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Bromodomain inhibitors and uses thereof Grant 8,796,261 - Albrecht , et al. August 5, 2 | 2014-08-05 |
Bromodomain Inhibitors And Uses Thereof App 20120157428 - Albrecht; Brian K. ;   et al. | 2012-06-21 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20070203108 - Thorsett; Eugene D. ;   et al. | 2007-08-30 |
Methods and compounds for inhibiting beta-amyloid peptide release and/or its synthesis App 20060223761 - Audia; James E. ;   et al. | 2006-10-05 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20050267150 - Thompson, Richard C. ;   et al. | 2005-12-01 |
Polycyclic .alpha.-amino-.epsilon.-caprolactams and related compounds Grant 6,958,330 - Audia , et al. October 25, 2 | 2005-10-25 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20050192269 - Thompson, Richard C. ;   et al. | 2005-09-01 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20050192265 - Thompson, Richard C. ;   et al. | 2005-09-01 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds Grant 6,906,056 - Thompson , et al. June 14, 2 | 2005-06-14 |
Methods and compounds for inhibiting .beta.-amyloid peptide release and/or its synthesis Grant 6,888,022 - Audia , et al. May 3, 2 | 2005-05-03 |
Methods and compounds for inhibiting .beta.-amyloid peptide release and/or its synthesis Grant 6,861,558 - Audia , et al. March 1, 2 | 2005-03-01 |
Heterocyclic compounds, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds Grant 6,849,650 - Thorsett , et al. February 1, 2 | 2005-02-01 |
Deoxyamino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds Grant 6,838,455 - Audia , et al. January 4, 2 | 2005-01-04 |
Deoxyamino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds Grant 6,774,125 - Audia , et al. August 10, 2 | 2004-08-10 |
N-(aryl/heteroarylacetyl) amino acid esters, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds Grant 6,767,918 - Wu , et al. July 27, 2 | 2004-07-27 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting Beta-amyloid peptide release and/or its synthesis by use of such compounds App 20040106598 - Thompson, Richard C. ;   et al. | 2004-06-03 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20040043977 - Wu, Jing ;   et al. | 2004-03-04 |
Cyclic amino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds Grant 6,696,438 - Audia , et al. February 24, 2 | 2004-02-24 |
Methods and compounds for inhibiting beta-amyloid peptide release and/or its synthesis App 20030229024 - Audia, James E. ;   et al. | 2003-12-11 |
N-(aryl/heteroarylacety) amino acid esters, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds Grant 6,642,261 - Wu , et al. November 4, 2 | 2003-11-04 |
N-(aryl/heteroarylacetyl) amino acid esters, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20030191119 - Wu, Jing ;   et al. | 2003-10-09 |
Cyclic amino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20030162768 - Audia, James E. ;   et al. | 2003-08-28 |
Deoxyamino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20030153550 - Audia, James E. ;   et al. | 2003-08-14 |
Deoxyamino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20030149022 - Audia, James E. ;   et al. | 2003-08-07 |
Heterocyclic compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20030130188 - Thorsett, Eugene D. ;   et al. | 2003-07-10 |
Biological reagents and methods for determining the mechanism in the generation of beta-amyloid peptide App 20030069445 - Audia, James E. ;   et al. | 2003-04-10 |
Deoxyamino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds Grant 6,509,331 - Audia , et al. Ja | 2003-01-21 |
Heterocyclic compounds, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds Grant 6,506,782 - Thorsett , et al. January 14, 2 | 2003-01-14 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting B-amyloid peptide release and/or its synthesis by use of such compounds App 20020173504 - Wu, Jing ;   et al. | 2002-11-21 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20020137738 - Wu, Jing ;   et al. | 2002-09-26 |
N-(aryl/heteroarylacetyl) amino acid esters, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20020137743 - Wu, Jing ;   et al. | 2002-09-26 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20020123486 - Wu, Jing ;   et al. | 2002-09-05 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20020115652 - Wu, Jing ;   et al. | 2002-08-22 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-Amyloid peptide release and/or its synthesis by use of such compounds App 20020111343 - Wu, Jing ;   et al. | 2002-08-15 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds App 20020068741 - Wu, Jing ;   et al. | 2002-06-06 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting B-amyloid peptide release and/or its synthesis by use of such compounds App 20020055500 - Wu, Jing ;   et al. | 2002-05-09 |
Methods and compounds for inhibiting beta-amyloid peptide release and/or its synthesis App 20020052322 - Audia, James E. ;   et al. | 2002-05-02 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting B-amyloid peptide release and/or its synthesis by use of such compounds App 20020052359 - Wu, Jing ;   et al. | 2002-05-02 |
N-(aryl/heteroaryl) Amino Acid Derivatives, Pharmaceutical Compositions Comprising Same, And Methods For Inhibiting Beta-amyloid Peptide Release And/or Its Synthesis By Use Of Such Compounds App 20010020097 - AUDIA, JAMES E. ;   et al. | 2001-09-06 |
N-(aryl/heteroaryl/alkylacetyl) amino acid amides, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds Grant 6,262,302 - Wu , et al. July 17, 2 | 2001-07-17 |
Compounds for inhibiting .beta.-amyloid peptide release and/or its synthesis Grant 6,211,235 - Wu , et al. April 3, 2 | 2001-04-03 |
Compounds having effects on serotonin-related systems Grant 6,172,073 - Audia , et al. January 9, 2 | 2001-01-09 |
N-(aryl/heteroarylacetyl) amino acid esters, pharmaceutical compositions comprising same, and methods for use Grant 6,117,901 - Wu , et al. September 12, 2 | 2000-09-12 |
Tetrahydro-beta-carbolines Grant 6,090,945 - Audia , et al. July 18, 2 | 2000-07-18 |
N-(aryl/heteroaryl) amino acid esters, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds Grant 5,965,614 - Audia , et al. October 12, 1 | 1999-10-12 |
Tetrahydrobetacarboline compounds Grant 5,886,004 - Audia , et al. March 23, 1 | 1999-03-23 |
Aminoalkyl-indoles Grant 5,869,691 - Audia , et al. February 9, 1 | 1999-02-09 |
Tetrahydro-beta-carbolines Grant 5,861,409 - Audia , et al. January 19, 1 | 1999-01-19 |
Inhibition of serotonin reuptake Grant 5,846,982 - Audia , et al. December 8, 1 | 1998-12-08 |
Compounds having effects on serotonin-related systems Grant 5,789,402 - Audia , et al. August 4, 1 | 1998-08-04 |
Tetrahydro-beta-carbolines Grant 5,760,051 - Audia , et al. June 2, 1 | 1998-06-02 |
Naphthylpiperazinyl compounds useful for treating 5HT.sub.2B receptor mediated conditions Grant 5,736,544 - Audia , et al. April 7, 1 | 1998-04-07 |
5HT.sub.1F agonists for the treatment of migraine Grant 5,721,252 - Audia , et al. February 24, 1 | 1998-02-24 |
Method for treating 5-HT.sub.2B receptor related conditions Grant 5,705,519 - Audia , et al. January 6, 1 | 1998-01-06 |
5-HT.sub.1F mediated inhibition of neurogenic meningeal extravasation: a method for the treatment of migraine Grant 5,698,571 - Audia , et al. December 16, 1 | 1997-12-16 |
Method for treating 5HT.sub.2B receptor related conditions Grant 5,688,807 - Audia , et al. November 18, 1 | 1997-11-18 |
Compositions for inhibiting bone loss Grant 5,670,514 - Audia , et al. September 23, 1 | 1997-09-23 |
Treatment and prevention of prostatic cancer metastasis Grant 5,635,197 - Audia , et al. June 3, 1 | 1997-06-03 |
Intermediates to tetrahydro-beta-carbolines Grant 5,635,528 - Audia , et al. June 3, 1 | 1997-06-03 |
8-substituted tetrahydro-beta-carbolines Grant 5,631,265 - Audia , et al. May 20, 1 | 1997-05-20 |
Compounds having effects on serotonin-related systems Grant 5,614,523 - Audia , et al. March 25, 1 | 1997-03-25 |
3-<1-alkylenearyl>-4-<1,2,3,6-tetrahydropyridinyl>-and 3-<1-alkylenearyl>-4-piperidinyl-1h-indoles: new 5-HT.sub.1F agonists Grant 5,521,197 - Audia May 28, 1 | 1996-05-28 |
Tetrahydro-beta-carbolines Grant 5,508,284 - Audia , et al. April 16, 1 | 1996-04-16 |
Tetrahydro-pyrido-indole Grant 5,300,645 - Audia , et al. April 5, 1 | 1994-04-05 |