Patent | Date |
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Crystalline forms of (2R,5S,13aR)-8-hydroxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13- ,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-1- 0-carboxamide Grant 11,202,780 - Carra , et al. December 21, 2 | 2021-12-21 |
Crystalline Forms Of (s)-2-ethylbutyl 2-(((s)-(((2r,3s,4r,5r)-5- (4-aminopyrrolo[2,1-f] [1,2,4]triazin-7-yl)-5-cyano-3,4-dihydroxytetrahydrofuran-2-yl)methoxy) (phenoxy) Phosphoryl)amino)propanoate App 20210163523 - Brak; Katrien ;   et al. | 2021-06-03 |
Solid forms of an ASK1 inhibitor Grant 10,946,004 - Andres , et al. March 16, 2 | 2021-03-16 |
Crystalline Forms Of (2r,5s,13ar)-8-hydroxy-7,9-dioxo-n-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13- ,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-1- 0-carboxamide App 20200390775 - Carra; Ernest A. ;   et al. | 2020-12-17 |
Crystalline forms of (S)-2-ethylbutyl 2-(((S)-(((2R,3S,4R,5R)-5- (4-aminopyrrolo[2,1-f] [1,2,4]triazin-7-yl)-5-cyano-3,4-dihydroxytetrahydrofuran-2-yl)methoxy)(p- henoxy) phosphoryl)amino)propanoate Grant 10,836,787 - Brak , et al. November 17, 2 | 2020-11-17 |
N-(cyanomethyl)-4-(2-(4-morpholinophenylamino)pyrimidin-4-yl)benzamide Grant RE48,285 - Brown , et al. October 27, 2 | 2020-10-27 |
Solid Forms Of An Ask1 Inhibitor App 20200061042 - Andres; Mark ;   et al. | 2020-02-27 |
Sodium (2R,5S,13aR)-7,9-dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,- 5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxa- zepin-8-olate Grant 10,385,067 - Carra , et al. A | 2019-08-20 |
Crystalline Forms Of (2r,5s,13ar)-8-hydroxy-7,9-dioxo-n-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13- ,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-1- 0-carboxamide App 20190015420 - Carra; Ernest A. ;   et al. | 2019-01-17 |
Crystalline Forms Of (s)-2-ethylbutyl 2-(((s)-(((2r,3s,4r,5r)-5- (4-aminopyrrolo[2,1-f] [1,2,4]triazin-7-yl)-5-cyano-3,4-dihydroxytetrahydrofuran-2-yl)methoxy) (phenoxy) Phosphoryl)amino)propanoate App 20180346504 - Brak; Katrien ;   et al. | 2018-12-06 |
Crystalline forms of (2R,5S,13AR)-8-hydroxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13- ,13A- octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-B] [1,3] oxazepine-10-carboxamide Grant 10,098,886 - Carra , et al. October 16, 2 | 2018-10-16 |
Sodium (2r,5s,13ar)-7,9-dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,- 5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxa- Zepin-8-olate App 20180065986 - CARRA; ERNEST A. ;   et al. | 2018-03-08 |
Crystalline Forms Of (2r,5s,13ar)-8-hydroxy-7,9-dioxo-n-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13- ,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-1- 0-carboxamide App 20170333438 - Carra; Ernest A. ;   et al. | 2017-11-23 |
(N-(cyanomethyl)-4-(2-(4-morpholinophenylamino)pyrimidin-4-yl)benzamide Grant 9,809,559 - Brown , et al. November 7, 2 | 2017-11-07 |
Sodium (2R,5S,13aR)-7,9-dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,- 5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2, 1-b][1, 3]oxazepin-8-olate Grant 9,708,342 - Carra , et al. July 18, 2 | 2017-07-18 |
Sodium (2r,5s,13ar)-7,9-dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,- 5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxa- Zepin-8-olate App 20170197985 - Carra; Ernest A. ;   et al. | 2017-07-13 |
Crystalline forms of (2R,5S,13AR)-8-hydroxy-7,9,-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,1- 3,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-- 10-carboxamide Grant 9,682,084 - Carra , et al. June 20, 2 | 2017-06-20 |
Solid forms of an ASK1 inhibitor Grant 9,643,956 - Andres , et al. May 9, 2 | 2017-05-09 |
(n-(cyanomethyl)-4-(2-(4-morpholinophenylamino)pyrimidin-4-yl)benzamide App 20160347719 - Brown; Brandon H. ;   et al. | 2016-12-01 |
(N-(cyanomethyl)-4-(2-(4-morpholinophenylamino)pyrimidin-4-yl)benzamide Grant 9,469,613 - Brown , et al. October 18, 2 | 2016-10-18 |
Solid Forms Of An Ask1 Inhibitor App 20160280683 - Andres; Mark ;   et al. | 2016-09-29 |
Sodium (2r,5s,13ar)-7,9-dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,- 5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b]oxazepin- -8-olate App 20160016973 - Carra; Ernest A. ;   et al. | 2016-01-21 |
Crystalline Forms Of (2r,5s,13ar)-8-hydroxy-7,9-dioxo-n-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13- ,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-1- 0-carboxamide App 20150366872 - Carra; Ernest A. ;   et al. | 2015-12-24 |
(n-(cyanomethyl)-4-(2-(4-morpholinophenylamino)pyrimidin-4-yl)benzamide App 20150361050 - Brown; Brandon H. ;   et al. | 2015-12-17 |