Patent | Date |
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Pyrrolotriazinones And Imidazotriazinones As Ubiquitin-specific Protease 7 Inhibitors App 20220033403 - Ioannidis; Stephanos ;   et al. | 2022-02-03 |
Pyrrolo And Pyrazolopyrimidines As Ubiquitin-specific Protease 7 Inhibitors App 20210332052 - Ioannidis; Stephanos ;   et al. | 2021-10-28 |
Isothiazolopyrimidinones, Pyrazolopyrimidinones, And Pyrrolopyrimidinones As Ubiquitin-specific Protease 7 Inhibitors App 20210323978 - Ioannidis; Stephanos ;   et al. | 2021-10-21 |
Thienopyrimidinones As Ubiquitin-specific Protease 7 Inhibitors App 20210292337 - Ioannidis; Stephanos ;   et al. | 2021-09-23 |
Quinazolinones And Azaquinazolinones As Ubiquitin-specific Protease 7 Inhibitors App 20210130321 - Ioannidis; Stephanos ;   et al. | 2021-05-06 |
Pyrrolotriazinones and imidazotriazinones as ubiquitin-specific protease 7 inhibitors Grant 10,981,915 - Ioannidis , et al. April 20, 2 | 2021-04-20 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20210078973 - Lin; Jian ;   et al. | 2021-03-18 |
Pyrrolo and pyrazolopyrimidines as ubiquitin-specific protease 7 inhibitors Grant 10,934,299 - Ioannidis , et al. March 2, 2 | 2021-03-02 |
Isothiazolopyrimidinones, pyrazolopyrimidinones, and pyrrolopyrimidinones as ubiquitin-specific protease 7 inhibitors Grant 10,927,130 - Ioannidis , et al. February 23, 2 | 2021-02-23 |
Thienopyrimidinones as ubiquitin-specific protease 7 inhibitors Grant 10,906,916 - Ioannidis , et al. February 2, 2 | 2021-02-02 |
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,889,567 - Lin , et al. January 12, 2 | 2021-01-12 |
Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors Grant 10,836,741 - Ioannidis , et al. November 17, 2 | 2020-11-17 |
Quinolinone five-membered heterocyclic compounds as mutant-isocitrate dehydrogenase inhibitors Grant 10,807,976 - Lin , et al. October 20, 2 | 2020-10-20 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20200223822 - Lin; Jian ;   et al. | 2020-07-16 |
Fused-bicyclic Aryl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20200115343 - Lin; Jian ;   et al. | 2020-04-16 |
Quinazolinones And Azaquinazolinones As Ubiquitin-specific Protease 7 Inhibitors App 20200087280 - Ioannidis; Stephanos ;   et al. | 2020-03-19 |
Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,577,329 - Lin , et al. | 2020-03-03 |
Quinolinone pyrimidines compositions as mutant-isocitrate dehydrogenase inhibitors Grant 10,550,099 - Lin , et al. Fe | 2020-02-04 |
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,550,098 - Lin , et al. Fe | 2020-02-04 |
Quinolinone Five-membered Heterocyclic Compounds As Mutant-isocitrate Dehydrogenase Inhibitors App 20200010464 - Lin; Jian ;   et al. | 2020-01-09 |
Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors Grant 10,519,127 - Ioannidis , et al. Dec | 2019-12-31 |
Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors Grant 10,519,129 - Ioannidis , et al. Dec | 2019-12-31 |
Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors Grant 10,519,130 - Ioannidis , et al. Dec | 2019-12-31 |
Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors Grant 10,519,128 - Ioannidis , et al. Dec | 2019-12-31 |
Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors Grant 10,513,508 - Ioannidis , et al. Dec | 2019-12-24 |
Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors Grant 10,513,507 - Ioannidis , et al. Dec | 2019-12-24 |
Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors Grant 10,508,098 - Ioannidis , et al. Dec | 2019-12-17 |
Pyrrolo And Pyrazolopyrimidines As Ubiquitin-specific Protease 7 Inhibitors App 20190367525 - Ioannidis; Stephanos ;   et al. | 2019-12-05 |
Isothiazolopyrimidinones, Pyrazolopyrimidinones, And Pyrrolopyrimidinones As Ubiquitin-specific Protease 7 Inhibitors App 20190359635 - Ioannidis; Stephanos ;   et al. | 2019-11-28 |
Thienopyrimidinones As Ubiquitin-specific Protease 7 Inhibitors App 20190359629 - Ioannidis; Stephanos ;   et al. | 2019-11-28 |
Pyrrolotriazinones And Imidazotriazinones As Ubiquitin-specific Protease 7 Inhibitors App 20190308980 - Ioannidis; Stephanos ;   et al. | 2019-10-10 |
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,414,752 - Lin , et al. Sept | 2019-09-17 |
Quinolinone five-membered heterocyclic compounds as mutant-isocitrate dehydrogenase inhibitors Grant 10,407,419 - Lin , et al. Sept | 2019-09-10 |
Quinolinone Pyrimidines Compositions As Mutant-isocitrate Dehydrogenase Inhibitors App 20190263779 - Lin; Jian ;   et al. | 2019-08-29 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20190263778 - Lin; Jian ;   et al. | 2019-08-29 |
Isothiazolopyrimidinones, pyrazolopyrimidinones, and pyrrolopyrimidinones as ubiquitin-specific protease 7 inhibitors Grant 10,377,773 - Ioannidis , et al. A | 2019-08-13 |
Thienopyrimidinones as ubiquitin-specific protease 7 inhibitors Grant 10,377,767 - Ioannidis , et al. A | 2019-08-13 |
Pyrrolo and pyrazolopyrimidines as ubiquitin-specific protease 7 inhibitors Grant 10,377,760 - Ioannidis , et al. A | 2019-08-13 |
Pyrrolotriazinones and imidazotriazinones as ubiquitin-specific protease 7 inhibitors Grant 10,351,571 - Ioannidis , et al. July 16, 2 | 2019-07-16 |
Phenyl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20190210970 - Lin; Jian ;   et al. | 2019-07-11 |
Quinolinone Pyrimidines Compositions As Mutant-isocitrate Dehydrogenase Inhibitors App 20190210995 - Lin; Jian ;   et al. | 2019-07-11 |
Fused-bicyclic Aryl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20190202790 - Lin; Jian ;   et al. | 2019-07-04 |
Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,294,206 - Lin , et al. | 2019-05-21 |
Pyridinyl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20190135781 - Lin; Jian ;   et al. | 2019-05-09 |
Quinolinone pyrimidines compositions as mutant-isocitrate dehydrogenase inhibitors Grant 10,280,150 - Lin , et al. | 2019-05-07 |
Phenyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,266,495 - Lin , et al. | 2019-04-23 |
Pyridinyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,253,015 - Lin , et al. | 2019-04-09 |
Quinazolinones And Azaquinazolinones As Ubiquitin-specific Protease 7 Inhibitors App 20190071421 - Ioannidis; Stephanos ;   et al. | 2019-03-07 |
Quinazolinones And Azaquinazolinones As Ubiquitin-specific Protease 7 Inhibitors App 20190071419 - Ioannidis; Stephanos ;   et al. | 2019-03-07 |
Quinazolinones And Azaquinazolinones As Ubiquitin-specific Protease 7 Inhibitors App 20190071420 - Ioannidis; Stephanos ;   et al. | 2019-03-07 |
Quinazolinones And Azaquinazolinones As Ubiquitin-specific Protease 7 Inhibitors App 20190071418 - Ioannidis; Stephanos ;   et al. | 2019-03-07 |
Quinazolinones And Azaquinazolinones As Ubiquitin-specific Protease 7 Inhibitors App 20190071423 - Ioannidis; Stephanos ;   et al. | 2019-03-07 |
Quinazolinones And Azaquinazolinones As Ubiquitin-specific Protease 7 Inhibitors App 20190071422 - Ioannidis; Stephanos ;   et al. | 2019-03-07 |
Thienopyrimidinones As Ubiquitin-specific Protease 7 Inhibitors App 20180346480 - Ioannidis; Stephanos ;   et al. | 2018-12-06 |
Isothiazolopyrimidinones, Pyrazolopyrimidinones, And Pyrrolopyrimidinones As Ubiquitin-specific Protease 7 Inhibitors App 20180346485 - Ioannidis; Stephanos ;   et al. | 2018-12-06 |
Pyrrolotriazinones And Imidazotriazinones As Ubiquitin-specific Protease 7 Inhibitors App 20180339991 - Ioannidis; Stephanos ;   et al. | 2018-11-29 |
Pyrrolo And Pyrazolopyrimidines As Ubiquitin-specific Protease 7 Inhibitors App 20180339988 - Ioannidis; Stephanos ;   et al. | 2018-11-29 |
Pyridinyl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20180327382 - Lin; Jian ;   et al. | 2018-11-15 |
Phenyl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20180327361 - Lin; Jian ;   et al. | 2018-11-15 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20180312487 - Lin; Jian ;   et al. | 2018-11-01 |
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,005,734 - Lin , et al. June 26, 2 | 2018-06-26 |
Pyrrolotriazinones and imidazotriazinones as ubiquitin-specific protease 7 inhibitors Grant 10,000,495 - Ioannidis , et al. June 19, 2 | 2018-06-19 |
Quinazolinones And Azaquinazolinones As Ubiquitin-specific Protease 7 Inhibitors App 20180162835 - Ioannidis; Stephanos ;   et al. | 2018-06-14 |
Fused-bicyclic Aryl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20180141910 - Lin; Jian ;   et al. | 2018-05-24 |
Substituted 2,3-dihydroimidazo[1,2-c]quinazoline derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis Grant RE46,856 - Hentemann , et al. May 22, 2 | 2018-05-22 |
Quinolinone Pyrimidines Compositions As Mutant-isocitrate Dehydrogenase Inhibitors App 20180134682 - Lin; Jian ;   et al. | 2018-05-17 |
Quinolinone Five-membered Heterocyclic Compounds As Mutant-isocitrate Dehydrogenase Inhibitors App 20180118732 - Lin; Jian ;   et al. | 2018-05-03 |
Isothiazolopyrimidinones, pyrazolopyrimidinones, and pyrrolopyrimidinones as ubiquitin-specific protease 7 inhibitors Grant 9,938,300 - Ioannidis , et al. April 10, 2 | 2018-04-10 |
Thienopyrimidinones as ubiquitin-specific protease 7 inhibitors Grant 9,932,351 - Ioannidis , et al. April 3, 2 | 2018-04-03 |
Pyridinyl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20180086733 - Lin; Jian ;   et al. | 2018-03-29 |
Pyrrolo and pyrazolopyrimidines as ubiquitin-specific protease 7 inhibitors Grant 9,902,728 - Ioannidis , et al. February 27, 2 | 2018-02-27 |
Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors Grant 9,840,491 - Ioannidis , et al. December 12, 2 | 2017-12-12 |
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 9,834,539 - Lin , et al. December 5, 2 | 2017-12-05 |
Quinolinone pyrimidines compositions as mutant-isocitrate dehydrogenase inhibitors Grant 9,815,817 - Lin , et al. November 14, 2 | 2017-11-14 |
Pyridinyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 9,771,349 - Lin , et al. September 26, 2 | 2017-09-26 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20170174658 - LIN; Jian ;   et al. | 2017-06-22 |
Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 9,624,175 - Lin , et al. April 18, 2 | 2017-04-18 |
Quinolinone five-membered heterocyclic compounds as mutant-isocitrate dehydrogenase inhibitors Grant 9,624,216 - Lin , et al. April 18, 2 | 2017-04-18 |
Quinolinone Five-membered Heterocyclic Compounds As Mutant-isocitrate Dehydrogenase Inhibitors App 20160311818 - Lin; Jian ;   et al. | 2016-10-27 |
Fused-bicyclic Aryl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20160311774 - Lin; Jian ;   et al. | 2016-10-27 |
Isothiazolopyrimidinones, Pyrazolopyrimidinones, And Pyrrolopyrimidinones As Ubiquitin-specific Protease 7 Inhibitors App 20160229872 - Ioannidis; Stephanos ;   et al. | 2016-08-11 |
Quinazolinones And Azaquinazolinones As Ubiquitin-specific Protease 7 Inhibitors App 20160229833 - Ioannidis; Stephanos ;   et al. | 2016-08-11 |
Thienopyrimidinones As Ubiquitin-specific Protease 7 Inhibitors App 20160229864 - Ioannidis; Stephanos ;   et al. | 2016-08-11 |
Pyrrolo And Pyrazolopyrimidines As Ubiquitin-specific Protease 7 Inhibitors App 20160185785 - Ioannidis; Stephanos ;   et al. | 2016-06-30 |
Pyrrolotriazinones And Imidazotriazinones As Ubiquitin-specific Protease 7 Inhibitors App 20160185786 - Ioannidis; Stephanos ;   et al. | 2016-06-30 |
Quinolinone Pyrimidines Compositions As Mutant-isocitrate Dehydrogenase Inhibitors App 20160083365 - Lin; Jian ;   et al. | 2016-03-24 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20160083349 - Lin; Jian ;   et al. | 2016-03-24 |
Pyridinyl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20160083367 - Lin; Jian ;   et al. | 2016-03-24 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20160083366 - Lin; Jian ;   et al. | 2016-03-24 |
Uses of substituted imidazoheterocycles Grant 8,859,538 - Beckett , et al. October 14, 2 | 2014-10-14 |
Substituted 2,3-dihydroimidazo[1,2-c]quinazoline Derivatives Useful For Treating Hyper-proliferative Disorders And Diseases Associated With Angiogenesis App 20130261113 - HENTEMANN; Martin ;   et al. | 2013-10-03 |
Substituted 2,3-dihydroimidazo[1,2-c]quinazoline derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis Grant 8,466,283 - Hentemann , et al. June 18, 2 | 2013-06-18 |
Substituted imidazoheterocycles Grant 8,431,565 - Beckett , et al. April 30, 2 | 2013-04-30 |
Preparation and use of aryl alkyl acid derivatives for the treatment of obesity Grant 8,013,166 - Smith , et al. September 6, 2 | 2011-09-06 |
Preparation and use of aryl alkyl acid derivatives for the treatment of obesity Grant 7,968,576 - Smith , et al. June 28, 2 | 2011-06-28 |
Preparation And Use Of Biphenyl-4-yl-carbonylamino Acid Derivatives For The Treatment Of Obesity App 20110118302 - Smith; Roger ;   et al. | 2011-05-19 |
Substituted 2,3-dihydroimidazo[1,2-c]quinazoline Derivatives Useful for Treating Hyper-Proliferative Disorders and Diseases Associated with Angiogenesis App 20110083984 - Hentemann; Martin ;   et al. | 2011-04-14 |
Uses Of Substituted Imidazoheterocycles App 20110034443 - Beckett; R. Paul ;   et al. | 2011-02-10 |
Preparation and use of biphenyl-4-yl-carbonylamino acid derivatives for the treatment of obesity Grant 7,759,376 - Smith , et al. July 20, 2 | 2010-07-20 |
Preparation and use of aryl alkyl acid derivatives for the treatment of obesity App 20090270468 - Smith; Roger ;   et al. | 2009-10-29 |
Preparation And Use Of Aryl Alkyl Acid Derivatives For The Treatment Of Obesity App 20090253762 - Smith; Roger ;   et al. | 2009-10-08 |
Preparation and Use of Aryl Alkyl Acid Derivatives for the Treatment of Obesity App 20090215780 - Smith; Roger ;   et al. | 2009-08-27 |
Preparation And Use Of Aryl Alkyl Acid Derivatives For The Treatment Of Obesity App 20090197795 - Smith; Roger ;   et al. | 2009-08-06 |
Substituted Imidazoheterocycles App 20090149450 - Beckett; R. Paul ;   et al. | 2009-06-11 |
Substituted imidazo[1,5-a][1,4]diazepines and imidazo[1,5-a]pyrazines as cannabinoid receptor agonists for the treatment of pain Grant 7,517,874 - Beckett , et al. April 14, 2 | 2009-04-14 |
Substituted Imidazoheterocycles App 20080318935 - Beckett; R. Paul ;   et al. | 2008-12-25 |
Preparation and use of aryl alkyl acid derivatives for the treatment of obesity Grant 7,423,156 - Smith , et al. September 9, 2 | 2008-09-09 |
Preparation and Use of Biphenyl-4-Yl-Carbonylamino Acid Derivatives for the Treatment of Obesity App 20070265298 - Smith; Roger ;   et al. | 2007-11-15 |
Preparation and use of aryl alkyl acid derivatives for the treatment of obesity App 20060194859 - Smith; Roger ;   et al. | 2006-08-31 |
Preparation and use of aryl alkyl acid derivatives for the treatment of obesity Grant 7,091,228 - Smith , et al. August 15, 2 | 2006-08-15 |
2,6-Substituted chroman derivatives useful as beta-3 adrenoreceptor agonists App 20050215594 - O'Connor, Stephen J. ;   et al. | 2005-09-29 |
2,6-substituted chroman derivatives useful as beta-3 adrenoreceptor agonists Grant 6,919,371 - O'Connor , et al. July 19, 2 | 2005-07-19 |
Sulfonamide substituted chroman derivatives Grant 6,903,218 - Ladouceur , et al. June 7, 2 | 2005-06-07 |
Preparation and use of aryl alkyl acid derivatives for the treatment of obesity App 20040224997 - Smith, Roger ;   et al. | 2004-11-11 |
Substituted indoles, pharmaceutical compounds containing such indoles and their use as PPAR-.gamma. binding agents Grant 6,787,651 - Stolle , et al. September 7, 2 | 2004-09-07 |
2,6-Substituted chroman derivatives useful as beta-3 adrenoreceptor agonists App 20040072828 - O'Connor, Stephen J. ;   et al. | 2004-04-15 |
Novel sulfonamide substituted chroman derivatives useful as beta 3 adrenoreceptor agonists App 20040072843 - Ladouceur, Gaetan H. ;   et al. | 2004-04-15 |
Di-substituted aminomethyl-chroman derivative beta-3 adrenoreceptor agonists Grant 6,699,860 - Ladouceur , et al. March 2, 2 | 2004-03-02 |
2,6-Substituted chroman derivatives useful as beta-3 adrenoreceptor agonists Grant 6,660,752 - O'Connor , et al. December 9, 2 | 2003-12-09 |
Substituted indoles, pharmaceutical compounds containing such indoles and their use as PPAR-gamma binding agents App 20030087902 - Stolle, Andreas ;   et al. | 2003-05-08 |
Di-substituted aminomethyl-chroman derivative beta-3 adrenoreceptor agonists App 20030078258 - Ladouceur, Gaetan H. ;   et al. | 2003-04-24 |
2,6-Substituted chroman derivatives useful as beta-3 adrenoreceptor agonists App 20030078260 - O'Connor, Stephen J. ;   et al. | 2003-04-24 |