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Spirocyclic Lactams As Jak2 V617f Inhibitors App 20220281887 - Shepard; Stacey ;   et al. | 2022-09-08 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20220251087 - Buesking; Andrew W. ;   et al. | 2022-08-11 |
Pyridine And Pyridimine Compounds As Pi3k-gamma Inhibitors App 20220227736 - Sparks; Richard B. ;   et al. | 2022-07-21 |
AMINOPYRAZINE DIOL COMPOUNDS AS PI3K-y INHIBITORS App 20220213065 - Shepard; Stacey ;   et al. | 2022-07-07 |
TERTIARY ALCOHOLS AS PI3K-y INHIBITORS App 20220213107 - Douty; Brent ;   et al. | 2022-07-07 |
Pyridine and pyridimine compounds as PI3K-gamma inhibitors Grant 11,352,340 - Sparks , et al. June 7, 2 | 2022-06-07 |
3-(5-amino-pyrazin-2-yl)-benzenesulfonamide derivatives and related compounds as PI3K-gamma kinase inhibitors Grant 11,306,079 - Shvartsbart , et al. April 19, 2 | 2022-04-19 |
Tertiary alcohols as PI3K-.gamma. inhibitors Grant 11,225,486 - Douty , et al. January 18, 2 | 2022-01-18 |
Heterocyclic Derivatives As Pi3k Inhibitors App 20210395258 - Shepard; Stacey ;   et al. | 2021-12-23 |
1H-PYRROLO[2,3-c]PYRIDIN-7(6H)-ONES AND PYRAZOLO[3,4-c]PYRIDIN-7(6H)-ONES AS INHIBITORS OF BET PROTEINS App 20210300925 - Combs; Andrew P. ;   et al. | 2021-09-30 |
Heterocyclic compounds as PI3K-y inhibitors Grant 11,091,491 - Shvartsbart , et al. August 17, 2 | 2021-08-17 |
Heterocyclic derivatives as PI3K inhibitors Grant 11,078,204 - Shepard , et al. August 3, 2 | 2021-08-03 |
1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins Grant 11,059,821 - Combs , et al. July 13, 2 | 2021-07-13 |
Aminopyrazine derivatives as PI3K-.gamma. inhibitors Grant 11,046,658 - Douty , et al. June 29, 2 | 2021-06-29 |
Imidazo[2,1-f][1,2,4]triazine compounds as pi3k-y inhibitors Grant 10,975,088 - Buesking , et al. April 13, 2 | 2021-04-13 |
TERTIARY ALCOHOLS AS PI3K-y INHIBITORS App 20200385392 - Douty; Brent ;   et al. | 2020-12-10 |
1H-PYRROLO[2,3-c]PYRIDIN-7(6H)-ONES AND PYRAZOLO[3,4-c]PYRIDIN-7(6H)-ONES AS INHIBITORS OF BET PROTEINS App 20200377502 - Combs; Andrew P. ;   et al. | 2020-12-03 |
AMINOPYRAZINE DIOL COMPOUNDS AS PI3K-y INHIBITORS App 20200339542 - Shepard; Stacey ;   et al. | 2020-10-29 |
3-(5-amino-pyrazin-2-yl)-benzenesulfonamide Derivatives And Related Compounds As Pi3k-gamma Kinase Inhibitors For Treating E.g. Cancer App 20200331903 - SHVARTSBART; Artem ;   et al. | 2020-10-22 |
1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins Grant 10,781,209 - Combs , et al. Sept | 2020-09-22 |
Tertiary alcohols as PI3K-.gamma. inhibitors Grant 10,738,057 - Douty , et al. A | 2020-08-11 |
Aminopyrazine diol compounds as PI3K-.gamma. inhibitors Grant 10,669,262 - Shepard , et al. | 2020-06-02 |
Heterocyclic Derivatives As Pi3k Inhibitors App 20200148689 - Shepard; Stacey ;   et al. | 2020-05-14 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20200102315 - Buesking; Andrew W. ;   et al. | 2020-04-02 |
1H-PYRROLO[2,3-c]PYRIDIN-7(6H)-ONES AND PYRAZOLO[3,4-c]PYRIDIN-7(6H)-ONES AS INHIBITORS OF BET PROTEINS App 20200048251 - Combs; Andrew P. ;   et al. | 2020-02-13 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20200031837 - Shvartsbart; Artem ;   et al. | 2020-01-30 |
AMINOPYRAZINE DERIVATIVES AS PI3K-y INHIBITORS App 20200002295 - Douty; Brent ;   et al. | 2020-01-02 |
Pyridine And Pyridimine Compounds As Pi3k-gamma Inhibitors App 20190359592 - Sparks; Richard B. ;   et al. | 2019-11-28 |
Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines and substituted imidazo[1,2-b]pyridazines as PI3K-gamma inhibitors Grant 10,479,795 - Buesking , et al. Nov | 2019-11-19 |
Heterocyclic compounds as PI3K-.gamma. inhibitors Grant 10,472,368 - Shvartsbart , et al. Nov | 2019-11-12 |
1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins Grant 10,472,358 - Combs , et al. Nov | 2019-11-12 |
AMINOPYRAZINE DIOL COMPOUNDS AS PI3K-y INHIBITORS App 20190276435 - Shepard; Stacey ;   et al. | 2019-09-12 |
TERTIARY ALCOHOLS AS PI3K-y INHIBITORS App 20190152975 - Douty; Brent ;   et al. | 2019-05-23 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20190119287 - Buesking; Andrew W. ;   et al. | 2019-04-25 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20190062336 - Shvartsbart; Artem ;   et al. | 2019-02-28 |
Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines, substituted imidazo[1,2-b]pyridazines and substituted imidazo[1,2-a]pyrazines as PI3K-.gamma. inhibitors Grant 10,138,248 - Buesking , et al. Nov | 2018-11-27 |
1H-PYRROLO[2,3-c]PYRIDIN-7(6H)-ONES AND PYRAZOLO[3,4-c]PYRIDIN-7(6H)-ONES AS INHIBITORS OF BET PROTEINS App 20180312506 - Combs; Andrew P. ;   et al. | 2018-11-01 |
Heterocyclic compounds as PI3K-.gamma. inhibitors Grant 10,065,963 - Shvartsbart , et al. September 4, 2 | 2018-09-04 |
1H-pyrrolo[2,3,c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins Grant 9,957,268 - Combs , et al. May 1, 2 | 2018-05-01 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20180009816 - Buesking; Andrew W. ;   et al. | 2018-01-11 |
Pyridine And Pyridimine Compounds As Pi3k-gamma Inhibitors App 20170190689 - Sparks; Richard B. ;   et al. | 2017-07-06 |
1H-PYRROLO[2,3-c]PYRIDIN-7(6H)-ONES AND PYRAZOLO[3,4-c]PYRIDIN-7(6H)-ONES AS INHIBITORS OF BET PROTEINS App 20170158689 - Combs; Andrew P. ;   et al. | 2017-06-08 |
HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS App 20170129899 - Shvartsbart; Artem ;   et al. | 2017-05-11 |
1H-PYRROLO[2,3-c]PYRIDIN-7(6H)-ONES AND PYRAZOLO[3,4-c]PYRIDIN-7(6H)-ONES AS INHIBITORS OF BET PROTEINS App 20150307493 - Combs; Andrew P. ;   et al. | 2015-10-29 |
Heteroaryl Substituted Pyrrolo[2,3-B] Pyridines And Pyrrolo[2,3-B] Pyrimidines As Janus Kinase Inhibitors App 20140005210 - Rodgers; James D. ;   et al. | 2014-01-02 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20130137681 - Rodgers; James D. ;   et al. | 2013-05-30 |
Pyrazolyl substituted pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors Grant 8,415,362 - Rodgers , et al. April 9, 2 | 2013-04-09 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20110223210 - Rodgers; James D. ;   et al. | 2011-09-15 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20110224157 - Rodgers; James D. ;   et al. | 2011-09-15 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20100022522 - Rodgers; James D. ;   et al. | 2010-01-28 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20090181959 - Rodgers; James D. ;   et al. | 2009-07-16 |
Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as janus kinase inhibitors App 20070135461 - Rodgers; James D. ;   et al. | 2007-06-14 |