Patent | Date |
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Inhibiting mutant IDH-1 Grant 11,376,246 - Kelly , et al. July 5, 2 | 2022-07-05 |
Inhibiting mutant isocitrate dehydrogenase 1 (mIDH-1) Grant 11,311,527 - Kelly , et al. April 26, 2 | 2022-04-26 |
INHIBITING MUTANT ISOCITRATE DEHYDROGENASE 1 (mIDH-1) App 20210244727 - ASHWELL; Susan ;   et al. | 2021-08-12 |
Inhibiting Mutant Idh-1 App 20210196701 - Kelly; Patrick F. ;   et al. | 2021-07-01 |
Treating patients harboring an isocitrate dehydrogenase-1 (IDH-1) mutation Grant 11,013,734 - Kelly , et al. May 25, 2 | 2021-05-25 |
Inhibiting mutant isocitrate dehydrogenase 1 (mlDH-1) Grant 11,013,733 - Ashwell , et al. May 25, 2 | 2021-05-25 |
Treating Patients Harboring An Isocitrate Dehydrogenase 1 (idh-1) Mutation App 20210085669 - Kelly; Patrick F. ;   et al. | 2021-03-25 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20210078973 - Lin; Jian ;   et al. | 2021-03-18 |
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,889,567 - Lin , et al. January 12, 2 | 2021-01-12 |
Quinolinone five-membered heterocyclic compounds as mutant-isocitrate dehydrogenase inhibitors Grant 10,807,976 - Lin , et al. October 20, 2 | 2020-10-20 |
INHIBITING MUTANT ISOCITRATE DEHYDROGENASE 1 (mIDH-1) App 20200297717 - Kelly; Patrick F. ;   et al. | 2020-09-24 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20200223822 - Lin; Jian ;   et al. | 2020-07-16 |
Fused-bicyclic Aryl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20200115343 - Lin; Jian ;   et al. | 2020-04-16 |
Inhibiting Mutant Idh-1 App 20200108060 - Kelly; Patrick F. ;   et al. | 2020-04-09 |
Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,577,329 - Lin , et al. | 2020-03-03 |
Quinolinone pyrimidines compositions as mutant-isocitrate dehydrogenase inhibitors Grant 10,550,099 - Lin , et al. Fe | 2020-02-04 |
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,550,098 - Lin , et al. Fe | 2020-02-04 |
Quinolinone Five-membered Heterocyclic Compounds As Mutant-isocitrate Dehydrogenase Inhibitors App 20200010464 - Lin; Jian ;   et al. | 2020-01-09 |
INHIBITING MUTANT ISOCITRATE DEHYDROGENASE 1 (mIDH-1) App 20190350921 - Ashwell; Susan | 2019-11-21 |
Inhibiting Mutant Idh-1 App 20190350919 - Kelly; Patrick F. ;   et al. | 2019-11-21 |
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,414,752 - Lin , et al. Sept | 2019-09-17 |
Quinolinone five-membered heterocyclic compounds as mutant-isocitrate dehydrogenase inhibitors Grant 10,407,419 - Lin , et al. Sept | 2019-09-10 |
Quinolinone Pyrimidines Compositions As Mutant-isocitrate Dehydrogenase Inhibitors App 20190263779 - Lin; Jian ;   et al. | 2019-08-29 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20190263778 - Lin; Jian ;   et al. | 2019-08-29 |
Quinolinone Pyrimidines Compositions As Mutant-isocitrate Dehydrogenase Inhibitors App 20190210995 - Lin; Jian ;   et al. | 2019-07-11 |
Phenyl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20190210970 - Lin; Jian ;   et al. | 2019-07-11 |
Fused-bicyclic Aryl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20190202790 - Lin; Jian ;   et al. | 2019-07-04 |
Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,294,206 - Lin , et al. | 2019-05-21 |
Pyridinyl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20190135781 - Lin; Jian ;   et al. | 2019-05-09 |
Quinolinone pyrimidines compositions as mutant-isocitrate dehydrogenase inhibitors Grant 10,280,150 - Lin , et al. | 2019-05-07 |
Phenyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,266,495 - Lin , et al. | 2019-04-23 |
Pyridinyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,253,015 - Lin , et al. | 2019-04-09 |
Pyridinyl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20180327382 - Lin; Jian ;   et al. | 2018-11-15 |
Phenyl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20180327361 - Lin; Jian ;   et al. | 2018-11-15 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20180312487 - Lin; Jian ;   et al. | 2018-11-01 |
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 10,005,734 - Lin , et al. June 26, 2 | 2018-06-26 |
Fused-bicyclic Aryl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20180141910 - Lin; Jian ;   et al. | 2018-05-24 |
Quinolinone Pyrimidines Compositions As Mutant-isocitrate Dehydrogenase Inhibitors App 20180134682 - Lin; Jian ;   et al. | 2018-05-17 |
Quinolinone Five-membered Heterocyclic Compounds As Mutant-isocitrate Dehydrogenase Inhibitors App 20180118732 - Lin; Jian ;   et al. | 2018-05-03 |
Pyridinyl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20180086733 - Lin; Jian ;   et al. | 2018-03-29 |
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 9,834,539 - Lin , et al. December 5, 2 | 2017-12-05 |
Quinolinone pyrimidines compositions as mutant-isocitrate dehydrogenase inhibitors Grant 9,815,817 - Lin , et al. November 14, 2 | 2017-11-14 |
Pyridinyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 9,771,349 - Lin , et al. September 26, 2 | 2017-09-26 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20170174658 - LIN; Jian ;   et al. | 2017-06-22 |
Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors Grant 9,624,175 - Lin , et al. April 18, 2 | 2017-04-18 |
Quinolinone five-membered heterocyclic compounds as mutant-isocitrate dehydrogenase inhibitors Grant 9,624,216 - Lin , et al. April 18, 2 | 2017-04-18 |
Fused-bicyclic Aryl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20160311774 - Lin; Jian ;   et al. | 2016-10-27 |
Quinolinone Five-membered Heterocyclic Compounds As Mutant-isocitrate Dehydrogenase Inhibitors App 20160311818 - Lin; Jian ;   et al. | 2016-10-27 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20160083349 - Lin; Jian ;   et al. | 2016-03-24 |
Pyridinyl Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20160083367 - Lin; Jian ;   et al. | 2016-03-24 |
Pyridin-2(1h)-one Quinolinone Derivatives As Mutant-isocitrate Dehydrogenase Inhibitors App 20160083366 - Lin; Jian ;   et al. | 2016-03-24 |
Quinolinone Pyrimidines Compositions As Mutant-isocitrate Dehydrogenase Inhibitors App 20160083365 - Lin; Jian ;   et al. | 2016-03-24 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,973,044 - Konradi , et al. July 5, 2 | 2011-07-05 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,968,547 - Konradi , et al. June 28, 2 | 2011-06-28 |
Alpha amino acid derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 Grant 7,745,454 - Konradi , et al. June 29, 2 | 2010-06-29 |
Heteroaryl, Heterocyclic And Aryl Compounds Which Inhibit Leukocyte Adhesion Mediated By Vla-4 App 20100160341 - Konradi; Andrei W. ;   et al. | 2010-06-24 |
Heteroaryl, Heterocyclic And Aryl Compounds Which Inhibit Leukocyte Adhesion Mediated By Vla-4 App 20100160343 - Konradi; Andrei W. ;   et al. | 2010-06-24 |
Substituted Thiophenes And Uses Thereof App 20090054396 - Ashwell; Susan ;   et al. | 2009-02-26 |
Substitute thiophenes and uses thereof Grant 7,423,061 - Ashwell , et al. September 9, 2 | 2008-09-09 |
3-(heteroaryl)alanine Derivatives-inhibitors Of Leukocyte Adhesion Mediated By Vla-4 App 20080182850 - Konradi; Andrei W. ;   et al. | 2008-07-31 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,378,529 - Konradi , et al. May 27, 2 | 2008-05-27 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,320,960 - Thorsett , et al. January 22, 2 | 2008-01-22 |
Phenylalanine derivatives as alpha 4 integrin inhibitors Grant 7,291,645 - Konradi , et al. November 6, 2 | 2007-11-06 |
Novel fused triazolones and the uses thereof App 20070149560 - Ashwell; Susan ;   et al. | 2007-06-28 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 7,229,970 - Thorsett , et al. June 12, 2 | 2007-06-12 |
Beta-amino acid derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 Grant 7,223,762 - Konradi , et al. May 29, 2 | 2007-05-29 |
Thiophene derivatives as chk 1 inhibitors App 20070010556 - Ashwell; Susan ;   et al. | 2007-01-11 |
Substitute thiophenes and uses therof App 20060281666 - Ashwell; Susan ;   et al. | 2006-12-14 |
Heteroaryl-.beta.-alanine derivatives as alpha 4 integrin inhibitors Grant 7,015,216 - Konradi , et al. March 21, 2 | 2006-03-21 |
Compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20050261293 - Konradi, Andrei W. ;   et al. | 2005-11-24 |
Beta-amino acid derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 Grant 6,953,802 - Konradi , et al. October 11, 2 | 2005-10-11 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20050222119 - Thorsett, Eugene D. ;   et al. | 2005-10-06 |
Compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,949,570 - Ashwell , et al. September 27, 2 | 2005-09-27 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20050203093 - Konradi, Andrei W. ;   et al. | 2005-09-15 |
Beta-amino acid derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 App 20050192280 - Konradi, Andrei W. ;   et al. | 2005-09-01 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,911,439 - Konradi , et al. June 28, 2 | 2005-06-28 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,900,179 - Thorsett , et al. May 31, 2 | 2005-05-31 |
Alpha amino acid derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 App 20050085459 - Konradi, Andrei W. ;   et al. | 2005-04-21 |
3-(heteroaryl) alanine derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 App 20040266763 - Konradi, Andrei W. ;   et al. | 2004-12-30 |
Alpha amino acid derivatives--inhibitors of leukocyte adhesion mediated by VLA-4 Grant 6,803,370 - Konradi , et al. October 12, 2 | 2004-10-12 |
3-(heteroaryl) alanine derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 Grant 6,794,506 - Konradi , et al. September 21, 2 | 2004-09-21 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20040147512 - Konradi, Andrei W. ;   et al. | 2004-07-29 |
Phenylalanine derivatives as alpha 4 integrin inhibitors App 20040127486 - Konradi, Andrei W. ;   et al. | 2004-07-01 |
Phenylalanine derivatives as alpha 4 integrin inhibitors Grant 6,689,781 - Konradi , et al. February 10, 2 | 2004-02-10 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20040014677 - Thorsett, Eugene D. ;   et al. | 2004-01-22 |
Compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20030144328 - Konradi, Andrei W. ;   et al. | 2003-07-31 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated byVLA-4 App 20030139402 - Konradi, Andrei W. ;   et al. | 2003-07-24 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20030125324 - Konradi, Andrei W. ;   et al. | 2003-07-03 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,525,026 - Thorsett , et al. February 25, 2 | 2003-02-25 |
Compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20030027850 - Ashwell, Susan ;   et al. | 2003-02-06 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20030017993 - Thorsett, Eugene D. ;   et al. | 2003-01-23 |
Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 App 20020193312 - Thorsett, Eugene D. ;   et al. | 2002-12-19 |
Substituted phenylalanine type compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,492,421 - Thorsett , et al. December 10, 2 | 2002-12-10 |
Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,492,372 - Konradi , et al. December 10, 2 | 2002-12-10 |
Compounds which inhibit leukocyte adhesion mediated by VLA-4 Grant 6,436,904 - Ashwell , et al. August 20, 2 | 2002-08-20 |
Heteroaryl-beta-alanine derivatives as alpha 4 integrin inhibitors App 20020086882 - Konradi, Andrei W. ;   et al. | 2002-07-04 |
Beta-amino acid derivatives--inhibitors of leukocyte adhesion mediated by VLA-4 App 20020058664 - Konradi, Andrei W. ;   et al. | 2002-05-16 |
Phenylalanine derivatives as alpha 4 integrin inhibitors App 20020055509 - Konradi, Andrei W. ;   et al. | 2002-05-09 |
3-(Heteroaryal) alanine derivatives-inhibitors of leukocyte adhesion mediated by VLA-4 App 20020052375 - Konradi, Andrei W. ;   et al. | 2002-05-02 |
Alpha amino acid derivatives--inhibitors of leukocyte adhesion mediated by VLA-4 App 20020052470 - Konradi, Andrei W. ;   et al. | 2002-05-02 |