Patent | Date |
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Carbamoyloxymethyl Triazole Cyclohexyl Acids As Lpa Antagonists App 20220249443 - Cheng; Peter Tai Wah ;   et al. | 2022-08-11 |
Cyclohexyl acid pyrazole azoles as LPA antagonists Grant 11,352,345 - Shi , et al. June 7, 2 | 2022-06-07 |
Cyclohexyl acid triazole azoles as LPA antagonists Grant 11,319,315 - Shi , et al. May 3, 2 | 2022-05-03 |
Cyclohexyl acid triazole azines as LPA antagonists Grant 11,267,800 - Shi , et al. March 8, 2 | 2022-03-08 |
Pyrimidinones As Factor Xia Inhibitors App 20220041601 - Dilger; Andrew K. ;   et al. | 2022-02-10 |
Radioligands For Imaging The Lpa1 Receptor App 20210379210 - Cheng; Peter Tai Wah ;   et al. | 2021-12-09 |
Macrocycles as factor XIA inhibitors Grant 11,136,327 - Corte , et al. October 5, 2 | 2021-10-05 |
Carbamoyloxymethyl Triazole Cyclohexyl Acids As Lpa Antagonists App 20210244711 - CHENG; PETER TAI WAH ;   et al. | 2021-08-12 |
Cyclohexyl Acid Triazole Azines As Lpa Antagonists App 20210230143 - Shi; Yan ;   et al. | 2021-07-29 |
Pyrimidinones as factor XIA inhibitors Grant 11,053,247 - Dilger , et al. July 6, 2 | 2021-07-06 |
Cyclohexyl Acid Triazole Azoles As Lpa Antagonists App 20210163470 - Shi; Yan ;   et al. | 2021-06-03 |
Triazole n-linked carbamoyl cyclohexyl acids as LPA antagonists Grant 11,008,300 - Shi , et al. May 18, 2 | 2021-05-18 |
Carbamoyloxymethyl triazole cyclohexyl acids as LPA antagonists Grant 11,007,180 - Cheng , et al. May 18, 2 | 2021-05-18 |
Cyclohexyl Acid Pyrazole Azoles As Lpa Antagonists App 20210078982 - Shi; Yan ;   et al. | 2021-03-18 |
Triazole N-linked carbamoyl cyclohexyl acids as LPA antagonists Grant 10,662,172 - Shi , et al. | 2020-05-26 |
Triazole N-linked Carbamoyl Cyclohexyl Acids As Lpa Antagonists App 20200148665 - Shi; Yan ;   et al. | 2020-05-14 |
Carbamoyloxymethyl Triazole Cyclohexyl Acids As Lpa Antagonists App 20200138789 - Cheng; Peter Tai Wah ;   et al. | 2020-05-07 |
Macrocycles As Factor Xia Inhibitors App 20200087312 - Corte; James R. ;   et al. | 2020-03-19 |
Carbamoyloxymethyl triazole cyclohexyl acids as LPA antagonists Grant 10,576,062 - Cheng , et al. | 2020-03-03 |
Pyrimidinones As Factor Xia Inhibitors App 20200055854 - Dilger; Andrew K. ;   et al. | 2020-02-20 |
Novel Substituted Glycine Derived Fxia Inhibitors App 20190382378 - Corte; James R. ;   et al. | 2019-12-19 |
Macrocycles as factor XIa inhibitors Grant 10,487,086 - Corte , et al. Nov | 2019-11-26 |
Pyrimidinones as factor XIa inhibitors Grant 10,336,754 - Dilger , et al. | 2019-07-02 |
Substituted glycine derived FXIA inhibitors Grant 10,336,730 - Corte , et al. | 2019-07-02 |
Triazole N-linked Carbamoyl Cyclohexyl Acids As Lpa Antagonists App 20190185446 - SHI; YAN ;   et al. | 2019-06-20 |
Factor Xia Macrocycles With Novel P1 Groups App 20190144393 - Corte; James R. ;   et al. | 2019-05-16 |
Factor XIa macrocyclic inhibitors bearing alkyl or cycloalkyl P2' moieties Grant 10,287,288 - Pabbisetty , et al. | 2019-05-14 |
Macrocyclic factor XIa inhibitors bearing heterocyclic groups Grant 10,273,236 - Dilger , et al. | 2019-04-30 |
Macrocycles as factor XIa inhibitors Grant 10,208,068 - Pinto , et al. Feb | 2019-02-19 |
Diamide macrocycles as factor XIa inhibitors Grant 10,160,750 - Smith, II , et al. Dec | 2018-12-25 |
Carbamoyloxymethyl Triazole Cyclohexyl Acids As Lpa Antagonists App 20180333395 - Cheng; Peter Tai Wah ;   et al. | 2018-11-22 |
Five-membered heterocycles useful as serine protease inhibitors Grant 10,112,936 - Hangeland , et al. October 30, 2 | 2018-10-30 |
Substituted Tetrahydroisoquinoline Compounds As Factor Xia Inhibitors App 20180265494 - Orwat; Michael J. ;   et al. | 2018-09-20 |
Carbamoyloxymethyl triazole cyclohexyl acids as LPA antagonists Grant 10,071,078 - Cheng , et al. September 11, 2 | 2018-09-11 |
Novel Substituted Glycine Derived Fxia Inhibitors App 20180222889 - Corte; James R. ;   et al. | 2018-08-09 |
Macrocyclic Factor Xia Inhibitors Bearing Heterocyclic Groups App 20180222907 - Dilger; Andrew K. ;   et al. | 2018-08-09 |
Factor Xia Macrocyclic Inhibitors Bearing Alkyl Or Cycloalkyl P2' Moieties App 20180215755 - Pabbisetty; Kumar Balashanmuga ;   et al. | 2018-08-02 |
Pyrimidinones As Factor Xia Inhibitors App 20180186795 - Dilger; Andrew K. ;   et al. | 2018-07-05 |
Substituted 4,5,6,7-tetrahydropyrazolo[3,4-c]pyridines as factor XIa inhibitors Grant 10,000,466 - Orwat , et al. June 19, 2 | 2018-06-19 |
Factor Xia Macrocycles With Novel P1 Groups App 20180162821 - Corte; James R. ;   et al. | 2018-06-14 |
Novel Macrocycles As Factor Xia Inhibitors App 20180148461 - Pinto; Donald J.P. ;   et al. | 2018-05-31 |
Diamide Macrocycles As Factor Xia Inhibitors App 20180141932 - Smith II; Leon ;   et al. | 2018-05-24 |
Dihydropyridone P1 as factor XIa inhibitors Grant 9,951,071 - Yang , et al. April 24, 2 | 2018-04-24 |
Macrocycles as factor XIa inhibitors Grant 9,902,742 - Pinto , et al. February 27, 2 | 2018-02-27 |
Macrocycles As Factor Xia Inhibitors App 20180022753 - Corte; James R. ;   et al. | 2018-01-25 |
Carbamoyloxymethyl Triazole Cyclohexyl Acids As Lpa Antagonists App 20170360759 - Cheng; Peter Tai Wah ;   et al. | 2017-12-21 |
Macrocyclic Factor Xia Inhibitors Condensed With Heterocycles App 20170342071 - Dilger; Andrew K. ;   et al. | 2017-11-30 |
Macrocycles as factor XIa inhibitors Grant 9,802,939 - Corte , et al. October 31, 2 | 2017-10-31 |
Substituted Tetrahydroisoquinoline Compounds As Factor Xia Inhibitors App 20170305880 - Orwat; Michael J. ;   et al. | 2017-10-26 |
Macrocycles with aromatic P2' groups as factor xia inhibitors Grant 9,777,001 - Corte , et al. October 3, 2 | 2017-10-03 |
Macrocycles as factor XIa inhibitors Grant 9,745,313 - Quan , et al. August 29, 2 | 2017-08-29 |
Tetrahydroisoquinolines containing substituted azoles as factor XIa inhibitors Grant 9,738,655 - Pinto , et al. August 22, 2 | 2017-08-22 |
Substituted 4,5,6,7-tetrahydropyrazolo[4,3-c]pyridines as factor XIa inhibitors Grant 9,725,435 - Orwat , et al. August 8, 2 | 2017-08-08 |
Five-membered Heterocycles Useful As Serine Protease Inhibitors App 20170166560 - Hangeland; Jon J. ;   et al. | 2017-06-15 |
Novel Macrocycles As Factor Xia Inhibitors App 20170158712 - Pinto; Donald J. P. ;   et al. | 2017-06-08 |
Five-membered heterocycles useful as serine protease inhibitors Grant 9,617,224 - Hangeland , et al. April 11, 2 | 2017-04-11 |
Macrocycles With Aromatic P2' Groups As Factor Xia Inhibitors App 20170096429 - Corte; James R. ;   et al. | 2017-04-06 |
Macrocycles as factor XIa inhibitors Grant 9,611,274 - Pinto , et al. April 4, 2 | 2017-04-04 |
Macrocyclic Factor Xia Inhibitors Condensed With Heterocycles App 20170057961 - Dilger; Andrew K. ;   et al. | 2017-03-02 |
Macrocycles With Hetrocyclic P2' Groups As Factor Xia Inhibitors App 20170002006 - Corte; James R. ;   et al. | 2017-01-05 |
Pyrimidinones As Factor Xia Inhibitors App 20160368923 - Dilger; Andrew K. ;   et al. | 2016-12-22 |
Macrocycles As Factor Xia Inhibitors App 20160362414 - Quan; Mimi L. ;   et al. | 2016-12-15 |
Dihydropyridone P1 As Factor Xia Inhibitors App 20160340360 - Yang; Wu ;   et al. | 2016-11-24 |
Substituted Tetrahydroisoquinoline Compounds As Factor Xia Inhibitors App 20160289209 - Orwat; Michael J. ;   et al. | 2016-10-06 |
Macrocycles as factor XIa inhibitors Grant 9,453,029 - Quan , et al. September 27, 2 | 2016-09-27 |
Pyrimidinones as factor XIa inhibitors Grant 9,453,018 - Dilger , et al. September 27, 2 | 2016-09-27 |
Dihydropyridone p1 as factor XIa inhibitors Grant 9,409,908 - Yang , et al. August 9, 2 | 2016-08-09 |
Substituted 1,2,3,4-tetrahydro-2,6-naphthyridines as factor XIa inhibitors Grant 9,394,276 - Orwat , et al. July 19, 2 | 2016-07-19 |
Dihydropyridone P1 as factor XIa inhibitors Grant 9,376,444 - Yang , et al. June 28, 2 | 2016-06-28 |
Tetrahydroisoquinolines Containing Substituted Azoles As Factor Xia Inhibitors App 20160145263 - Pinto; Donald J. P. ;   et al. | 2016-05-26 |
Pyrimidinones As Factor Xia Inhibitors App 20160096839 - Dilger; Andrew K. ;   et al. | 2016-04-07 |
Novel Macrocycles As Factor Xia Inhibitors App 20160068544 - Pinto; Donald J. P. ;   et al. | 2016-03-10 |
Macrocycles as factor XIa inhibitors Grant 9,221,818 - Pinto , et al. December 29, 2 | 2015-12-29 |
Substituted Tetrahydroisoquinoline Compounds As Factor Xia Inhibitors App 20150315200 - Orwat; Michael J. ;   et al. | 2015-11-05 |
Macrocycles As Factor Xia Inhibitors App 20150266894 - Quan; Mimi L. ;   et al. | 2015-09-24 |
Five-membered Heterocycles Useful As Serine Protease Inhibitors App 20150259297 - Hangeland; Jon J. ;   et al. | 2015-09-17 |
Cyclic P1 linkers as factor XIa inhibitors Grant 9,108,981 - Lam , et al. August 18, 2 | 2015-08-18 |
Substituted 5,6,7,8-tetrahydro-1,6-naphthyridines as factor XIa inhibitors Grant 9,108,951 - Orwat , et al. August 18, 2 | 2015-08-18 |
Dihydropyridone P1 As Factor Xia Inhibitors App 20150203492 - Yang; Wu ;   et al. | 2015-07-23 |
Five-membered heterocycles useful as serine protease inhibitors Grant 9,079,860 - Hangeland , et al. July 14, 2 | 2015-07-14 |
Macrocycles as factor XIa inhibitors Grant 9,079,918 - Quan , et al. July 14, 2 | 2015-07-14 |
Dihydropyridone P1 As Factor Xia Inhibitors App 20150166550 - Yang; Wu ;   et al. | 2015-06-18 |
Macrocycles As Factor Xia Inhibitors App 20150112058 - Corte; James R. ;   et al. | 2015-04-23 |
Cyclic P1 Linkers As Factor Xia Inhibitors App 20150057262 - Lam; Patrick Y.S. ;   et al. | 2015-02-26 |
Macrocycles as factor XIa inhibitors Grant 8,940,720 - Corte , et al. January 27, 2 | 2015-01-27 |
Cyclic P1 linkers as factor XIa inhibitors Grant 8,901,115 - Lam , et al. December 2, 2 | 2014-12-02 |
Macrocycles As Factor Xia Inhibitors App 20140343276 - Quan; Mimi L. ;   et al. | 2014-11-20 |
Substituted Tetrahydroisoquinoline Compounds As Factor Xia Inhibitors App 20140275061 - Orwat; Michael J. ;   et al. | 2014-09-18 |
Macrocycles as factor XIa inhibitors Grant 8,828,983 - Quan , et al. September 9, 2 | 2014-09-09 |
Novel Macrocycles As Factor Xia Inhibitors App 20140221338 - Pinto; Donald J. P. ;   et al. | 2014-08-07 |
Five-membered Heterocycles Useful As Serine Protease Inhibitors App 20140206706 - Hangeland; Jon J. ;   et al. | 2014-07-24 |
Cyclic P1 Linkers As Factor Xia Inhibitors App 20140163002 - Lam; Patrick Y.S. ;   et al. | 2014-06-12 |
Five-membered heterocycles useful as serine protease inhibitors Grant 8,716,492 - Hangeland , et al. May 6, 2 | 2014-05-06 |
Dihydropyridone P1 As Factor Xia Inhibitors App 20140038969 - Yang; Wu ;   et al. | 2014-02-06 |
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 8,604,056 - Pinto , et al. December 10, 2 | 2013-12-10 |
Macrocycles As Factor Xia Inhibitors App 20120309960 - Quan; Mimi L. ;   et al. | 2012-12-06 |
Pyridazine derivatives as factor xia inhibitors Grant 8,324,199 - Corte , et al. December 4, 2 | 2012-12-04 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20120270853 - Pinto; Donald J.P. ;   et al. | 2012-10-25 |
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 8,252,830 - Pinto , et al. August 28, 2 | 2012-08-28 |
Six-membered heterocycles useful as serine protease inhibitors Grant 8,163,749 - Corte April 24, 2 | 2012-04-24 |
Five-membered Heterocycles Useful As Serine Protease Inhibitors App 20120088758 - Hangeland; Jon J. ;   et al. | 2012-04-12 |
Macrocycles As Factor Xia Inhibitors App 20120041190 - Corte; James R. ;   et al. | 2012-02-16 |
Five-membered heterocycles useful as serine protease inhibitors Grant 8,101,778 - Hangeland , et al. January 24, 2 | 2012-01-24 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20110028446 - Pinto; Donald J.P. ;   et al. | 2011-02-03 |
Pyridazine Derivatives As Factor Xia Inhibitors App 20110021492 - Corte; James R. ;   et al. | 2011-01-27 |
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 7,842,708 - Pinto , et al. November 30, 2 | 2010-11-30 |
Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function Grant 7,655,689 - Salvati , et al. February 2, 2 | 2010-02-02 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20100022506 - Pinto; Donald J.P. ;   et al. | 2010-01-28 |
Substituted biaryl compounds as factor XIa inhibitors Grant 7,645,799 - Corte , et al. January 12, 2 | 2010-01-12 |
Arylpropionamide, arylacrylamide, ayrlpropynamide, or arylmethylurea analogs as factor XIa inhibitors Grant 7,626,039 - Pinto , et al. December 1, 2 | 2009-12-01 |
Six-membered Heterocycles Useful As Serine Protease Inhibitors App 20090181983 - Corte; James R. | 2009-07-16 |
Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function Grant 7,517,904 - Salvati , et al. April 14, 2 | 2009-04-14 |
Substituted Biaryl Compounds As Factor Xia Inhibitors App 20090062287 - Corte; James R. ;   et al. | 2009-03-05 |
Five-membered Heterocycles Useful As Serine Protease Inhibitors App 20090036438 - Hangeland; Jon J. ;   et al. | 2009-02-05 |
Substituted biaryl compounds as factor XIa inhibitors Grant 7,459,564 - Corte , et al. December 2, 2 | 2008-12-02 |
C-5 substituted quinazolinone derivatives as selective estrogen receptor beta modulators Grant 7,456,188 - Corte , et al. November 25, 2 | 2008-11-25 |
Five-membered heterocycles useful as serine protease inhibitors Grant 7,453,002 - Hangeland , et al. November 18, 2 | 2008-11-18 |
Six-membered heterocycles useful as serine protease inhibitors Grant 7,429,604 - Corte , et al. September 30, 2 | 2008-09-30 |
Bicyclic heterocycles useful as serine protease inhibitors Grant 7,417,063 - Smallheer , et al. August 26, 2 | 2008-08-26 |
Arylpropionamide, Arylacrylamide, Arylpropynamide, Or Arylmethylurea Analogs As Factor Xia Inhibitors App 20080161373 - Pinto; Donald J.P. ;   et al. | 2008-07-03 |
3-arylquinazoline derivatives as selective estrogen receptor beta modulators Grant 7,381,730 - Gungor , et al. June 3, 2 | 2008-06-03 |
Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function Grant 7,141,578 - Salvati , et al. November 28, 2 | 2006-11-28 |
Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function App 20060264459 - Salvati; Mark E. ;   et al. | 2006-11-23 |
Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function App 20060223832 - Salvati; Mark E. ;   et al. | 2006-10-05 |
2-substituted cyclic amines as calcium sensing receptor modulators Grant 7,105,537 - Gavai , et al. September 12, 2 | 2006-09-12 |
Substituted biaryl compounds as factor XIa inhibitors App 20060154915 - Corte; James R. ;   et al. | 2006-07-13 |
Cyclic beta-amino acid derivatives as factor Xa inhibitors App 20060074103 - Corte; James R. ;   et al. | 2006-04-06 |
Six-membered heterocycles useful as serine protease inhibitors App 20060009455 - Corte; James R. ;   et al. | 2006-01-12 |
Five-membered heterocycles useful as serine protease inhibitors App 20050282805 - Hangeland, Jon J. ;   et al. | 2005-12-22 |
Fused Heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function App 20050272799 - Salvati, Mark E. ;   et al. | 2005-12-08 |
Bicyclic heterocycles useful as serine protease inhibitors App 20050228000 - Smallheer, Joanne M. ;   et al. | 2005-10-13 |
Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function App 20050192253 - Salvati, Mark E. ;   et al. | 2005-09-01 |
Novel 2-substituted cyclic amines as calcium sensing receptor modulators App 20040229860 - Gavai, Ashvinikumar V. ;   et al. | 2004-11-18 |
Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function App 20040077605 - Salvati, Mark E. ;   et al. | 2004-04-22 |
3-Arylquinazoline derivatives as selective estrogen receptor beta modulators App 20030220227 - Gungor, Timur ;   et al. | 2003-11-27 |