | 2014-11-27 |
New Somatostatin receptor subtype 4 (SSTR4) agonists App 20140343065 - GIOVANNINI; Riccardo ;   et al. | 2014-11-20 |
Process And Intermediates For The Production Of Ccr2 Antagonists App 20140336374 - EBEL; Heiner ;   et al. | 2014-11-13 |
CCR2 receptor antagonists, method for producing the same, and use thereof as medicaments Grant 8,877,745 - Ebel , et al. November 4, 2 | 2014-11-04 |
Ccr2 Receptor Antagonists App 20140323492 - Ebel; Heiner ;   et al. | 2014-10-30 |
CCR2 antagonists and uses thereof Grant 8,841,313 - Ebel , et al. September 23, 2 | 2014-09-23 |
Cyclic pyrimidin-4-carboxamides as CCR2 receptor antagonists for treatment of inflammation, asthma and COPD Grant 8,835,440 - Ebel , et al. September 16, 2 | 2014-09-16 |
6-cycloalkyl-pyrazolopyrimidinones for the treatment of CNS disorders Grant 8,809,345 - Heine , et al. August 19, 2 | 2014-08-19 |
CCR2 receptor antagonists and uses thereof Grant 8,765,949 - Ebel , et al. July 1, 2 | 2014-07-01 |
Tricyclic pyridine derivatives, medicaments containing such compounds, their use and process for their preparation Grant 8,703,793 - Wagner , et al. April 22, 2 | 2014-04-22 |
1-heterocyclyl-1,5-dihydro-pyrazolo[3,4-d] Pyrimidin-4-one Derivatives And Their Use As Pde9a Modulators App 20140073641 - GIOVANNINI; Riccardo ;   et al. | 2014-03-13 |
Therapeutic methods employing substituted piperidines which are CCR3 antagonists Grant 8,653,075 - Grundl , et al. February 18, 2 | 2014-02-18 |
4-Methyl-2,3,5,9,9b-pentaaza-cyclopenta[a]naphthalenes App 20140045856 - GIOVANNINI; Riccardo ;   et al. | 2014-02-13 |
4-Methyl-2,3,5,9,9b-pentaaza-cyclopenta[a]naphthalenes App 20140045857 - GIOVANNINI; Riccardo ;   et al. | 2014-02-13 |
Bicyclic ring system substituted amide functionalised phenols as medicaments Grant 8,648,118 - Giovannini , et al. February 11, 2 | 2014-02-11 |
1, 5-dihydro-pyrazolo (3, 4-D) pyrimidin-4-one derivatives and their use as PDE9A mudulators for the treatment of CNS disorders Grant 8,648,085 - Eickmeier , et al. February 11, 2 | 2014-02-11 |
Bicyclic ring system substituted sulfonamide functionalised phenols as medicaments Grant 8,648,070 - Giovannini , et al. February 11, 2 | 2014-02-11 |
Compounds for the treatment of CNS disorders Grant 8,623,901 - Giovannini , et al. January 7, 2 | 2014-01-07 |
1-heterocyclyl-1,5-dihydro-pyrazolo[3,4-D] pyrimidin-4-one derivates and their use as PDE9A modulators Grant 8,623,879 - Giovannini , et al. January 7, 2 | 2014-01-07 |
Cyclic Pyrimidin-4-carboxamides As Ccr2 Receptor Antagonists For Treatment Of Inflammation, Asthma And Copd App 20130324517 - EBEL; Heiner ;   et al. | 2013-12-05 |
New Ccr2 Antagonists App 20130217728 - Ebel; Heiner ;   et al. | 2013-08-22 |
Phenyl-3-aza-bicyclo[3.1.0]hex-3-yl-methanones and the use thereof as medicament App 20130197011 - GIOVANNINI; Riccardo ;   et al. | 2013-08-01 |
Ccr2 Antagonists And Uses Thereof App 20130184299 - Ebel; Heiner ;   et al. | 2013-07-18 |
Novel And Selective Ccr2 Antagonists App 20130172348 - EBEL; Heiner ;   et al. | 2013-07-04 |
New Selective Ccr2 Antagonists App 20130150354 - EBEL; Heiner ;   et al. | 2013-06-13 |
Novel Antagonists For Ccr2 And Uses Thereof App 20130143905 - Ebel; Heiner ;   et al. | 2013-06-06 |
Novel Ccr2 Receptor Antagonists, Method For Producing The Same, And Use Thereof As Medicaments App 20130123241 - Ebel; Heiner ;   et al. | 2013-05-16 |
New Ccr2 Receptor Antagonists, Method For Producing The Same, And Use Thereof As Medicaments App 20130090338 - Ebel; Heiner ;   et al. | 2013-04-11 |
Pteridinone derivatives as PI3-kinases inhibitors Grant 8,410,100 - Giovannini , et al. April 2, 2 | 2013-04-02 |
Tricyclic pyridine derivatives, medicaments containing such compounds, their use and process for their preparation App 20130053404 - Wagner; Holger ;   et al. | 2013-02-28 |
6-cycloalkyl-pyrazolopyrimidinones For The Treatment Of Cns Disorders App 20130040971 - HEINE; Niklas ;   et al. | 2013-02-14 |
6-cycloalkyl-pyrazolopyrimidinones For The Treatment Of Cns Disorders App 20130040955 - HEINE; Niklas ;   et al. | 2013-02-14 |
Therapeutic methods employing substituted piperidines which are CCR3 antagonists App 20130023517 - GRUNDL; Marc ;   et al. | 2013-01-24 |
Bicyclic Ring System Substituted Amide Functionalised Phenols As Medicaments App 20120329773 - GIOVANNINI; Riccardo ;   et al. | 2012-12-27 |
Bicyclic Ring System Substituted Sulfonamide Functionalised Phenols As Medicaments App 20120316159 - GIOVANNINI; Riccardo ;   et al. | 2012-12-13 |
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Compounds For The Treatment Of Cns Disorders App 20120115863 - Fuchs; Klaus ;   et al. | 2012-05-10 |
Method of treating epilepsy by administering 5-(4{[(2-fluorophenyl)methyl]oxy}phenyl)prolinamide Grant 8,153,681 - Alvaro , et al. April 10, 2 | 2012-04-10 |
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Tricyclic Pyridine Derivatives, Medicaments Containing Such Compounds, Their Use And Process For Their Preparation App 20120053197 - WAGNER; Holger ;   et al. | 2012-03-01 |
Tricyclic Pyridine Derivatives, Medicaments Containing Such Compounds, Their Use And Process For Their Preparation App 20120046304 - WAGNER; Holger ;   et al. | 2012-02-23 |
New Ccr2 Receptor Antagonists And Uses Thereof App 20120004252 - Ebel; Heiner ;   et al. | 2012-01-05 |
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1-heterocyclyl-1,5-dihydro-pyrazolo[3,4-d] Pyrimidin-4-one Derivates And Their Use As Pde9a Modulators App 20110184000 - Giovannini; Riccardo ;   et al. | 2011-07-28 |
Novel Compounds App 20110098335 - Alvaro; Giuseppe ;   et al. | 2011-04-28 |
New Compounds For The Treatment Of Cns Disorders App 20110082137 - GIOVANNINI; Riccardo ;   et al. | 2011-04-07 |
Tricyclic pyridine derivatives, medicaments containing such compounds, their use and process for their preparation App 20110021550 - Wagner; Holger ;   et al. | 2011-01-27 |
1, 5-dihydro-pyrazolo (3, 4-d) Pyrimidin-4-one Derivatives And Their Use As Pde9a Mudulators For The Treatment Of Cns Disorders App 20110015193 - Eickmeier; Christian ;   et al. | 2011-01-20 |
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Pyridine Derivatives and Their Use in The Treatment of Psychotic Disorders App 20100152175 - Alvaro; Giuseppe ;   et al. | 2010-06-17 |
5-(4phenyl)prolinamide For Treatment Of Epilepsy App 20100105754 - Alvaro; Giuseppe ;   et al. | 2010-04-29 |
Pteridinone Derivatives As P13-kinases Inhibitors App 20100099680 - Giovannini; Riccardo ;   et al. | 2010-04-22 |
Compounds Grant 7,655,693 - Alvaro , et al. February 2, 2 | 2010-02-02 |
Methods for the treatment of sleep disorders Grant 7,625,904 - Alvaro , et al. December 1, 2 | 2009-12-01 |
Cyclic Amine Derivatives, Processes For Their Preparation, And Pharmaceutical Compositions Containing Them App 20090192194 - Alvaro; Giuseppe ;   et al. | 2009-07-30 |
Novel Compounds App 20080306122 - Alvaro; Giuseppe ;   et al. | 2008-12-11 |
Novel Compounds App 20080280969 - Alvaro; Giuseppe ;   et al. | 2008-11-13 |
Pyridine Derivatives and Their Use in the Treatment of Psychotic Disorders App 20080269208 - Alvaro; Giuseppe ;   et al. | 2008-10-30 |
Beta-Lactams for Treatment of Cns Disorders App 20080262041 - Alvaro; Giuseppe ;   et al. | 2008-10-23 |
Chemical Compounds App 20080249108 - Alvaro; Giuseppe ;   et al. | 2008-10-09 |
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Chemical compounds Grant 7,071,196 - Alvaro , et al. July 4, 2 | 2006-07-04 |
Chemical compounds App 20060128752 - Alvaro; Giuseppe ;   et al. | 2006-06-15 |
Chemical compounds App 20060122192 - Alvaro; Giuseppe ;   et al. | 2006-06-08 |
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Chemical compounds App 20040209893 - Alvaro, Giuseppe ;   et al. | 2004-10-21 |
Chemical compounds App 20040048862 - Alvaro, Giuseppe ;   et al. | 2004-03-11 |
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Chemical compounds App 20030028021 - Alvaro, Giuseppe ;   et al. | 2003-02-06 |