Patent | Date |
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Pyridone-pyrimidine derivative acting as KRASG12C mutein inhibitor Grant 11,453,667 - Cai , et al. September 27, 2 | 2022-09-27 |
Pyrimidine Compound Acting On Egfr And Erbb2 App 20220289714 - DING; Charles Z. ;   et al. | 2022-09-15 |
Crystal Forms C And E Of Pyrazin-2(1h)-one Compound And Preparation Method Therefor App 20220289722 - HONG; Fei ;   et al. | 2022-09-15 |
Salt form and crystal form of compound as FGFR4 inhibitor and preparation method thereof Grant 11,440,903 - Long , et al. September 13, 2 | 2022-09-13 |
Compound As Porcupine Inhibitor And Use Thereof App 20220281873 - XU; Xiongbin ;   et al. | 2022-09-08 |
Crystalline Form Of Atr Inhibitor And Use Thereof App 20220281858 - WANG; Jian ;   et al. | 2022-09-08 |
Pyrrolotriazine Compounds Acting As Mnk Inhibitor App 20220281895 - WU; Lingyun ;   et al. | 2022-09-08 |
Crystal Form D Of Pyrazine-2(1h)-ketone Compound And Preparation Method Therefor App 20220281853 - CHEN; Zhiliang ;   et al. | 2022-09-08 |
Macrocyclic Derivatives As Factor Xia Inhibitors App 20220281868 - CAI; Yaxian ;   et al. | 2022-09-08 |
ATR inhibitor and application thereof Grant 11,434,232 - Qian , et al. September 6, 2 | 2022-09-06 |
Bicyclic compound as a caspase inhibitor Grant 11,434,212 - Mou , et al. September 6, 2 | 2022-09-06 |
LSD1 inhibitor and preparation method and application thereof Grant 11,433,053 - Wu , et al. September 6, 2 | 2022-09-06 |
JAK inhibitor and use thereof Grant 11,427,581 - Mao , et al. August 30, 2 | 2022-08-30 |
Azaindole Pyrazole Compounds As Cdk9 Inhibitors App 20220267321 - LIU; Yingchun ;   et al. | 2022-08-25 |
Oxazole Compound As Multi-targeted Inhibitor Of Irak4 And Btk App 20220267322 - WANG; Jianfei ;   et al. | 2022-08-25 |
Quinazoline And Cinnoline Derivatives As Dna-pk Inhibitor App 20220267310 - Chen; Kevin X ;   et al. | 2022-08-25 |
Pyridine Derivative As Fgfr And Vegfr Dual Inhibitors App 20220267324 - CHEN; Zhengxia ;   et al. | 2022-08-25 |
Sglts/dpp4 Inhibitor And Application Thereof App 20220259247 - MAO; Qinghua ;   et al. | 2022-08-18 |
Benzimidazole derivatives and use thereof as IDH1 inhibitors Grant 11,407,717 - Wang , et al. August 9, 2 | 2022-08-09 |
Bicyclic Compound As Rip-1 Kinase Inhibitor And Application Thereof App 20220242877 - WEI; Wei ;   et al. | 2022-08-04 |
Sglt2/dpp4 Inhibitor And Application Thereof App 20220242898 - MAO; Qinghua ;   et al. | 2022-08-04 |
Tetracyclic Compounds As Cdc7 Inhibitors App 20220235068 - Li; Gang ;   et al. | 2022-07-28 |
Amorphous pyrrolidine derivative as PPAR agonist and preparation method thereof Grant 11,396,493 - Yuan , et al. July 26, 2 | 2022-07-26 |
Pyrrolopyrimidine Compound And Use Thereof App 20220227788 - QIAN; Wenyuan ;   et al. | 2022-07-21 |
Imidazopyridine Compound As Irak4 Inhibitor App 20220227758 - WANG; Jianfei ;   et al. | 2022-07-21 |
Antibacterial Aminoglycoside Derivatives App 20220227802 - TANG; Dongdong ;   et al. | 2022-07-21 |
Aryl-phosphorus-oxygen compound as EGFR kinase inhibitor Grant 11,390,625 - Wu , et al. July 19, 2 | 2022-07-19 |
Pyrazolopyridine Compound As Ret Inhibitor And Application Thereof App 20220220104 - WANG; Jiansong ;   et al. | 2022-07-14 |
Crystal Form Of Wee1 Inhibitor Compound And Use Thereof App 20220220120 - QIAN; Wenyuan ;   et al. | 2022-07-14 |
Hydroxyl purine compounds and applications thereof Grant RE49,128 - Wu , et al. July 12, 2 | 2022-07-12 |
Heterocyclic compound as CSF-1R inhibitor and use thereof Grant 11,384,065 - Qian , et al. July 12, 2 | 2022-07-12 |
Pyridopyrimidine compounds acting as mTORC 1/2 dual inhibitors Grant 11,377,444 - Chen , et al. July 5, 2 | 2022-07-05 |
Nitrogen-containing Spiro Derivative As Ret Inhibitor App 20220204507 - WANG; Jiansong ;   et al. | 2022-06-30 |
Macrocyclic Derivatives Acting As Xia Factor Inhibitor App 20220204508 - Cai; Yaxian ;   et al. | 2022-06-30 |
2,3-dihydro-1h-pyrrolizine-7-formamide Derivative And Application Thereof App 20220204510 - HE; Haiying ;   et al. | 2022-06-30 |
Crystal Form Of Egfr Inhibitor And Preparation Method Thereof App 20220194959 - LIU; Xile ;   et al. | 2022-06-23 |
SMAC mimetics used as IAP inhibitors and use thereof Grant 11,358,950 - Liu , et al. June 14, 2 | 2022-06-14 |
Fgfr Inhibitor Compound In Solid Form And Preparation Method Therefor App 20220177475 - FU; Zhifei ;   et al. | 2022-06-09 |
Crystallization Of Smac Mimic Used As Iap Inhibitor And Preparation Method Thereof App 20220177453 - Liu; Yingchun ;   et al. | 2022-06-09 |
Application Of Combination Of Quinoline Derivative And Immunomodulator In Preparation Of Antitumor Drugs App 20220175756 - ZHANG; Yang ;   et al. | 2022-06-09 |
Compounds Having Both Effects Of Bet Bromodomain Protein Inhibition And Pd-l1 Gene Regulation App 20220177490 - SHEN; Chunli ;   et al. | 2022-06-09 |
Crystal and salt of 4-(naphthalen-1-yl)-4H-1,2,4-triazole compound and preparation method therefor Grant 11,352,331 - Wang , et al. June 7, 2 | 2022-06-07 |
Benzopyrazole compound used as RHO kinase inhibitor Grant 11,345,678 - Wu , et al. May 31, 2 | 2022-05-31 |
Lactam compound as FXR receptor agonist Grant 11,339,147 - He , et al. May 24, 2 | 2022-05-24 |
Glucoside Derivative That Acts As Sglt1 Inhibitor And Application Thereof App 20220153772 - LI; Yi ;   et al. | 2022-05-19 |
Diarylthiohydantoin compound as androgen receptor antagonist Grant 11,332,465 - Shen , et al. May 17, 2 | 2022-05-17 |
Vinylpyridine Carboxamide Compound As Pd-l1 Immunomodulator App 20220144806 - Zhang; Yang ;   et al. | 2022-05-12 |
Indolo Heptamyl Oxime Analogue As Parp Inhibitor App 20220144850 - Hu; Yanbin ;   et al. | 2022-05-12 |
Anti-influenza Virus Pyrimidine Derivative App 20220135558 - Xiong; Jian ;   et al. | 2022-05-05 |
Five-Membered Heteroaryl-Fused Imidazole Compound And Application Thereof App 20220135588 - YU; Tao ;   et al. | 2022-05-05 |
Pyrimidine sulfamide derivative and preparation method and medical application thereof Grant 11,319,305 - Luo , et al. May 3, 2 | 2022-05-03 |
Tricyclic furan-substituted piperidinedione compound Grant 11,319,330 - Lei , et al. May 3, 2 | 2022-05-03 |
Compound For Use In Retinal Diseases App 20220127243 - LI; Peng ;   et al. | 2022-04-28 |
Thienodiazepine derivatives and application thereof Grant 11,312,726 - Shen , et al. April 26, 2 | 2022-04-26 |
Fused ring derivative as A.sub.2A receptor inhibitor Grant 11,312,715 - Chen , et al. April 26, 2 | 2022-04-26 |
Fluorovinylbenzamide Compound As Pd-l1 Immunomodulator App 20220119368 - Zhang; Yang ;   et al. | 2022-04-21 |
Tricyclic Compounds Acting On Crbn Proteins App 20220119376 - Lei; Maoyi ;   et al. | 2022-04-21 |
Salt Of Egfr Inhibitor, Crystal Form, And Preparation Method Therefor App 20220119431 - WU; Lingyun ;   et al. | 2022-04-21 |
Cyclopropylamine Compound As Lsd1 Inhibitor And Use Thereof App 20220119401 - WU; Lingyun ;   et al. | 2022-04-21 |
Pyrazolopyrimidine Derivative And Use Thereof As Pi3k Inhibitor App 20220112217 - WU; Chengde ;   et al. | 2022-04-14 |
Prostacyclin receptor agonist Grant 11,299,475 - Qian , et al. April 12, 2 | 2022-04-12 |
5-(4-pyridyloxy)pyrazole Compounds Serving As Tgf- R1 Kinase Inhibitor App 20220098171 - FU; Xiangyu ;   et al. | 2022-03-31 |
Pyrazine-2(1H)-ketone compound acting as FGFR inhibitor Grant 11,286,248 - Zhang , et al. March 29, 2 | 2022-03-29 |
Pyrazole Compounds As LSD1 Inhibitors And Applications Thereof App 20220064126 - WU; Lingyun ;   et al. | 2022-03-03 |
Application Of Monocyclic -lactam Compound In Pharmacy App 20220062244 - WEI; Xiawei ;   et al. | 2022-03-03 |
Compound as GLS1 inhibitor Grant 11,254,666 - Liao , et al. February 22, 2 | 2022-02-22 |
Encryption and decryption method and system with continuous-variable quantum neural network Grant 11,251,948 - Shi , et al. February 15, 2 | 2022-02-15 |
Estrogen Receptor Antagonist App 20220033376 - DUAN; Shuwen ;   et al. | 2022-02-03 |
Crystal form and salt form of TGF-.beta.RI inhibitor and preparation method therefor Grant 11,236,112 - Wu , et al. February 1, 2 | 2022-02-01 |
Crystal of tricyclic compound Grant 11,236,107 - Liu , et al. February 1, 2 | 2022-02-01 |
Substituted pyrrolo[2,1-f][1,2,4]triazines as FGFR inhibitors Grant 11,236,094 - Wang , et al. February 1, 2 | 2022-02-01 |
Process Route Of Compound Of Formula (iv), Crystal Form And Preparation Method Therefor App 20220024880 - LUO; Zhi ;   et al. | 2022-01-27 |
Quinolino-pyrrolidin-2-one derivative and application thereof Grant 11,230,549 - Qian , et al. January 25, 2 | 2022-01-25 |
Substituted 1,3,4-thiadiazoles as GLS1 inhibitors Grant 11,230,544 - Liao , et al. January 25, 2 | 2022-01-25 |
Pyrazolopyrimidine Derivative As Selective Trk Inhibitor App 20210403485 - WANG; Jianfei ;   et al. | 2021-12-30 |
Pyrimidopyrazolone Derivative As Wee1 Inhibitor And Use Thereof App 20210403451 - QIAN; Wenyuan ;   et al. | 2021-12-30 |
Tricyclic Compund As Crth2 Inhibitor App 20210403466 - CHEN; Bin ;   et al. | 2021-12-30 |
3,9-diazaspiro[5,5]undecane Compound As Flt3 And Axl Inhibitors App 20210395252 - FU; Xiangyu ;   et al. | 2021-12-23 |
Crystal form and salt form of pyridone compound and preparation method therefor Grant 11,198,686 - Zhang , et al. December 14, 2 | 2021-12-14 |
Quinolino-pyrrolidin-2-one Derivative And Application Thereof App 20210380599 - QIAN; Wenyuan ;   et al. | 2021-12-09 |
S1P1 agonist and application thereof Grant 11,192,886 - Wu , et al. December 7, 2 | 2021-12-07 |
Benzopyrazole Compound Used As Rho Kinase Inhibitor App 20210371393 - WU; Lingyun ;   et al. | 2021-12-02 |
Pyridone-pyrimidine Derivative Acting As Krasg12c Mutein Inhibitor App 20210371411 - CAI; Yaxian ;   et al. | 2021-12-02 |
Smac Mimetics Used As Iap Inhibitors And Use Thereof App 20210371400 - Liu; Yingchun ;   et al. | 2021-12-02 |
Tlr8 Agonist App 20210371414 - Cai; Zhe ;   et al. | 2021-12-02 |
Uracil Compound As C-met/axl Inhibitor App 20210371395 - LI; Jinping ;   et al. | 2021-12-02 |
Crystal form of 3,4-dihydrothieno[3,2-d]pyrimidine compound and preparation method thereof Grant 11,174,270 - Xiong , et al. November 16, 2 | 2021-11-16 |
Tlr8 Agonist App 20210340141 - SUN; Fei ;   et al. | 2021-11-04 |
Quinoline derivative and use thereof as tyrosine kinase inhibitor Grant 11,161,817 - Zhang , et al. November 2, 2 | 2021-11-02 |
Bicyclic Compound as a Caspase Inhibitor App 20210332019 - MOU; Jianfeng ;   et al. | 2021-10-28 |
Biphenyl compound as CCR2/CCR5 receptor antagonist Grant 11,155,523 - Luo , et al. October 26, 2 | 2021-10-26 |
Sulfonyl-substituted isoquinolines as inhibitors of RHO kinase and hERG potassium channel activity Grant 11,155,559 - Yao , et al. October 26, 2 | 2021-10-26 |
Fused Tri-cyclic Compound As Pde3/pde4 Dual Inhibitor App 20210323960 - LUO; Yunfu ;   et al. | 2021-10-21 |
Pyrrolo[2,1-f][1,2,4]triazine Derivatives Serving As Selective Her2 Inhibitors And Application Thereof App 20210323979 - CHEN; Kevin X ;   et al. | 2021-10-21 |
Crystal form of lanosterol prodrug compound and application thereof Grant 11,149,055 - Liu , et al. October 19, 2 | 2021-10-19 |
Salt Of Lsd1 Inhibitor And A Polymorph Thereof App 20210317096 - ZHAO; Lele ;   et al. | 2021-10-14 |
Tricyclic Furan-substituted Piperidinedione Compound App 20210317138 - LEI; Maoyi ;   et al. | 2021-10-14 |
Tricyclic Substituted Piperidine Dione Compound App 20210317109 - LUO; Yunfu ;   et al. | 2021-10-14 |
CXCR2 antagonist Grant 11,136,315 - Chen , et al. October 5, 2 | 2021-10-05 |
Anti-influenza virus pyrimidine derivative Grant 11,136,319 - Xiong , et al. October 5, 2 | 2021-10-05 |
S1p1 Agonist And Application Thereof App 20210300908 - WU; Lingyun ;   et al. | 2021-09-30 |
Substituted pyrrolo[2,1-f][1,2,4]triazines as FGFR inhibitors Grant 11,130,761 - Zhang , et al. September 28, 2 | 2021-09-28 |
2,6-dioxaspiro [4,5] decane derivatives and preparation method therefor and pharmaceutical applications thereof Grant 11,124,523 - Zhang , et al. September 21, 2 | 2021-09-21 |
[1,2,4]triazolo[1,5-c]pyrimidine derivative as A.sub.2A receptor inhibitor Grant 11,117,899 - Chen , et al. September 14, 2 | 2021-09-14 |
Isothiazolo[5,4-d]pyrimidine Compound As Irak4 Inhibitor App 20210269459 - ZHANG; Yang ;   et al. | 2021-09-02 |
Azaindole Derivative And Use Thereof As Fgfr And C-met Inhibitor App 20210253571 - ZHANG; Yang ;   et al. | 2021-08-19 |
Syk inhibitor and use method therefor Grant 11,091,460 - Liu , et al. August 17, 2 | 2021-08-17 |
Crystal Form Of Lanosterol Prodrug Compound And Application Thereof App 20210246158 - LIU; Yizhi ;   et al. | 2021-08-12 |
Thieno[2,3-c]pyridazin-4(1h)-one Derivative And Application Thereof App 20210238190 - ZHENG; Xiaoping ;   et al. | 2021-08-05 |
Salt form and crystal form serving as FGFR and VEGFR inhibitor compounds, and preparation method therefor Grant 11,078,194 - Chen , et al. August 3, 2 | 2021-08-03 |
Imidaxopyrolone Compound And Application Thereof App 20210230164 - CHEN; Kevin X ;   et al. | 2021-07-29 |
[1,2,4]triazolo[1,5-c]pyrimidine derivative as A.sub.2A receptor inhibitor Grant 11,066,411 - Chen , et al. July 20, 2 | 2021-07-20 |
Crystal Form And Salt Form Of Pyridone Compound And Preparation Method Therefor App 20210206753 - ZHANG; Lei ;   et al. | 2021-07-08 |
Benzimidazole Derivatives And Use Thereof As Idh1 Inhibitors App 20210206728 - WANG; Dahai ;   et al. | 2021-07-08 |
Tri-cycle compound and applications thereof Grant 11,053,260 - He , et al. July 6, 2 | 2021-07-06 |
Ssao Inhibitor App 20210198220 - LUO; Zhi ;   et al. | 2021-07-01 |
Dimethylphosphine oxide compound Grant 11,046,720 - Wu , et al. June 29, 2 | 2021-06-29 |
Quinazoline compound for EGFR inhibition Grant 11,040,984 - Liu , et al. June 22, 2 | 2021-06-22 |
Pyridine derivative as ASK1 inhibitor and preparation method and use thereof Grant 11,040,968 - Wu , et al. June 22, 2 | 2021-06-22 |
Crystal form of indole derivative and preparation method and use thereof Grant 11,034,681 - Yao , et al. June 15, 2 | 2021-06-15 |
Borate Of Azetidine Derivative App 20210163507 - Xiong; Jian ;   et al. | 2021-06-03 |
Carboxylic acid derivative as AT.sub.2R receptor antagonist Grant 11,021,445 - Zhang , et al. June 1, 2 | 2021-06-01 |
Coumarin-like cyclic compound as MEK inhibitor and use thereof Grant 11,021,486 - Mao , et al. June 1, 2 | 2021-06-01 |
[1,2,4]triazolo[1,5-a]pyridine Compound As Jak Inhibitor And Use Thereof App 20210155621 - MAO; Weiwei ;   et al. | 2021-05-27 |
Azetidine derivative Grant 11,014,943 - Xiong , et al. May 25, 2 | 2021-05-25 |
Pyrrolidinyl Urea Derivatives And Application Thereof In Trka-related Diseases App 20210147436 - ZHANG; Yang ;   et al. | 2021-05-20 |
Pyridone-Pyrimidine Derivative Acting As KRASG12C Mutein Inhibitor App 20210147418 - CAI; Yaxian ;   et al. | 2021-05-20 |
Dimethylphosphine Oxide Compound App 20210147453 - WU; Lingyun ;   et al. | 2021-05-20 |
FGFR4 inhibitor and preparation method and use thereof Grant 11,008,292 - Chen , et al. May 18, 2 | 2021-05-18 |
SSAO inhibitor Grant 11,001,563 - Luo , et al. May 11, 2 | 2021-05-11 |
Fgfr Inhibitor App 20210130357 - ZHANG; Yang ;   et al. | 2021-05-06 |
Crystal form of URAT1 inhibitor, and preparation method therefor Grant 10,995,087 - Wang , et al. May 4, 2 | 2021-05-04 |
Monocyclic B-lactam Compound For Treating Bacterial Infection App 20210115035 - GU; Lianghu ;   et al. | 2021-04-22 |
Caspase inhibitor and pharmaceutical composition, use and therapeutic method thereof Grant 10,981,860 - He , et al. April 20, 2 | 2021-04-20 |
Spiro compound and use thereof Grant 10,981,900 - Zhang , et al. April 20, 2 | 2021-04-20 |
Heterocyclic Compound As Csf-1r Inhibitor And Use Thereof App 20210107894 - QIAN; Wenyuan ;   et al. | 2021-04-15 |
Salt Form And Crystal Form Of Compound As Fgfr4 Inhibitor And Preparation Method Thereof App 20210087181 - LONG; Chaofeng ;   et al. | 2021-03-25 |
Prostacyclin Receptor Agonist App 20210087168 - QIAN; Wenyuan ;   et al. | 2021-03-25 |
1,2-dihydro-3H-pyrazolo[3,4-d]pyrimidin-3-one derivative as Wee1 inhibitor Grant 10,954,253 - Qian , et al. March 23, 2 | 2021-03-23 |
Crystal And Salt Of 4-(naphthalen-1-yl)-4h-1,2,4-triazole Compound And Preparation Method Therefor App 20210078960 - WANG; Jianfei ;   et al. | 2021-03-18 |
Quinazoline Derivative And Use Thereof App 20210078958 - CHEN; Kevin X. ;   et al. | 2021-03-18 |
Crystal Form And Salt Form Of Tgf-bri Inhibitor And Preparation Method Therefor App 20210079021 - WU; Lifang ;   et al. | 2021-03-18 |
Jak Inhibitor And Use Thereof App 20210070754 - MAO; Weiwei ;   et al. | 2021-03-11 |
Salt type and crystal type of 4h-pyrazolo [1, 5-alpha] benzimidazole compound and preparation method and intermediate thereof Grant 10,941,150 - Wang , et al. March 9, 2 | 2021-03-09 |
Steroid Derivative FXR Agonist App 20210040140 - HE; Haiying ;   et al. | 2021-02-11 |
Pyrazine-2(1h)-ketone Compound Acting As Fgfr Inhibitor App 20210040070 - ZHANG; Yang ;   et al. | 2021-02-11 |
Anti-influenza Virus Pyrimidine Derivative App 20210032238 - Xiong; Jian ;   et al. | 2021-02-04 |
Crystal Form of 3,4-Dihydrothieno[3,2-D]Pyrimidine Compound and Preparation Method Thereof App 20210024538 - Xiong; Jian ;   et al. | 2021-01-28 |
Thienodiazepine Derivatives And Application Thereof App 20210017190 - SHEN; Chunli ;   et al. | 2021-01-21 |
Pyrazolopyrimidine Derivative And Use Thereof App 20200405725 - WANG; Jianfei ;   et al. | 2020-12-31 |
Encryption And Decryption Method And System With Continuous-variable Quantum Neural Network App 20200412532 - SHI; Jinjing ;   et al. | 2020-12-31 |
Crystal Form And Salt Form Of Pyridoimidazole Compound And Preparation Method Therefor App 20200407354 - Xiong; Jian ;   et al. | 2020-12-31 |
Steroid derivative FXR agonist Grant 10,875,888 - He , et al. December 29, 2 | 2020-12-29 |
Atr Inhibitor And Application Thereof App 20200399260 - QIAN; Wenyuan ;   et al. | 2020-12-24 |
Anti-hbvtetrahydroisoxazolo[4,3-c]pyridine Compounds App 20200377517 - WU; Lifang ;   et al. | 2020-12-03 |
Anti-HCMV virus compound Grant 10,851,112 - Xiong , et al. December 1, 2 | 2020-12-01 |
Crystal Form Of Urat1 Inhibitor, And Preparation Method Therefor App 20200361917 - Wang; Jianfei ;   et al. | 2020-11-19 |
Salt Form And Crystal Form Serving As Fgfr And Vegfr Inhibitor Compounds, And Preparation Method Therefor App 20200361913 - CHEN; Zhengxia ;   et al. | 2020-11-19 |
Thiophene, manufacturing method thereof, and pharmaceutical application of same Grant 10,829,483 - Wang , et al. November 10, 2 | 2020-11-10 |
Crystal Form Of Indole Derivative And Preparation Method And Use Thereof App 20200347040 - Yao; Yuanshan ;   et al. | 2020-11-05 |
Lsd1 Inhibitor And Preparation Method And Application Thereof App 20200345700 - WU; Lingyun ;   et al. | 2020-11-05 |
SGLTS inhibitor and application thereof Grant 10,822,365 - Wu , et al. November 3, 2 | 2020-11-03 |
Pyridopyrimidine Compounds Acting As Mtorc 1/2 Double-kinase Inhibitors App 20200339568 - CHEN; Kevin X ;   et al. | 2020-10-29 |
Cxcr2 Antagonist App 20200339549 - CHEN; Bin ;   et al. | 2020-10-29 |
Amorphous Pyrrolidine Derivative As Ppar Agonist And Preparation Method Thereof App 20200339508 - Yuan; Zhiliang ;   et al. | 2020-10-29 |
Sglts Inhibitor And Application Thereof App 20200331950 - WU; CHENGDE ;   et al. | 2020-10-22 |
Macrocyclic Compound Serving As Wee1 Inhibitor And Applications Thereof App 20200325145 - QIAN; Wenyuan ;   et al. | 2020-10-15 |
Indole derivative used as CRTH2 inhibitor Grant 10,800,765 - Yao , et al. October 13, 2 | 2020-10-13 |
Quinazolinone Compound and Application Thereof App 20200317660 - WU; Chengde ;   et al. | 2020-10-08 |
ASK1 inhibitor and preparation method and use thereof Grant 10,787,435 - Wu , et al. September 29, 2 | 2020-09-29 |
Indolo substituted piperidine compound as estrogen receptor down-regulator Grant 10,774,081 - Lu , et al. Sept | 2020-09-15 |
Pyrimidine Sulfamide Derivative And Preparation Method And Medical Application Thereof App 20200283425 - LUO; Yunfu ;   et al. | 2020-09-10 |
Crystal form and salt form of and preparation method for tyrosine kinase inhibitor Grant 10,766,862 - Long , et al. Sep | 2020-09-08 |
Diarylthiohydantoin Compound As Androgen Receptor Antagonist App 20200277290 - SHEN; Chunli ;   et al. | 2020-09-03 |
Quinoline Derivative And Use Thereof As Tyrosine Kinase Inhibitor App 20200262791 - ZHANG; Yang ;   et al. | 2020-08-20 |
HDAC6 selective inhibitors, preparation method therefor, and application thereof Grant 10,745,389 - Wu , et al. A | 2020-08-18 |
2,6-dioxaspiro [4,5] Decane Derivatives And Preparation Method Therefor And Pharmaceutical Applications Thereof App 20200255444 - Kind Code | 2020-08-13 |
Crystal Of Tricyclic Compound App 20200255449 - Kind Code | 2020-08-13 |
Lanosterol prodrug compound and preparation method therefor and use thereof Grant 10,738,076 - Liu , et al. A | 2020-08-11 |
.beta.-lactamase inhibitors Grant 10,738,051 - Hu , et al. A | 2020-08-11 |
Tri-cycle Compound And Applications Thereof App 20200247819 - Kind Code | 2020-08-06 |
Fused Ring Derivative As A2a Receptor Inhibitor App 20200239465 - CHEN; Kevin X ;   et al. | 2020-07-30 |
Modified compound of andrographolide Grant 10,717,720 - He , et al. | 2020-07-21 |
Biphenyl Compound As CCR2/CCR5 Receptor Antagonist App 20200223801 - LUO; Yunfu ;   et al. | 2020-07-16 |
Compound As Gls1 Inhibitor App 20200216436 - LIAO; Yonggang ;   et al. | 2020-07-09 |
Aryl-Phosphorus-Oxygen Compound As EGFR Kinase Inhibitor App 20200207768 - WU; Lingyun ;   et al. | 2020-07-02 |
Fgfr Inhibitor And Medical Application Thereof App 20200207773 - WANG; Yikai ;   et al. | 2020-07-02 |
Isoquinolinylsulfonyl Derivative And Use Thereof App 20200207772 - YAO; Yuanshan ;   et al. | 2020-07-02 |
Syk Inhibitor And Use Method Therefor App 20200199101 - LIU; Shilan ;   et al. | 2020-06-25 |
Hepatitis B Virus Surface Antigen Inhibitor App 20200197409 - DING; Charles Z. ;   et al. | 2020-06-25 |
Lactam Compound As Fxr Receptor Agonist App 20200190074 - HE; Haiying ;   et al. | 2020-06-18 |
Quinazoline Compound For Egfr Inhibition App 20200190107 - LIU; Xile ;   et al. | 2020-06-18 |
1,6-naphthyridine derivatives as CDK4/6 inhibitor Grant 10,676,474 - Xu , et al. | 2020-06-09 |
7-(thiazol-5-yl) pyrrolopyrimidine compound as TLR7 agonist Grant 10,676,478 - Ding , et al. | 2020-06-09 |
PDE4 inhibitor Grant 10,662,189 - Luo , et al. | 2020-05-26 |
BTK inhibitor Grant 10,662,174 - Wang , et al. | 2020-05-26 |
Dihydropyrazole azepine compound serving as Akt inhibitor Grant 10,654,868 - Lu , et al. | 2020-05-19 |
Tyrosine kinase inhibitor and pharmaceutical composition comprising same Grant 10,654,808 - Long , et al. | 2020-05-19 |
Coumarin-like Cyclic Compound As Mek Inhibitor And Use Thereof App 20200148695 - MAO; Qinghua ;   et al. | 2020-05-14 |
Thiazole derivative and applications thereof Grant 10,647,710 - He , et al. | 2020-05-12 |
Thiophene, Manufacturing Method Thereof, And Pharmaceutical Application Of Same App 20200140423 - WANG; Jianfei ;   et al. | 2020-05-07 |
[1,2,4]triazolo[1,5-c]pyrimidine Derivative As A2a Receptor Inhibitor App 20200131184 - CHEN; KEVIN X ;   et al. | 2020-04-30 |
Halogenated compound and axially chiral isomer thereof Grant 10,633,351 - Wang , et al. | 2020-04-28 |
Crystal form, salt type of substituted 2-hydro-pyrazole derivative and preparation method therefor Grant 10,626,107 - Ding , et al. | 2020-04-21 |
Azetidine Derivative App 20200115392 - XIONG; Jian ;   et al. | 2020-04-16 |
Ssao Inhibitor App 20200115352 - LUO; Zhi ;   et al. | 2020-04-16 |
Hydroxyl purine compounds and use thereof Grant 10,618,898 - Wu , et al. | 2020-04-14 |
JAK inhibitor Grant 10,617,690 - Wu , et al. | 2020-04-14 |
Carboxylic Acid Derivative As At2r Receptor Antagonist App 20200102275 - ZHANG; Yang ;   et al. | 2020-04-02 |
Pyridone derivative comprising heteroatomic ring butane substituent, for treating fibrosis and inflammatory diseases Grant 10,604,513 - Shih , et al. | 2020-03-31 |
Fgfr4 Inhibitor And Preparation Method And Use Thereof App 20200062716 - CHEN; Zhengxia ;   et al. | 2020-02-27 |
Spiro Compound And Use Thereof App 20200048235 - ZHANG; Peng ;   et al. | 2020-02-13 |
Benzotriazole-derived .alpha. and .beta.-unsaturated amide compound used as TGF-.beta. RI inhibitor Grant 10,548,883 - Sun , et al. Fe | 2020-02-04 |
Pyridine Derivative As Ask1 Inhibitor And Preparation Method And Use Thereof App 20200031823 - WU; Chengde ;   et al. | 2020-01-30 |
Crystal Form And Salt Form Of And Preparation Method For Tyrosine Kinase Inhibitor App 20200024235 - Long; Chaofeng ;   et al. | 2020-01-23 |
1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one Derivative As Wee1 Inhibitor App 20200017528 - QIAN; Wenyuan ;   et al. | 2020-01-16 |
Cyclic compound acting as PDE4 inhibitor Grant 10,532,986 - Luo , et al. Ja | 2020-01-14 |
Novel Beta-lactamase Inhibitors App 20200010467 - HU; Boyu ;   et al. | 2020-01-09 |
Pyrrolidine derivatives as PPAR agonists Grant 10,526,320 - Yuan , et al. J | 2020-01-07 |
Vinyl compounds as FGFR and VEGFR inhibitors Grant 10,519,133 - Chen , et al. Dec | 2019-12-31 |
Substituted-indole-compounds as estrogen receptor down-regulators Grant 10,519,143 - Lu , et al. Dec | 2019-12-31 |
Piperidine compounds as PCSK9 inhibitors Grant 10,513,514 - Wu , et al. Dec | 2019-12-24 |
Steroid Derivative FXR Agonist App 20190382437 - HE; Haiying ;   et al. | 2019-12-19 |
Benzimidazole-linked indole compound acting as novel divalent IAP antagonist Grant 10,508,103 - Sun , et al. Dec | 2019-12-17 |
Ask1 Inhibitor And Preparation Method And Use Thereof App 20190375728 - Wu; Chengde ;   et al. | 2019-12-12 |
HDAC6 Selective Inhibitors, Preparation Method Therefor, and Application Thereof App 20190375735 - Wu; Hao ;   et al. | 2019-12-12 |
Thiazole Derivative And Applications Thereof App 20190375744 - He; Haiying ;   et al. | 2019-12-12 |
Salt Type And Crystal Type Of 4h-Pyrazolo [1, 5-Alpha] Benzimidazole Compound And Preparation Method And Intermediate Thereof App 20190375756 - WANG; Xuehai ;   et al. | 2019-12-12 |
Pyridone compound as c-met inhibitor Grant 10,501,443 - Xu , et al. Dec | 2019-12-10 |
Fused-ring or tricyclic aryl pyrimidine compound used as kinase inhibitor Grant 10,494,373 - Ding , et al. De | 2019-12-03 |
Tricyclic compound serving as immunomodulator Grant 10,487,088 - Liu , et al. Nov | 2019-11-26 |
Halogenated Compound And Axially Chiral Isomer Thereof App 20190337904 - WANG; Jianfei ;   et al. | 2019-11-07 |
Indolo Substituted Piperidine Compound As Estrogen Receptor Degrading Agent App 20190337938 - LU; Jianyu ;   et al. | 2019-11-07 |
Cdk4/6 Inhibitor App 20190315745 - XU; Zhaobing ;   et al. | 2019-10-17 |
Salt type and crystal type of 4H-pyrazolo [1, 5-alpha] benzimidazole compound and preparation method and intermediate thereof Grant 10,428,073 - Wang , et al. October 1, 2 | 2019-10-01 |
Dezocine analogue Grant 10,414,718 - Zhang , et al. Sept | 2019-09-17 |
Crystal form A of 7-(cyclopropylmethyl)-1-(((cis )-4-hydroxy-4-methylcyclohexyl)methyl)-3-methyl-1H-purine-2,6-(3H,7H)-dio- ne for treating liver diseases Grant 10,399,981 - Wu , et al. Sep | 2019-09-03 |
Lanosterol Prodrug Compound And Preparation Method Therefor And Use Thereof App 20190256548 - LIU; Yizhi ;   et al. | 2019-08-22 |
Pyridone Compound As C-met Inhibitor App 20190248763 - XU; Xiongbin ;   et al. | 2019-08-15 |
Indole Derivative Used As Crth2 Inhibitor App 20190248770 - YAO; Yuanshan ;   et al. | 2019-08-15 |
Dihydropyrazole Azepine Compound Serving As Akt Inhibitor App 20190233434 - LU; Lun ;   et al. | 2019-08-01 |
Pyrrolidine Derivatives As Ppar Agonists App 20190225597 - Yuan; Zhiliang ;   et al. | 2019-07-25 |
Cyclic Compound Acting As Pde4 Inhibitor App 20190210975 - LUO; Yunfu ;   et al. | 2019-07-11 |
Anti-hcmv Virus Compound App 20190202838 - XIONG; Jian ;   et al. | 2019-07-04 |
Crystal Form, Salt Type Of Substituted 2-hydro-pyrazole Derivative And Preparation Method Therefor App 20190194168 - Ding; Charles Z. ;   et al. | 2019-06-27 |
Pde4 Inhibitor App 20190177318 - LUO; Yunfu ;   et al. | 2019-06-13 |
Ido1 Inhibitor And Preparation Method And Application Thereof App 20190169140 - ZHANG; Yang ;   et al. | 2019-06-06 |
Benzotriazole-derived Alpha And Beta-unsaturated Amide Compound Used As Tgf-beta Ri Inhibitor App 20190151299 - SUN; Fei ;   et al. | 2019-05-23 |
Caspase Inhibitor And Pharmaceutical Composition, Use And Therapeutic Method Thereof App 20190135733 - He; Haiying ;   et al. | 2019-05-09 |
Benzimidazole-linked Indole Compound Acting As Novel Divalent Iap Antagonist App 20190135794 - SUN; Fei ;   et al. | 2019-05-09 |
Linkers and their application towards ADC Grant 10,280,229 - Li , et al. | 2019-05-07 |
Hydroxyl purine compounds and use thereof Grant 10,278,973 - Wu , et al. | 2019-05-07 |
Tyrosine Kinase Inhibitor And Pharmaceutical Composition Comprising Same App 20190119217 - LONG; Chaofeng ;   et al. | 2019-04-25 |
Substituted-indole-compounds As Estrogen Receptor Down-regulators App 20190106414 - LU; Jianyu ;   et al. | 2019-04-11 |
Step gap inductor apparatus and methods Grant 10,256,025 - Ma , et al. | 2019-04-09 |
Salt form and crystal form of 1,2,5-thiadiazolidin-1,1-dioxide, preparation method thereof and intermediate Grant 10,227,339 - Li , et al. | 2019-03-12 |
Anti-pulmonary tuberculosis nitroimidazole derivative Grant 10,227,362 - Luo , et al. | 2019-03-12 |
Tricyclic Compound Serving As Immunomodulator App 20190062338 - Liu; Shilan ;   et al. | 2019-02-28 |
Pyridone Derivative Comprising Heteroatomic Ring Butane Substituent, For Treating Fibrosis And Inflammatory Diseases App 20190062315 - SHIH; Neng-yang ;   et al. | 2019-02-28 |
Axially chiral isomers, and preparation methods therefor and pharmaceutical uses thereof Grant 10,183,915 - Wang , et al. Ja | 2019-01-22 |
Dezocine Analogue App 20190010114 - ZHANG; Yang ;   et al. | 2019-01-10 |
Substituted pyrazoles as JAK inhibitors Grant 10,174,036 - Wu , et al. J | 2019-01-08 |
Substituted pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors Grant 10,174,056 - Wu , et al. J | 2019-01-08 |
7-(thiazol-5-yl) Pyrrolopyrimidine Compound As Tlr7 Agonist App 20180370976 - DING; Zhaozhong ;   et al. | 2018-12-27 |
Hepatitis C virus inhibitors and uses thereof in preparation of drugs Grant 10,160,771 - Zhang , et al. Dec | 2018-12-25 |
Fused-ring Or Tricyclic Aryl Pyrimidine Compound Used As Kinase Inhibitor App 20180354953 - DING; Charles Z. ;   et al. | 2018-12-13 |
Modified Compound Of Andrographolide App 20180346438 - HE; Haiying ;   et al. | 2018-12-06 |
CRYSTAL FORM OF 4H-PYRAZOLO[1,5-alpha]BENZOIMIDAZOLE COMPOUND, PREPARATION METHOD THEREOF AND INTERMEDIATE THEREOF App 20180305361 - WU; Lingyun ;   et al. | 2018-10-25 |
Piperidine Compounds As Pcsk9 Inhibitors App 20180305346 - Wu; Chengde ;   et al. | 2018-10-25 |
Preparation method for benzoxazoleoxazine ketone compound and intermediate and crystal form thereof Grant 10,106,557 - Chen , et al. October 23, 2 | 2018-10-23 |
Piperidine derivatives as orexin receptor antagonist Grant 10,100,047 - He , et al. October 16, 2 | 2018-10-16 |
Hydroxyl purine compounds and applications thereof Grant 10,098,885 - Wu , et al. October 16, 2 | 2018-10-16 |
Benzofuran analogue as NS4B inhibitor Grant 10,100,027 - Zhang , et al. October 16, 2 | 2018-10-16 |
Fused-ring or tricyclic aryl pyrimidine compound used as kinase inhibitor Grant 10,093,656 - Ding , et al. October 9, 2 | 2018-10-09 |
Salt Type And Crystal Type Of 4h-pyrazolo [1, 5-alpha] Benzimidazole Compound And Preparation Method And Intermediate Thereof App 20180258093 - WANG; Xuehai ;   et al. | 2018-09-13 |
Spirocyclic aryl phosphorus oxide and aryl phosphorus sulfide Grant 10,053,477 - Ding , et al. August 21, 2 | 2018-08-21 |
Vinyl Compounds As Fgfr And Vegfr Inhibitors App 20180222886 - CHEN; Shuhui ;   et al. | 2018-08-09 |
Resorcinol derivative as HSP90 inhibitor Grant 10,035,792 - Chen , et al. July 31, 2 | 2018-07-31 |
Imidazole derivative used as antiviral agent and use thereof in preparation of medicament Grant 10,030,029 - He , et al. July 24, 2 | 2018-07-24 |
Jak Inhibitors App 20180179209 - WU; Hao ;   et al. | 2018-06-28 |
Anti-pulmonary Tuberculosis Nitroimidazole Derivative App 20180162878 - LUO; Wei ;   et al. | 2018-06-14 |
Janus Kinase Inhibitor App 20180162879 - WU; Hao ;   et al. | 2018-06-14 |
Anti-enterovirus 71 thiadiazolidine derivative Grant 9,988,361 - Li , et al. June 5, 2 | 2018-06-05 |
Hydroxyl Purine Compounds And Use Thereof App 20180148451 - WU; Linyun ;   et al. | 2018-05-31 |
Hydroxyl Purine Compounds And Use Thereof App 20180140607 - WU; Lingyun ;   et al. | 2018-05-24 |
Salt Form And Crystal Form Of 1,2,5-thiadiazolidin-1,1-dioxide, Preparation Method Thereof And Intermediate App 20180141940 - LI; Peng ;   et al. | 2018-05-24 |
Substituted 2-hydrogen-pyrazole derivative serving as anticancer drug Grant 9,969,719 - Ding , et al. May 15, 2 | 2018-05-15 |
Imidazole Compound App 20180104220 - CHEN; Shuhui ;   et al. | 2018-04-19 |
Quinoline derivatives as SMO inhibitors Grant 9,938,292 - Wu , et al. April 10, 2 | 2018-04-10 |
Hydrazine compound as blood coagulation factor Xa inhibitor Grant 9,938,272 - Ding , et al. April 10, 2 | 2018-04-10 |
Dihydropyrimido fused ring derivative as HBV inhibitor Grant 9,938,301 - He , et al. April 10, 2 | 2018-04-10 |
Axially Chiral Isomers, And Preparation Methods Therefor And Pharmaceutical Uses Thereof App 20180079731 - WANG; Jianfei ;   et al. | 2018-03-22 |
Fused-Ring Or Tricyclic Aryl Pyrimidine Compound Used As Kinase Inhibitor App 20180072704 - DING; Charles Z. ;   et al. | 2018-03-15 |
Substituted 2-hydrogen-pyrazole Derivative Serving As Anticancer Drug App 20180072707 - Ding; Charles Z. ;   et al. | 2018-03-15 |
Pyridine derivatives and anti-mycobacterial use thereof Grant 9,878,982 - Ding , et al. January 30, 2 | 2018-01-30 |
Pyridino[1,2-A]pyrimidone analogue used as MTOR/P13K inhibitor Grant 9,868,737 - Guan , et al. January 16, 2 | 2018-01-16 |
Imidazole Derivative Used As Antiviral Agent And Use Thereof In Preparation Of Medicament App 20180009820 - He; Haiying ;   et al. | 2018-01-11 |
Resorcinol Derivative As HSP90 Inhibitor App 20180009794 - CHEN; Shuhui ;   et al. | 2018-01-11 |
Pyridino[1,2-A]pyrimidone analogue used as P13K inhibitor Grant 9,856,256 - Wu , et al. January 2, 2 | 2018-01-02 |
Isoquinolinesulfonyl derivative as RHO kinase inhibitor Grant 9,856,264 - Wu , et al. January 2, 2 | 2018-01-02 |
Analogues of 4H-pyrazolo[1,5-a] benzimidazole compound as PARP inhibitors Grant 9,856,262 - Wang , et al. January 2, 2 | 2018-01-02 |
Imidazole derivative used as antiviral agent and use therof in preparation of medicament Grant 9,850,251 - He , et al. December 26, 2 | 2017-12-26 |
Jak Inhibitor App 20170360794 - WU; Hao ;   et al. | 2017-12-21 |
Hydroxyl Purine Compounds And Applications Thereof App 20170326149 - WU; Lingyun ;   et al. | 2017-11-16 |
Btk Inhibitor App 20170313683 - Wang; Xuehai ;   et al. | 2017-11-02 |
Preparation Method For Benzoxazoleoxazine Ketone Compound And Intermediate And Crystal Form Thereof App 20170275299 - CHEN; Shuhui ;   et al. | 2017-09-28 |
Hepatitis C Virus Inhibitors And Uses Thereof In Preparation Of Drugs App 20170253614 - ZHANG; Yang ;   et al. | 2017-09-07 |
Benzofuran Analogue As Ns4b Inhibitor App 20170240519 - ZHANG; Yang ;   et al. | 2017-08-24 |
Piperidine Derivatives As Orexin Receptor Antagonist App 20170233385 - HE; Haiying ;   et al. | 2017-08-17 |
Linkers And Their Application Towards Adc App 20170202974 - LI; Chun Sing ;   et al. | 2017-07-20 |
Dihydropyrimido Loop Derivative As Hbv Inhibitor App 20170197986 - HE; Haiying ;   et al. | 2017-07-13 |
Pyridine Derivatives And Anti-mycobacterial Use Thereof App 20170174628 - DING; Zhaozhong ;   et al. | 2017-06-22 |
Quinoline Derivatives As Smo Inhibitors App 20170174703 - WU; Hao ;   et al. | 2017-06-22 |
HYDRAZINE COMPOUND AS BLOOD COAGULATION FACTOR Xa INHIBITOR App 20170152259 - DING; Zhaozhong ;   et al. | 2017-06-01 |
Pyridino[1,2-a]pyrimidone Analogue Used As P13k Inhibitor App 20170137420 - WU; Chengde ;   et al. | 2017-05-18 |
Spirocyclic Aryl Phosphorus Oxide And Aryl Phosphorus Sulfide App 20170129909 - DING; Zhaozhong ;   et al. | 2017-05-11 |
Pyridino[1,2-a]pyrimidone Analogue Used As Mtor/p13k Inhibitor App 20170129888 - GUAN; Huiping ;   et al. | 2017-05-11 |
Anti-enterovirus 71 Thiadiazolidine Derivative App 20170066732 - LI; Peng ;   et al. | 2017-03-09 |
Isoquinolinesulfonyl Derivative As Rho Kinase Inhibitor App 20170037050 - WU; Lingyun ;   et al. | 2017-02-09 |
ANALOGUES OF 4H-PYRAZOLO[1,5-a] BENZIMIDAZOLE COMPOUND AS PARP INHIBITORS App 20170029430 - WANG; Xuehai ;   et al. | 2017-02-02 |
Step Gap Inductor Apparatus And Methods App 20170011836 - Ma; Hongzhong ;   et al. | 2017-01-12 |
Imidazole Derivative Used As Antiviral Agent And Use Therof In Preparation Of Medicament App 20160318943 - He; Haiying ;   et al. | 2016-11-03 |
Self-leaded Inductive Device And Methods App 20160307692 - Zhou; Shuizhen ;   et al. | 2016-10-20 |
Parasiticidal dihydroisoxazole compounds Grant 9,255,111 - An , et al. February 9, 2 | 2016-02-09 |
Tricyclic Sulfonamide Derivatives App 20150183802 - CHEN; Shuhui ;   et al. | 2015-07-02 |
Parasiticidal dihydroisoxazole compounds Grant 8,889,710 - An , et al. November 18, 2 | 2014-11-18 |
Analgesic compounds, methods, and formulations Grant 8,802,728 - Defauw , et al. August 12, 2 | 2014-08-12 |
Parasiticidal dihydroisoxazole compounds Grant 8,648,081 - An , et al. February 11, 2 | 2014-02-11 |