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name:-0.16951298713684
name:-0.05758810043335
name:-0.011425018310547
Gijsen; Henricus Jacobus Maria Patent Filings

Gijsen; Henricus Jacobus Maria

Patent Applications and Registrations

Patent applications and USPTO patent grants for Gijsen; Henricus Jacobus Maria.The latest application filed is for "inhibitors of beta secretase".

Company Profile
8.52.52
  • Gijsen; Henricus Jacobus Maria - Breda NL
  • GIJSEN; Henricus Jacobus Maria - Beerse BE
  • Gijsen; Henricus Jacobus Maria - Turnhoutseweg BE
*profile and listings may contain filings by different individuals or companies with the same name. Review application materials to confirm ownership/assignment.
Patent Activity
PatentDate
[1,2,4]triazolo[1,5-a]pyrimidine compounds as PDE2 inhibitors
Grant 11,319,321 - Van Roosbroeck , et al. May 3, 2
2022-05-03
Inhibitors Of Beta Secretase
App 20210284659 - Vos; Ann Marleen ;   et al.
2021-09-16
[1,2,4]triazolo[1,5-a]pyrimidine compounds as PDE2 inhibitors
Grant 11,053,248 - Van Roosbroeck , et al. July 6, 2
2021-07-06
[1,2,4]triazolo[1,5-a]pyrimidin-7-yl compound
Grant 10,947,239 - Buijnsters , et al. March 16, 2
2021-03-16
[1,2,4]triazolo[1,5and#8208;A]pyrimidine compounds as PDE2 inhibitors
Grant 10,947,242 - Van Roosbroeck , et al. March 16, 2
2021-03-16
Substituted imidazoles as N-type calcium channel blockers
Grant 10,653,673 - Ahmad , et al.
2020-05-19
[1,2,4]triazolo[1,5-a]pyrimidine Compounds As Pde2 Inhibitors
App 20200055858 - Van Roosbroeck; Yves Emiel Maria ;   et al.
2020-02-20
Substituted 3,4-dihydro-2H-pyrido[1,2-a]pyrazine-1,6-diones as gamma secretase modulators
Grant 10,562,897 - Bischoff , et al. Feb
2020-02-18
[1,2,4]triazolo[1,5-a]pyrimidine Compounds As Pde2 Inhibitors
App 20200048260 - Van Roosbroeck; Yves Emiel Maria ;   et al.
2020-02-13
Inhibitors Of Beta Secretase
App 20200010482 - Vos; Ann Marleen ;   et al.
2020-01-09
Inhibitors Of Beta Secretase
App 20190389882 - Van Brandt; Sven Franciscus Anna ;   et al.
2019-12-26
[1,2,4]triazolo[1,5‐a]pyrimidine Compounds As Pde2 Inhibitors
App 20190276462 - Van Roosbroeck; Yves Emiel Maria ;   et al.
2019-09-12
Substituted 3,4-dihydro-2H-pyrido[1,2-a]pyrazine-1,6-diones as gamma secretase modulators
Grant 10,246,454 - Bischoff , et al.
2019-04-02
2,3,4,5-tetrahydropyridin-6-amine Derivatives
App 20180334447 - ROMBOUTS; Frederik Jan Rita ;   et al.
2018-11-22
[1,2,4]TRIAZOLO[1,5-a]PYRIMIDIN-7-YL COMPOUND
App 20180327408 - BUIJNSTERS; Petrus Jacobus Johannes Antonius ;   et al.
2018-11-15
Novel Substituted Pyrido-piperazinone Derivatives As Gamma Secretase Modulators
App 20180319797 - Bischoff; Francois Paul ;   et al.
2018-11-08
Substituted imidazoles as gamma secretase modulators
Grant 10,112,943 - Bischoff , et al. October 30, 2
2018-10-30
2,3,4,5-tetrahydropyridin-6-amine and 3,4-dihydro-2H-pyrrol-5-amine compound inhibitors of beta-secretase
Grant 10,106,524 - Trabanco-Suarez , et al. October 23, 2
2018-10-23
Substituted Imidazoles As N-type Calcium Channel Blockers
App 20180161312 - Ahmad; Ishtiyaque ;   et al.
2018-06-14
Substituted imidazoles as N-type calcium channel blockers
Grant 9,974,775 - Ahmad , et al. May 22, 2
2018-05-22
2,3,4,5-tetrahydropyridin-6-amine And 3,4-dihydro-2h-pyrrol-5-amine Compound Inhibitors Of Beta-secretase
App 20170362198 - Trabanco-Suarez; Andres Avelino ;   et al.
2017-12-21
5,6-dihydro-imidazo[1,2-a]pyrazin-8-ylamine derivatives useful as inhibitors of beta-secretase (BACE)
Grant 9,840,507 - Trabanco-Suarez , et al. December 12, 2
2017-12-12
4-Amino-6-phenyl-5,6-dihydroimidazo[1,5-a]pyrazin-3(2H)-one derivatives as inhibitors of beta-secretase (BACE)
Grant 9,834,559 - Oehlrich , et al. December 5, 2
2017-12-05
5,6-dihydro-2H-[1,4]oxazin-3-yl-amine derivatives useful as inhibitors of beta-secretase (BACE)
Grant 9,828,350 - Trabanco-Suarez , et al. November 28, 2
2017-11-28
4-amino-6-phenyl-6,7-dihydro[1,2,3]triazolo[1,5-A]pyrazine derivatives as inhibitors of beta-secretase (BACE)
Grant 9,751,886 - Oehlrich , et al. September 5, 2
2017-09-05
4-amino-6-phenyl-5,6-dihydroimidazo[1,5-A]pyrazine derivatives as inhibitors of beta-secretase (BACE)
Grant 9,580,433 - Oehlrich , et al. February 28, 2
2017-02-28
Substituted Imidazoles As N-type Calcium Channel Blockers
App 20160310468 - Ahmad; Ishtiyaque ;   et al.
2016-10-27
Substituted imidazoles as N-type calcium channel blockers
Grant 9,453,002 - Ahmad , et al. September 27, 2
2016-09-27
5,6-dihydro-2h-[1,4]oxazin-3-yl-amine Derivatives Useful As Inhibitors Of Beta-secretase (bace)
App 20160152581 - Trabanco-Suarez; Andres Avelino ;   et al.
2016-06-02
6,7-dihydro-pyrazolo[1,5-a]pyrazin-4-ylamine derivatives useful as inhibitors of beta-secretase (BACE)
Grant 9,346,811 - Trabanco-Suarez , et al. May 24, 2
2016-05-24
4-amino-6-phenyl-6,7-dihydro[1,2,3]triazolo[1,5-a]pyrazine Derivatives As Inhibitors Of Beta-secretase (bace)
App 20160130274 - Oehlrich; Daniel ;   et al.
2016-05-12
4-amino-6-phenyl-5,6-dihydroimidazo[1,5-a]pyrazin-3(2h)-one Derivatives As Inhibitors Of Beta-secretase (bace)
App 20160115171 - Oehlrich; Daniel ;   et al.
2016-04-28
4-amino-6-phenyl-5,6-dihydroimidazo[1,5-a]pyrazine Derivatives As Inhibitors Of Beta-secretase (bace)
App 20160115170 - Oehlrich; Daniel ;   et al.
2016-04-28
Benzimidazole cannabinoid agonists bearing a substituted heterocyclic group
Grant 9,284,303 - Gijsen , et al. March 15, 2
2016-03-15
Novel Substituted Pyrido-piperazinone Derivatives As Gamma Secretase Modulators
App 20150353544 - Bischoff; Francois Paul ;   et al.
2015-12-10
Substituted pyrido[1,2-a]pyrazines and substituted pyrido[1,2-a][1,4]diazepines for the treatment of (inter alia) Alzheimer's disease
Grant 9,181,245 - Rombouts , et al. November 10, 2
2015-11-10
NOVEL TRICYCLIC 3,4-DIHYDRO-2H-PYRIDO[1,2-a]PYRAZINE-1,6-DIONE DERIVATIVES AS GAMMA SECRETASE MODULATORS
App 20150307496 - Bischoff; Francois Paul ;   et al.
2015-10-29
Substituted bicyclic triazole derivatives as gamma secretase modulators
Grant 9,145,399 - De Cleyn , et al. September 29, 2
2015-09-29
Substituted indole derivatives as gamma secretase modulators
Grant 9,115,143 - Minne , et al. August 25, 2
2015-08-25
Substituted triazole derivatives as gamma secretase modulators
Grant 9,079,886 - Van Brandt , et al. July 14, 2
2015-07-14
Substituted 3,4-dihydro-2h-pyrido[1,2-a]pyrazine-1,6-dione Derivatives Useful For The Treatment Of (inter Alia) Alzheimer's Disease
App 20150141411 - Rombouts; Frederik Jan Rita ;   et al.
2015-05-21
Novel Substituted Bicyclic Heterocyclic Compounds As Gamma Secretase Modulators
App 20150094311 - GIJSEN; HENRICUS JACOBUS MARIA ;   et al.
2015-04-02
Substituted Imidazoles As N-type Calcium Channel Blockers
App 20150051225 - Ahmad; Ishtiyaque ;   et al.
2015-02-19
Substituted bicyclic heterocyclic compounds as gamma secretase modulators
Grant 8,946,426 - Gijsen , et al. February 3, 2
2015-02-03
Substituted triazole and imidazole derivatives as gamma secretase modulators
Grant 8,946,266 - Wu , et al. February 3, 2
2015-02-03
5-(3-aminophenyl)-5-alkyl-5,6-dihydro-2h-[1,4]oxazin-3-amine Derivatives
App 20140364428 - Gijsen; Henricus Jacobus Maria ;   et al.
2014-12-11
6-difluoromethyl-5,6-dihydro-2h-[1,4]oxazin-3-amine Derivatives
App 20140343048 - Trabanco-Suarez; Andres Avelino ;   et al.
2014-11-20
Substituted indazole and aza-indazole derivatives as gamma secretase modulators
Grant 8,835,482 - Bischoff , et al. September 16, 2
2014-09-16
Substituted benzoxazole, benzimidazole, oxazolopyridine and imidazopyridine derivatives as gamma secretase modulators
Grant 8,772,504 - Gijsen , et al. July 8, 2
2014-07-08
Novel Substituted Indole Derivatives As Gamma Secretase Modulators
App 20140148450 - Minne; Garrett Berlond ;   et al.
2014-05-29
6,7-DIHYDRO-PYRAZOLO[1,5-a]PYRAZIN-4-YLAMINE DERIVATIVES USEFUL AS INHIBITORS OF BETA-SECRETASE (BACE)
App 20140005200 - Trabanco-Suarez; Andres Avelino ;   et al.
2014-01-02
Heterocyclic amides as modulators of TRPA1
Grant 8,614,201 - Berthelot , et al. December 24, 2
2013-12-24
Benzimidazole Cannabinoid Agonists Bearing A Substituted Heterocyclic Group
App 20130324529 - Gijsen; Henricus Jacobus Maria ;   et al.
2013-12-05
5,6-DIHYDRO-IMIDAZO[1,2-a]PYRAZIN-8-YLAMINE DERIVATIVES USEFUL AS INHIBITORS OF BETA-SECRETASE (BACE)
App 20130274266 - Trabanco-Suarez; Andres Avelino ;   et al.
2013-10-17
Substituted bicyclic imidazole derivatives as gamma secretase modulators
Grant 8,546,440 - Gijsen , et al. October 1, 2
2013-10-01
Benzimidazole cannabinoid agonists bearing a substituted heterocyclic group
Grant 8,524,757 - Gijsen , et al. September 3, 2
2013-09-03
Dibenzoazepine and dibenzooxazepine TRPA1 agonists
Grant 8,461,145 - Gijsen , et al. June 11, 2
2013-06-11
5,6-dihydro-2h-[1,4]oxazin-3-yl-amine Derivatives Useful As Inhibitors Of Beta-secretase (bace)
App 20130109683 - Trabanco-Suarez; Andres Avelino ;   et al.
2013-05-02
Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT.sub.4-antagonists
Grant 8,334,304 - Bosmans , et al. December 18, 2
2012-12-18
Novel Substituted Bicyclic Triazole Derivatives As Gamma Secretase Modulators
App 20120295901 - De Cleyn; Michel Anna Jozef ;   et al.
2012-11-22
Novel Substituted Triazole Derivatives As Gamma Secretase Modulators
App 20120295891 - Van Brandt; Sven Franciscus Anna ;   et al.
2012-11-22
Benzimidazole cannabinoid agonists
Grant 8,193,369 - Gijsen , et al. June 5, 2
2012-06-05
Novel Substituted Triazole And Imidazole Derivatives As Gamma Secretase Modulators
App 20120135981 - Wu; Tongfei ;   et al.
2012-05-31
Novel Substituted Indazole And Aza-indazole Derivatives As Gamma Secretase Modulators
App 20120095036 - Bischoff; Francois Paul ;   et al.
2012-04-19
Heterocyclic Amides As Modulators Of Trpa1
App 20120083474 - Berthelot; Didier Jean-Claude ;   et al.
2012-04-05
Novel Substituted Bicyclic Heterocyclic Compounds As Gamma Secretase Modulators
App 20110281881 - Gijsen; Henricus, Jacobus, Maria ;   et al.
2011-11-17
Substituted Bicyclic Imidazole Derivatives As Gamma Secretase Modulators
App 20110237580 - Gijsen; Henricus Jacobus Maria ;   et al.
2011-09-29
3,4-dihydropyrimidine Trpa1 Antagonists
App 20110124666 - Gijsen; Henricus Jacobus Maria ;   et al.
2011-05-26
Dibenzoazepine And Dibenzooxazepine Trpa1 Agonists
App 20100273773 - Gijsen; Henricus Jacobus Maria ;   et al.
2010-10-28
Fluoro Alkyl Substituted Benzimidazole Cannabinoid Agonists
App 20100273831 - Gijsen; Henricus Jacobus Maria ;   et al.
2010-10-28
Heterocyclic substituted 4-(aminomethyl)-piperidine benzamides as 5HT.sub.4-antagonists
Grant 7,732,464 - Bosmans , et al. June 8, 2
2010-06-08
Aminosulfonyl Substituted 4-(Aminomethyl)-Piperidine Benzamides As 5HT 4-Antagonists
App 20100087483 - BOSMANS; Jean-Paul Rene Marie Andre ;   et al.
2010-04-08
Benzimidazole Cannabinoid Agonists
App 20100041702 - Gijsen; Henricus Jacobus Maria ;   et al.
2010-02-18
Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT.sub.4-antagonists
Grant 7,652,040 - Bosmans , et al. January 26, 2
2010-01-26
4-(aminomethyl)-piperidine benzamides as 5HT.sub.4-antagonists
Grant 7,638,535 - Bosmans , et al. December 29, 2
2009-12-29
5HT.sub.4-antagonistic 4-(aminomethyl)-piperidine benzamides
Grant 7,635,706 - Bosmans , et al. December 22, 2
2009-12-22
Benzimidazole Cannabinoid Agonists Bearing A Substituted Heterocyclic Group
App 20090312339 - Gijsen; Henricus Jacobus Maria ;   et al.
2009-12-17
Hydroxycarbonylphenyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT.sub.4 antagonists
Grant 7,498,347 - Bosmans , et al. March 3, 2
2009-03-03
Heterocyclic substituted 4-(aminomethyl)-piperidine benzamides as 5ht4-antagonists
App 20070197600 - Bosmans; Jean-Paul Rene Marie Andre ;   et al.
2007-08-23
4-(aminomethyl)-piperidine benzamides for treating gastrointestinal disorders
Grant 7,205,410 - Bosmans , et al. April 17, 2
2007-04-17
5Ht4-antagonistic 4-(aminomethyl)-piperidine benzamides
App 20070032486 - Bosmans; Jean-Paul Rene Marie Andre ;   et al.
2007-02-08
4-(Aminomethyl)-piperidine benzamides as 5ht4 - antagonists
App 20060281753 - Bosmans; Jean-Paul Rene Marie Andre ;   et al.
2006-12-14
Chimeric gaba receptor
App 20060216749 - Smans; Karine Alfonsine Astrid ;   et al.
2006-09-28
Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5ht 4-antagonists
App 20060142339 - Bosmans; Jean-Paul Rene Marie Andre ;   et al.
2006-06-29
Hydroxycarbonylphenyl substituted 4-(aminomethyl)-piperidine benzamides as 5ht4 antagonists
App 20060142340 - Bosmans; Jean-Paul Rene Marie Andre ;   et al.
2006-06-29
4-(aminomethyl)-piperidine benzamides for treating gastrointestinal disorders
App 20030181456 - Bosmans, Jean-Paul Rene Marie Andre ;   et al.
2003-09-25
4-(aminomethyl)-piperidine benzamides for treating gastrointestinal disorders
Grant 6,544,997 - Bosmans , et al. April 8, 2
2003-04-08

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