loadpatents
name:-0.036454916000366
name:-0.033586025238037
name:-0.0011141300201416
Gilligan; Paul J. Patent Filings

Gilligan; Paul J.

Patent Applications and Registrations

Patent applications and USPTO patent grants for Gilligan; Paul J..The latest application filed is for "novel macrocycles as factor xia inhibitors".

Company Profile
0.33.31
  • Gilligan; Paul J. - Wilmington DE
  • Gilligan; Paul J - Wilmington DE
  • Gilligan, Paul J. - US
  • Gilligan; Paul J. - Claymont DE
  • Gilligan; Paul J. - New Haven CT
*profile and listings may contain filings by different individuals or companies with the same name. Review application materials to confirm ownership/assignment.
Patent Activity
PatentDate
Dihydropyridone P1 as factor XIa inhibitors
Grant 9,951,071 - Yang , et al. April 24, 2
2018-04-24
Macrocycles as factor XIa inhibitors
Grant 9,902,742 - Pinto , et al. February 27, 2
2018-02-27
Novel Macrocycles As Factor Xia Inhibitors
App 20170158712 - Pinto; Donald J. P. ;   et al.
2017-06-08
Macrocycles as factor XIa inhibitors
Grant 9,611,274 - Pinto , et al. April 4, 2
2017-04-04
Dihydropyridone P1 As Factor Xia Inhibitors
App 20160340360 - Yang; Wu ;   et al.
2016-11-24
Dihydropyridone p1 as factor XIa inhibitors
Grant 9,409,908 - Yang , et al. August 9, 2
2016-08-09
Dihydropyridone P1 as factor XIa inhibitors
Grant 9,376,444 - Yang , et al. June 28, 2
2016-06-28
Novel Macrocycles As Factor Xia Inhibitors
App 20160068544 - Pinto; Donald J. P. ;   et al.
2016-03-10
Macrocycles as factor XIa inhibitors
Grant 9,221,818 - Pinto , et al. December 29, 2
2015-12-29
Cyclic P1 linkers as factor XIa inhibitors
Grant 9,108,981 - Lam , et al. August 18, 2
2015-08-18
Dihydropyridone P1 As Factor Xia Inhibitors
App 20150203492 - Yang; Wu ;   et al.
2015-07-23
Dihydropyridone P1 As Factor Xia Inhibitors
App 20150166550 - Yang; Wu ;   et al.
2015-06-18
Cyclic P1 Linkers As Factor Xia Inhibitors
App 20150057262 - Lam; Patrick Y.S. ;   et al.
2015-02-26
Cyclic P1 linkers as factor XIa inhibitors
Grant 8,901,115 - Lam , et al. December 2, 2
2014-12-02
Novel Macrocycles As Factor Xia Inhibitors
App 20140221338 - Pinto; Donald J. P. ;   et al.
2014-08-07
Cyclic P1 Linkers As Factor Xia Inhibitors
App 20140163002 - Lam; Patrick Y.S. ;   et al.
2014-06-12
Dihydropyridone P1 As Factor Xia Inhibitors
App 20140038969 - Yang; Wu ;   et al.
2014-02-06
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors
Grant 8,604,056 - Pinto , et al. December 10, 2
2013-12-10
Dipeptide analogs as coagulation factor inhibitors
Grant 8,367,709 - Pinto , et al. February 5, 2
2013-02-05
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors
App 20120270853 - Pinto; Donald J.P. ;   et al.
2012-10-25
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors
Grant 8,252,830 - Pinto , et al. August 28, 2
2012-08-28
2-Aryl Glycinamide Derivatives
App 20110059940 - Gilligan; Paul J. ;   et al.
2011-03-10
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors
App 20110028446 - Pinto; Donald J.P. ;   et al.
2011-02-03
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors
Grant 7,842,708 - Pinto , et al. November 30, 2
2010-11-30
Dipeptide Analogs As Coagulation Factor Inhibitors
App 20100173899 - Pinto; Donald J.P. ;   et al.
2010-07-08
4-(2-Butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl)pyrazolo-[1,- 5-A]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands
Grant 7,662,817 - Gilligan February 16, 2
2010-02-16
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors
App 20100022506 - Pinto; Donald J.P. ;   et al.
2010-01-28
Arylpropionamide, arylacrylamide, ayrlpropynamide, or arylmethylurea analogs as factor XIa inhibitors
Grant 7,626,039 - Pinto , et al. December 1, 2
2009-12-01
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors
App 20080161373 - Pinto; Donald J.P. ;   et al.
2008-07-03
4-(2-Butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl)pyrazolo-[1,- 5-A]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands
App 20080139567 - Gilligan; Paul J.
2008-06-12
4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl)pyrazolo-[1,- 5-a]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands
Grant 7,358,252 - Gilligan April 15, 2
2008-04-15
Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands
Grant 7,319,100 - Arvanitis , et al. January 15, 2
2008-01-15
Substituted Pyrazinones, Pyridines And Pyrimidines As Corticotropin Releasing Factor Ligands
App 20070155740 - Arvanitis; Argyrios G. ;   et al.
2007-07-05
Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands
Grant 7,205,306 - Arvanitis , et al. April 17, 2
2007-04-17
4-(2-Butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl)pyrazolo-[1,- 5-a]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands
App 20070054913 - Gilligan; Paul J.
2007-03-08
4-(2-butylamino)-2, 7-dimethyl-8-(2-methyl-6-methoxypyrid-3-YL) pyrazolo-[1,5-A]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands
Grant 7,157,578 - Gilligan January 2, 2
2007-01-02
Salt and crystalline form thereof of a corticotropin releasing factor receptor antagonist
Grant 7,153,961 - Gilligan , et al. December 26, 2
2006-12-26
Sulfonamide bicyclic compounds
Grant 7,144,894 - Gilligan December 5, 2
2006-12-05
Pyrazolotriazines as CRF antagonists
Grant 7,026,317 - Gilligan , et al. April 11, 2
2006-04-11
Sulfonamide bicyclic compounds
App 20060063799 - Gilligan; Paul J.
2006-03-23
Pyrazolotriazines as CRF antagonists
Grant 6,960,583 - Gilligan , et al. November 1, 2
2005-11-01
Pyrazolopyrimidines as CRF antagonists
Grant 6,958,341 - Wilde , et al. October 25, 2
2005-10-25
Salt and crystalline form thereof of a corticotropin releasing factor receptor antagonist
App 20050113375 - Gilligan, Paul J. ;   et al.
2005-05-26
Pyrazolotriazines as CRF antagonists
App 20040176376 - Gilligan, Paul J. ;   et al.
2004-09-09
4- (2-butylamino) -2, 7-dimethyl-8- (2-methyl-6-methoxypyrid-3-YL) pyrazolo- [1,5-A] -1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands
App 20040014760 - Gilligan, Paul J.
2004-01-22
Imidazo[1, 2-a] pyrazines for the treatment of irritable bowel syndrome
App 20030220342 - Bakthavatchalam, Rajagopal ;   et al.
2003-11-27
Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands
App 20030171380 - Arvanitis, Argyrios G. ;   et al.
2003-09-11
Pyrazolopyrimidines as CRF antagonists
App 20030139426 - Wilde, Richard G. ;   et al.
2003-07-24
Imidazo[1,2-a]pyrazines for the treatment of neurological disorders
Grant 6,589,952 - Bakthavatchalam , et al. July 8, 2
2003-07-08
4 - (2-butylamino) - 2, 7-dimethyl-8- (2-methyl-6-methoxypyrid-3-yl) pyrazolo- [1,5-A] - 1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands
App 20030125330 - Gilligan, Paul J.
2003-07-03
Pyrazolotriazines as CRF antagonists
App 20020147338 - Gilligan, Paul J. ;   et al.
2002-10-10
Imidazo[1,2-a]pyrazines for the treatment of neurological disorders
App 20020049208 - Bakthavatchalam, Rajagopal ;   et al.
2002-04-25
Heterocyclyl-substituted ring-fused pyridines and pyrimidines as corticotropin releasing hormone (CRH) antagonists, useful for treating cns and stress-related disorders
App 20010025042 - Arvanitis, Argyrios ;   et al.
2001-09-27
Nitrogen substituted imidazo[4,5-C]pyrazoles as corticotropin releasing hormone antagonists
Grant 6,174,912 - Beck , et al. January 16, 2
2001-01-16
Aryl- and arylamino- substituted heterocycles as corticotropin releasing hormone antagonists
Grant 6,103,737 - Cocuzza , et al. August 15, 2
2000-08-15
Antipsychotic nitrogen-containing bicyclic compounds
Grant 5,532,243 - Gilligan July 2, 1
1996-07-02
Antipsychotic 1-cycloalkylpiperidines
Grant 5,109,002 - Cain , et al. April 28, 1
1992-04-28
Antibiotic derivatives of 7-phenyl-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids
Grant 4,623,650 - Gilligan , et al. November 18, 1
1986-11-18

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