Patent | Date |
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Pyrazolyl Quinoxaline Kinase Inhibitors App 20220135544 - SAXTY; Gordon ;   et al. | 2022-05-05 |
Benzolactam compounds as protein kinase inhibitors Grant 11,001,575 - Berdini , et al. May 11, 2 | 2021-05-11 |
Pyrazolyl Quinoxaline Kinase Inhibitors App 20200131153 - SAXTY; Gordon ;   et al. | 2020-04-30 |
Pyrazolyl quinoxaline kinase inhibitors Grant 10,519,137 - Saxty , et al. Dec | 2019-12-31 |
Benzolactam compounds as protein kinase inhibitors Grant 10,457,669 - Berdini , et al. Oc | 2019-10-29 |
Pteridines as FGFR inhibitors Grant 10,272,087 - Saxty , et al. | 2019-04-30 |
Benzolactam Compounds As Protein Kinase Inhibitors App 20190047990 - BERDINI; Valerio ;   et al. | 2019-02-14 |
Substituted quinoxalines as FGFR kinase inhibitors Grant 10,052,320 - Woodhead , et al. August 21, 2 | 2018-08-21 |
Substituted pyrido[2,3-b]pyrazines as FGFR kinase inhibitors Grant 10,045,982 - Berdini , et al. August 14, 2 | 2018-08-14 |
Quinolines as FGFR kinase modulators Grant 10,039,759 - Berdini , et al. August 7, 2 | 2018-08-07 |
Pyrazolyl Quinoxaline Kinase Inhibitors App 20180127397 - SAXTY; Gordon ;   et al. | 2018-05-10 |
Substituted quinoxalines as FGFR kinase inhibitors Grant 9,856,236 - Saxty , et al. January 2, 2 | 2018-01-02 |
Pyrazolyl quinoxaline kinase inhibitors Grant 9,850,228 - Saxty , et al. December 26, 2 | 2017-12-26 |
Pteridines As Fgfr Inhibitors App 20170000796 - SAXTY; Gordon ;   et al. | 2017-01-05 |
Quinolines As Fgfr Kinase Modulators App 20170000781 - BERDINI; Valerio ;   et al. | 2017-01-05 |
Omega-aminoalkylamides of R-2-aryl-propionic acids as inhibitors of the chemotaxis of polymorphonucleate and mononucleate cells Grant 9,493,402 - Allegretti , et al. November 15, 2 | 2016-11-15 |
Pyrazolyl Quinoxaline Kinase Inhibitors App 20160311800 - SAXTY; Gordon ;   et al. | 2016-10-27 |
Pyrazolyl quinoxaline kinase inhibitors Grant 9,464,071 - Saxty , et al. October 11, 2 | 2016-10-11 |
Pteridines as FGFR inhibitors Grant 9,447,098 - Saxty , et al. September 20, 2 | 2016-09-20 |
Quinolines as FGFR kinase modulators Grant 9,439,896 - Berdini , et al. September 13, 2 | 2016-09-13 |
Pyrazole Derivatives As Protein Kinase Modulators App 20160250187 - BERDINI; Valerio ;   et al. | 2016-09-01 |
SUBSTITUTED PYRIDO[2,3-b]PYRAZINES AS FGFR KINASE INHIBITORS App 20160235744 - BERDINI; Valerio ;   et al. | 2016-08-18 |
Substitutued Quinoxalines As Fgfr Kinase Inhibitors App 20160220564 - WOODHEAD; Steven John ;   et al. | 2016-08-04 |
Substituted pyrido[2,3-b]pyrazines as FGFR kinase inhibitors Grant 9,309,242 - Berdini , et al. April 12, 2 | 2016-04-12 |
Substituted quinoxalines as FGFR kinase inhibitors Grant 9,303,029 - Woodhead , et al. April 5, 2 | 2016-04-05 |
Substituted quinoxalines as FGFR kinase inhibitors Grant 9,290,478 - Saxty , et al. March 22, 2 | 2016-03-22 |
Pyrazole derivatives as protein kinase modulators Grant 9,283,226 - Berdini , et al. March 15, 2 | 2016-03-15 |
Substituted Quinoxalines As Fgfr Kinase Inhibitors App 20160031856 - SAXTY; Gordon ;   et al. | 2016-02-04 |
Pteridines As Fgfr Inhibitors App 20150291589 - Saxty; Gordon ;   et al. | 2015-10-15 |
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators Grant 9,051,278 - Berdini , et al. June 9, 2 | 2015-06-09 |
Pyrazolyl Quinoxaline Kinase Inhibitors App 20150105368 - SAXTY; Gordon ;   et al. | 2015-04-16 |
Ortho-condensed pyridine and pyrimidine derivatives (e.g., purines) as protein Grant 9,006,430 - Berdini , et al. April 14, 2 | 2015-04-14 |
Anticancer Benzopyrazines Via The Inhibition Of Fgfr Kinases App 20150031669 - Woodhead; Steven John ;   et al. | 2015-01-29 |
3,4-disubstituted 1h-pyrazole Compounds And Their Use As Cyclin Dependent Kinase And Glycogen Synthase Kinase-3 Modulators App 20140371213 - BERDINI; Valerio ;   et al. | 2014-12-18 |
Bicyclic heterocyclic compounds as FGFR inhibitors Grant 8,895,745 - Berdini , et al. November 25, 2 | 2014-11-25 |
Pyrazolyl quinoxaline kinase inhibitors Grant 8,895,601 - Saxty , et al. November 25, 2 | 2014-11-25 |
Bicyclic heterocyclic compounds as protein tyrosine kinase inhibitors Grant 8,859,582 - Saxty , et al. October 14, 2 | 2014-10-14 |
Bicyclic heterocyclic compounds as protein tyrosine kinase inhibitors Grant 8,859,583 - Saxty , et al. October 14, 2 | 2014-10-14 |
Ortho-condensed Pyridine And Pyrimidine Derivatives (e.g., Purines) As Protein Kinases Inhibitors App 20140303177 - BERDINI; Valerio ;   et al. | 2014-10-09 |
Quinolines As Fgfr Kinase Modulators App 20140296236 - Berdini; Valerio ;   et al. | 2014-10-02 |
Anticancer Pyridopyrazines Via The Inhibition Of Fgfr Kinases App 20140288053 - Berdini; Valerio ;   et al. | 2014-09-25 |
Pyrazole Derivatives As Protein Kinase Modulators App 20140271662 - BERDINI; Valerio ;   et al. | 2014-09-18 |
Ortho-condensed pyridine and pyrimidine derivatives (e.g., purines) as protein kinases inhibitors Grant 8,809,336 - Berdini , et al. August 19, 2 | 2014-08-19 |
Imidazopyridine derivatives as inhibitors of receptor tyrosine kinases Grant 8,796,244 - Berdini , et al. August 5, 2 | 2014-08-05 |
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators Grant 8,779,147 - Berdini , et al. July 15, 2 | 2014-07-15 |
Pyrazole compounds that modulate the activity of CDK, GSK and aurora kinases Grant 8,778,936 - Berdini , et al. July 15, 2 | 2014-07-15 |
Imidazo [1,2-A]pyridine derivatives as FGFR kinase inhibitors for use in therapy Grant 8,722,687 - Saxty , et al. May 13, 2 | 2014-05-13 |
Ortho-Condensed Pyridine and Pyrimidine Derivatives (e.g., Purines) as Protein Kinases Inhibitors App 20140107137 - BERDINI; Valerio ;   et al. | 2014-04-17 |
Pyrazole derivatives as protein kinase modulators Grant 8,691,806 - Berdini , et al. April 8, 2 | 2014-04-08 |
Benzimidazole Derivatives And Their Use As Protein Kinase Inhibitors App 20140010892 - BERDINI; Valerio ;   et al. | 2014-01-09 |
Substituted Benzopyrazin Derivatives As Fgfr Kinase Inhibitors For The Treatment Of Cancer Diseases App 20130267525 - Saxty; Gordon ;   et al. | 2013-10-10 |
Ortho-condensed pyridine and pyrimidine derivatives (e.g., purines) as protein kinases inhibitors Grant 8,546,407 - Berdini , et al. October 1, 2 | 2013-10-01 |
Imidazo[1,2-a]pyridine compounds for use in treating cancer Grant 8,513,276 - Berdini , et al. August 20, 2 | 2013-08-20 |
Bicyclic heterocyclyl derivatives as FGFR kinase inhibitors for therapeutic use Grant 8,481,531 - Saxty , et al. July 9, 2 | 2013-07-09 |
"omega-aminoalkylamides Of R-2-aryl-propionic Acids Asinhibitors Of The Chemotaxis Of Polymorphonucleate Andmononucleate Cells" App 20130079514 - ALLEGRETTI; Marcello ;   et al. | 2013-03-28 |
Pyrazolyl Quinazoline Kinase Inhibitors App 20130072457 - Saxty; Gordon ;   et al. | 2013-03-21 |
Pharmaceutical compounds Grant 8,399,442 - Berdini , et al. March 19, 2 | 2013-03-19 |
Pyrazole Derivatives As Protein Kinase Modulators App 20130005702 - BERDINI; Valerio ;   et al. | 2013-01-03 |
Omega aminoalkylamides of R-2 aryl propionic acids as inhibitors of the chemotaxis of polymorphonucleate and mononucleate cells Grant 8,288,368 - Allegretti , et al. October 16, 2 | 2012-10-16 |
3,4-disubstituted 1h-pyrazole Compounds And Their Use As Cyclin Dependent Kinase And Glycogen Synthase Kinase-3 Modulators App 20120213791 - BERDINI; Valerio ;   et al. | 2012-08-23 |
Pyrazole derivatives as protein kinase modulators Grant 8,247,576 - Berdini , et al. August 21, 2 | 2012-08-21 |
Imidazopyridine Derivatives As Inhibitors Of Receptor Tyrosine Kinases App 20120208791 - Berdini; Valerio ;   et al. | 2012-08-16 |
Pyrazole Compounds That Modulate The Activity Of Cdk, Gsk And Aurora Kinases App 20120190673 - BERDINI; Valerio ;   et al. | 2012-07-26 |
FGFR pharmacophore compounds Grant 8,131,527 - Saxty , et al. March 6, 2 | 2012-03-06 |
Imidazo [1,2-a]pyridine Derivatives As Fgfr Kinase Inhibitors For Use In Therapy App 20120041000 - Saxty; Gordon ;   et al. | 2012-02-16 |
Bicyclic Heterocyclic Compounds As Protein Tyrosine Kinase Inhibitors App 20120035153 - SAXTY; Gordon ;   et al. | 2012-02-09 |
Bicyclic Heterocyclyl Derivatives As Fgfr Kinase Inhibitors For Therapeutic Use App 20120035171 - Saxty; Gordon ;   et al. | 2012-02-09 |
Bicyclic Heterocyclic Compounds As Protein Tyrosine Kinase Inhibitors App 20120035152 - SAXTY; Gordon ;   et al. | 2012-02-09 |
Pyrazole compounds that modulate the activity of CDK, GSK and aurora kinases Grant 8,110,573 - Berdini , et al. February 7, 2 | 2012-02-07 |
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators Grant 8,080,666 - Berdini , et al. December 20, 2 | 2011-12-20 |
Bicyclic heterocyclic compounds as protein tyrosine kinase inhibitors Grant 8,076,354 - Saxty , et al. December 13, 2 | 2011-12-13 |
Bicyclic heterocyclic compounds as protein tyrosine kinase inhibitors Grant 8,071,614 - Saxty , et al. December 6, 2 | 2011-12-06 |
Benzimidazole Derivatives And Their Use As Protein Kinase Inhibitors App 20110224203 - BERDINI; Valerio ;   et al. | 2011-09-15 |
Benzimidazole derivatives and their use as protein kinase inhibitors Grant 7,977,477 - Berdini , et al. July 12, 2 | 2011-07-12 |
Pyrazole Derivatives As Protein Kinase Modulators App 20110144080 - Berdini; Valerio ;   et al. | 2011-06-16 |
3,4-disubstituted 1h-pyrazole Compounds And Their Use As Cyclin Dependent Kinase And Glycogen Synthase Kinase-3 Modulators App 20110003799 - BERDINI; Valerio ;   et al. | 2011-01-06 |
Bicyclic Heterocyclic Compounds As Protein Tyrosine Kinase Inhibitors App 20100331296 - Saxty; Gordon ;   et al. | 2010-12-30 |
Bicyclic Heterocyclic Compounds As Protein Tyrosine Kinase Inhibitors App 20100286113 - Saxty; Gordon ;   et al. | 2010-11-11 |
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators Grant 7,825,140 - Berdini , et al. November 2, 2 | 2010-11-02 |
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators Grant 7,745,638 - Berdini , et al. June 29, 2 | 2010-06-29 |
Pyrazole Derivatives As That Modulate The Activity Of Cdk, Gsk And Aurora Kinases App 20100160324 - Berdini; Valerio ;   et al. | 2010-06-24 |
Bicyclic Heterocyclic Compounds as FGFR Inhibitors App 20100120761 - Berdini; Valerio ;   et al. | 2010-05-13 |
Compounds App 20100093718 - Berdini; Valerio ;   et al. | 2010-04-15 |
Pharmaceutical Compounds App 20100004232 - Berdini; Valerio ;   et al. | 2010-01-07 |
Ortho-Condensed Pyridine and Pyrimidine Derivatives (e.g., Purines) as Protein Kinases Inhibitors App 20090247538 - Berdini; Valerio ;   et al. | 2009-10-01 |
Ortho-Condensed Pyridine and Pyrimidine Derivatives (e.g., Purines) as Protein Kinases Inhibitors App 20090099213 - Berdini; Valerio ;   et al. | 2009-04-16 |
Thiazole And Isothiazole Derivatives That Modulate The Activity Of CDK, GSK And Aurora Kinases App 20080312223 - Berdini; Valerio ;   et al. | 2008-12-18 |
Pyrazole Derivatives for the Inhibition of CDK'S and GSK'S App 20080306069 - Wyatt; Paul Graham ;   et al. | 2008-12-11 |
Compounds for Treating Protein-Kinase Mediated Disorders App 20080275029 - Berdini; Valerio ;   et al. | 2008-11-06 |
3,4-disubstituted 1h-pyrazole Compounds And Their Use As Cyclin Dependent Kinase And Glycogen Synthase Kinase-3 Modulators App 20080269207 - Berdini; Valerio ;   et al. | 2008-10-30 |
3,4-disubstituted 1h-pyrazole Compounds And Their Use As Cyclin Dependent Kinase And Glycogen Synthase Kinase-3 Modulators App 20080200509 - Berdini; Valerio ;   et al. | 2008-08-21 |
Pyrazole Derivatives For The Inhibition Of Cdk's And Gsk's App 20080194562 - Wyatt; Paul Graham ;   et al. | 2008-08-14 |
Pharmaceutical Compounds App 20080167309 - Berdini; Valerio ;   et al. | 2008-07-10 |
Pyrazole Derivatives For The Inhibition Of Cdk's And Gsk's App 20080139620 - Wyatt; Paul Graham ;   et al. | 2008-06-12 |
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators Grant 7,385,059 - Berdini , et al. June 10, 2 | 2008-06-10 |
Pyrazole Compounds that Modulate the Activity of Cdk, Gsk and Aurora Kinases App 20080132495 - Berdini; Valerio ;   et al. | 2008-06-05 |
Omega-aminoalkylamides Of R-2-aryl-propionic Acids As Inhibitors Of The Chemotaxis Of Polymorphonucleate And Mononucleate Cells App 20080045522 - ALLEGRETTI; Marcello ;   et al. | 2008-02-21 |
3,4-Disubstituted Pyrazoles as Cyclin Dependent Kinases (Cdk) or Aurora Kinase or Glycogen Synthase 3 (Gsk-3) Inhibitors App 20080004270 - Gill; Adrian Liam ;   et al. | 2008-01-03 |
Benzimidazole derivatives and their use as protein kinases inhibitors App 20070135477 - Berdini; Valerio ;   et al. | 2007-06-14 |
Pharmaceutical compounds App 20070105900 - Berdini; Valerio ;   et al. | 2007-05-10 |
3,4-Disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators App 20060194843 - Berdini; Valerio ;   et al. | 2006-08-31 |
3-(Carbonyl) 1h-indazole compounds as cyclin dependent kinases (cdk) inhibitors App 20060135516 - Berdini; Valerio ;   et al. | 2006-06-22 |
Omega aminoalkylamides of R-2 aryl propionic acids as inhibitors of the chemotaxis of polymorphonucleate and mononucleate cells App 20050080067 - Allegretti, Marcello ;   et al. | 2005-04-14 |