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Dihydropyridone P1 as factor XIa inhibitors Grant 9,951,071 - Yang , et al. April 24, 2 | 2018-04-24 |
Macrocycles as factor XIa inhibitors Grant 9,902,742 - Pinto , et al. February 27, 2 | 2018-02-27 |
Novel Macrocycles As Factor Xia Inhibitors App 20170158712 - Pinto; Donald J. P. ;   et al. | 2017-06-08 |
Macrocycles as factor XIa inhibitors Grant 9,611,274 - Pinto , et al. April 4, 2 | 2017-04-04 |
Dihydropyridone P1 As Factor Xia Inhibitors App 20160340360 - Yang; Wu ;   et al. | 2016-11-24 |
Dihydropyridone p1 as factor XIa inhibitors Grant 9,409,908 - Yang , et al. August 9, 2 | 2016-08-09 |
Dihydropyridone P1 as factor XIa inhibitors Grant 9,376,444 - Yang , et al. June 28, 2 | 2016-06-28 |
Novel Macrocycles As Factor Xia Inhibitors App 20160068544 - Pinto; Donald J. P. ;   et al. | 2016-03-10 |
Macrocycles as factor XIa inhibitors Grant 9,221,818 - Pinto , et al. December 29, 2 | 2015-12-29 |
Cyclic P1 linkers as factor XIa inhibitors Grant 9,108,981 - Lam , et al. August 18, 2 | 2015-08-18 |
Dihydropyridone P1 As Factor Xia Inhibitors App 20150203492 - Yang; Wu ;   et al. | 2015-07-23 |
Dihydropyridone P1 As Factor Xia Inhibitors App 20150166550 - Yang; Wu ;   et al. | 2015-06-18 |
Cyclic P1 Linkers As Factor Xia Inhibitors App 20150057262 - Lam; Patrick Y.S. ;   et al. | 2015-02-26 |
Cyclic P1 linkers as factor XIa inhibitors Grant 8,901,115 - Lam , et al. December 2, 2 | 2014-12-02 |
Novel Macrocycles As Factor Xia Inhibitors App 20140221338 - Pinto; Donald J. P. ;   et al. | 2014-08-07 |
Cyclic P1 Linkers As Factor Xia Inhibitors App 20140163002 - Lam; Patrick Y.S. ;   et al. | 2014-06-12 |
Dihydropyridone P1 As Factor Xia Inhibitors App 20140038969 - Yang; Wu ;   et al. | 2014-02-06 |
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 8,604,056 - Pinto , et al. December 10, 2 | 2013-12-10 |
Dipeptide analogs as coagulation factor inhibitors Grant 8,367,709 - Pinto , et al. February 5, 2 | 2013-02-05 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20120270853 - Pinto; Donald J.P. ;   et al. | 2012-10-25 |
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 8,252,830 - Pinto , et al. August 28, 2 | 2012-08-28 |
2-Aryl Glycinamide Derivatives App 20110059940 - Gilligan; Paul J. ;   et al. | 2011-03-10 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20110028446 - Pinto; Donald J.P. ;   et al. | 2011-02-03 |
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 7,842,708 - Pinto , et al. November 30, 2 | 2010-11-30 |
Dipeptide Analogs As Coagulation Factor Inhibitors App 20100173899 - Pinto; Donald J.P. ;   et al. | 2010-07-08 |
4-(2-Butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl)pyrazolo-[1,- 5-A]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands Grant 7,662,817 - Gilligan February 16, 2 | 2010-02-16 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20100022506 - Pinto; Donald J.P. ;   et al. | 2010-01-28 |
Arylpropionamide, arylacrylamide, ayrlpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 7,626,039 - Pinto , et al. December 1, 2 | 2009-12-01 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20080161373 - Pinto; Donald J.P. ;   et al. | 2008-07-03 |
4-(2-Butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl)pyrazolo-[1,- 5-A]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands App 20080139567 - Gilligan; Paul J. | 2008-06-12 |
4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl)pyrazolo-[1,- 5-a]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands Grant 7,358,252 - Gilligan April 15, 2 | 2008-04-15 |
Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands Grant 7,319,100 - Arvanitis , et al. January 15, 2 | 2008-01-15 |
Substituted Pyrazinones, Pyridines And Pyrimidines As Corticotropin Releasing Factor Ligands App 20070155740 - Arvanitis; Argyrios G. ;   et al. | 2007-07-05 |
Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands Grant 7,205,306 - Arvanitis , et al. April 17, 2 | 2007-04-17 |
4-(2-Butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl)pyrazolo-[1,- 5-a]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands App 20070054913 - Gilligan; Paul J. | 2007-03-08 |
4-(2-butylamino)-2, 7-dimethyl-8-(2-methyl-6-methoxypyrid-3-YL) pyrazolo-[1,5-A]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands Grant 7,157,578 - Gilligan January 2, 2 | 2007-01-02 |
Salt and crystalline form thereof of a corticotropin releasing factor receptor antagonist Grant 7,153,961 - Gilligan , et al. December 26, 2 | 2006-12-26 |
Sulfonamide bicyclic compounds Grant 7,144,894 - Gilligan December 5, 2 | 2006-12-05 |
Pyrazolotriazines as CRF antagonists Grant 7,026,317 - Gilligan , et al. April 11, 2 | 2006-04-11 |
Sulfonamide bicyclic compounds App 20060063799 - Gilligan; Paul J. | 2006-03-23 |
Pyrazolotriazines as CRF antagonists Grant 6,960,583 - Gilligan , et al. November 1, 2 | 2005-11-01 |
Pyrazolopyrimidines as CRF antagonists Grant 6,958,341 - Wilde , et al. October 25, 2 | 2005-10-25 |
Salt and crystalline form thereof of a corticotropin releasing factor receptor antagonist App 20050113375 - Gilligan, Paul J. ;   et al. | 2005-05-26 |
Pyrazolotriazines as CRF antagonists App 20040176376 - Gilligan, Paul J. ;   et al. | 2004-09-09 |
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Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands App 20030171380 - Arvanitis, Argyrios G. ;   et al. | 2003-09-11 |
Pyrazolopyrimidines as CRF antagonists App 20030139426 - Wilde, Richard G. ;   et al. | 2003-07-24 |
Imidazo[1,2-a]pyrazines for the treatment of neurological disorders Grant 6,589,952 - Bakthavatchalam , et al. July 8, 2 | 2003-07-08 |
4 - (2-butylamino) - 2, 7-dimethyl-8- (2-methyl-6-methoxypyrid-3-yl) pyrazolo- [1,5-A] - 1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands App 20030125330 - Gilligan, Paul J. | 2003-07-03 |
Pyrazolotriazines as CRF antagonists App 20020147338 - Gilligan, Paul J. ;   et al. | 2002-10-10 |
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Heterocyclyl-substituted ring-fused pyridines and pyrimidines as corticotropin releasing hormone (CRH) antagonists, useful for treating cns and stress-related disorders App 20010025042 - Arvanitis, Argyrios ;   et al. | 2001-09-27 |
Nitrogen substituted imidazo[4,5-C]pyrazoles as corticotropin releasing hormone antagonists Grant 6,174,912 - Beck , et al. January 16, 2 | 2001-01-16 |
Aryl- and arylamino- substituted heterocycles as corticotropin releasing hormone antagonists Grant 6,103,737 - Cocuzza , et al. August 15, 2 | 2000-08-15 |
Antipsychotic nitrogen-containing bicyclic compounds Grant 5,532,243 - Gilligan July 2, 1 | 1996-07-02 |
Antipsychotic 1-cycloalkylpiperidines Grant 5,109,002 - Cain , et al. April 28, 1 | 1992-04-28 |
Antibiotic derivatives of 7-phenyl-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids Grant 4,623,650 - Gilligan , et al. November 18, 1 | 1986-11-18 |