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Bicyclic heterocycle derivatives and their use as modulators of the activity of GPR119 Grant 8,907,095 - Xia , et al. December 9, 2 | 2014-12-09 |
Bicyclic heterocycle derivatives and use thereof as GPR119 modulators Grant 8,822,480 - Neelamkavil , et al. September 2, 2 | 2014-09-02 |
Bicyclic heterocycle derivatives and methods of use thereof Grant 8,815,876 - Neelamkavil , et al. August 26, 2 | 2014-08-26 |
Substituted bicyclic piperidinyl- and piperazinyl-sulfonamides useful to inhibit 11.beta.-hydroxysteroid dehydrogenase type-1 Grant 8,604,195 - Shah , et al. December 10, 2 | 2013-12-10 |
Bicyclic piperidine and piperazine derivatives as GPCR modulators for the treatment of obesity, diabetes and other metabolic disorders Grant 8,580,807 - Boyle , et al. November 12, 2 | 2013-11-12 |
6-substituted sulfonyl azabicyclo[3.2.1]octanes useful to inhibit 11.beta.-hydroxysteroid dehydrogenase type-I Grant 8,466,149 - Boyle , et al. June 18, 2 | 2013-06-18 |
Adenosine A.sub.2a receptor antagonists Grant RE44,205 - Neustadt , et al. May 7, 2 | 2013-05-07 |
7-[2-[4-(6-fluoro-3-methyl-1,2-benzisoxazol-5-yl)-1-piperazinyl]ethyl]-2-(- 1-propynyl)-7H-pyrazolo-[4,3-E]-[1,2,4]-triazolo-[1,5-C]-pyrimidin-5-amine Grant 8,389,532 - Boyle , et al. March 5, 2 | 2013-03-05 |
Pyrimidinone derivatives and methods of use thereof Grant 8,318,751 - Boyle , et al. November 27, 2 | 2012-11-27 |
Substituted Biaryl Derivatives And Methods Of Use Thereof App 20120220614 - Boyle; Craig D. ;   et al. | 2012-08-30 |
Bridged Bicyclic Heterocycle Derivatives And Methods Of Use Thereof App 20120040975 - Neelamkavil; Santhosh Francis ;   et al. | 2012-02-16 |
Bicyclic Piperidine And Piperazine Derivatives As Gpcr Modulators For The Treatment Of Obesity, Diabetes And Other Metabolic Disorders App 20120021976 - Boyle; Craig D. ;   et al. | 2012-01-26 |
6-SUBSTITUTED SULFONYL AZABICYCLO[3.2.1]OCTANES USEFUL TO INHIBIT 11Beta-HYDROXYSTEROID DEHYDROGENASE TYPE-1 App 20110237559 - Boyle; Craig D. ;   et al. | 2011-09-29 |
Bicyclic Heterocycle Derivatives And Their Use As Modulators Of The Activity Of Gpr119 App 20110212938 - Xia; Yan ;   et al. | 2011-09-01 |
Bicyclic Heterocycle Derivatives And Methods Of Use Thereof App 20110166167 - Neelamkavil; Santhosh Francis ;   et al. | 2011-07-07 |
Bicyclic Heterocycle Derivatives And Use Thereof As Gpr119 Modulators App 20110166165 - Neelamkavil; Santhosh Francis ;   et al. | 2011-07-07 |
Substituted Azepine- And Diazepine-sulfonamides Useful To Inhibit 11beta-hydroxysteroid Dehydrogenase Type-1 App 20110129542 - Neelamkavil; Santhosh ;   et al. | 2011-06-02 |
Bicyclic Heterocycle Derivatives And Their Use As Gpcr Modulators App 20110118286 - Neelamkavil; Santhosh Francis ;   et al. | 2011-05-19 |
Bicyclic Heterocycle Derivatives And Use Thereof As Gpr119 Modulators App 20110065671 - Harris; Joel M. ;   et al. | 2011-03-17 |
SUBSTITUTED BICYCLIC PIPERIDINYL-AND PIPERAZINYL- SULFONAMIDES USEFUL TO INHIBIT 11beta-HYDROXYSTEROID DEHYDROGENASE TYPE-1 App 20110059929 - Shah; Unmesh ;   et al. | 2011-03-10 |
Pyrimidinone Derivatives And Methods Of Use Thereof App 20100190687 - Boyle; Craig D. ;   et al. | 2010-07-29 |
Pyrimidinone Derivatives And Methods Of Use Thereof App 20100113487 - Boyle; Craig D ;   et al. | 2010-05-06 |
Tetrahydropyrido[4,3-d]pyrimidinone Derivatives And Methods Of Use Thereof App 20100113330 - Boyle; Craig D. ;   et al. | 2010-05-06 |
Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A.sub.2a receptor antagonists Grant 7,709,492 - Neustadt , et al. May 4, 2 | 2010-05-04 |
7-[2-[4-(6-FLUORO-3-METHYL-1,2-BENZISOXAZOL-5-YL)-1-PIPERAZINYL]ETHYL]-2-(- 1-PROPYNYL)-7H-PYRAZOLO-[4,3-e]-[1,2,4]-TRIAZOLO-[1,5-c]-PYRIMIDIN-5-AMINE App 20090270432 - Boyle; Craig D. ;   et al. | 2009-10-29 |
7-[2-[4-(6-fluoro-3-methyl-1,2-benzisoxazol-5-yl)-1-piperazinyl]ethyl]-2-(- 1-propynyl)-7H-pyrazolo-[4,3-e]-[1,2,4]-triazolo-[1,5-C]-pyrimidin-5-amine Grant 7,572,802 - Boyle , et al. August 11, 2 | 2009-08-11 |
Xanthine phosphodiesterase V inhibitors Grant 7,531,544 - Chackalamannil , et al. May 12, 2 | 2009-05-12 |
2-heteroaryl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists Grant 7,465,740 - Neustadt , et al. December 16, 2 | 2008-12-16 |
2-alkynyl- and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A.sub.2a receptor antagonists Grant 7,368,449 - Neustadt , et al. May 6, 2 | 2008-05-06 |
Xanthine Phosphodiesterase V Inhibitors App 20080058354 - Chackalamannil; Samuel ;   et al. | 2008-03-06 |
Metabolite of xanthine Phosphodiesterase 5 inhibitor and derivatives thereof useful for treatment of erectile dysfunction Grant 7,312,223 - Ghosal , et al. December 25, 2 | 2007-12-25 |
7-[2-[4-(6-fluoro-3-methyl-1,2-benzisoxazol-5-YL)-1-piperazinyl]ethyl]-2-(- 1-propynyl)-7H-pyrazolo-[4,3-e]-[1,2,4]-triazolo-[1,5-c]-pyrimidin-5amine App 20070072867 - Boyle; Craig D. ;   et al. | 2007-03-29 |
2-Heteroaryl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists App 20070066620 - Neustadt; Bernard R. ;   et al. | 2007-03-22 |
Xanthine phosphodiesterase V inhibitor polymorphs Grant 7,192,962 - Dahanukar , et al. March 20, 2 | 2007-03-20 |
Method and system for ad hoc networking of computer users Grant 7,120,667 - Derocher , et al. October 10, 2 | 2006-10-10 |
Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists App 20050239795 - Neustadt, Bernard R. ;   et al. | 2005-10-27 |
2-alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists App 20050222164 - Neustadt, Bernard R. ;   et al. | 2005-10-06 |
Xanthine phosphodiesterase V inhibitors App 20050182077 - Chackalamannil, Samuel ;   et al. | 2005-08-18 |
Adenosine A2a receptor antagonists Grant 6,916,811 - Boyle , et al. July 12, 2 | 2005-07-12 |
Adenosine A2a receptor antagonists Grant 6,897,216 - Neustadt , et al. May 24, 2 | 2005-05-24 |
2-Alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists Grant 6,897,217 - Neustadt , et al. May 24, 2 | 2005-05-24 |
Muscarinic antagonists Grant 6,890,936 - Boyle , et al. May 10, 2 | 2005-05-10 |
Xanthine phosphodiesterase V inhibitors App 20050075349 - Chackalamannil, Samuel ;   et al. | 2005-04-07 |
Metabolite of xanthine phosphodiesterase 5 inhibitor and derivatives thereof useful for treatment of erectile dysfunction App 20050026939 - Ghosal, Anima ;   et al. | 2005-02-03 |
Xanthine phosphodiesterase V inhibitors Grant 6,821,978 - Chackalamannil , et al. November 23, 2 | 2004-11-23 |
Xanthine phosphodiesterase V inhibitors App 20040229885 - Chackalamannil, Samuel ;   et al. | 2004-11-18 |
2-Alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists App 20040220194 - Neustadt, Bernard R. ;   et al. | 2004-11-04 |
Xanthine phosphodiesterase V inhibitors App 20040167137 - Chackalamannil, Samuel ;   et al. | 2004-08-26 |
Muscarinic antagonists App 20040067972 - Boyle, Craig D. ;   et al. | 2004-04-08 |
Adenosine A2a receptor antagonists App 20040023997 - Neustadt, Bernard R. ;   et al. | 2004-02-05 |
Xanthine phosphodiesterase V inhibitor polymorphs App 20030232845 - Dahanukar, Vilas H. ;   et al. | 2003-12-18 |
Adenosine A2a receptor antagonists App 20030212059 - Boyle, Craig D. ;   et al. | 2003-11-13 |
Substituted imidazole neuropeptide Y Y5 receptor antagonists Grant 6,632,828 - Stamford , et al. October 14, 2 | 2003-10-14 |
Adenosine A2a receptor antagonists Grant 6,630,475 - Neustadt , et al. October 7, 2 | 2003-10-07 |
Substituted imidazole neuropeptide Y Y5 receptor antagonists App 20030114465 - Stamford, Andrew W. ;   et al. | 2003-06-19 |
Method and system for ad hoc networking of computer users App 20030097449 - Derocher, Michael D. ;   et al. | 2003-05-22 |
Xanthine phosphodiesterase V inhibitors App 20020169174 - Chackalamannil, Samuel ;   et al. | 2002-11-14 |
Adenosine A2a receptor antagonists App 20020099061 - Neustadt, Bernard R. ;   et al. | 2002-07-25 |
Muscarinic antagonists Grant 6,043,255 - Lowe , et al. March 28, 2 | 2000-03-28 |
Muscarinic antagonists Grant 5,889,006 - Lowe , et al. March 30, 1 | 1999-03-30 |