Patent | Date |
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Pyrimidine derivatives Grant 11,446,298 - Boss , et al. September 20, 2 | 2022-09-20 |
Inhibitors Of Indoleamine 2,3-dioxygenase And/or Tryptophan 2,3-dioxygenase App 20220259212 - BOSS; Christoph ;   et al. | 2022-08-18 |
Benzofurane and benzothiophene derivatives as PGE2 receptor modulators Grant 11,325,899 - Boss , et al. May 10, 2 | 2022-05-10 |
Inhibitors of indoleamine 2,3-dioxygenase and/or tryptophan 2,3-dioxygenase Grant 11,267,824 - Boss , et al. March 8, 2 | 2022-03-08 |
Nadph Oxidase 4 Inhibitors App 20210395238 - AISSAOUI; Hamed ;   et al. | 2021-12-23 |
NADPH oxidase 4 inhibitors Grant 11,136,317 - Aissaoui , et al. October 5, 2 | 2021-10-05 |
Benzimidazole-proline derivatives Grant 11,040,966 - Boss , et al. June 22, 2 | 2021-06-22 |
Pyrimidine Derivatives As Pge2 Receptor Modulators App 20210113559 - BOSS; Christoph ;   et al. | 2021-04-22 |
Benzofurane And Benzothiophene Derivatives As Pge2 Receptor Modulators App 20210115031 - BOSS; Christoph ;   et al. | 2021-04-22 |
Inhibitors Of Indoleamine 2,3-dioxygenase And/or Tryptophan 2,3-dioxygenase App 20200405696 - BOSS; Christoph ;   et al. | 2020-12-31 |
Inhibitors Of Indoleamine 2,3-dioxygenase And/or Tryptophan 2,3-dioxygenase App 20200216467 - BOSS; Christoph ;   et al. | 2020-07-09 |
Phenyl Derivatives As Pge2 Receptor Modulators App 20200179383 - BOSS; Christoph ;   et al. | 2020-06-11 |
Nadph Oxidase 4 Inhibitors App 20200165235 - Aissaoui; Hamed ;   et al. | 2020-05-28 |
Pyrimidine Derivatives App 20200108068 - BOSS; Christoph ;   et al. | 2020-04-09 |
NADPH oxidase 4 inhibitors Grant 10,584,118 - Aissaoui , et al. | 2020-03-10 |
Benzimidazole-proline Derivatives App 20190263797 - BOSS; Christoph ;   et al. | 2019-08-29 |
Crystalline forms Grant 10,351,560 - Aissaoui , et al. July 16, 2 | 2019-07-16 |
Benzimidazole-proline derivatives Grant 10,329,287 - Boss , et al. | 2019-06-25 |
Azaindole acetic acid derivatives and their use as prostaglandin D2 receptor modulators Grant 10,301,309 - Aissaoui , et al. | 2019-05-28 |
Crystalline Forms App 20190047996 - AISSAOUI; Hamed ;   et al. | 2019-02-14 |
Crystalline salt form of (S)-(2-(6 chloro-7-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-yl)(5-meth- oxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone as orexin receptor antagonist Grant 10,023,560 - Boss , et al. July 17, 2 | 2018-07-17 |
Nadph Oxidase 4 Inhibitors App 20180179194 - AISSAOUI; Hamed ;   et al. | 2018-06-28 |
Azaindole Acetic Acid Derivatives And Their Use As Prostaglandin D2 Receptor Modulators App 20180105520 - Aissaoui; Hamed ;   et al. | 2018-04-19 |
Use of benzimidazole-proline derivatives Grant 9,914,721 - Boss , et al. March 13, 2 | 2018-03-13 |
Crystalline form of (S)-(2-(6-chloro-7-methyl-1H-benzo[D]imidazol-2-yl)-2-methylpyrrolidin-1-- yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone and its use as orexin receptor antagonists Grant 9,914,720 - Boss , et al. March 13, 2 | 2018-03-13 |
Azaindole acetic acid derivatives and their use as prostaglandin D.sub.2 receptor modulators Grant 9,879,006 - Aissaoui , et al. January 30, 2 | 2018-01-30 |
Crystalline Salt Form Of (s)-(2-(6-chloro-7-methyl-1h-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-- Yl)(5-methoxy-2-(2h-1,2,3-triazol-2-yl)phenyl)methanone As Orexin Receptor Antagonist App 20180002317 - BOSS; Christoph ;   et al. | 2018-01-04 |
Azaindole acetic acid derivatives and their use as prostaglandin D2 receptor modulators Grant 9,850,241 - Aissaoui , et al. December 26, 2 | 2017-12-26 |
Benzimidazole-proline Derivatives App 20170305897 - BOSS; Christoph ;   et al. | 2017-10-26 |
Crystalline salt form of (S)-(2-(6-chloro-7-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-- yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone as orexin receptor antagonist Grant 9,790,208 - Boss , et al. October 17, 2 | 2017-10-17 |
Benzimidazole-proline derivatives Grant 9,732,075 - Boss , et al. August 15, 2 | 2017-08-15 |
Azaindole Acetic Acid Derivatives And Their Use As Prostaglandin D2 Receptor Modulators App 20170129884 - AISSAOUI; Hamed ;   et al. | 2017-05-11 |
Acrylamide derivatives as antimalarial agents Grant 9,637,473 - Aissaoui , et al. May 2, 2 | 2017-05-02 |
Azaindole Acetic Acid Derivatives And Their Use As Prostaglandin D2 Receptor Modulators App 20170022196 - AISSAOUI; Hamed ;   et al. | 2017-01-26 |
Use Of Benzimidazole-proline Derivatives App 20170001985 - BOSS; Christoph ;   et al. | 2017-01-05 |
Crystalline Form Of (s)-(2-(6-chloro-7-methyl-1h-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1 -yl)(5-methoxy-2-(2h-1,2,3-triazol-2-yl)phenyl)methanone And Its Use As Orexin Receptor Antagonists App 20160368901 - BOSS; Christoph ;   et al. | 2016-12-22 |
Crystalline Salt Form Of (s)-(2-(6-chloro-7-methyl-1h-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-- Yl)(5-methoxy-2-(2h-1,2,3-triazol-2-yl)phenyl)methanone As Orexin Receptor Antagonist App 20160355506 - BOSS; Christoph ;   et al. | 2016-12-08 |
Orexin receptor antagonists which are [ortho bi-(hetero-)aryl]-[2-(meta bi-(hetero-)aryl)-pyrrolidin-1-yl]-methanone derivatives Grant 9,493,446 - Bolli , et al. November 15, 2 | 2016-11-15 |
Azetidine amide derivatives as orexin receptor antagonists Grant 9,403,813 - Bolli , et al. August 2, 2 | 2016-08-02 |
Pyrazole and imidazole derivatives useful as orexin antagonists Grant 9,303,023 - Bolli , et al. April 5, 2 | 2016-04-05 |
Heterocyclyl derivatives and their use as prostaglandin D2 receptor modulators Grant 9,255,090 - Aissaoui , et al. February 9, 2 | 2016-02-09 |
Novel Acrylamide Derivatives As Antimalarial Agents App 20160024050 - AISSAOUI; Hamed ;   et al. | 2016-01-28 |
Azetidine Amide Derivatives As Orexin Receptor Antagonists App 20160024064 - BOLLI; Martin ;   et al. | 2016-01-28 |
Proline sulfonamide derivatives as orexin receptor antagonists Grant 9,211,279 - Boss , et al. December 15, 2 | 2015-12-15 |
1-phenyl-substituted heterocyclyl derivatives and their use as prostaglandin D2 receptor modulators Grant 9,169,270 - Aissaoui , et al. October 27, 2 | 2015-10-27 |
2-(1,2,3-triazol-2-yl)benzamide and 3-(1,2,3-triazol-2-YL)picolinamide derivatives as orexin receptor antagonists Grant 9,150,566 - Bolli , et al. October 6, 2 | 2015-10-06 |
Heterocyclyl Derivatives and their use as Prostaglandin D2 Receptor Modulators App 20150252036 - Aissaoui; Hamed ;   et al. | 2015-09-10 |
Orexin Receptor Antagonists Which Are [ortho Bi-(hetero-)aryl]-[2-(meta Bi-(hetero-)aryl)-pyrrolidin-1-yl]-methanone Derivatives App 20150252032 - Bolli; Martin ;   et al. | 2015-09-10 |
Proline Sulfonamide Derivatives As Orexin Receptor Antagonists App 20150246021 - BOSS; Christoph ;   et al. | 2015-09-03 |
7-(heteroaryl-amino)-6,7,8,9-tetrahydropyrido[1,2-a]indol acetic acid derivatives and their use as prostaglandin D2 receptor modulators Grant 9,096,595 - Aissaoui , et al. August 4, 2 | 2015-08-04 |
Benzimidazole-proline Derivatives App 20150166527 - Boss; Christoph ;   et al. | 2015-06-18 |
1-phenyl-substituted Heterocyclyl Derivatives And Their Use As Prostaglandin D2 Receptor Modulators App 20150158883 - Aissaoui; Hamed ;   et al. | 2015-06-11 |
2-(1,2,3-triazol-2-yl)benzamide And 3-(1,2,3-triazol-2-yl)picolinamide Derivatives As Orexin Receptor Antagonists App 20150158855 - Bolli; Martin ;   et al. | 2015-06-11 |
Proline sulfonamide derivatives as orexin receptor antagonists Grant 9,000,029 - Boss , et al. April 7, 2 | 2015-04-07 |
Proline Sulfonamide Derivatives As Orexin Receptor Antagonists App 20150057328 - BOSS; Christoph ;   et al. | 2015-02-26 |
Proline sulfonamide derivatives as orexin receptor antagonists Grant 8,895,606 - Boss , et al. November 25, 2 | 2014-11-25 |
Piperazines as antimalarial agents Grant 8,889,688 - Aissaoui , et al. November 18, 2 | 2014-11-18 |
7-(Heteroaryl-Amino)-6,7,8,9-Tetrahydropyrido[1,2-A]Indol Acetic Acid Derivatives and Their Use as Prostaglandin D2 Receptor Modulators App 20140045870 - Aissaoui; Hamed ;   et al. | 2014-02-13 |
Novel Pyrazole And Imidazole Derivatives Useful As Orexin Antagonists App 20130324579 - Bolli; Martin ;   et al. | 2013-12-05 |
1-phenyl-substituted heterocyclyl derivatives and their use as prostaglandin D.sub.2 receptor modulators Grant 8,575,158 - Aissaoui , et al. November 5, 2 | 2013-11-05 |
Lactam Derivatives Useful As Orexin Receptor Antagonists App 20130237525 - Aissaoui; Hamed ;   et al. | 2013-09-12 |
Proline Sulfonamide Derivatives As Orexin Receptor Antagonists App 20130150424 - Boss; Christoph ;   et al. | 2013-06-13 |
1-phenyl-substituted Heterocyclyl Derivatives And Their Use As Prostaglandin D2 Receptor Modulators App 20130109685 - Aissaoui; Hamed ;   et al. | 2013-05-02 |
Piperazines As Antimalarial Agents App 20120316178 - Aissaoui; Hamed ;   et al. | 2012-12-13 |
Oxazolidinone derivatives Grant 8,329,706 - Aissaoui , et al. December 11, 2 | 2012-12-11 |
4-pyrimidinesulfamide derivative Grant 8,324,232 - Bolli , et al. December 4, 2 | 2012-12-04 |
Pyrrolidines and piperidines as orexin receptor antagonists Grant 8,288,411 - Aissaoui , et al. October 16, 2 | 2012-10-16 |
2-aza-bicyclo[3.1.0]hexane derivatives as orexin receptor antagonists Grant 8,288,435 - Aissaoui , et al. October 16, 2 | 2012-10-16 |
2-aza-bicyclo[3.3.0]octane derivatives Grant 8,288,429 - Aissaoui , et al. October 16, 2 | 2012-10-16 |
2-aza-bicyclo[2.2.1]heptane derivatives Grant 8,236,801 - Aissaoui , et al. August 7, 2 | 2012-08-07 |
Thiazolidine derivatives as orexin receptor antagonists Grant 8,236,964 - Aissaoui , et al. August 7, 2 | 2012-08-07 |
4-pyrimidinesulfamide Derivative App 20120142716 - Bolli; Martin ;   et al. | 2012-06-07 |
5,6,7,8-tetrahydro-imidazo[1,5-.alpha.]pyrazine derivatives Grant 8,188,082 - Aissaoui , et al. May 29, 2 | 2012-05-29 |
Novel Oxazolidinone Deriviatives App 20120101111 - Aissaoui; Hamed ;   et al. | 2012-04-26 |
Thiazolidin-4-one And [1,3]-thiazinan-4-one Compounds As Orexin Receptor Antagonists App 20120088759 - Aissaoui; Hamed ;   et al. | 2012-04-12 |
Bicyclononene derivatives Grant 8,138,340 - Bezencon , et al. March 20, 2 | 2012-03-20 |
3-heteroaryl (amino or amido)-1-(biphenyl or phenylthiazolyl) carbonylpiperidine derivatives as orexin receptor inhibitors Grant 8,133,901 - Aissaoui , et al. March 13, 2 | 2012-03-13 |
3-aza-bicyclo[3.3.0]octane compounds Grant 8,106,215 - Aissaoui , et al. January 31, 2 | 2012-01-31 |
Piperazines as antimalarial agents Grant 8,067,419 - Binkert , et al. November 29, 2 | 2011-11-29 |
Trans-3-aza-bicyclo[3.1.0]hexane derivatives Grant 8,063,099 - Aissaoui , et al. November 22, 2 | 2011-11-22 |
Tetrahydroisoquinolines As Antimalarial Agents App 20110281869 - Aissaoui; Hamed ;   et al. | 2011-11-17 |
1,2-diamido-ethylene Derivatives As Orexin Antagonists App 20110263662 - Aissaoui; Hamed ;   et al. | 2011-10-27 |
Novel Bis-amides As Anti-malarial Agents App 20110224210 - Aissaoui; Hamed ;   et al. | 2011-09-15 |
Phenethylamide Derivatives And Their Heterocyclic Analogues App 20110212968 - Aissaoui; Hamed ;   et al. | 2011-09-01 |
N-glycinsulfonamide derivatives and uses as orexin receptor antagonists Grant 8,003,654 - Aissaoui , et al. August 23, 2 | 2011-08-23 |
Azetidine compounds as orexin receptor antagonists Grant 7,994,336 - Aissaoui , et al. August 9, 2 | 2011-08-09 |
2-aza-bicyclo[3.1.0]hexane Derivatives As Orexin Receptor Antagonists App 20110124636 - Aissaoui; Hamed ;   et al. | 2011-05-26 |
5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine Compounds App 20110105514 - Aissaoui; Hamed ;   et al. | 2011-05-05 |
Thiazolidine Compounds As Orexin Receptor Antagonists App 20110105491 - Aissaoui; Hamed ;   et al. | 2011-05-05 |
Tetrazole Compounds As Orexin Receptor Antagonists App 20110086889 - Aissaoui; Hamed ;   et al. | 2011-04-14 |
Piperidine And Pyroolidine Compounds App 20110039857 - Aissaoui; Hamed ;   et al. | 2011-02-17 |
2-aza-bicyclo[3.3.0]octane Derivatives App 20110009461 - Aissaoui; Hamed ;   et al. | 2011-01-13 |
2-aza-bicyclo[2.2.1]heptane Derivatives App 20110009401 - Aissaoui; Hamed ;   et al. | 2011-01-13 |
Sulfamides as endothelin receptor antagonists for the treatment of cardiovascular diseases Grant 7,868,012 - Bolli , et al. January 11, 2 | 2011-01-11 |
Novel Piperidine Carboxylic Acid Amine Derivatives App 20100324052 - Bezencon; Olivier ;   et al. | 2010-12-23 |
Pyrazolo-tetrahydro pyridine derivatives as orexin receptor antagonists Grant 7,834,028 - Aissaoui , et al. November 16, 2 | 2010-11-16 |
Piperidine carboxylic acid amide derivatives Grant 7,799,805 - Bezencon , et al. September 21, 2 | 2010-09-21 |
2-cyclopropyl-thiazole Derivatives App 20100222328 - Aissaoui; Hamed ;   et al. | 2010-09-02 |
Azetidine Compounds As Orexin Receptor Antagonists App 20100222600 - Aissaoui; Hamed ;   et al. | 2010-09-02 |
Trans-3-aza-bicyclo[3.1.0]hexane Derivatives App 20100204285 - Aissaoui; Hamed ;   et al. | 2010-08-12 |
Pyrrolidines And Piperidines As Orexin Receptor Antagonists App 20100197733 - Aissaoui; Hamed ;   et al. | 2010-08-05 |
3-aza-bicyclo[3.3.0]octane Compounds App 20100184808 - Aissaoui; Hamed ;   et al. | 2010-07-22 |
Thiazolidine Derivatives As Orexin Receptor Antagonists App 20100113531 - Aissaoui; Hamed ;   et al. | 2010-05-06 |
5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine Derivatives App 20100093740 - Aissaoui; Hamed ;   et al. | 2010-04-15 |
3-heteroaryl (amino Or Amido)-1-(biphenyl Or Phenylthiazolyl) Carbonylpiperidine Derivatives As Orexin Receptor Inhibitors App 20100069418 - Aissaoui; Hamed ;   et al. | 2010-03-18 |
1,4,5,6,7,8-hexahydro-1,2,5-triaza-azulene Derivatives As Orexin Receptor Antagonists App 20100029617 - Aissaoui; Hamed ;   et al. | 2010-02-04 |
3-aza-bicyclo[3.1.0]hexane Derivatives App 20100016401 - Aissaoui; Hamed ;   et al. | 2010-01-21 |
Bicyclononene derivaties App 20090306123 - Bezencon; Olivier ;   et al. | 2009-12-10 |
Novel Sulfonamide Compounds App 20090275588 - Aissaoui; Hamed ;   et al. | 2009-11-05 |
Pyrazolo-tetrahydro Pyridine Derivatives As Orexin Receptor Antagonists App 20090099228 - Aissaoui; Hamed ;   et al. | 2009-04-16 |
Pyrimidine-sulfamides and their use as endothelian receptor antagonist Grant 7,452,896 - Bolli , et al. November 18, 2 | 2008-11-18 |
Novel Piperazines as Antimalarial Agents App 20080234272 - Binkert; Christoph ;   et al. | 2008-09-25 |
Novel Piperidine Carboxylic Acid Amide Derivatives App 20080214598 - Bezencon; Olivier ;   et al. | 2008-09-04 |
Novel 4-Aminopiperidine Derivatives App 20080076762 - Boss; Christoph ;   et al. | 2008-03-27 |
Alkansulfonamides as endothelin antagonists Grant 7,323,465 - Bolli , et al. January 29, 2 | 2008-01-29 |
Sulfamides as Endothelin Receptor Antagonists for the Treatment of Cardiovascular Diseases App 20080004298 - Bolli; Martin ;   et al. | 2008-01-03 |
Sulfamides and their use as endothelin receptor antagonists Grant 7,285,549 - Bolli , et al. October 23, 2 | 2007-10-23 |
Novel sulfamides App 20070167472 - Bolli; Martin ;   et al. | 2007-07-19 |
Benzo-fused heterocycles as endothelin antagonists Grant 7,238,685 - Bolli , et al. July 3, 2 | 2007-07-03 |
Sliding roof system Grant 7,234,767 - Boss , et al. June 26, 2 | 2007-06-26 |
Sulfamides and their use as endothelin receptor antagonists Grant 7,094,781 - Bolli , et al. August 22, 2 | 2006-08-22 |
Arylalkane-sulfonamides having endothelin-antagonist activity Grant 7,091,201 - Weller , et al. August 15, 2 | 2006-08-15 |
Novel sulfamides App 20060178365 - Bolli; Martin ;   et al. | 2006-08-10 |
Sliding roof system App 20060049671 - Boss; Christoph ;   et al. | 2006-03-09 |
Arylethene-sulfonamides Grant 6,951,856 - Boss , et al. October 4, 2 | 2005-10-04 |
Novel benzo-fused heterocycles as endothelin antagonisits App 20050124605 - Bolli, Martin ;   et al. | 2005-06-09 |
Novel alkansulfonamides as endothelin antagonists App 20050085639 - Bolli, Martin ;   et al. | 2005-04-21 |
Roof module with moveable lid and rigid sealing strip Grant 6,854,796 - Boss , et al. February 15, 2 | 2005-02-15 |
Wind deflector for a vehicle roof Grant 6,834,914 - Bohm , et al. December 28, 2 | 2004-12-28 |
Substituted amino-aza-cycloalkanes useful against malaria App 20040102431 - Boss, Christoph ;   et al. | 2004-05-27 |
Arylalkane-sulfonamides having endothelin-antagonist activity App 20040102464 - Weller, Thomas ;   et al. | 2004-05-27 |
Novel sulfamides and their use as endothelin receptor antagonists App 20040077670 - Bolli, Martin ;   et al. | 2004-04-22 |
Roof module with moveable lid and rigid sealing strip App 20040070234 - Boss, Christoph ;   et al. | 2004-04-15 |
Butyne diol derivatives Grant 6,720,322 - Bolli , et al. April 13, 2 | 2004-04-13 |
Substituted alkyldiamines App 20040067927 - Boss, Christoph ;   et al. | 2004-04-08 |
Novel arylethene-sulfonamides App 20030220359 - Boss, Christoph ;   et al. | 2003-11-27 |
Wind deflector for a vehicle roof App 20030168892 - Bohm, Horst ;   et al. | 2003-09-11 |
6 alkoxy-4-pyrimidinyl bis-sulfonamides Grant 6,596,719 - Bolli , et al. July 22, 2 | 2003-07-22 |
Butyne diol derivatives App 20030087920 - Bolli, Martin ;   et al. | 2003-05-08 |