Patent | Date |
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Crystal Forms of (S)-4-(8-amino-3-(1-(but-2-ynoyl)-pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1- -yl)-n-(pyridin-2-yl)benzamide App 20220177476 - Blatter; Frtiz ;   et al. | 2022-06-09 |
PROCESSES FOR THE PREPARATION OF 4-{8-AMINO-3-[(2S)-1-(BUT-2-YNOYL)-PYRROLIDIN-2-YL]IMIDAZO[1,5-a]-PYRAZIN- -1-YL}N-(PYRIDIN-2-YL)-BENZAMIDE App 20220127270 - BETHEL; Paul Allen ;   et al. | 2022-04-28 |
Crystal forms of (S)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-- yl)-N-(pyridin-2-yl)benzamide maleate Grant 11,059,829 - Blatter , et al. July 13, 2 | 2021-07-13 |
Process methods for phosphatidylinositol 3-kinase inhibitors Grant 10,954,199 - Bremner , et al. March 23, 2 | 2021-03-23 |
Imidazopyrazine inhibitors of Bruton's tyrosine kinase Grant 10,858,364 - Podoll , et al. December 8, 2 | 2020-12-08 |
Crystal Forms of (S)-4-(8-amino-3-(1-(but-2-ynoyl)-pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1- -yl)-N-(pyridin-2-yl)benzamide malea App 20200255437 - Kind Code | 2020-08-13 |
Pharmaceutical composition comprising a crystal form of (S)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-- yl)-N-(pyridin-2-yl)benzamide for treating diffuse large B-cell lymphoma Grant 10,640,509 - Blatter , et al. | 2020-05-05 |
Process Methods For Phosphatidylinositol 3-kinase Inhibitors App 20200102277 - BREMNER; Stacy ;   et al. | 2020-04-02 |
Imidazopyrazine Inhibitors of Bruton's Tyrosine Kinase App 20190345164 - Podoll; Terry ;   et al. | 2019-11-14 |
Solid Forms and Formulations of Imidazopyrazine Compound App 20190337949 - Blatter; Fritz ;   et al. | 2019-11-07 |
Polymorphic forms of a hydrochloride salt of (S)-2-(1-(9H-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3H)-on- e Grant 10,442,805 - Buttar , et al. Oc | 2019-10-15 |
Phosphatidylinositol 3-kinase inhibitors Grant 10,308,639 - Evarts , et al. | 2019-06-04 |
Phosphatidylinositol 3-kinase inhibitors Grant 10,221,197 - Du , et al. | 2019-03-05 |
Pharmaceutical composition comprising a crystal form of (S)-4-(8-amino-3-(1-(but-2-ynoyl) pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide Grant 10,167,291 - Blatter , et al. J | 2019-01-01 |
Process for preparing phosphatidylinositol 3-kinase inhibitors and intermediates thereof Grant 10,059,677 - Bremner , et al. August 28, 2 | 2018-08-28 |
Process methods for phosphatidylinositol 3-kinase inhibitors Grant 10,047,060 - Bremner , et al. August 14, 2 | 2018-08-14 |
Solid Forms and Formulations of Imidazopyrazine Compound App 20180208596 - Blatter; Fritz ;   et al. | 2018-07-26 |
Process Methods For Phosphatidylinositol 3-kinase Inhibitors App 20180162826 - BREMNER; Stacy ;   et al. | 2018-06-14 |
Phosphatidylinositol 3-kinase Inhibitors App 20180065953 - Evarts; Jerry ;   et al. | 2018-03-08 |
Polymorphic Forms Of A Hydrochloride Salt Of (s)-2-(1-(9h-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3h)-on- E App 20180009811 - BUTTAR; Suzanne ;   et al. | 2018-01-11 |
Crystal forms of (S)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-- yl)-N-(pyridin-2-yl)benzamide Grant 9,796,721 - Blatter , et al. October 24, 2 | 2017-10-24 |
Phosphatidylinositol 3-kinase inhibitors Grant 9,765,060 - Evarts , et al. September 19, 2 | 2017-09-19 |
Polymorphic forms of a hydrochloride salt of (S)-2-(1-(9H-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3H)-on- e Grant 9,708,327 - Buttar , et al. July 18, 2 | 2017-07-18 |
Process Methods For Phosphatidylinositol 3-kinase Inhibitors App 20170107187 - BREMNER; Stacy ;   et al. | 2017-04-20 |
Process methods for phosphatidylinositol 3-kinase inhibitors Grant 9,567,337 - Bremner , et al. February 14, 2 | 2017-02-14 |
Solid Forms and Formulations of Imidazopyrazine Compound App 20170029428 - Blatter; Fritz ;   et al. | 2017-02-02 |
Polymorphic Forms Of (s)-2-(1-(9h-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3h)-on- E App 20160376274 - Carra; Ernest ;   et al. | 2016-12-29 |
Phosphatidylinositol 3-kinase inhibitors Grant 9,266,878 - Evarts , et al. February 23, 2 | 2016-02-23 |
Phosphatidylinositol 3-kinase Inhibitors App 20160039793 - Evarts; Jerry ;   et al. | 2016-02-11 |
Phosphatidylinositol 3-kinase Inhibitors App 20160024054 - Evarts; Jerry ;   et al. | 2016-01-28 |
Phosphatidylinositol 3-kinase Inhibitors App 20160016915 - Evarts; Jerry ;   et al. | 2016-01-21 |
Phosphatidylinositol 3-kinase inhibitors Grant 9,221,795 - Evarts , et al. December 29, 2 | 2015-12-29 |
Phosphatidylinositol 3-kinase Inhibitors App 20150361095 - Du; Zhimin ;   et al. | 2015-12-17 |
Phosphatidylinositol 3-kinase Inhibitors App 20150361070 - Evarts; Jerry ;   et al. | 2015-12-17 |
Phosphatidylinositol 3-kinase Inhibitors App 20150218154 - Evarts; Jerry ;   et al. | 2015-08-06 |
Process Methods For Phosphatidylinositol 3-kindase Inhibitors App 20150175605 - Bremner; Stacy ;   et al. | 2015-06-25 |
Phosphatidylinositol 3-kinase inhibitors Grant 9,029,384 - Evarts , et al. May 12, 2 | 2015-05-12 |
Phosphatidylinositol 3-kinase inhibitors Grant 9,018,221 - Evarts , et al. April 28, 2 | 2015-04-28 |
Phosphatidylinositol 3-kinase Inhibitors App 20140371246 - Evarts; Jerry ;   et al. | 2014-12-18 |
Phosphatidylinositol 3-kinase Inhibitors App 20140179718 - EVARTS; Jerry ;   et al. | 2014-06-26 |
Phosphatidylinositol 3-kinase Inhibitors App 20140179673 - EVARTS; Jerry ;   et al. | 2014-06-26 |
Atropisomers Of P13k-inhibiting Compounds App 20130324561 - Evarts; Jerry ;   et al. | 2013-12-05 |