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2,3-dihydrobenzohurans as bromodomain inhibitors Grant 11,319,307 - Atkinson , et al. May 3, 2 | 2022-05-03 |
Benzofuran derivatives and their use as bromodomain inhibitors Grant 11,273,146 - Atkinson , et al. March 15, 2 | 2022-03-15 |
Furan Derivatives As Bromodomain Inhibitors App 20210346336 - DEMONT; Emmanuel Hubert ;   et al. | 2021-11-11 |
Pyrazole derivatives as bromodomain inhibitors Grant 10,966,961 - Atkinson , et al. April 6, 2 | 2021-04-06 |
Pyridyl derivatives as bromodomain inhibitors Grant 10,934,272 - Atkinson , et al. March 2, 2 | 2021-03-02 |
Pyridinone dicarboxamide for use as bromodomain inhibitors Grant 10,927,080 - Atkinson , et al. February 23, 2 | 2021-02-23 |
Pyridyl derivatives as bromodomain inhibitors Grant 10,849,897 - Atkinson , et al. December 1, 2 | 2020-12-01 |
Pyridine dicarboxamide derivatives as bromodomain inhibitors Grant 10,844,015 - Atkinson , et al. November 24, 2 | 2020-11-24 |
2,3-dihydrobenzofurans As Bromodomain Inhibitors App 20200291009 - ATKINSON; Stephen John ;   et al. | 2020-09-17 |
Benzofuran Derivatives And Their Use As Bromodomain Inhibitors App 20200289464 - ATKINSON; Stephen John ;   et al. | 2020-09-17 |
Benzo[b]furans as bromodomain inhibitors Grant 10,583,112 - Atkinson , et al. | 2020-03-10 |
Pyridyl Derivatives As Bromodomain Inhibitors App 20200009140 - ATKINSON; Stephen John ;   et al. | 2020-01-09 |
Pyrazole Derivatives As Bromodomain Inhibitors App 20190381010 - ATKINSON; Stephen John ;   et al. | 2019-12-19 |
Pyridinone Dicarboxamide For Use As Bromodomain Inhibitors App 20190359572 - ATKINSON; Stephen John ;   et al. | 2019-11-28 |
2-OXO-1,2-dihydropyridine-3,5-dicarboxamide compounds as bromodomain inhibitors Grant 10,471,050 - Atkinson , et al. Nov | 2019-11-12 |
Pyridinone dicarboxamide for use as bromodomain inhibitors Grant 10,428,026 - Atkinson , et al. October 1, 2 | 2019-10-01 |
Pyridinone dicarboxamide for use as bromodomain inhibitors Grant 10,370,356 - Atkinson , et al. | 2019-08-06 |
Pyridine Dicarboxamide Derivatives As Bromodomain Inhibitors App 20190202786 - ATKINSON; Stephen John ;   et al. | 2019-07-04 |
Benzo[b]furans As Bromodomain Inhibitors App 20190151279 - ATKINSON; Stephen John ;   et al. | 2019-05-23 |
Pyridyl Derivatives As Bromodomain Inhibitors App 20190119248 - ATKINSON; Stephen John ;   et al. | 2019-04-25 |
2-oxo-1,2-dihydropyridine-3,5-dicarboxamide Compounds As Bromodomain Inhibitors App 20180280368 - ATKINSON; Stephen John ;   et al. | 2018-10-04 |
Pyridinone Dicarboxamide For Use As Bromodomain Inhibitors App 20180258044 - ATKINSON; Stephen John ;   et al. | 2018-09-13 |
4-(8-methoxy-1-((1-methoxypropan-2-yl)-2-(tetrahydro-2H-pyran-4-yl)-1 H-imidazo[4,5-C]quinolin-7-yl)-3,5-dimethylisoxazole and its use as bromodomain inhibitor Grant 9,861,627 - Demont , et al. January 9, 2 | 2018-01-09 |
4-(8-methoxy-1-((1-methoxypropan-2-yl)-2-(tetrahydro-2h-pyran-4-yl)-1 H-imidazo[4,5-c]quinolin-7-yl)-3,5-dimethylisoxazole And Its Use As Bromodomain Inhibitor App 20170157113 - Demont; Emmanuel Hubert ;   et al. | 2017-06-08 |
4-(8-methoxy-1-((1-methoxypropan-2-yl)-2-(tetrahydro-2H-pyran-4-yl)-1H-imi- dazo[4,5-c]quinolin-7-yl)-3,5-dimethylisoxazole and its use as bromodomain inhibitor Grant 9,610,284 - Demont , et al. April 4, 2 | 2017-04-04 |
4-(8-methoxy-1-((1-methoxypropan-2-yl)-2-(tetrahydro-2h-pyran-4-yl)-1 H-imidazo[4,5-c]quinolin-7-yl)-3,5-dimethylisoxazole And Its Use As Bromodomain Inhibitor App 20160317529 - Demont; Emmanuel Hubert ;   et al. | 2016-11-03 |
4-(8-methoxy-1-((1-methoxypropan-2-yl)-2-(tetrahydro-2H-pyran-4-yl)-1 H-imidazo[4,5-C]quinolin-7-yl)-3,5-dimethylisoxazole and its use as bromodomain inhibitor Grant 9,416,130 - Demont , et al. August 16, 2 | 2016-08-16 |
Tetrahydroquinoline derivatives useful as bromodomain inhibitors Grant 9,315,487 - Amans , et al. April 19, 2 | 2016-04-19 |
4-(8-methoxy-1-((1-methoxypropan-2-yl)-2-(tetrahydro-2h-pyran-4-yl)-1 H-imidazo[4,5-c]quinolin-7-yl)-3,5-dimethylisoxazole And Its Use As Bromodomain Inhibitor App 20150315184 - Demont; Emmanuel Hubert ;   et al. | 2015-11-05 |
4-(8-methoxy-1-((1-methoxypropan-2-yl)-2-(tetrahydro-2H-pyran-4-yl)-1 H-imidazo[4,5-C]quinolin-7-yl)-3,5-dimethylisoxazole and its use as bromodomain inhibitor Grant 9,067,936 - Demont , et al. June 30, 2 | 2015-06-30 |
Tetrahydroquinoline derivatives useful as bromodomain inhibitors Grant 9,029,395 - Amans , et al. May 12, 2 | 2015-05-12 |
Tetrahydroquinoline derivatives useful as bromodomain inhibitors Grant 8,993,554 - Amans , et al. March 31, 2 | 2015-03-31 |
7-(3,5-dimethyl-4-isoxazolyl)-8-(methyloxy)-1H-imidazo[4,5-C]quinoline derivatives Grant 8,846,709 - Demont , et al. September 30, 2 | 2014-09-30 |
4-(8-methoxy-1-((1-methoxypropan-2-yl)-2-(tetrahydro-2h-pyran-4-yl)-1 H-imidazo[4,5-c]quinolin-7-yl)-3,5-dimethylisoxazole And Its Use As Bromodomain Inhibitor App 20140171462 - Demont; Emmanuel Hubert ;   et al. | 2014-06-19 |
Tetrahydroquinoline derivatives and their pharmaceutical use Grant 8,697,725 - Demont , et al. April 15, 2 | 2014-04-15 |
Tetrahydroquinoline Derivatives Useful As Bromodomain Inhibitors App 20140066459 - Amans; Dominique ;   et al. | 2014-03-06 |
7-(3,5-Dimethyl-4-Isoxazolyl)-8-(Methyloxy)-1H-Imidazo[4,5-C]Quinoline Derivatives App 20140045834 - Demont; Emmanuel Hubert ;   et al. | 2014-02-13 |
Tetrahydroquinoline Derivatives Useful As Bromodomain Inhibitors App 20140039006 - Amans; Dominique ;   et al. | 2014-02-06 |
Tetrahydroquinoline Derivatives Useful As Bromodomain Inhibitors App 20140031336 - Amans; Dominique ;   et al. | 2014-01-30 |
Thetrahydroquinolines derivatives as bromodomain inhibitors Grant 8,580,957 - Demont , et al. November 12, 2 | 2013-11-12 |
Thetrahydroquinolines Derivatives As Bromodomain Inhibitors App 20120208814 - Demont; Emmanuel Hubert ;   et al. | 2012-08-16 |
Tetrahydroquinoline Derivatives And Their Pharmaceutical Use App 20120208798 - Demont; Emmanuel Hubert ;   et al. | 2012-08-16 |
Oxadiazole derivatives active on sphingosine-1-phosphate (S1P) Grant 8,222,245 - Demont , et al. July 17, 2 | 2012-07-17 |
S1p1 Agonists Comprising A Bicyclic N-containing Ring App 20120101083 - Bailey; James Matthew ;   et al. | 2012-04-26 |
Thiadiazole Derivatives And Their Use For The Treatment Of Disorders Mediated By S1p1 Receptors App 20120101086 - Bailey; James Matthew ;   et al. | 2012-04-26 |
Thiazole Or Thiadizaloe Derivatives For Use As Sphingosine 1-phosphate 1 (s1p1) Receptor Agonists App 20120094979 - Bailey; James Matthew ;   et al. | 2012-04-19 |
Pyrazole Derivatives as P2X7 Modulators App 20110046137 - Beswick; Paul John ;   et al. | 2011-02-24 |
Oxadiazole Derivatives Active On Sphingosine-1-phosphate (sip) App 20100273771 - Demont; Emmanuel Hubert ;   et al. | 2010-10-28 |
N-(Phenylmethyl)-2-(1H-Pyrazol-4-yl) Acetamide Derivatives as P2X7 Antagonists for the Treatment of Pain, Inflammation and Neurodegeneration App 20090149524 - Beswick; Paul John ;   et al. | 2009-06-11 |
Derivatives of Imidazo [1,2-A] Pyridine Useful as Medicaments For Treating Gastrointestinal Diseases App 20080255358 - Bamford; Mark James ;   et al. | 2008-10-16 |
Tricycle indole hydroxyethlamine derivatives and their use in the treatment of alzheimer's disease App 20070073060 - Demont; Emmanuel Hubert ;   et al. | 2007-03-29 |
Tricyclic indole derivatives and their use in the treatment of alzheimer's disease App 20060229302 - Demont; Emmanuel Hubert ;   et al. | 2006-10-12 |
Novel compounds App 20060211740 - Demont; Emmanuel Hubert ;   et al. | 2006-09-21 |