Patent | Date |
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Process for the preparation of 7-(4,7-diazaspiro[2.5]octan-7-yl)-2-(2,8-dimethylimidazo [1,2-B]pyridazin-6-yl)pyrido[1,2-a]pyrimidin-4-one derivatives Grant 11,390,632 - Adam , et al. July 19, 2 | 2022-07-19 |
Synthesis Of Trans-8-chloro-5-methyl-1 -[4-(pyridin-2-yloxy)-cyclohexyl]-5,6-dihydro-4h-2,3,5,10b-tetraaza-benzo- [e]azulene And Crytalline Forms Thereof App 20210284648 - Rothenhaeusler; Benno ;   et al. | 2021-09-16 |
Synthesis of trans-8-chloro-5-methyl-1-[4-(pyridin-2-yloxy)-cyclohexyl]-5,6-dihydro-4H- -2,3,5,10B-tetraaza-benzo[e]azulene and crytalline forms thereof Grant 11,040,977 - Rothenhaeusler , et al. June 22, 2 | 2021-06-22 |
Process For The Preparation Of 7-(4,7-diazaspiro[2.5]octan-7-yl)-2-(2,8-dimethylimidazo[1,2-b]pyridazin-- 6-yl)pyrido[1,2-a]pyri App 20200216472 - Adam; Jean-Michel ;   et al. | 2020-07-09 |
Process For The Preparation Of Hu-910 And Crystalline Structure Thereof App 20190315669 - ADAM; Jean-Michel ;   et al. | 2019-10-17 |
Synthesis Of Trans-8-chloro-5-methyl-1 -[4-(pyridin-2-yloxy)-cyclohexyl]-5,6-dihydro-4h-2,3,5,10b-tetraaza-benzo- [e]azulene And App 20190194210 - Rothenhaeusler; Benno ;   et al. | 2019-06-27 |
Synthesis of trans-8-chloro-5-methyl-1-[4-(pyridin-2-yloxy)-cyclohexyl]-5,6-dihydro-4H- -2,3,5,10B-tetraaza-benzo[E]azulene and crytalline forms thereof Grant 10,246,460 - Rothenhaeusler , et al. | 2019-04-02 |
(3,4-dichloro-phenyl)-((S)-3-propyl-pyrrolidin-3-yl)-methanone hydrochloride and manufacturing processes Grant 9,527,810 - Adam , et al. December 27, 2 | 2016-12-27 |
Synthesis Of Trans-8-chloro-5-methyl-1 -[4-(pyridin-2-yloxy)-cyclohexyl]-5,6-dihydro-4h-2,3,5,10b-tetraaza-benzo- [e]azulene And Crytalline Forms Thereof App 20160280712 - Rothenhaeusler; Benno ;   et al. | 2016-09-29 |
[1,2,3]triazolo[4,5-D]pyrimidine derivatives Grant 9,056,866 - Adam , et al. June 16, 2 | 2015-06-16 |
Process For The Preparation Of Pyrido [2,1-A] Isoquinoline Derivatives Comprising Optical Resolution Of An Enamine App 20150126743 - Abrecht; Stefan ;   et al. | 2015-05-07 |
(3,4-dichloro-phenyl)-((s)-3-propyl-pyrrolidin-3-yl)-methanone Hydrochloride And Manufacturing Processes App 20150045408 - Adam; Jean-Michel ;   et al. | 2015-02-12 |
Novel [1,2,3]triazolo[4,5-d]pyrimidine Derivatives App 20140288046 - Adam; Jean-Michel ;   et al. | 2014-09-25 |
Synthesis of Cyclosporin Analogs App 20140288266 - Naicker; Selvaraj A. ;   et al. | 2014-09-25 |
[1,2,3]triazolo[4,5-D]pyrimidine derivatives Grant 8,741,906 - Adam , et al. June 3, 2 | 2014-06-03 |
Process For The Preparation Of Pyrido [2,1-a] Isoquinoline Derivatives Comprising Optical Resolution Of An Enamine App 20130338366 - Abrecht; Stefan ;   et al. | 2013-12-19 |
Novel [1,2,3]triazolo[4,5-d]pyrimidine Derivatives App 20130116236 - Adam; Jean-Michel ;   et al. | 2013-05-09 |
Process for the preparation of pyrido[2,1-a] isoquinoline derivatives Grant 8,420,818 - Abrecht , et al. April 16, 2 | 2013-04-16 |
Process For The Preparation Of Pyrido [2,1-a] Isoquinoline Derivatives Comprising Optical Resolution Of An Enamine App 20130018191 - Abrecht; Stefan ;   et al. | 2013-01-17 |
Heteroaryl carboxamide derivatives Grant 8,227,613 - Adam , et al. July 24, 2 | 2012-07-24 |
Heterocyclyl compounds Grant 8,138,175 - Adam , et al. March 20, 2 | 2012-03-20 |
PROCESS FOR THE PREPARATION OF PYRIDO[2,1-a] ISOQUINOLINE DERIVATIVES App 20120035368 - Abrecht; Stefan ;   et al. | 2012-02-09 |
PROCESS FOR THE PREPARATION OF PYRIDO [2,1-a] ISOQUINOLINE DERIVATIVES COMPRISING OPTICAL RESOLUTION OF AN ENAMINE App 20120022260 - Abrecht; Stefan ;   et al. | 2012-01-26 |
Synthesis Of Cyclosporin Analogs App 20110092669 - Naicker; Selvaraj A. ;   et al. | 2011-04-21 |
Processes for the manufacture of a pyrrolidine-3,4-dicarboxamide derivative Grant 7,872,141 - Adam , et al. January 18, 2 | 2011-01-18 |
Synthesis of Cyclosporin Analogs App 20100062976 - Naicker; Selvaraj A. ;   et al. | 2010-03-11 |
Novel Heterocyclyl Compounds App 20100022518 - Adam; Jean-Michel ;   et al. | 2010-01-28 |
Novel Heteroaryl Carboxamide Derivatives App 20090318467 - Adam; Jean-Michel ;   et al. | 2009-12-24 |
Process for the preparation of (S)-4-fluoromethyl-dihydro-furan-2-one useful in the preparation of the DPP-IV inhibitor (S)-1 ((2S,3S,11bS)-2-amino-9,10-dimethoxy-1,3,4,6,7, 11b-hexahydro-2H-pyrido[2,1-a] isoquinolin-3-yl)-4-fluoromethyl-pyrrolidin-2-one Grant 7,619,101 - Abrecht , et al. November 17, 2 | 2009-11-17 |
Solid Forms Of A Pyrrolidine-3,4-dicarboxamide Derivative App 20090215826 - Adam; Jean-Michel ;   et al. | 2009-08-27 |
PROCESS FOR THE PREPARATION OF PYRIDO[2,1-a] ISOQUINOLINE DERIVATIVES App 20090163718 - Abrecht; Stefan ;   et al. | 2009-06-25 |
Processes For The Manufacture Of A Pyrrolidine-3,4-dicarboxamide Derivative App 20080214826 - Adam; Jean-Michel ;   et al. | 2008-09-04 |
PROCESS FOR THE PREPARATION OF PYRIDO [2,1-a] ISOQUINOLINE DERIVATIVES COMPRISING OPTICAL RESOLUTION OF AN ENAMINE App 20080071087 - Abrecht; Stefan ;   et al. | 2008-03-20 |
Synthesis of cyclosporin analogs App 20070087963 - Naicker; Selvaraj A. ;   et al. | 2007-04-19 |
Process for the preparation of (S)-4-fluoromethyl-dihydro-furan-2-one useful in the preparation of the DPP-IV inhibitor (S)-1 ((2S,3S,11bS)-2-amino-9,10-dimethoxy-1,3,4,6,7, 11b-hexahydro-2h-pyrido[2,1-a] isoquinolin-3-yl)-4-fluoromethyl-pyrrolidin-2-one App 20060270853 - Abrecht; Stefan ;   et al. | 2006-11-30 |
Synthesis of cyclosporin analogs Grant 7,141,648 - Naicker , et al. November 28, 2 | 2006-11-28 |
Process for preparation of cyclosporin A analogs App 20040220091 - Adam, Jean-Michel ;   et al. | 2004-11-04 |
Synthesis of cyclosporin analogs App 20030212249 - Naicker, Selvaraj A. ;   et al. | 2003-11-13 |