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[1,2,4]triazolo[1,5-a]pyrimidine compounds as PDE2 inhibitors Grant 11,319,321 - Van Roosbroeck , et al. May 3, 2 | 2022-05-03 |
Inhibitors Of Beta Secretase App 20210284659 - Vos; Ann Marleen ;   et al. | 2021-09-16 |
[1,2,4]triazolo[1,5-a]pyrimidine compounds as PDE2 inhibitors Grant 11,053,248 - Van Roosbroeck , et al. July 6, 2 | 2021-07-06 |
[1,2,4]triazolo[1,5-a]pyrimidin-7-yl compound Grant 10,947,239 - Buijnsters , et al. March 16, 2 | 2021-03-16 |
[1,2,4]triazolo[1,5and#8208;A]pyrimidine compounds as PDE2 inhibitors Grant 10,947,242 - Van Roosbroeck , et al. March 16, 2 | 2021-03-16 |
Substituted imidazoles as N-type calcium channel blockers Grant 10,653,673 - Ahmad , et al. | 2020-05-19 |
[1,2,4]triazolo[1,5-a]pyrimidine Compounds As Pde2 Inhibitors App 20200055858 - Van Roosbroeck; Yves Emiel Maria ;   et al. | 2020-02-20 |
Substituted 3,4-dihydro-2H-pyrido[1,2-a]pyrazine-1,6-diones as gamma secretase modulators Grant 10,562,897 - Bischoff , et al. Feb | 2020-02-18 |
[1,2,4]triazolo[1,5-a]pyrimidine Compounds As Pde2 Inhibitors App 20200048260 - Van Roosbroeck; Yves Emiel Maria ;   et al. | 2020-02-13 |
Inhibitors Of Beta Secretase App 20200010482 - Vos; Ann Marleen ;   et al. | 2020-01-09 |
Inhibitors Of Beta Secretase App 20190389882 - Van Brandt; Sven Franciscus Anna ;   et al. | 2019-12-26 |
[1,2,4]triazolo[1,5‐a]pyrimidine Compounds As Pde2 Inhibitors App 20190276462 - Van Roosbroeck; Yves Emiel Maria ;   et al. | 2019-09-12 |
Substituted 3,4-dihydro-2H-pyrido[1,2-a]pyrazine-1,6-diones as gamma secretase modulators Grant 10,246,454 - Bischoff , et al. | 2019-04-02 |
2,3,4,5-tetrahydropyridin-6-amine Derivatives App 20180334447 - ROMBOUTS; Frederik Jan Rita ;   et al. | 2018-11-22 |
[1,2,4]TRIAZOLO[1,5-a]PYRIMIDIN-7-YL COMPOUND App 20180327408 - BUIJNSTERS; Petrus Jacobus Johannes Antonius ;   et al. | 2018-11-15 |
Novel Substituted Pyrido-piperazinone Derivatives As Gamma Secretase Modulators App 20180319797 - Bischoff; Francois Paul ;   et al. | 2018-11-08 |
Substituted imidazoles as gamma secretase modulators Grant 10,112,943 - Bischoff , et al. October 30, 2 | 2018-10-30 |
2,3,4,5-tetrahydropyridin-6-amine and 3,4-dihydro-2H-pyrrol-5-amine compound inhibitors of beta-secretase Grant 10,106,524 - Trabanco-Suarez , et al. October 23, 2 | 2018-10-23 |
Substituted Imidazoles As N-type Calcium Channel Blockers App 20180161312 - Ahmad; Ishtiyaque ;   et al. | 2018-06-14 |
Substituted imidazoles as N-type calcium channel blockers Grant 9,974,775 - Ahmad , et al. May 22, 2 | 2018-05-22 |
2,3,4,5-tetrahydropyridin-6-amine And 3,4-dihydro-2h-pyrrol-5-amine Compound Inhibitors Of Beta-secretase App 20170362198 - Trabanco-Suarez; Andres Avelino ;   et al. | 2017-12-21 |
5,6-dihydro-imidazo[1,2-a]pyrazin-8-ylamine derivatives useful as inhibitors of beta-secretase (BACE) Grant 9,840,507 - Trabanco-Suarez , et al. December 12, 2 | 2017-12-12 |
4-Amino-6-phenyl-5,6-dihydroimidazo[1,5-a]pyrazin-3(2H)-one derivatives as inhibitors of beta-secretase (BACE) Grant 9,834,559 - Oehlrich , et al. December 5, 2 | 2017-12-05 |
5,6-dihydro-2H-[1,4]oxazin-3-yl-amine derivatives useful as inhibitors of beta-secretase (BACE) Grant 9,828,350 - Trabanco-Suarez , et al. November 28, 2 | 2017-11-28 |
4-amino-6-phenyl-6,7-dihydro[1,2,3]triazolo[1,5-A]pyrazine derivatives as inhibitors of beta-secretase (BACE) Grant 9,751,886 - Oehlrich , et al. September 5, 2 | 2017-09-05 |
4-amino-6-phenyl-5,6-dihydroimidazo[1,5-A]pyrazine derivatives as inhibitors of beta-secretase (BACE) Grant 9,580,433 - Oehlrich , et al. February 28, 2 | 2017-02-28 |
Substituted Imidazoles As N-type Calcium Channel Blockers App 20160310468 - Ahmad; Ishtiyaque ;   et al. | 2016-10-27 |
Substituted imidazoles as N-type calcium channel blockers Grant 9,453,002 - Ahmad , et al. September 27, 2 | 2016-09-27 |
5,6-dihydro-2h-[1,4]oxazin-3-yl-amine Derivatives Useful As Inhibitors Of Beta-secretase (bace) App 20160152581 - Trabanco-Suarez; Andres Avelino ;   et al. | 2016-06-02 |
6,7-dihydro-pyrazolo[1,5-a]pyrazin-4-ylamine derivatives useful as inhibitors of beta-secretase (BACE) Grant 9,346,811 - Trabanco-Suarez , et al. May 24, 2 | 2016-05-24 |
4-amino-6-phenyl-6,7-dihydro[1,2,3]triazolo[1,5-a]pyrazine Derivatives As Inhibitors Of Beta-secretase (bace) App 20160130274 - Oehlrich; Daniel ;   et al. | 2016-05-12 |
4-amino-6-phenyl-5,6-dihydroimidazo[1,5-a]pyrazin-3(2h)-one Derivatives As Inhibitors Of Beta-secretase (bace) App 20160115171 - Oehlrich; Daniel ;   et al. | 2016-04-28 |
4-amino-6-phenyl-5,6-dihydroimidazo[1,5-a]pyrazine Derivatives As Inhibitors Of Beta-secretase (bace) App 20160115170 - Oehlrich; Daniel ;   et al. | 2016-04-28 |
Benzimidazole cannabinoid agonists bearing a substituted heterocyclic group Grant 9,284,303 - Gijsen , et al. March 15, 2 | 2016-03-15 |
Novel Substituted Pyrido-piperazinone Derivatives As Gamma Secretase Modulators App 20150353544 - Bischoff; Francois Paul ;   et al. | 2015-12-10 |
Substituted pyrido[1,2-a]pyrazines and substituted pyrido[1,2-a][1,4]diazepines for the treatment of (inter alia) Alzheimer's disease Grant 9,181,245 - Rombouts , et al. November 10, 2 | 2015-11-10 |
NOVEL TRICYCLIC 3,4-DIHYDRO-2H-PYRIDO[1,2-a]PYRAZINE-1,6-DIONE DERIVATIVES AS GAMMA SECRETASE MODULATORS App 20150307496 - Bischoff; Francois Paul ;   et al. | 2015-10-29 |
Substituted bicyclic triazole derivatives as gamma secretase modulators Grant 9,145,399 - De Cleyn , et al. September 29, 2 | 2015-09-29 |
Substituted indole derivatives as gamma secretase modulators Grant 9,115,143 - Minne , et al. August 25, 2 | 2015-08-25 |
Substituted triazole derivatives as gamma secretase modulators Grant 9,079,886 - Van Brandt , et al. July 14, 2 | 2015-07-14 |
Substituted 3,4-dihydro-2h-pyrido[1,2-a]pyrazine-1,6-dione Derivatives Useful For The Treatment Of (inter Alia) Alzheimer's Disease App 20150141411 - Rombouts; Frederik Jan Rita ;   et al. | 2015-05-21 |
Novel Substituted Bicyclic Heterocyclic Compounds As Gamma Secretase Modulators App 20150094311 - GIJSEN; HENRICUS JACOBUS MARIA ;   et al. | 2015-04-02 |
Substituted Imidazoles As N-type Calcium Channel Blockers App 20150051225 - Ahmad; Ishtiyaque ;   et al. | 2015-02-19 |
Substituted bicyclic heterocyclic compounds as gamma secretase modulators Grant 8,946,426 - Gijsen , et al. February 3, 2 | 2015-02-03 |
Substituted triazole and imidazole derivatives as gamma secretase modulators Grant 8,946,266 - Wu , et al. February 3, 2 | 2015-02-03 |
5-(3-aminophenyl)-5-alkyl-5,6-dihydro-2h-[1,4]oxazin-3-amine Derivatives App 20140364428 - Gijsen; Henricus Jacobus Maria ;   et al. | 2014-12-11 |
6-difluoromethyl-5,6-dihydro-2h-[1,4]oxazin-3-amine Derivatives App 20140343048 - Trabanco-Suarez; Andres Avelino ;   et al. | 2014-11-20 |
Substituted indazole and aza-indazole derivatives as gamma secretase modulators Grant 8,835,482 - Bischoff , et al. September 16, 2 | 2014-09-16 |
Substituted benzoxazole, benzimidazole, oxazolopyridine and imidazopyridine derivatives as gamma secretase modulators Grant 8,772,504 - Gijsen , et al. July 8, 2 | 2014-07-08 |
Novel Substituted Indole Derivatives As Gamma Secretase Modulators App 20140148450 - Minne; Garrett Berlond ;   et al. | 2014-05-29 |
6,7-DIHYDRO-PYRAZOLO[1,5-a]PYRAZIN-4-YLAMINE DERIVATIVES USEFUL AS INHIBITORS OF BETA-SECRETASE (BACE) App 20140005200 - Trabanco-Suarez; Andres Avelino ;   et al. | 2014-01-02 |
Heterocyclic amides as modulators of TRPA1 Grant 8,614,201 - Berthelot , et al. December 24, 2 | 2013-12-24 |
Benzimidazole Cannabinoid Agonists Bearing A Substituted Heterocyclic Group App 20130324529 - Gijsen; Henricus Jacobus Maria ;   et al. | 2013-12-05 |
5,6-DIHYDRO-IMIDAZO[1,2-a]PYRAZIN-8-YLAMINE DERIVATIVES USEFUL AS INHIBITORS OF BETA-SECRETASE (BACE) App 20130274266 - Trabanco-Suarez; Andres Avelino ;   et al. | 2013-10-17 |
Substituted bicyclic imidazole derivatives as gamma secretase modulators Grant 8,546,440 - Gijsen , et al. October 1, 2 | 2013-10-01 |
Benzimidazole cannabinoid agonists bearing a substituted heterocyclic group Grant 8,524,757 - Gijsen , et al. September 3, 2 | 2013-09-03 |
Dibenzoazepine and dibenzooxazepine TRPA1 agonists Grant 8,461,145 - Gijsen , et al. June 11, 2 | 2013-06-11 |
5,6-dihydro-2h-[1,4]oxazin-3-yl-amine Derivatives Useful As Inhibitors Of Beta-secretase (bace) App 20130109683 - Trabanco-Suarez; Andres Avelino ;   et al. | 2013-05-02 |
Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT.sub.4-antagonists Grant 8,334,304 - Bosmans , et al. December 18, 2 | 2012-12-18 |
Novel Substituted Bicyclic Triazole Derivatives As Gamma Secretase Modulators App 20120295901 - De Cleyn; Michel Anna Jozef ;   et al. | 2012-11-22 |
Novel Substituted Triazole Derivatives As Gamma Secretase Modulators App 20120295891 - Van Brandt; Sven Franciscus Anna ;   et al. | 2012-11-22 |
Benzimidazole cannabinoid agonists Grant 8,193,369 - Gijsen , et al. June 5, 2 | 2012-06-05 |
Novel Substituted Triazole And Imidazole Derivatives As Gamma Secretase Modulators App 20120135981 - Wu; Tongfei ;   et al. | 2012-05-31 |
Novel Substituted Indazole And Aza-indazole Derivatives As Gamma Secretase Modulators App 20120095036 - Bischoff; Francois Paul ;   et al. | 2012-04-19 |
Heterocyclic Amides As Modulators Of Trpa1 App 20120083474 - Berthelot; Didier Jean-Claude ;   et al. | 2012-04-05 |
Novel Substituted Bicyclic Heterocyclic Compounds As Gamma Secretase Modulators App 20110281881 - Gijsen; Henricus, Jacobus, Maria ;   et al. | 2011-11-17 |
Substituted Bicyclic Imidazole Derivatives As Gamma Secretase Modulators App 20110237580 - Gijsen; Henricus Jacobus Maria ;   et al. | 2011-09-29 |
3,4-dihydropyrimidine Trpa1 Antagonists App 20110124666 - Gijsen; Henricus Jacobus Maria ;   et al. | 2011-05-26 |
Dibenzoazepine And Dibenzooxazepine Trpa1 Agonists App 20100273773 - Gijsen; Henricus Jacobus Maria ;   et al. | 2010-10-28 |
Fluoro Alkyl Substituted Benzimidazole Cannabinoid Agonists App 20100273831 - Gijsen; Henricus Jacobus Maria ;   et al. | 2010-10-28 |
Heterocyclic substituted 4-(aminomethyl)-piperidine benzamides as 5HT.sub.4-antagonists Grant 7,732,464 - Bosmans , et al. June 8, 2 | 2010-06-08 |
Aminosulfonyl Substituted 4-(Aminomethyl)-Piperidine Benzamides As 5HT 4-Antagonists App 20100087483 - BOSMANS; Jean-Paul Rene Marie Andre ;   et al. | 2010-04-08 |
Benzimidazole Cannabinoid Agonists App 20100041702 - Gijsen; Henricus Jacobus Maria ;   et al. | 2010-02-18 |
Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT.sub.4-antagonists Grant 7,652,040 - Bosmans , et al. January 26, 2 | 2010-01-26 |
4-(aminomethyl)-piperidine benzamides as 5HT.sub.4-antagonists Grant 7,638,535 - Bosmans , et al. December 29, 2 | 2009-12-29 |
5HT.sub.4-antagonistic 4-(aminomethyl)-piperidine benzamides Grant 7,635,706 - Bosmans , et al. December 22, 2 | 2009-12-22 |
Benzimidazole Cannabinoid Agonists Bearing A Substituted Heterocyclic Group App 20090312339 - Gijsen; Henricus Jacobus Maria ;   et al. | 2009-12-17 |
Hydroxycarbonylphenyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT.sub.4 antagonists Grant 7,498,347 - Bosmans , et al. March 3, 2 | 2009-03-03 |
Heterocyclic substituted 4-(aminomethyl)-piperidine benzamides as 5ht4-antagonists App 20070197600 - Bosmans; Jean-Paul Rene Marie Andre ;   et al. | 2007-08-23 |
4-(aminomethyl)-piperidine benzamides for treating gastrointestinal disorders Grant 7,205,410 - Bosmans , et al. April 17, 2 | 2007-04-17 |
5Ht4-antagonistic 4-(aminomethyl)-piperidine benzamides App 20070032486 - Bosmans; Jean-Paul Rene Marie Andre ;   et al. | 2007-02-08 |
4-(Aminomethyl)-piperidine benzamides as 5ht4 - antagonists App 20060281753 - Bosmans; Jean-Paul Rene Marie Andre ;   et al. | 2006-12-14 |
Chimeric gaba receptor App 20060216749 - Smans; Karine Alfonsine Astrid ;   et al. | 2006-09-28 |
Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5ht 4-antagonists App 20060142339 - Bosmans; Jean-Paul Rene Marie Andre ;   et al. | 2006-06-29 |
Hydroxycarbonylphenyl substituted 4-(aminomethyl)-piperidine benzamides as 5ht4 antagonists App 20060142340 - Bosmans; Jean-Paul Rene Marie Andre ;   et al. | 2006-06-29 |
4-(aminomethyl)-piperidine benzamides for treating gastrointestinal disorders App 20030181456 - Bosmans, Jean-Paul Rene Marie Andre ;   et al. | 2003-09-25 |
4-(aminomethyl)-piperidine benzamides for treating gastrointestinal disorders Grant 6,544,997 - Bosmans , et al. April 8, 2 | 2003-04-08 |