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METABOLITES OF THE JANUS KINASE INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYL- PROPANENITR App 20200038404 - Rodgers; James D. ;   et al. | 2020-02-06 |
Metabolites of the janus kinase inhibitor (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentyl- propanenitrile Grant 10,463,667 - Rodgers , et al. No | 2019-11-05 |
METABOLITES OF THE JANUS KINASE INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYL- PROPANENITRILE App 20170326144 - Rodgers; James D. ;   et al. | 2017-11-16 |
Hydroxyl, keto, and glucuronide derivatives of 3-(4-(7H-pyrrolo[2,3-D]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylprop- anenitrile Grant 9,512,161 - Rodgers , et al. December 6, 2 | 2016-12-06 |
Cyclohexyl azetidine derivatives as JAK inhibitors Grant 9,359,358 - Rodgers , et al. June 7, 2 | 2016-06-07 |
N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors Grant 9,334,274 - Rodgers , et al. May 10, 2 | 2016-05-10 |
METABOLITES OF THE JANUS KINASE INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYL- PROPANENITRILE App 20150164900 - Rodgers; James D. ;   et al. | 2015-06-18 |
HYDROXYL, KETO, AND GLUCURONIDE DERIVATIVES OF 3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROP- ANENITRILE App 20140378400 - Rodgers; James D. ;   et al. | 2014-12-25 |
Metabolites of the janus kinase inhibitor (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentyl- propanenitrile Grant 8,889,697 - Rodgers , et al. November 18, 2 | 2014-11-18 |
Substituted heterocycles as janus kinase inhibitors Grant 8,841,318 - Arvanitis , et al. September 23, 2 | 2014-09-23 |
Azepine inhibitors of janus kinases Grant 8,835,423 - Arvanitis , et al. September 16, 2 | 2014-09-16 |
N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-d]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20140221379 - Rodgers; James D ;   et al. | 2014-08-07 |
Hydroxyl, keto, and glucuronide derivatives of 3-(4-(7H pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitril- e Grant 8,748,401 - Rodgers , et al. June 10, 2 | 2014-06-10 |
N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors Grant 8,716,303 - Rodgers , et al. May 6, 2 | 2014-05-06 |
Azepine Inhibitors Of Janus Kinases App 20140031344 - Arvanitis; Argyrios G. ;   et al. | 2014-01-30 |
Heteroaryl Substituted Pyrrolo[2,3-B] Pyridines And Pyrrolo[2,3-B] Pyrimidines As Janus Kinase Inhibitors App 20140005210 - Rodgers; James D. ;   et al. | 2014-01-02 |
HYDROXYL, KETO, AND GLUCURONIDE DERIVATIVES OF 3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROP- ANENITRILE App 20130345157 - Rodgers; James D. ;   et al. | 2013-12-26 |
Azepine inhibitors of Janus kinases Grant 8,563,541 - Arvanitis , et al. October 22, 2 | 2013-10-22 |
Substituted Heterocycles As Janus Kinase Inhibitors App 20130274257 - Arvanitis; Argyrios G. ;   et al. | 2013-10-17 |
Substituted heterocycles as Janus kinase inhibitors Grant 8,513,270 - Arvanitis , et al. August 20, 2 | 2013-08-20 |
Hydroxyl, keto, and glucuronide derivatives of 3-(4-(7H-pyrrolo[2,3-d] pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile Grant 8,486,902 - Rodgers , et al. July 16, 2 | 2013-07-16 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20130137681 - Rodgers; James D. ;   et al. | 2013-05-30 |
Pyrazolyl substituted pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors Grant 8,415,362 - Rodgers , et al. April 9, 2 | 2013-04-09 |
Cyclohexyl Azetidine Derivatives as JAK Inhibitors App 20130045963 - Rodgers; James D. ;   et al. | 2013-02-21 |
Azepine Inhibitors Of Janus Kinases App 20120329782 - Arvanitis; Argyrios G. ;   et al. | 2012-12-27 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20110224157 - Rodgers; James D. ;   et al. | 2011-09-15 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20110223210 - Rodgers; James D. ;   et al. | 2011-09-15 |
HYDROXYL, KETO, AND GLUCURONIDE DERIVATIVES OF 3-(4-(7H-PYRROLO[2,3-d] PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROPANENITRILE App 20110086810 - RODGERS; James D. ;   et al. | 2011-04-14 |
METABOLITES OF THE JANUS KINASE INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYL- PROPANENITRILE App 20110082159 - RODGERS; James D. ;   et al. | 2011-04-07 |
N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-d]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20100298334 - Rodgers; James D. ;   et al. | 2010-11-25 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20100022522 - Rodgers; James D. ;   et al. | 2010-01-28 |
Tetracyclic Inhibitors Of Janus Kinases App 20090215766 - Rodgers; James D. ;   et al. | 2009-08-27 |
Azepine Inhibitors Of Janus Kinases App 20090197869 - Arvanitis; Argyrios G. ;   et al. | 2009-08-06 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS App 20090181959 - Rodgers; James D. ;   et al. | 2009-07-16 |
METABOLITES OF THE JANUS KINASE INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYL- PROPANENITRILE App 20080312258 - Rodgers; James D. ;   et al. | 2008-12-18 |
Substituted Heterocycles As Janus Kinase Inhibitors App 20080188500 - Arvanitis; Argyrios G. ;   et al. | 2008-08-07 |
Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands Grant 7,319,100 - Arvanitis , et al. January 15, 2 | 2008-01-15 |
Substituted Pyrazinones, Pyridines And Pyrimidines As Corticotropin Releasing Factor Ligands App 20070155740 - Arvanitis; Argyrios G. ;   et al. | 2007-07-05 |
Azepine inhibitors of Janus kinases App 20070149506 - Arvanitis; Argyrios G. ;   et al. | 2007-06-28 |
Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as janus kinase inhibitors App 20070135461 - Rodgers; James D. ;   et al. | 2007-06-14 |
Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands Grant 7,205,306 - Arvanitis , et al. April 17, 2 | 2007-04-17 |
Pyrimidine derivatives as corticotropin releasing factor inhibitors Grant 7,112,585 - Hartz , et al. September 26, 2 | 2006-09-26 |
Pyridinyl derivatives for the treatment of depression Grant 7,030,145 - Hartz , et al. April 18, 2 | 2006-04-18 |
Pyrimidine derivatives as corticotropin releasing factor inhibitors App 20040229891 - Hartz, Richard A. ;   et al. | 2004-11-18 |
Pyridinyl derivatives for the treatment of depression App 20040209917 - Hartz, Richard A. ;   et al. | 2004-10-21 |
Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands App 20030171380 - Arvanitis, Argyrios G. ;   et al. | 2003-09-11 |