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Oga Inhibitor Compounds App 20210300900 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2021-09-30 |
Oga Inhibitor Compounds App 20210300943 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2021-09-30 |
Oga Inhibitor Compounds App 20210277003 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2021-09-09 |
Oga Inhibitor Compounds App 20210277015 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2021-09-09 |
Oga Inhibitor Compounds App 20210261527 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2021-08-26 |
Oga Inhibitor Compounds App 20210130352 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2021-05-06 |
Oga Inhibitor Compounds App 20210122763 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2021-04-29 |
Oga Inhibitor Compounds App 20210115040 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2021-04-22 |
[1,2,4]-triazolo [1,5-a]-pyrimidinyl Derivatives Substituted With Piperidine, Morpholine Or Piperazine As Oga Inhibitors App 20200157092 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2020-05-21 |
Monocyclic Oga Inhibitor Compounds App 20200079766 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2020-03-12 |
Oga Inhibitor Compounds App 20200048267 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2020-02-13 |
Bicyclic Oga Inhibitor Compounds App 20190359609 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2019-11-28 |
Inhibitors of phosphodiesterase 10 enzyme Grant 9,550,784 - Leclercq , et al. January 24, 2 | 2017-01-24 |
Fast-dissociating dopamine 2 receptor antagonists Grant 9,422,296 - Macdonald , et al. August 23, 2 | 2016-08-23 |
Substituted pyrazolo[1,5-a]pyrazines as mGluR5 receptor modulators Grant 9,255,103 - Conn , et al. February 9, 2 | 2016-02-09 |
Substituted Bicyclic Alkoxy Pyrazole Analogs As Allosteric Modulators Of Mglur5 Receptors App 20150216863 - Conn; P. Jeffrey ;   et al. | 2015-08-06 |
Bicyclic oxazole and thiazole compounds and their use as allosteric modulators of mGluR5 receptors Grant 9,090,632 - Conn , et al. July 28, 2 | 2015-07-28 |
Inhibitors Of Phosphodiesterase 10 Enzyme App 20150203498 - Leclercq; Laurent Christian L. ;   et al. | 2015-07-23 |
Bicyclic thiazoles as allosteric modulators of mGluR5 receptors Grant 9,040,707 - MacDonald , et al. May 26, 2 | 2015-05-26 |
Substituted bicyclic alkoxy pyrazole analogs as allosteric modulators of mGluR5 receptors Grant 9,029,366 - Conn , et al. May 12, 2 | 2015-05-12 |
Substituted 6-methylnicotinamides as mGluR5 positive allosteric modulators Grant 8,969,389 - Conn , et al. March 3, 2 | 2015-03-03 |
Thia(dia)zoles as fast dissociating dopamine 2 receptor antagonists Grant 8,933,101 - MacDonald , et al. January 13, 2 | 2015-01-13 |
4-alkoxypyridazine derivatives as fast dissociating dopamine 2 receptor antagonists Grant 8,906,921 - MacDonald , et al. December 9, 2 | 2014-12-09 |
Substituted bicyclic alkoxy pyrazole analogs as allosteric modulators of mGluR5 receptors Grant 8,901,125 - Conn , et al. December 2, 2 | 2014-12-02 |
Piperazin-1-yl-trifluoromethyl-substituted-pyridines as fast dissociating dopamine 2 receptor antagonists Grant 8,895,562 - Bartolome-Nebreda , et al. November 25, 2 | 2014-11-25 |
Fast-dissociating Dopamine 2 Receptor Antagonists App 20140336381 - Macdonald; Gregor James ;   et al. | 2014-11-13 |
Substituted Imidazopyrimidin-5(6h)-ones As Allosteric Modulators Of Mglur5 Receptors App 20140329838 - Conn; P. Jeffrey ;   et al. | 2014-11-06 |
Substituted imidazopyrimidin-5(6H)-ones as allosteric modulators of MGLUR5 receptors Grant 8,865,725 - Conn , et al. October 21, 2 | 2014-10-21 |
Imidazo[1,2-a]pyrazine derivatives and their use for the prevention or treatment of neurological, psychiatric and metabolic disorders and diseases Grant 8,859,543 - Bartolome-Nebreda , et al. October 14, 2 | 2014-10-14 |
Naphthyridinone analogs as mGluR5 positive allosteric modulators Grant 8,853,237 - Conn , et al. October 7, 2 | 2014-10-07 |
Bicyclic Pyrazole Compounds As Allosteric Modulators Of Mglur5 Receptors App 20140213593 - Conn; P. Jeffrey ;   et al. | 2014-07-31 |
Fast-dissociating dopamine 2 receptor antagonists Grant 8,791,120 - MacDonald , et al. July 29, 2 | 2014-07-29 |
Imidazo[1,2-b]pyridazine derivatives and their use as PDE10 inhibitors Grant 8,716,282 - Pastor-Fernandez , et al. May 6, 2 | 2014-05-06 |
Dihydronaphthyridinyl(organo)methanone analogs as positive allosteric mGluR5 modulators Grant 8,710,074 - Conn , et al. April 29, 2 | 2014-04-29 |
Substituted pyrazolo[1,5-A]pyrazine compounds as allosteric modulators of mGluR5 receptors Grant 8,703,946 - Conn , et al. April 22, 2 | 2014-04-22 |
Bicyclic Triazole And Pyrazole Lactams As Allosteric Modulators Of Mglur5 Receptors App 20140057870 - Conn; P. Jeffrey ;   et al. | 2014-02-27 |
Substituted Bicyclic Cycloalkyl Pyrazole Lactam Analogs As Allosteric Modulators Of Mglur5 Receptors App 20130345204 - Conn; P. Jeffrey ;   et al. | 2013-12-26 |
Substituted Bicyclic Alkoxy Pyrazole Analogs As Allosteric Modulators Of Mglur5 Receptors App 20130345203 - Conn; P. Jeffrey ;   et al. | 2013-12-26 |
Substituted Bicyclic Alkoxy Pyrazole Analogs As Allosteric Modulators Of Mglur5 Receptors App 20130345206 - Conn; P. Jeffrey ;   et al. | 2013-12-26 |
Substituted Bicyclic Aralkyl Pyrazole Lactam Analogs As Allosteric Modulators Of Mglur5 Receptors App 20130345205 - Conn; P. Jeffrey ;   et al. | 2013-12-26 |
Bicyclic triazole and pyrazole lactams as allosteric modulators of mGluR5 receptors Grant 8,592,422 - Conn , et al. November 26, 2 | 2013-11-26 |
Bicyclic Oxazole And Thiazole Compounds And Their Use As Allosteric Modulators Of Mglur5 Receptors App 20130261107 - Conn; P. Jeffrey ;   et al. | 2013-10-03 |
Bicyclic Oxazole Lactams As Allosteric Modulators Of Mglur5 Receptors App 20130252943 - Conn; P. Jeffrey ;   et al. | 2013-09-26 |
Substituted Imidazopyrimidin-5(6h)-ones As Allosteric Modulators Of Mglur5 Receptors App 20130245043 - Conn; P. Jeffrey ;   et al. | 2013-09-19 |
Substituted 6-(1-piperazinyl)-pyridazines as 5-HT.sub.6 receptor antagonists Grant 8,530,474 - Bartolome-Nebreda , et al. September 10, 2 | 2013-09-10 |
Piperidinylamino-pyridazines and their use as fast dissociating dopamine 2 receptor antagonists Grant 8,466,153 - MacDonald , et al. June 18, 2 | 2013-06-18 |
IMIDAZO[1,2-a]PYRAZINE DERIVATIVES AND THEIR USE FOR THE PREVENTION OR TREATMENT OF NEUROLOGICAL, PSYCHIATRIC AND METABOLIC DISORDERS AND DISEASES App 20120329792 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2012-12-27 |
Bicyclic Pyrazole Compounds As Allosteric Modulators Of Mglur5 Receptors App 20120295913 - Conn; P. Jeffrey ;   et al. | 2012-11-22 |
Bicyclic Thiazoles As Allosteric Modulators Of Mglur5 Receptors App 20120258955 - MacDonald; Gregor James ;   et al. | 2012-10-11 |
Bicyclic Triazole And Pyrazole Lactams As Allosteric Modulators Of Mglur5 Receptors App 20120225844 - Conn; P. Jeffrey ;   et al. | 2012-09-06 |
IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AND THEIR USE AS PDE10 INHIBITORS App 20120220581 - Pastor-Fernandez; Joaquin ;   et al. | 2012-08-30 |
Dihydronaphthyridinyl(organo)methanone Analogs As Positive Allosteric Mglur5 Modulators App 20120178776 - Conn; P. Jeffrey ;   et al. | 2012-07-12 |
Naphthyridinone Analogs As Mglur5 Positive Allosteric Modulators App 20120172391 - Conn; P. Jeffrey ;   et al. | 2012-07-05 |
Substituted 6-methylnicotinamides As Mglur5 Positive Allosteric Modulators App 20110294858 - Conn; P. Jeffrey ;   et al. | 2011-12-01 |
IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AND THEIR USE AS PDE10 INHIBITORS App 20110269752 - Pastor-Fernandez; Joaquin ;   et al. | 2011-11-03 |
O-benzyl Nicotinamide Analogs As Mglur5 Positive Allosteric Modulators App 20110183980 - Conn; P. Jeffrey ;   et al. | 2011-07-28 |
Substituted 6-(1-piperazinyl)-pyridazines As 5-ht6 Receptor Antagonists App 20110112107 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2011-05-12 |
Use of anti-histaminics for acute reduction of elevated intracranial pressure Grant 7,732,437 - Tegtmeier , et al. June 8, 2 | 2010-06-08 |
Pyridine Derivatives As Fast Dissociating Dopamine 2 Receptor Antagonists App 20100137368 - MacDonald; Gregor James ;   et al. | 2010-06-03 |
Thia(dia)zoles As Fast Dissociating Dopamine 2 Receptor Antagonists App 20100120860 - MacDonald; Gregor James ;   et al. | 2010-05-13 |
Fast Dissociating Dopamine 2 Receptor Antagonists App 20100076187 - MacDonald; Gregor James ;   et al. | 2010-03-25 |
Fast-dissociating Dopamine 2 Receptor Antagonists App 20100069394 - MacDonald; Gregor James ;   et al. | 2010-03-18 |
4-alkoxypyridazine Derivatives As Fast Dissociating Dopamine 2 Receptor Antagonists App 20100063058 - MacDonald; Gregor James ;   et al. | 2010-03-11 |
Isoxazoline-indole derivatives with an improved antipsychotic and anxiolytic activity Grant 7,635,696 - Andres-Gil , et al. December 22, 2 | 2009-12-22 |
Fused heterocyclic isoxazoline derivatives and their use as anti-depressants Grant 7,501,418 - Andres-Gil , et al. March 10, 2 | 2009-03-10 |
Substituted tetracyclic imidazole derivatives, processes for their preparation, pharmaceutical compositions comprising them and their use as a medicine Grant 7,476,662 - Janssens , et al. January 13, 2 | 2009-01-13 |
C-substituted tricyclic isoxazoline derivatives and their use as anti-depressants Grant 7,465,741 - Andres-Gil , et al. December 16, 2 | 2008-12-16 |
Compounds for treating fundic disaccomodation Grant 7,423,048 - Van Emelen , et al. September 9, 2 | 2008-09-09 |
Isoxazoline-Indole Derivatives With an Improved Antipsychotic and Anxiolytic Activity App 20080113988 - Andres-Gil; Jose Ignacio ;   et al. | 2008-05-15 |
Novel indole derivatives with an improved antipsychotic activity App 20070066608 - Bartolome-Nebreda; Jose Manuel ;   et al. | 2007-03-22 |
Compounds for treating impaired fundic relaxation Grant 7,081,453 - Van Emelen , et al. July 25, 2 | 2006-07-25 |
Fused heterocyclic isoxazoline derivatives and their use as anti-derpressants App 20060116378 - Andres-Gil; Jose Ignacio ;   et al. | 2006-06-01 |
C-substituted tricyclic isoxazoline derivatives and their use as anti-depressants App 20050256119 - Andres-Gil, Jose Ignacio ;   et al. | 2005-11-17 |
Use of anti-histaminics for acute reduction of elevated intracranial pressure App 20050070525 - Tegtmeier, Frank ;   et al. | 2005-03-31 |
Novel substituted tetracyclic imidazole derivatives, processes for their preparation, pharamaceutical compositions comprising them and their use as a medicine App 20040167138 - Janssens, Frans Eduard ;   et al. | 2004-08-26 |
Compounds for treating impaired fundic relaxation App 20040019051 - Van Emelen, Kristof ;   et al. | 2004-01-29 |